Peringatan Keamanan

Symptoms of overdose include severe extrapyramidal manifestations, hypotension, lethargy and sedation.

Pipotiazine

DB01621

small molecule approved investigational

Deskripsi

Pipotiazine has actions similar to those of other phenothiazines. Among the different phenothiazine derivatives, it appears to be less sedating and to have a weak propensity for causing hypotension or potentiating the effects of CNS depressants and anesthetics. However, it produces a high incidence of extra pyramidal reactions. It is used for the maintenance treatment of chronic non-agitated schizophrenic patients. Symptoms of overdose include severe extrapyramidal manifestations, hypotension, lethargy and sedation.

Struktur Molekul 2D

Berat 475.667
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food. Food decreases irritation.

Interaksi Obat

1129 Data
Buprenorphine Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Hydrocodone Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Magnesium sulfate The therapeutic efficacy of Pipotiazine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Mirtazapine Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Orphenadrine Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Rotigotine Pipotiazine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Pipotiazine.
Sodium oxybate The risk or severity of CNS depression can be increased when Pipotiazine is combined with Sodium oxybate.
Suvorexant Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Thalidomide Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Amisulpride Pipotiazine may increase the antipsychotic activities of Amisulpride.
Methylphenidate The risk or severity of adverse effects can be increased when Pipotiazine is combined with Methylphenidate.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Pipotiazine is combined with Dexmethylphenidate.
Metoclopramide The risk or severity of adverse effects can be increased when Metoclopramide is combined with Pipotiazine.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with Pipotiazine.
Sulpiride Pipotiazine may increase the antipsychotic activities of Sulpiride.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Pipotiazine.
Lithium citrate Lithium citrate may increase the neurotoxic activities of Pipotiazine.
Lithium hydroxide Lithium hydroxide may increase the neurotoxic activities of Pipotiazine.
Mequitazine Pipotiazine may increase the arrhythmogenic activities of Mequitazine.
Thiopental The risk or severity of adverse effects can be increased when Pipotiazine is combined with Thiopental.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Pipotiazine.
Metyrosine The risk or severity of extrapyramidal symptoms and CNS depression can be increased when Metyrosine is combined with Pipotiazine.
Mirabegron The serum concentration of Pipotiazine can be increased when it is combined with Mirabegron.
Ethanol Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Pipotiazine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Pipotiazine.
Citalopram The risk or severity of adverse effects can be increased when Pipotiazine is combined with Citalopram.
Trazodone The risk or severity of adverse effects can be increased when Pipotiazine is combined with Trazodone.
Sertraline The risk or severity of adverse effects can be increased when Pipotiazine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Pipotiazine is combined with Sibutramine.
Zimelidine The risk or severity of adverse effects can be increased when Pipotiazine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Pipotiazine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Pipotiazine is combined with Milnacipran.
Desvenlafaxine The serum concentration of Pipotiazine can be increased when it is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Pipotiazine is combined with Seproxetine.
Levomilnacipran The risk or severity of adverse effects can be increased when Levomilnacipran is combined with Pipotiazine.
Indalpine The risk or severity of adverse effects can be increased when Pipotiazine is combined with Indalpine.
Alaproclate The risk or severity of adverse effects can be increased when Pipotiazine is combined with Alaproclate.
Esmolol The serum concentration of Esmolol can be increased when it is combined with Pipotiazine.
Betaxolol The serum concentration of Betaxolol can be increased when it is combined with Pipotiazine.
Atenolol The serum concentration of Atenolol can be increased when it is combined with Pipotiazine.
Propranolol The serum concentration of Propranolol can be increased when it is combined with Pipotiazine.
Labetalol The serum concentration of Labetalol can be increased when it is combined with Pipotiazine.
Bisoprolol The serum concentration of Bisoprolol can be increased when it is combined with Pipotiazine.
