Peringatan Keamanan

Overdosage may result in severe extrapyramidal symptoms with dysphagia, marked sialorrhea, persistent and rapidly increasing hyperthermia, pulmonary syndrome, state of shock with pallor and profuse sweating, which may be followed by collapse and coma. LD50 in mice is 70 mg/kg I.V., 120 mg/kg I.P., 500 mg/kg S.C. and 830 mg/kg P.O.

Thioproperazine

DB01622

small molecule experimental

Deskripsi

Thioproperazine is a potent neuroleptic with antipsychotic properties. Thioproperazine has a marked cataleptic and antiapomorphine activity associated with relatively slight sedative, hypothermic and spasmolytic effects. It is virtually without antiserotonin and hypotensive action and has no antihistaminic property. It is used for the treatment of all types of acute and chronic schizophrenia, including those which did not respond to the usual neuroleptics; manic syndromes.

Struktur Molekul 2D

Berat 446.629
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food. Food decreases irritation.

Interaksi Obat

1256 Data
Valsartan Thioproperazine may decrease the antihypertensive activities of Valsartan.
Ramipril Thioproperazine may decrease the antihypertensive activities of Ramipril.
Remikiren Thioproperazine may decrease the antihypertensive activities of Remikiren.
Torasemide Thioproperazine may decrease the antihypertensive activities of Torasemide.
Guanadrel Thioproperazine may decrease the antihypertensive activities of Guanadrel.
Olmesartan Thioproperazine may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Thioproperazine may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Thioproperazine may decrease the antihypertensive activities of Nitroprusside.
Minoxidil Thioproperazine may decrease the antihypertensive activities of Minoxidil.
Treprostinil Thioproperazine may decrease the antihypertensive activities of Treprostinil.
Bendroflumethiazide Thioproperazine may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Thioproperazine may decrease the antihypertensive activities of Fosinopril.
Trandolapril Thioproperazine may decrease the antihypertensive activities of Trandolapril.
Metolazone Thioproperazine may decrease the antihypertensive activities of Metolazone.
Benazepril Thioproperazine may decrease the antihypertensive activities of Benazepril.
Bosentan Thioproperazine may decrease the antihypertensive activities of Bosentan.
Enalapril Thioproperazine may decrease the antihypertensive activities of Enalapril.
Cyclothiazide Thioproperazine may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Thioproperazine may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Thioproperazine may decrease the antihypertensive activities of Mecamylamine.
Losartan Thioproperazine may decrease the antihypertensive activities of Losartan.
Moexipril Thioproperazine may decrease the antihypertensive activities of Moexipril.
Eplerenone Thioproperazine may decrease the antihypertensive activities of Eplerenone.
Lisinopril Thioproperazine may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Thioproperazine may decrease the antihypertensive activities of Nitroglycerin.
Hydroflumethiazide Thioproperazine may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Thioproperazine may decrease the antihypertensive activities of Cryptenamine.
Perindopril Thioproperazine may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Thioproperazine may decrease the antihypertensive activities of Candesartan cilexetil.
Indapamide Thioproperazine may decrease the antihypertensive activities of Indapamide.
Eprosartan Thioproperazine may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Thioproperazine may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Thioproperazine may decrease the antihypertensive activities of Quinapril.
Telmisartan Thioproperazine may decrease the antihypertensive activities of Telmisartan.
Hydrochlorothiazide Thioproperazine may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Thioproperazine may decrease the antihypertensive activities of Trichlormethiazide.
Irbesartan Thioproperazine may decrease the antihypertensive activities of Irbesartan.
Deserpidine Thioproperazine may decrease the antihypertensive activities of Deserpidine.
Pentolinium Thioproperazine may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Thioproperazine may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Thioproperazine may decrease the antihypertensive activities of Diazoxide.
Bretylium Thioproperazine may decrease the antihypertensive activities of Bretylium.
Guanethidine Thioproperazine may decrease the antihypertensive activities of Guanethidine.
Captopril Thioproperazine may decrease the antihypertensive activities of Captopril.
Epoprostenol Thioproperazine may decrease the antihypertensive activities of Epoprostenol.
Hydralazine Thioproperazine may decrease the antihypertensive activities of Hydralazine.
