Peringatan Keamanan

ORAL (LD50): Acute: >2000 mg/kg Rat.

Estriol

DB04573

small molecule approved investigational vet_approved

Deskripsi

A hydroxylated metabolite of estradiol or estrone that has a hydroxyl group at C3-beta, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen. During pregnancy, large amount of estriol is produced by the placenta. Isomers with inversion of the hydroxyl group or groups are called epiestriol. Though estriol is used as part of the primarily North American phenomenon of bioidentical hormone replacement therapy, it is not approved for use by the FDA or Health Canada. It is however available in the United States by prescription filled only by compounding pharmacies. It has also been approved and marketed throughout Europe and Asia for approximately 40 years for the treatment of post-menopausal hot flashes.

Struktur Molekul 2D

Berat 288.3814
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

562 Data
Prasterone The risk or severity of adverse effects can be increased when Prasterone is combined with Estriol.
Exemestane The therapeutic efficacy of Exemestane can be decreased when used in combination with Estriol.
Hyaluronidase (ovine) The therapeutic efficacy of Hyaluronidase (ovine) can be decreased when used in combination with Estriol.
Hyaluronidase (human recombinant) The therapeutic efficacy of Hyaluronidase (human recombinant) can be decreased when used in combination with Estriol.
Hyaluronidase The therapeutic efficacy of Hyaluronidase can be decreased when used in combination with Estriol.
Lenalidomide Estriol may increase the thrombogenic activities of Lenalidomide.
Ospemifene The risk or severity of adverse effects can be increased when Estriol is combined with Ospemifene.
Ropinirole Estriol may increase the excretion rate of Ropinirole which could result in a lower serum level and potentially a reduction in efficacy.
Thalidomide Estriol may increase the thrombogenic activities of Thalidomide.
Cetuximab Estriol may increase the thrombogenic activities of Cetuximab.
Human immunoglobulin G Estriol may increase the thrombogenic activities of Human immunoglobulin G.
Omalizumab Estriol may increase the thrombogenic activities of Omalizumab.
Adalimumab Estriol may increase the thrombogenic activities of Adalimumab.
Gemtuzumab ozogamicin Estriol may increase the thrombogenic activities of Gemtuzumab ozogamicin.
Indium In-111 satumomab pendetide Estriol may increase the thrombogenic activities of Indium In-111 satumomab pendetide.
Infliximab Estriol may increase the thrombogenic activities of Infliximab.
Trastuzumab Estriol may increase the thrombogenic activities of Trastuzumab.
Rituximab Estriol may increase the thrombogenic activities of Rituximab.
Basiliximab Estriol may increase the thrombogenic activities of Basiliximab.
Muromonab Estriol may increase the thrombogenic activities of Muromonab.
Digoxin Immune Fab (Ovine) Estriol may increase the thrombogenic activities of Digoxin Immune Fab (Ovine).
Ibritumomab tiuxetan Estriol may increase the thrombogenic activities of Ibritumomab tiuxetan.
Tositumomab Estriol may increase the thrombogenic activities of Tositumomab.
Alemtuzumab Estriol may increase the thrombogenic activities of Alemtuzumab.
Capromab pendetide Estriol may increase the thrombogenic activities of Capromab pendetide.
Efalizumab Estriol may increase the thrombogenic activities of Efalizumab.
Antithymocyte immunoglobulin (rabbit) Estriol may increase the thrombogenic activities of Antithymocyte immunoglobulin (rabbit).
Natalizumab Estriol may increase the thrombogenic activities of Natalizumab.
Palivizumab Estriol may increase the thrombogenic activities of Palivizumab.
Daclizumab Estriol may increase the thrombogenic activities of Daclizumab.
Bevacizumab Estriol may increase the thrombogenic activities of Bevacizumab.
Technetium Tc-99m arcitumomab Estriol may increase the thrombogenic activities of Technetium Tc-99m arcitumomab.
Eculizumab Estriol may increase the thrombogenic activities of Eculizumab.
Panitumumab Estriol may increase the thrombogenic activities of Panitumumab.
Ranibizumab Estriol may increase the thrombogenic activities of Ranibizumab.
Galiximab Estriol may increase the thrombogenic activities of Galiximab.
Pexelizumab Estriol may increase the thrombogenic activities of Pexelizumab.
Afelimomab Estriol may increase the thrombogenic activities of Afelimomab.
Epratuzumab Estriol may increase the thrombogenic activities of Epratuzumab.
Bectumomab Estriol may increase the thrombogenic activities of Bectumomab.
Oregovomab Estriol may increase the thrombogenic activities of Oregovomab.
IGN311 Estriol may increase the thrombogenic activities of IGN311.
Adecatumumab Estriol may increase the thrombogenic activities of Adecatumumab.
Labetuzumab Estriol may increase the thrombogenic activities of Labetuzumab.
Matuzumab Estriol may increase the thrombogenic activities of Matuzumab.
Fontolizumab Estriol may increase the thrombogenic activities of Fontolizumab.
Bavituximab Estriol may increase the thrombogenic activities of Bavituximab.
CR002 Estriol may increase the thrombogenic activities of CR002.
Rozrolimupab Estriol may increase the thrombogenic activities of Rozrolimupab.
Girentuximab Estriol may increase the thrombogenic activities of Girentuximab.
Obiltoxaximab Estriol may increase the thrombogenic activities of Obiltoxaximab.
XTL-001 Estriol may increase the thrombogenic activities of XTL-001.
NAV 1800 Estriol may increase the thrombogenic activities of NAV 1800.
Briakinumab Estriol may increase the thrombogenic activities of Briakinumab.
Otelixizumab Estriol may increase the thrombogenic activities of Otelixizumab.
AMG 108 Estriol may increase the thrombogenic activities of AMG 108.
Iratumumab Estriol may increase the thrombogenic activities of Iratumumab.
Enokizumab Estriol may increase the thrombogenic activities of Enokizumab.
Ramucirumab Estriol may increase the thrombogenic activities of Ramucirumab.
Farletuzumab Estriol may increase the thrombogenic activities of Farletuzumab.
Veltuzumab Estriol may increase the thrombogenic activities of Veltuzumab.
Ustekinumab Estriol may increase the thrombogenic activities of Ustekinumab.
PRO-542 Estriol may increase the thrombogenic activities of PRO-542.
TNX-901 Estriol may increase the thrombogenic activities of TNX-901.
RI 624 Estriol may increase the thrombogenic activities of RI 624.
Stamulumab Estriol may increase the thrombogenic activities of MYO-029.
CT-011 Estriol may increase the thrombogenic activities of CT-011.
Leronlimab Estriol may increase the thrombogenic activities of Leronlimab.
Glembatumumab vedotin Estriol may increase the thrombogenic activities of Glembatumumab vedotin.
Olaratumab Estriol may increase the thrombogenic activities of Olaratumab.
IPH 2101 Estriol may increase the thrombogenic activities of IPH 2101.
TB-402 Estriol may increase the thrombogenic activities of TB-402.
Caplacizumab Estriol may increase the thrombogenic activities of Caplacizumab.
IMC-1C11 Estriol may increase the thrombogenic activities of IMC-1C11.
Eldelumab Estriol may increase the thrombogenic activities of Eldelumab.
Lumiliximab Estriol may increase the thrombogenic activities of Lumiliximab.
Canakinumab Estriol may increase the thrombogenic activities of Canakinumab.
Ipilimumab Estriol may increase the thrombogenic activities of Ipilimumab.
Nimotuzumab Estriol may increase the thrombogenic activities of Nimotuzumab.
Clenoliximab Estriol may increase the thrombogenic activities of Clenoliximab.
Tocilizumab Estriol may increase the thrombogenic activities of Tocilizumab.
BIIB015 Estriol may increase the thrombogenic activities of BIIB015.
Sonepcizumab Estriol may increase the thrombogenic activities of Sonepcizumab.
Motavizumab Estriol may increase the thrombogenic activities of Motavizumab.
Elotuzumab Estriol may increase the thrombogenic activities of Elotuzumab.
AVE9633 Estriol may increase the thrombogenic activities of AVE9633.
Carotuximab Estriol may increase the thrombogenic activities of Carotuximab.
XmAb 2513 Estriol may increase the thrombogenic activities of XmAb 2513.
Coltuximab ravtansine Estriol may increase the thrombogenic activities of Coltuximab ravtansine.
Lucatumumab Estriol may increase the thrombogenic activities of Lucatumumab.
Pertuzumab Estriol may increase the thrombogenic activities of Pertuzumab.
Siplizumab Estriol may increase the thrombogenic activities of Siplizumab.
Apolizumab Estriol may increase the thrombogenic activities of Apolizumab.
Sibrotuzumab Estriol may increase the thrombogenic activities of Sibrotuzumab.
Bivatuzumab Estriol may increase the thrombogenic activities of Bivatuzumab.
Lerdelimumab Estriol may increase the thrombogenic activities of Lerdelimumab.
Lexatumumab Estriol may increase the thrombogenic activities of Lexatumumab.
Reslizumab Estriol may increase the thrombogenic activities of Reslizumab.
Teplizumab Estriol may increase the thrombogenic activities of Teplizumab.
Catumaxomab Estriol may increase the thrombogenic activities of Catumaxomab.

