Peringatan Keamanan

Drowsiness and ataxia are dose related. Central nervous system toxicity may result in respiratory depression and loss of consciousness. As such, pre-existing central nervous system depression and severe hepatic impairment are two particular contraindications for use.

Cloxazolam

DB01553

small molecule experimental

Deskripsi

Cloxazolam is a benzodiazepine with anxiolytic, sedative/hypnotic, muscle relaxant, and antiepileptic effects. It is marketed in the Argentina, Australia, Portugal, Belgium, Switzerland, Luxembourg, Germany, Taiwan and Japan -- mainly for anti-anxiety. The usual dose of cloxazolam in adults is 3-12mg/day for anti-anxiety. Although less commonly noted, it has also been reported as clinically effective in the treatment of depression, schizophrenia, and neurosis. As well, it has also been studied in Japan in doses of 15-30mg/day as an adjunct in the treatment of intractable epilepsy, for which it has demonstrated effectiveness.

Struktur Molekul 2D

Berat 349.211
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 65 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Cloxazolam is metabolised by the liver into the active metabolite chlordesmethyldiazepam (delorazepam). 5

Rute Eliminasi

Renal elimination.

Interaksi Makanan

1 Data
  • 1. Avoid alcohol. Alcohol can increase CNS depressant effects, such as fatal respiratory or cardiac depression.

Interaksi Obat

711 Data
Buprenorphine Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Hydrocodone Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Magnesium sulfate The therapeutic efficacy of Cloxazolam can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Cloxazolam may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Mirtazapine Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Orphenadrine Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Pramipexole Cloxazolam may increase the sedative activities of Pramipexole.
Ropinirole Cloxazolam may increase the sedative activities of Ropinirole.
Rotigotine Cloxazolam may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Cloxazolam.
Suvorexant Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Thalidomide Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Clozapine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Clozapine.
Methadone Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Methadone.
Phenytoin The serum concentration of Phenytoin can be increased when it is combined with Cloxazolam.
Fosphenytoin The serum concentration of Fosphenytoin can be increased when it is combined with Cloxazolam.
Sodium oxybate Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Teduglutide The serum concentration of Cloxazolam can be increased when it is combined with Teduglutide.
Yohimbine The therapeutic efficacy of Cloxazolam can be increased when used in combination with Yohimbine.
Ethanol Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Cloxazolam may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Cloxazolam.
Fluvoxamine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Cloxazolam is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Cloxazolam is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Cloxazolam is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Cloxazolam is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Cloxazolam is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Cloxazolam is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Cloxazolam is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Cloxazolam is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Cloxazolam is combined with Alaproclate.
Amitriptyline The risk or severity of CNS depression can be increased when Amitriptyline is combined with Cloxazolam.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Cloxazolam.
Imipramine The risk or severity of CNS depression can be increased when Imipramine is combined with Cloxazolam.
Nortriptyline The risk or severity of CNS depression can be increased when Nortriptyline is combined with Cloxazolam.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Cloxazolam.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Cloxazolam.
Maprotiline The risk or severity of CNS depression can be increased when Maprotiline is combined with Cloxazolam.
Doxepin The risk or severity of CNS depression can be increased when Doxepin is combined with Cloxazolam.
Desipramine The risk or severity of CNS depression can be increased when Desipramine is combined with Cloxazolam.
Pizotifen The risk or severity of CNS depression can be increased when Cloxazolam is combined with Pizotifen.
Dosulepin The risk or severity of CNS depression can be increased when Cloxazolam is combined with Dosulepin.
Olanzapine The risk or severity of CNS depression can be increased when Olanzapine is combined with Cloxazolam.
Zopiclone The risk or severity of adverse effects can be increased when Cloxazolam is combined with Zopiclone.
Caffeine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Caffeine.
Theophylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Theophylline.
Dyphylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Dyphylline.
Pentoxifylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Pentoxifylline.
Mercaptopurine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Mercaptopurine.
Aminophylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Aminophylline.
Oxtriphylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Oxtriphylline.
Theobromine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Theobromine.
Fenethylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Fenethylline.
8-azaguanine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 8-azaguanine.
7,9-Dimethylguanine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 7,9-Dimethylguanine.
Xanthine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Xanthine.
7-Deazaguanine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 7-Deazaguanine.
Guanine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Guanine.
9-Methylguanine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 9-Methylguanine.
Peldesine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Peldesine.
Hypoxanthine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Hypoxanthine.
9-Deazaguanine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 9-Deazaguanine.
Propentofylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Propentofylline.
Valomaciclovir The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Valomaciclovir.
3-isobutyl-1-methyl-7H-xanthine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 3-isobutyl-1-methyl-7H-xanthine.
Uric acid The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Uric acid.
Doxofylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Doxofylline.
6-O-benzylguanine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 6-O-benzylguanine.
Lisofylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Lisofylline.
Lobucavir The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Lobucavir.
Cafedrine The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Cafedrine.
Theodrenaline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Theodrenaline.
Bamifylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Bamifylline.
Proxyphylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Proxyphylline.
Acefylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Acefylline.
Etamiphylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Etamiphylline.
Pentifylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Pentifylline.
Bufylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Bufylline.
Bromotheophylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Bromotheophylline.
Furafylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with Furafylline.
8-chlorotheophylline The therapeutic efficacy of Cloxazolam can be decreased when used in combination with 8-chlorotheophylline.

Target Protein

GABA(A) Receptor GABRA1
GABA(A) Receptor Benzodiazepine Binding Site GABRA1

Referensi & Sumber

Synthesis reference: Tachikawa, R., Takagi, H., Kamioka, T., Fukunaga, M., Kawano, Y. and Miyadera, T.; US. Patents 3,696,094; October 3,1972; and 3,772,371; November 13, 1973; both assigned to Sankyo Company Limited, Japan.
Artikel (PubMed)

Contoh Produk & Brand

Produk: 0 • International brands: 7
International Brands
  • Akton — Nycomed
  • Cloxam — Jaba Recordati
  • Clozal — Sankyo Pharma Brasil Ltda
  • Elum — Farmasa
  • Olcadil — Novartis
  • Sepazon — Daiichi Sankyo
  • Tolestan — Roemmers

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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