Carfentanil

DB01535

small molecule illicit investigational vet_approved

Deskripsi

Carfentanil or carfentanyl (Wildnil) is an analogue of the popular synthetic opioid analgesic fentanyl, and is one of the most potent opioids known (also the most potent opioid used commercially). Carfentanil was first synthesized in 1974 by a team of chemists at Janssen Pharmaceutica which included Paul Janssen. It has a quantitative potency approximately 10,000 times that of morphine and 100 times that of fentanyl, with activity in humans starting at about 1 microgram. It is marketed under the trade name Wildnil as a general anaesthetic agent for large animals. Carfentanil is intended for large-animal use only as its extreme potency makes it inappropriate for use in humans. Currently sufentanil, approximately 10–20 times less potent (500 to 1000 times the efficacy of morphine per weight) than carfentanil, is the maximum strength fentanyl analog for use in humans.

Struktur Molekul 2D

Berat 394.5066
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

916 Data
Buprenorphine Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Hydrocodone Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Magnesium sulfate The therapeutic efficacy of Carfentanil can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Carfentanil may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Orphenadrine Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Pramipexole Carfentanil may increase the sedative activities of Pramipexole.
Ropinirole Carfentanil may increase the sedative activities of Ropinirole.
Rotigotine Carfentanil may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Carfentanil.
Sodium oxybate Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Thalidomide Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Alvimopan The risk or severity of adverse effects can be increased when Carfentanil is combined with Alvimopan.
Desmopressin The risk or severity of hyponatremia can be increased when Carfentanil is combined with Desmopressin.
Morphine The risk or severity of adverse effects can be increased when Morphine is combined with Carfentanil.
Codeine The risk or severity of adverse effects can be increased when Codeine is combined with Carfentanil.
Hydromorphone The risk or severity of adverse effects can be increased when Hydromorphone is combined with Carfentanil.
Meperidine The risk or severity of adverse effects can be increased when Meperidine is combined with Carfentanil.
Oxycodone The risk or severity of adverse effects can be increased when Oxycodone is combined with Carfentanil.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Dextropropoxyphene is combined with Carfentanil.
Naltrexone The therapeutic efficacy of Carfentanil can be decreased when used in combination with Naltrexone.
Sufentanil The risk or severity of adverse effects can be increased when Sufentanil is combined with Carfentanil.
Alfentanil The risk or severity of adverse effects can be increased when Alfentanil is combined with Carfentanil.
Fentanyl The risk or severity of adverse effects can be increased when Fentanyl is combined with Carfentanil.
Levorphanol The risk or severity of adverse effects can be increased when Levorphanol is combined with Carfentanil.
Remifentanil The risk or severity of adverse effects can be increased when Remifentanil is combined with Carfentanil.
Diphenoxylate The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Carfentanil.
Oxymorphone The risk or severity of adverse effects can be increased when Oxymorphone is combined with Carfentanil.
Dezocine The risk or severity of adverse effects can be increased when Dezocine is combined with Carfentanil.
Methadyl acetate The risk or severity of adverse effects can be increased when Methadyl acetate is combined with Carfentanil.
Dihydroetorphine The risk or severity of adverse effects can be increased when Dihydroetorphine is combined with Carfentanil.
Diamorphine The risk or severity of adverse effects can be increased when Diamorphine is combined with Carfentanil.
Bezitramide The risk or severity of adverse effects can be increased when Bezitramide is combined with Carfentanil.
Ethylmorphine The risk or severity of adverse effects can be increased when Ethylmorphine is combined with Carfentanil.
Etorphine The risk or severity of adverse effects can be increased when Etorphine is combined with Carfentanil.
Dextromoramide The risk or severity of adverse effects can be increased when Dextromoramide is combined with Carfentanil.
Desomorphine The risk or severity of adverse effects can be increased when Desomorphine is combined with Carfentanil.
Dihydrocodeine The risk or severity of adverse effects can be increased when Carfentanil is combined with Dihydrocodeine.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Carfentanil is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Carfentanil is combined with Dihydromorphine.
Ketobemidone The risk or severity of adverse effects can be increased when Carfentanil is combined with Ketobemidone.
DPDPE The risk or severity of adverse effects can be increased when Carfentanil is combined with DPDPE.
Lofentanil The risk or severity of adverse effects can be increased when Carfentanil is combined with Lofentanil.
Opium The risk or severity of adverse effects can be increased when Carfentanil is combined with Opium.
Normethadone The risk or severity of adverse effects can be increased when Carfentanil is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Carfentanil is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Carfentanil is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Carfentanil is combined with Nicomorphine.
Meptazinol The therapeutic efficacy of Carfentanil can be decreased when used in combination with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Carfentanil is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Carfentanil is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Carfentanil is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Carfentanil is combined with Carfentanil, C-11.
Naloxegol The risk or severity of adverse effects can be increased when Carfentanil is combined with Naloxegol.
Benzhydrocodone The risk or severity of adverse effects can be increased when Carfentanil is combined with Benzhydrocodone.
Pegvisomant The therapeutic efficacy of Pegvisomant can be decreased when used in combination with Carfentanil.
Succinylcholine The risk or severity of bradycardia can be increased when Succinylcholine is combined with Carfentanil.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Carfentanil.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Carfentanil.
Mirtazapine Carfentanil may increase the serotonergic activities of Mirtazapine.
Fluvoxamine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Fluvoxamine.
Citalopram The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Citalopram.
Duloxetine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Duloxetine.
Paroxetine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Paroxetine.
Sertraline The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Sertraline.
Sibutramine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Sibutramine.
Nefazodone The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Nefazodone.
Zimelidine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Zimelidine.
Dapoxetine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Dapoxetine.
Milnacipran The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Milnacipran.
Desvenlafaxine The risk or severity of serotonin syndrome can be increased when Desvenlafaxine is combined with Carfentanil.
Seproxetine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Seproxetine.
Levomilnacipran The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Levomilnacipran.
Indalpine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Indalpine.
Ritanserin The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Ritanserin.
Alaproclate The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Alaproclate.
Ethanol Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Carfentanil may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Carfentanil.
Phentermine Phentermine may increase the analgesic activities of Carfentanil.
Pseudoephedrine Pseudoephedrine may increase the analgesic activities of Carfentanil.
Benzphetamine Benzphetamine may increase the analgesic activities of Carfentanil.
Diethylpropion Diethylpropion may increase the analgesic activities of Carfentanil.
Lisdexamfetamine The risk or severity of serotonin syndrome can be increased when Carfentanil is combined with Lisdexamfetamine.
Mephentermine Mephentermine may increase the analgesic activities of Carfentanil.
MMDA MMDA may increase the analgesic activities of Carfentanil.
Midomafetamine Midomafetamine may increase the analgesic activities of Carfentanil.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may increase the analgesic activities of Carfentanil.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may increase the analgesic activities of Carfentanil.

Target Protein

Mu-type opioid receptor OPRM1
Delta-type opioid receptor OPRD1
Kappa-type opioid receptor OPRK1

Referensi & Sumber

Synthesis reference: Louis P. Reiff, Paul B. Sollman, "Process of making carfentanil and related analgesics." U.S. Patent US5106983, issued January, 1981.
Artikel (PubMed)
  • PMID: 12712038
    Wax PM, Becker CE, Curry SC: Unexpected "gas" casualties in Moscow: a medical toxicology perspective. Ann Emerg Med. 2003 May;41(5):700-5.

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Sekuens Gen/Protein (FASTA)

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