Trioxsalen

DB04571

small molecule approved

Deskripsi

Trioxsalen (trimethylpsoralen, trioxysalen or trisoralen) is a furanocoumarin and a psoralen derivative obtained from several plants, mainly Psoralea corylifolia. Like other psoralens it causes photosensitization of the skin. It is administered either topically or orally in conjunction with UV-A (the least damaging form of ultraviolet light) for phototherapy treatment of vitiligo and hand eczema. The photoactivated form produces interstrand linkages in DNA resulting in cell apoptosis. In research it can be conjugated to dyes for confocal microscopy and used to visualize sites of DNA damage.3 The compound is has been explored for development of antisense oligonucleotides that can be cross-linked specifically to a mutant mRNA sequence without affecting normal transcripts differing at even a single base pair.

Struktur Molekul 2D

Berat 228.2433
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Avoid foods high in furanocoumarins. Eating these foods while you are taking trioxsalen may increase your skin's sensitivity to sunlight. Examples include limes, figs, parsley, parsnips, mustard, carrots, and celery.

Interaksi Obat

21 Data
Porfimer sodium Trioxsalen may increase the photosensitizing activities of Porfimer sodium.
Verteporfin Trioxsalen may increase the photosensitizing activities of Verteporfin.
Dexmethylphenidate The serum concentration of the active metabolites of Trioxsalen can be increased when Trioxsalen is used in combination with Dexmethylphenidate.
Glimepiride The therapeutic efficacy of Glimepiride can be increased when used in combination with Trioxsalen.
Acetohexamide The therapeutic efficacy of Acetohexamide can be increased when used in combination with Trioxsalen.
Chlorpropamide The therapeutic efficacy of Chlorpropamide can be increased when used in combination with Trioxsalen.
Tolazamide The therapeutic efficacy of Tolazamide can be increased when used in combination with Trioxsalen.
Glyburide The therapeutic efficacy of Glyburide can be increased when used in combination with Trioxsalen.
Glipizide The therapeutic efficacy of Glipizide can be increased when used in combination with Trioxsalen.
Gliclazide The therapeutic efficacy of Gliclazide can be increased when used in combination with Trioxsalen.
Tolbutamide The therapeutic efficacy of Tolbutamide can be increased when used in combination with Trioxsalen.
Gliquidone The therapeutic efficacy of Gliquidone can be increased when used in combination with Trioxsalen.
Glisoxepide The therapeutic efficacy of Glisoxepide can be increased when used in combination with Trioxsalen.
Glibornuride The therapeutic efficacy of Glibornuride can be increased when used in combination with Trioxsalen.
Carbutamide The therapeutic efficacy of Carbutamide can be increased when used in combination with Trioxsalen.
Metahexamide The therapeutic efficacy of Metahexamide can be increased when used in combination with Trioxsalen.
Tretinoin The risk or severity of adverse effects can be increased when Tretinoin is combined with Trioxsalen.
Padeliporfin Trioxsalen may increase the photosensitizing activities of Padeliporfin.
Lepirudin The risk or severity of bleeding can be increased when Trioxsalen is combined with Lepirudin.
Doxycycline The therapeutic efficacy of Trioxsalen can be increased when used in combination with Doxycycline.
Diazoxide The serum concentration of Trioxsalen can be increased when it is combined with Diazoxide.

Target Protein

DNA

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15611423
    van Coevorden AM, Kamphof WG, van Sonderen E, Bruynzeel DP, Coenraads PJ: Comparison of oral psoralen-UV-A with a portable tanning unit at home vs hospital-administered bath psoralen-UV-A in patients with chronic hand eczema: an open-label randomized controlled trial of efficacy. Arch Dermatol. 2004 Dec;140(12):1463-6.
  • PMID: 17373769
    Thazhathveetil AK, Liu ST, Indig FE, Seidman MM: Psoralen conjugates for visualization of genomic interstrand cross-links localized by laser photoactivation. Bioconjug Chem. 2007 Mar-Apr;18(2):431-7.
  • PMID: 17150768
    Higuchi M, Yamayoshi A, Kobori A, Yamaoka T, Murakami A: Synthesis and properties of photo-reactive antisense oligonucleotides containing 2'-O-psoralen-conjugated adenosine. Nucleic Acids Symp Ser (Oxf). 2005;(49):331-2.

Contoh Produk & Brand

Produk: 1 • International brands: 0
Produk
  • Trisoralen Tab 5mg
    Tablet • 5 mg • Oral • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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