Alprenolol The serum concentration of Alprenolol can be increased when it is combined with Pipotiazine.
Pindolol The serum concentration of Pindolol can be increased when it is combined with Pipotiazine.
Carvedilol The serum concentration of Carvedilol can be increased when it is combined with Pipotiazine.
Acebutolol The serum concentration of Acebutolol can be increased when it is combined with Pipotiazine.
Nadolol The serum concentration of Nadolol can be increased when it is combined with Pipotiazine.
Bevantolol The serum concentration of Bevantolol can be increased when it is combined with Pipotiazine.
Practolol The serum concentration of Practolol can be increased when it is combined with Pipotiazine.
Penbutolol The serum concentration of Penbutolol can be increased when it is combined with Pipotiazine.
Oxprenolol The serum concentration of Oxprenolol can be increased when it is combined with Pipotiazine.
Dexpropranolol The serum concentration of Dexpropranolol can be increased when it is combined with Pipotiazine.
Celiprolol The serum concentration of Celiprolol can be increased when it is combined with Pipotiazine.
Nebivolol The serum concentration of Nebivolol can be increased when it is combined with Pipotiazine.
Bufuralol The serum concentration of Bufuralol can be increased when it is combined with Pipotiazine.
Bopindolol The serum concentration of Bopindolol can be increased when it is combined with Pipotiazine.
Bupranolol The serum concentration of Bupranolol can be increased when it is combined with Pipotiazine.
Indenolol The serum concentration of Indenolol can be increased when it is combined with Pipotiazine.
Arotinolol The serum concentration of Arotinolol can be increased when it is combined with Pipotiazine.
Levobetaxolol The serum concentration of Levobetaxolol can be increased when it is combined with Pipotiazine.
Talinolol The serum concentration of Talinolol can be increased when it is combined with Pipotiazine.
Anisodamine The serum concentration of Anisodamine can be increased when it is combined with Pipotiazine.
Bucindolol The serum concentration of Bucindolol can be increased when it is combined with Pipotiazine.
Esatenolol The serum concentration of Esatenolol can be increased when it is combined with Pipotiazine.
Cloranolol The serum concentration of Cloranolol can be increased when it is combined with Pipotiazine.
Mepindolol The serum concentration of Mepindolol can be increased when it is combined with Pipotiazine.
Epanolol The serum concentration of Epanolol can be increased when it is combined with Pipotiazine.
Tertatolol The serum concentration of Tertatolol can be increased when it is combined with Pipotiazine.
Morphine The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Morphine.
Codeine The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Codeine.
Hydromorphone The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Hydromorphone.
Oxycodone The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Oxycodone.
Butorphanol The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Butorphanol.
Dextropropoxyphene The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Dextropropoxyphene.
Pentazocine The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Pentazocine.
Naltrexone The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Naltrexone.
Sufentanil The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Sufentanil.
Nalbuphine The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Nalbuphine.
Levorphanol The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Levorphanol.
Remifentanil The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Remifentanil.
Diphenoxylate The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Diphenoxylate.
Oxymorphone The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Oxymorphone.
Dezocine The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Dezocine.
Methadyl acetate The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Dihydroetorphine.
Diamorphine The risk or severity of hypotension and CNS depression can be increased when Pipotiazine is combined with Diamorphine.

Target Protein

D(2) dopamine receptor DRD2
D(1A) dopamine receptor DRD1
5-hydroxytryptamine receptor 2A HTR2A
5-hydroxytryptamine receptor 1A HTR1A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 6143579
    Bechelli LP, Ruffino-Netto A, Hetem G: A double-blind controlled trial of pipotiazine, haloperidol and placebo in recently-hospitalized acute schizophrenic patients. Braz J Med Biol Res. 1983 Dec;16(4):305-11.

Contoh Produk & Brand

Produk: 2 • International brands: 0
Produk
  • Piportil L4
    Solution • 25 mg / mL • Intramuscular • Canada • Approved
  • Piportil L4
    Solution • 50 mg / mL • Intramuscular • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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