Peringatan Keamanan

Acute oral toxicity (LD50) in mouse: 50.1 mg/kg

Camptothecin

DB04690

small molecule experimental

Deskripsi

Camptothecin is an alkaloid isolated from the stem wood of the Chinese tree, Camptotheca acuminata. This compound selectively inhibits the nuclear enzyme DNA topoisomerase, type I. Several semisynthetic analogs of camptothecin have demonstrated antitumor activity.

Struktur Molekul 2D

Berat 348.352
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

157 Data
Pravastatin Pravastatin may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Diethylstilbestrol Diethylstilbestrol may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Estradiol Estradiol may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Sulfasalazine Sulfasalazine may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Novobiocin Novobiocin may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Hesperetin Hesperetin may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Rabeprazole Rabeprazole may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Dexamethasone Dexamethasone may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Dasatinib Dasatinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Topiroxostat Topiroxostat may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Daidzin Daidzin may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Fusidic acid Fusidic acid may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Naringenin Naringenin may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Vandetanib Vandetanib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Eltrombopag Eltrombopag may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Safinamide Safinamide may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Vismodegib Vismodegib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Teriflunomide Teriflunomide may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Dabrafenib Dabrafenib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Cannabidiol Cannabidiol may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Palbociclib Palbociclib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Dasabuvir Dasabuvir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Dacomitinib Dacomitinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Glasdegib Glasdegib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Fostamatinib Fostamatinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Gilteritinib Gilteritinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Brigatinib Brigatinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Estradiol acetate Estradiol acetate may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Estradiol benzoate Estradiol benzoate may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Estradiol cypionate Estradiol cypionate may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Estradiol dienanthate Estradiol dienanthate may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Estradiol valerate Estradiol valerate may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Nabiximols Nabiximols may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Fedratinib Fedratinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Istradefylline Istradefylline may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Caffeine Caffeine may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Vemurafenib Vemurafenib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Isavuconazole Isavuconazole may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Cyclosporine Cyclosporine may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Pantoprazole Pantoprazole may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Nelfinavir Nelfinavir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Gefitinib Gefitinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Beclomethasone dipropionate Beclomethasone dipropionate may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Progesterone Progesterone may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Lansoprazole Lansoprazole may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Ritonavir Ritonavir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Erlotinib Erlotinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Imatinib Imatinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Buprenorphine Buprenorphine may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Telmisartan Telmisartan may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Saquinavir Saquinavir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Sunitinib Sunitinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Genistein Genistein may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Quercetin Quercetin may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Taurocholic acid Taurocholic acid may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Nilotinib Nilotinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Elacridar Elacridar may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Dovitinib Dovitinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Simeprevir Simeprevir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Rilpivirine Rilpivirine may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Regorafenib Regorafenib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Ponatinib Ponatinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Afatinib Afatinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Cobicistat Cobicistat may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Daclatasvir Daclatasvir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Rolapitant Rolapitant may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Paritaprevir Paritaprevir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Alectinib Alectinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Venetoclax Venetoclax may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Velpatasvir Velpatasvir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Abemaciclib Abemaciclib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Voxilaprevir Voxilaprevir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Rucaparib Rucaparib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Enasidenib Enasidenib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Pibrentasvir Pibrentasvir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Glecaprevir Glecaprevir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Ripretinib Ripretinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Fostemsavir Fostemsavir may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Pralsetinib Pralsetinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Clofazimine Clofazimine may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Dexamethasone acetate Dexamethasone acetate may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Avanafil Avanafil may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Tepotinib Tepotinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Tivozanib Tivozanib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Osimertinib Osimertinib may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Belumosudil Belumosudil may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Venlafaxine Venlafaxine may increase the excretion rate of Camptothecin which could result in a lower serum level and potentially a reduction in efficacy.
Cholesterol Cholesterol may increase the excretion rate of Camptothecin which could result in a lower serum level and potentially a reduction in efficacy.
Apalutamide The serum concentration of Camptothecin can be decreased when it is combined with Apalutamide.
Lasmiditan The serum concentration of Camptothecin can be increased when it is combined with Lasmiditan.
Darolutamide The serum concentration of Camptothecin can be increased when it is combined with Darolutamide.
Tafamidis The serum concentration of Camptothecin can be increased when it is combined with Tafamidis.
Capmatinib The serum concentration of Camptothecin can be increased when it is combined with Capmatinib.
Febuxostat The excretion of Camptothecin can be decreased when combined with Febuxostat.
Darbepoetin alfa The risk or severity of Thrombosis can be increased when Darbepoetin alfa is combined with Camptothecin.
Erythropoietin The risk or severity of Thrombosis can be increased when Erythropoietin is combined with Camptothecin.
Peginesatide The risk or severity of Thrombosis can be increased when Peginesatide is combined with Camptothecin.
Methoxy polyethylene glycol-epoetin beta The risk or severity of Thrombosis can be increased when Methoxy polyethylene glycol-epoetin beta is combined with Camptothecin.
Itraconazole Itraconazole may decrease the excretion rate of Camptothecin which could result in a higher serum level.
Ledipasvir Ledipasvir may decrease the excretion rate of Camptothecin which could result in a higher serum level.

Target Protein

DNA topoisomerase 1 TOP1

Referensi & Sumber

Synthesis reference: Tadashi Miyasaka, Seigo Sawada, Kenichiro Nokata, Masahiko Mutai, "Photochemical process for preparing camptothecin derivatives." U.S. Patent US4545880, issued March, 1976.
Artikel (PubMed)
  • PMID: 9213622
    Wall ME, Wani MC: Camptothecin and taxol: from discovery to clinic. J Ethnopharmacol. 1996 Apr;51(1-3):239-53; discussion 253-4.
  • PMID: 5357525
    Kepler JA, Wani MC, McNaull JN, Wall ME, Levine SG: Plant antitumor agents. IV. An approach toward the synthesis of camptothecin. J Org Chem. 1969 Dec;34(12):3853-8.

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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