Alvocidib

DB03496

small molecule experimental investigational

Deskripsi

Alvocidib is a synthetic flavonoid based on an extract from an Indian plant for the potential treatment of cancer. It works by inhibiting cyclin-dependent kinases, arresting cell division and causing apoptosis in non-small lung cancer cells.

Struktur Molekul 2D

Berat 401.84
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

191 Data
Nelfinavir The metabolism of Alvocidib can be increased when combined with Nelfinavir.
Phenytoin The metabolism of Alvocidib can be increased when combined with Phenytoin.
Desogestrel The metabolism of Alvocidib can be increased when combined with Desogestrel.
Zidovudine The metabolism of Alvocidib can be increased when combined with Zidovudine.
Ritonavir The metabolism of Alvocidib can be increased when combined with Ritonavir.
Lamotrigine The metabolism of Alvocidib can be increased when combined with Lamotrigine.
Carbamazepine The metabolism of Alvocidib can be increased when combined with Carbamazepine.
Efavirenz The metabolism of Alvocidib can be increased when combined with Efavirenz.
Primidone The metabolism of Alvocidib can be increased when combined with Primidone.
Tipranavir The metabolism of Alvocidib can be increased when combined with Tipranavir.
Ethinylestradiol The metabolism of Alvocidib can be increased when combined with Ethinylestradiol.
Rifampin The metabolism of Alvocidib can be increased when combined with Rifampicin.
Phenobarbital The metabolism of Alvocidib can be increased when combined with Phenobarbital.
Testosterone propionate The metabolism of Alvocidib can be increased when combined with Testosterone propionate.
Cyclosporine Cyclosporine may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Pravastatin Pravastatin may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Pantoprazole Pantoprazole may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Diethylstilbestrol Diethylstilbestrol may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Gefitinib Gefitinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Beclomethasone dipropionate Beclomethasone dipropionate may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Progesterone Progesterone may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Lansoprazole Lansoprazole may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Imatinib Imatinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Estradiol Estradiol may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Sulfasalazine Sulfasalazine may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Buprenorphine Buprenorphine may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Telmisartan Telmisartan may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Novobiocin Novobiocin may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Hesperetin Hesperetin may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Rabeprazole Rabeprazole may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Saquinavir Saquinavir may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Dexamethasone Dexamethasone may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Dasatinib Dasatinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Sunitinib Sunitinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Genistein Genistein may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Topiroxostat Topiroxostat may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Daidzin Daidzin may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Fusidic acid Fusidic acid may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Naringenin Naringenin may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Quercetin Quercetin may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Taurocholic acid Taurocholic acid may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Elacridar Elacridar may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Vandetanib Vandetanib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Dovitinib Dovitinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Simeprevir Simeprevir may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Safinamide Safinamide may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Vismodegib Vismodegib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Rilpivirine Rilpivirine may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Teriflunomide Teriflunomide may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Vemurafenib Vemurafenib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Ponatinib Ponatinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Dabrafenib Dabrafenib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Afatinib Afatinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Cannabidiol Cannabidiol may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Cobicistat Cobicistat may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Palbociclib Palbociclib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Daclatasvir Daclatasvir may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Rolapitant Rolapitant may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Alectinib Alectinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Venetoclax Venetoclax may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Velpatasvir Velpatasvir may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Isavuconazole Isavuconazole may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Glasdegib Glasdegib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Abemaciclib Abemaciclib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Voxilaprevir Voxilaprevir may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Gilteritinib Gilteritinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Brigatinib Brigatinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Estradiol acetate Estradiol acetate may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Estradiol benzoate Estradiol benzoate may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Estradiol cypionate Estradiol cypionate may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Estradiol dienanthate Estradiol dienanthate may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Estradiol valerate Estradiol valerate may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Nabiximols Nabiximols may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Fedratinib Fedratinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Istradefylline Istradefylline may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Caffeine Caffeine may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Ripretinib Ripretinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Fostemsavir Fostemsavir may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Pralsetinib Pralsetinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Clofazimine Clofazimine may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Dexamethasone acetate Dexamethasone acetate may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Avanafil Avanafil may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Tepotinib Tepotinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Tivozanib Tivozanib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Osimertinib Osimertinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Belumosudil Belumosudil may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Venlafaxine Venlafaxine may increase the excretion rate of Alvocidib which could result in a lower serum level and potentially a reduction in efficacy.
Cholesterol Cholesterol may increase the excretion rate of Alvocidib which could result in a lower serum level and potentially a reduction in efficacy.
Apalutamide The serum concentration of Alvocidib can be decreased when it is combined with Apalutamide.
Adenine The metabolism of Alvocidib can be decreased when combined with Adenine.
Indinavir The metabolism of Alvocidib can be decreased when combined with Indinavir.
Valproic acid The metabolism of Alvocidib can be decreased when combined with Valproic acid.
Amitriptyline The metabolism of Alvocidib can be decreased when combined with Amitriptyline.
Indomethacin The metabolism of Alvocidib can be decreased when combined with Indomethacin.
Sorafenib The metabolism of Alvocidib can be decreased when combined with Sorafenib.
Erlotinib Erlotinib may decrease the excretion rate of Alvocidib which could result in a higher serum level.
Flurbiprofen The metabolism of Alvocidib can be decreased when combined with Flurbiprofen.
Propofol The metabolism of Alvocidib can be decreased when combined with Propofol.
Ketoconazole The metabolism of Alvocidib can be decreased when combined with Ketoconazole.
Probenecid The metabolism of Alvocidib can be decreased when combined with Probenecid.

Target Protein

Glycogen phosphorylase, muscle form PYGM
Cyclin-dependent kinase 9 CDK9
Glycogen phosphorylase, brain form PYGB
Glycogen phosphorylase, liver form PYGL
Cyclin-dependent kinase 7 CDK7
Cyclin-dependent kinase 5 CDK5
Cyclin-dependent kinase 1 CDK1
Cyclin-dependent kinase 6 CDK6
Epidermal growth factor receptor EGFR
Cyclin-dependent kinase 4 CDK4
Cyclin-dependent kinase 8 CDK8
Cyclin-dependent kinase 2 CDK2

Referensi & Sumber

Synthesis reference: Kyoung Soon Kim, "Process for the preparation of chiral ketone intermediates useful for the preparation of flavopiridol and analogs." U.S. Patent US5908934, issued March, 1998.

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