Polythiazide Thioproperazine may decrease the antihypertensive activities of Polythiazide.
Cilazapril Thioproperazine may decrease the antihypertensive activities of Cilazapril.
Saprisartan Thioproperazine may decrease the antihypertensive activities of Saprisartan.
Spirapril Thioproperazine may decrease the antihypertensive activities of Spirapril.
Tienilic acid Thioproperazine may decrease the antihypertensive activities of Tienilic acid.
Debrisoquine Thioproperazine may decrease the antihypertensive activities of Debrisoquine.
Sitaxentan Thioproperazine may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Thioproperazine may decrease the antihypertensive activities of Ambrisentan.
Diethylnorspermine Thioproperazine may decrease the antihypertensive activities of Diethylnorspermine.
Pinacidil Thioproperazine may decrease the antihypertensive activities of Pinacidil.
Temocapril Thioproperazine may decrease the antihypertensive activities of Temocapril.
Riociguat Thioproperazine may decrease the antihypertensive activities of Riociguat.
Macitentan Thioproperazine may decrease the antihypertensive activities of Macitentan.
Aliskiren Thioproperazine may decrease the antihypertensive activities of Aliskiren.
Nicorandil Thioproperazine may decrease the antihypertensive activities of Nicorandil.
Rauwolfia serpentina root Thioproperazine may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Thioproperazine may decrease the antihypertensive activities of Enalaprilat.
Selexipag Thioproperazine may decrease the antihypertensive activities of Selexipag.
Angiotensin 1-7 Thioproperazine may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Thioproperazine may decrease the antihypertensive activities of Imidapril.
BQ-123 Thioproperazine may decrease the antihypertensive activities of BQ-123.
Cicletanine Thioproperazine may decrease the antihypertensive activities of Cicletanine.
Dihydralazine Thioproperazine may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Thioproperazine may decrease the antihypertensive activities of Zofenopril.
Guanoxan Thioproperazine may decrease the antihypertensive activities of Guanoxan.
Delapril Thioproperazine may decrease the antihypertensive activities of Delapril.
Vincamine Thioproperazine may decrease the antihypertensive activities of Vincamine.
Linsidomine Thioproperazine may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Thioproperazine may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Thioproperazine may decrease the antihypertensive activities of Tolonidine.
Endralazine Thioproperazine may decrease the antihypertensive activities of Endralazine.
Cadralazine Thioproperazine may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Thioproperazine may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Thioproperazine may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Thioproperazine may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Thioproperazine may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Thioproperazine may decrease the antihypertensive activities of Guanoclor.
Muzolimine Thioproperazine may decrease the antihypertensive activities of Muzolimine.
Xipamide Thioproperazine may decrease the antihypertensive activities of Xipamide.
Candesartan Thioproperazine may decrease the antihypertensive activities of Candesartan.
Tocopherylquinone Thioproperazine may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Thioproperazine may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Thioproperazine may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Thioproperazine may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Thioproperazine may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Thioproperazine may decrease the antihypertensive activities of Quinaprilat.
Furosemide Thioproperazine may decrease the antihypertensive activities of Furosemide.
Levamlodipine Thioproperazine may decrease the antihypertensive activities of Levamlodipine.
Buthiazide Thioproperazine may decrease the antihypertensive activities of Buthiazide.
Azilsartan medoxomil Thioproperazine may decrease the antihypertensive activities of Azilsartan medoxomil.
Buprenorphine Thioproperazine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Thioproperazine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Thioproperazine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Thioproperazine.

Target Protein

D(2) dopamine receptor DRD2
Alpha-1A adrenergic receptor ADRA1A
Alpha-1B adrenergic receptor ADRA1B
D(1A) dopamine receptor DRD1

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 1 • International brands: 1
Produk
  • Majeptil Tab 10mg
    Tablet • 10 mg • Oral • Canada • Approved
International Brands
  • Majeptil

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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