Target Protein

Estrogen receptor ESR1
Estrogen receptor beta ESR2
Sex hormone-binding globulin SHBG

Referensi & Sumber

Synthesis reference: James V. Freeman, Gary M. Johnson, "Synthesis of 6.alpha.-functionalized estriol haptens and protein conjugates thereof." U.S. Patent US5902888, issued June, 1973.
Artikel (PubMed)
  • PMID: 14634144
    Soldan SS, Alvarez Retuerto AI, Sicotte NL, Voskuhl RR: Immune modulation in multiple sclerosis patients treated with the pregnancy hormone estriol. J Immunol. 2003 Dec 1;171(11):6267-74.
Link

Contoh Produk & Brand

Produk: 6 • International brands: 5
Produk
  • Advanced Formula Estro-Life
    Cream • 1.69 mg/1mL • Topical • US • OTC
  • BiEST 2.5 Estrogen Cream
    Cream • - • Transdermal • US • OTC
  • BiEST 2.5 Estrogen Cream (Lavender scented)
    Cream • - • Transdermal • US • OTC
  • BiEST 5.0 Estrogen Cream
    Cream • - • Transdermal • US • OTC
  • Estriol 5.0 Cream
    Cream • 5 mg/85g • Transdermal • US • OTC
  • Estro-Life
    Cream • 1.69 mg/1mL • Topical • US • OTC
International Brands
  • Aacifemine — Organon
  • Colpoestriol — Temis-Lostalo
  • Estriel
  • Ovestin — Merck Sharp & Dohme
  • Synapause E — Organon

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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