Peringatan Keamanan

Oral LD50 (rat):5628 mg/kg; Skin LD50 (rabbit): 15800 mg/kg; Subcutaneous LD50 (mouse):9800 mg/kg; Intraperitoneal LD50 (rabbit):1826 mg/kg

Hyperforin

DB01892

small molecule nutraceutical

Deskripsi

Hyperforin is a phytochemical generated by the plants of the Hypericum family. One of the most important members of this family, due to its medical properties, is Hypericum perforatum, also known as St John's wort.

Struktur Molekul 2D

Berat 536.797
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 9 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

58 Data
Eluxadoline The serum concentration of Eluxadoline can be increased when it is combined with Hyperforin.
Pravastatin The excretion of Pravastatin can be decreased when combined with Hyperforin.
Valsartan The excretion of Valsartan can be decreased when combined with Hyperforin.
Erythromycin The excretion of Erythromycin can be decreased when combined with Hyperforin.
Torasemide The excretion of Torasemide can be decreased when combined with Hyperforin.
Liothyronine The excretion of Liothyronine can be decreased when combined with Hyperforin.
Conjugated estrogens The excretion of Conjugated estrogens can be decreased when combined with Hyperforin.
Digoxin The excretion of Digoxin can be decreased when combined with Hyperforin.
Cerivastatin The excretion of Cerivastatin can be decreased when combined with Hyperforin.
Raloxifene The excretion of Raloxifene can be decreased when combined with Hyperforin.
Caspofungin The excretion of Caspofungin can be decreased when combined with Hyperforin.
Bosentan The excretion of Bosentan can be decreased when combined with Hyperforin.
Methotrexate The excretion of Methotrexate can be decreased when combined with Hyperforin.
Enalapril The excretion of Enalapril can be decreased when combined with Hyperforin.
Simvastatin The excretion of Simvastatin can be decreased when combined with Hyperforin.
Sumatriptan The excretion of Sumatriptan can be decreased when combined with Hyperforin.
Mycophenolate mofetil The excretion of Mycophenolate mofetil can be decreased when combined with Hyperforin.
Penicillamine The excretion of Penicillamine can be decreased when combined with Hyperforin.
Repaglinide The excretion of Repaglinide can be decreased when combined with Hyperforin.
Dinoprostone The excretion of Dinoprostone can be decreased when combined with Hyperforin.
Fexofenadine The excretion of Fexofenadine can be decreased when combined with Hyperforin.
Ezetimibe The excretion of Ezetimibe can be decreased when combined with Hyperforin.
Benzylpenicillin The excretion of Benzylpenicillin can be decreased when combined with Hyperforin.
Atorvastatin The excretion of Atorvastatin can be decreased when combined with Hyperforin.
Ouabain The excretion of Ouabain can be decreased when combined with Hyperforin.
Fluvastatin The excretion of Fluvastatin can be decreased when combined with Hyperforin.
Rosuvastatin The excretion of Rosuvastatin can be decreased when combined with Hyperforin.
Liotrix The excretion of Liotrix can be decreased when combined with Hyperforin.
Cholic Acid The excretion of Cholic Acid can be decreased when combined with Hyperforin.
Taurocholic acid The excretion of Taurocholic acid can be decreased when combined with Hyperforin.
Atrasentan The excretion of Atrasentan can be decreased when combined with Hyperforin.
Simeprevir The excretion of Simeprevir can be decreased when combined with Hyperforin.
Ambrisentan The excretion of Ambrisentan can be decreased when combined with Hyperforin.
Axitinib The excretion of Axitinib can be decreased when combined with Hyperforin.
Gimatecan The excretion of Gimatecan can be decreased when combined with Hyperforin.
Temocapril The excretion of Temocapril can be decreased when combined with Hyperforin.
Cholecystokinin The excretion of Cholecystokinin can be decreased when combined with Hyperforin.
Gadoxetic acid The excretion of Gadoxetic acid can be decreased when combined with Hyperforin.
Technetium Tc-99m mebrofenin The excretion of Technetium Tc-99m mebrofenin can be decreased when combined with Hyperforin.
Fimasartan The excretion of Fimasartan can be decreased when combined with Hyperforin.
Paritaprevir The excretion of Paritaprevir can be decreased when combined with Hyperforin.
Tenofovir alafenamide The excretion of Tenofovir alafenamide can be decreased when combined with Hyperforin.
Selexipag The excretion of Selexipag can be decreased when combined with Hyperforin.
Grazoprevir The excretion of Grazoprevir can be decreased when combined with Hyperforin.
Asunaprevir The excretion of Asunaprevir can be decreased when combined with Hyperforin.
Elagolix The excretion of Elagolix can be decreased when combined with Hyperforin.
Voxilaprevir The excretion of Voxilaprevir can be decreased when combined with Hyperforin.
Letermovir The excretion of Letermovir can be decreased when combined with Hyperforin.
Levosalbutamol The excretion of Levosalbutamol can be decreased when combined with Hyperforin.
Glecaprevir The excretion of Glecaprevir can be decreased when combined with Hyperforin.
Belantamab mafodotin The excretion of Belantamab mafodotin can be decreased when combined with Hyperforin.
Revefenacin Hyperforin may decrease the excretion rate of Revefenacin which could result in a higher serum level.
Brincidofovir The serum concentration of Brincidofovir can be increased when it is combined with Hyperforin.
Atogepant The serum concentration of Atogepant can be increased when it is combined with Hyperforin.
Mesalazine The excretion of Mesalazine can be decreased when combined with Hyperforin.
Tezacaftor The excretion of Tezacaftor can be decreased when combined with Hyperforin.
Momelotinib The serum concentration of Momelotinib can be increased when it is combined with Hyperforin.
Resmetirom The serum concentration of Resmetirom can be increased when it is combined with Hyperforin.

Target Protein

Polyunsaturated fatty acid 5-lipoxygenase ALOX5
Prostaglandin G/H synthase 1 PTGS1
Nuclear receptor subfamily 1 group I member 2 NR1I2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 9718074
    Chatterjee SS, Bhattacharya SK, Wonnemann M, Singer A, Muller WE: Hyperforin as a possible antidepressant component of hypericum extracts. Life Sci. 1998;63(6):499-510.
  • PMID: 17666455
    Leuner K, Kazanski V, Muller M, Essin K, Henke B, Gollasch M, Harteneck C, Muller WE: Hyperforin--a key constituent of St. John's wort specifically activates TRPC6 channels. FASEB J. 2007 Dec;21(14):4101-11. Epub 2007 Jul 31.
  • PMID: 10852961
    Moore LB, Goodwin B, Jones SA, Wisely GB, Serabjit-Singh CJ, Willson TM, Collins JL, Kliewer SA: St. John's wort induces hepatic drug metabolism through activation of the pregnane X receptor. Proc Natl Acad Sci U S A. 2000 Jun 20;97(13):7500-2.

Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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