Ubenimex

DB03424

small molecule investigational

Deskripsi

Ubenimex (also known as bestatin) is a competitive protease inhibitor. It is an inhibitor of aminopeptidase B, leukotriene A4 hydrolase, aminopeptidase N. It is being studied for use in the treatment of acute myelocytic leukemia.

Struktur Molekul 2D

Berat 308.3728
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

55 Data
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Ubenimex.
BCG vaccine The therapeutic efficacy of BCG vaccine can be decreased when used in combination with Ubenimex.
Typhoid vaccine The therapeutic efficacy of Typhoid vaccine can be decreased when used in combination with Ubenimex.
Dicoumarol The risk or severity of bleeding can be increased when Ubenimex is combined with Dicoumarol.
Phenindione The risk or severity of bleeding can be increased when Ubenimex is combined with Phenindione.
Warfarin The risk or severity of bleeding can be increased when Ubenimex is combined with Warfarin.
Phenprocoumon The risk or severity of bleeding can be increased when Ubenimex is combined with Phenprocoumon.
Acenocoumarol The risk or severity of bleeding can be increased when Ubenimex is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of bleeding can be increased when Ubenimex is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of bleeding can be increased when Ubenimex is combined with Coumarin.
(R)-warfarin The risk or severity of bleeding can be increased when Ubenimex is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of bleeding can be increased when Ubenimex is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of bleeding can be increased when Ubenimex is combined with Fluindione.
Clorindione The risk or severity of bleeding can be increased when Ubenimex is combined with Clorindione.
Diphenadione The risk or severity of bleeding can be increased when Ubenimex is combined with Diphenadione.
Tioclomarol The risk or severity of bleeding can be increased when Ubenimex is combined with Tioclomarol.
(S)-Warfarin The risk or severity of bleeding can be increased when Ubenimex is combined with (S)-Warfarin.
Lactulose The therapeutic efficacy of Lactulose can be decreased when used in combination with Ubenimex.
Vibrio cholerae CVD 103-HgR strain live antigen The therapeutic efficacy of Vibrio cholerae CVD 103-HgR strain live antigen can be decreased when used in combination with Ubenimex.
Estetrol The therapeutic efficacy of Estetrol can be decreased when used in combination with Ubenimex.
Lidocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Lidocaine.
Ropivacaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Ropivacaine.
Bupivacaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Bupivacaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Cinchocaine.
Dyclonine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Dyclonine.
Procaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Procaine.
Prilocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Prilocaine.
Proparacaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Proparacaine.
Meloxicam The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Meloxicam.
Oxybuprocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Oxybuprocaine.
Cocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Cocaine.
Mepivacaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Mepivacaine.
Levobupivacaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Levobupivacaine.
Diphenhydramine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Diphenhydramine.
Benzocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Benzocaine.
Chloroprocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Chloroprocaine.
Phenol The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Phenol.
Tetrodotoxin The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Tetrodotoxin.
Benzyl alcohol The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Benzyl alcohol.
Capsaicin The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Capsaicin.
Etidocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Etidocaine.
Articaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Articaine.
Tetracaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Tetracaine.
Propoxycaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Propoxycaine.
Pramocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Pramocaine.
Butamben The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Butamben.
Butacaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Butacaine.
Oxetacaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Oxetacaine.
Ethyl chloride The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Ethyl chloride.
Butanilicaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Butanilicaine.
Metabutethamine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Metabutethamine.
Quinisocaine The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Quinisocaine.
Cisatracurium Ubenimex may increase the neuromuscular blocking activities of Cisatracurium.
Ambroxol The risk or severity of methemoglobinemia can be increased when Ubenimex is combined with Ambroxol.
Fecal microbiota The therapeutic efficacy of Fecal microbiota can be decreased when used in combination with Ubenimex.

Target Protein

Leukotriene A-4 hydrolase LTA4H
Bacterial leucyl aminopeptidase

Referensi & Sumber

Synthesis reference: Hamao Umezawa, Takaaki Aoyagi, Tomio Takeuchi, Masa Hamada, Yoshiro Okami, "Biologically active substance, bestatin, and production thereof." U.S. Patent US4052449, issued October 04, 1977.
Artikel (PubMed)
  • PMID: 11465152
    Scornik OA, Botbol V: Bestatin as an experimental tool in mammals. Curr Drug Metab. 2001 Mar;2(1):67-85.
  • PMID: 1733647
    Yoneda J, Saiki I, Fujii H, Abe F, Kojima Y, Azuma I: Inhibition of tumor invasion and extracellular matrix degradation by ubenimex (bestatin). Clin Exp Metastasis. 1992 Jan;10(1):49-59.
  • PMID: 16216010
    Bauvois B, Dauzonne D: Aminopeptidase-N/CD13 (EC 3.4.11.2) inhibitors: chemistry, biological evaluations, and therapeutic prospects. Med Res Rev. 2006 Jan;26(1):88-130.
  • PMID: 21205077
    Wickstrom M, Larsson R, Nygren P, Gullbo J: Aminopeptidase N (CD13) as a target for cancer chemotherapy. Cancer Sci. 2011 Mar;102(3):501-8. doi: 10.1111/j.1349-7006.2010.01826.x. Epub 2011 Jan 30.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Bestatin — Nippon Kayaku, Japan

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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