1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine

DB01562

small molecule experimental illicit

Deskripsi

1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine (PEPAP) is a synthetic analogue of meperidine. It is sold as a "synthetic heroin."

Struktur Molekul 2D

Berat 323.4287
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

245 Data
Fluvoxamine The metabolism of Fluvoxamine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Amphetamine The metabolism of Amphetamine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Cevimeline The metabolism of Cevimeline can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Esmolol The metabolism of Esmolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Bortezomib The metabolism of Bortezomib can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Tramadol The metabolism of Tramadol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Betaxolol The metabolism of Betaxolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Sildenafil The metabolism of Sildenafil can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Ticlopidine The metabolism of Ticlopidine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Citalopram The metabolism of Citalopram can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Eletriptan The metabolism of Eletriptan can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Nevirapine The metabolism of Nevirapine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Ranolazine The metabolism of Ranolazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Benzatropine The metabolism of Benzatropine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Metoprolol The metabolism of Metoprolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Lidocaine The metabolism of Lidocaine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Venlafaxine The metabolism of Venlafaxine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Bupivacaine The metabolism of Bupivacaine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Acetaminophen The metabolism of Acetaminophen can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Gefitinib The metabolism of Gefitinib can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Codeine The metabolism of Codeine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Methadone The metabolism of Methadone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Olanzapine The metabolism of Olanzapine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Atenolol The metabolism of Atenolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Terfenadine The metabolism of Terfenadine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Diltiazem The metabolism of Diltiazem can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Chlorzoxazone The metabolism of Chlorzoxazone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Clozapine The metabolism of Clozapine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Mirtazapine The metabolism of Mirtazapine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Timolol The metabolism of Timolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Palonosetron The metabolism of Palonosetron can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Mexiletine The metabolism of Mexiletine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Progesterone The metabolism of Progesterone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Remoxipride The metabolism of Remoxipride can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Promazine The metabolism of Promazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Zolpidem The metabolism of Zolpidem can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Prochlorperazine The metabolism of Prochlorperazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Quinine The metabolism of Quinine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Fluoxetine The metabolism of Fluoxetine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Duloxetine The metabolism of Duloxetine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Chlorpromazine The metabolism of Chlorpromazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Celecoxib The metabolism of Celecoxib can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Buspirone The metabolism of Buspirone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Darifenacin The metabolism of Darifenacin can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Oxycodone The metabolism of Oxycodone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Haloperidol The metabolism of Haloperidol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Ritonavir The metabolism of Ritonavir can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Dextromethorphan The metabolism of Dextromethorphan can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Cinnarizine The metabolism of Cinnarizine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Propranolol The metabolism of Propranolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Lisuride The metabolism of Lisuride can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Doxazosin The metabolism of Doxazosin can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Piperazine The metabolism of Piperazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Labetalol The metabolism of Labetalol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Chloroquine The metabolism of Chloroquine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Imatinib The metabolism of Imatinib can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Simvastatin The metabolism of Simvastatin can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Dextropropoxyphene The metabolism of Dextropropoxyphene can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Trazodone The metabolism of Trazodone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Galantamine The metabolism of Galantamine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Thioridazine The metabolism of Thioridazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Nicergoline The metabolism of Nicergoline can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Amprenavir The metabolism of Amprenavir can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Delavirdine The metabolism of Delavirdine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Tamsulosin The metabolism of Tamsulosin can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Paroxetine The metabolism of Paroxetine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Nateglinide The metabolism of Nateglinide can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Risperidone The metabolism of Risperidone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Meclizine The metabolism of Meclizine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Pentamidine The metabolism of Pentamidine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Dolasetron The metabolism of Dolasetron can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Minaprine The metabolism of Minaprine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Donepezil The metabolism of Donepezil can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Perphenazine The metabolism of Perphenazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Alprenolol The metabolism of Alprenolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Ondansetron The metabolism of Ondansetron can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Phenformin The metabolism of Phenformin can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Almotriptan The metabolism of Almotriptan can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Buprenorphine The metabolism of Buprenorphine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Tipranavir The metabolism of Tipranavir can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Mesoridazine The metabolism of Mesoridazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Maprotiline The metabolism of Maprotiline can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Hydrocodone The metabolism of Hydrocodone can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Pindolol The metabolism of Pindolol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Azelastine The metabolism of Azelastine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Formoterol The metabolism of Formoterol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Methoxyflurane The metabolism of Methoxyflurane can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Tolterodine The metabolism of Tolterodine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Selegiline The metabolism of Selegiline can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Promethazine The metabolism of Promethazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Mequitazine The metabolism of Mequitazine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Perhexiline The metabolism of Perhexiline can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Diphenhydramine The metabolism of Diphenhydramine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Tegaserod The metabolism of Tegaserod can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Fluvastatin The metabolism of Fluvastatin can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Sertraline The metabolism of Sertraline can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Chlorpheniramine The metabolism of Chlorpheniramine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Nifedipine The metabolism of Nifedipine can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.
Carvedilol The metabolism of Carvedilol can be decreased when combined with 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 12006905
    Pritzker D, Kanungo A, Kilicarslan T, Tyndale RF, Sellers EM: Designer drugs that are potent inhibitors of CYP2D6. J Clin Psychopharmacol. 2002 Jun;22(3):330-2. doi: 10.1097/00004714-200206000-00015.

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