Ajmaline

DB01426

small molecule approved experimental

Deskripsi

An alkaloid found in the root of Rauwolfia serpentina, among other plant sources. It is a class Ia antiarrhythmic agent that apparently acts by changing the shape and threshold of cardiac action potentials. Ajmaline produces potent sodium channel blocking effects and a very short half-life which makes it a very useful drug for acute intravenous treatments. The drug has been very popular in some countries for the treatment of atrial fibrillation in patients with the Wolff–Parkinson–White syndrome and in well tolerated monomorphic ventricular tachycardias. It has also been used for many years as a drug to challenge the conduction system of the heart in cases of bundle branch block and syncope. In these cases, abnormal prolongation of the HV interval has been taken as a proof for infrahisian conduction defects tributary for permanent pacemaker implantation.

Struktur Molekul 2D

Berat 326.4326
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

440 Data
Amiodarone Amiodarone may increase the QTc-prolonging activities of Ajmaline.
Fingolimod Fingolimod may increase the arrhythmogenic activities of Ajmaline.
Propafenone Propafenone may increase the arrhythmogenic activities of Ajmaline.
Metoprolol Metoprolol may increase the arrhythmogenic activities of Ajmaline.
Lidocaine Lidocaine may increase the arrhythmogenic activities of Ajmaline.
Atenolol Atenolol may increase the arrhythmogenic activities of Ajmaline.
Mexiletine Mexiletine may increase the arrhythmogenic activities of Ajmaline.
Nisoldipine Nisoldipine may increase the arrhythmogenic activities of Ajmaline.
Acetyldigitoxin Acetyldigitoxin may increase the arrhythmogenic activities of Ajmaline.
Lercanidipine Lercanidipine may increase the arrhythmogenic activities of Ajmaline.
Magnesium sulfate Magnesium sulfate may increase the arrhythmogenic activities of Ajmaline.
Alprenolol Alprenolol may increase the arrhythmogenic activities of Ajmaline.
Tocainide Tocainide may increase the arrhythmogenic activities of Ajmaline.
Deslanoside Deslanoside may increase the arrhythmogenic activities of Ajmaline.
Carvedilol Carvedilol may increase the arrhythmogenic activities of Ajmaline.
Nadolol Nadolol may increase the arrhythmogenic activities of Ajmaline.
Practolol Practolol may increase the arrhythmogenic activities of Ajmaline.
Carteolol Ajmaline may increase the arrhythmogenic activities of Carteolol.
Metipranolol Ajmaline may increase the arrhythmogenic activities of Metipranolol.
Aprindine Ajmaline may increase the arrhythmogenic activities of Aprindine.
Dexpropranolol Ajmaline may increase the arrhythmogenic activities of Dexpropranolol.
Nimesulide Ajmaline may increase the arrhythmogenic activities of Nimesulide.
Cyclandelate Ajmaline may increase the arrhythmogenic activities of Cyclandelate.
Flunarizine Ajmaline may increase the arrhythmogenic activities of Flunarizine.
Nebivolol Ajmaline may increase the arrhythmogenic activities of Nebivolol.
Clevidipine Ajmaline may increase the arrhythmogenic activities of Clevidipine.
Seletracetam Ajmaline may increase the arrhythmogenic activities of Seletracetam.
Nylidrin Ajmaline may increase the arrhythmogenic activities of Nylidrin.
Dotarizine Ajmaline may increase the arrhythmogenic activities of Dotarizine.
Xylometazoline Ajmaline may increase the arrhythmogenic activities of Xylometazoline.
Sparteine Ajmaline may increase the arrhythmogenic activities of Sparteine.
Tranilast Ajmaline may increase the arrhythmogenic activities of Tranilast.
Fasudil Ajmaline may increase the arrhythmogenic activities of Fasudil.
Agmatine Ajmaline may increase the arrhythmogenic activities of Agmatine.
Nicorandil Ajmaline may increase the arrhythmogenic activities of Nicorandil.
Barnidipine Ajmaline may increase the arrhythmogenic activities of Barnidipine.
Azelnidipine Ajmaline may increase the arrhythmogenic activities of Azelnidipine.
Cilnidipine Ajmaline may increase the arrhythmogenic activities of Cilnidipine.
Darodipine Ajmaline may increase the arrhythmogenic activities of Darodipine.
Manidipine Ajmaline may increase the arrhythmogenic activities of Manidipine.
Niludipine Ajmaline may increase the arrhythmogenic activities of Niludipine.
Tropisetron Ajmaline may increase the arrhythmogenic activities of Tropisetron.
Carboxyamidotriazole Ajmaline may increase the arrhythmogenic activities of Carboxyamidotriazole.
Naftopidil Ajmaline may increase the arrhythmogenic activities of Naftopidil.
Vinpocetine Ajmaline may increase the arrhythmogenic activities of Vinpocetine.
Landiolol Ajmaline may increase the arrhythmogenic activities of Landiolol.
Spiradoline Ajmaline may increase the arrhythmogenic activities of Spiradoline.
Cymarin Ajmaline may increase the arrhythmogenic activities of Cymarin.
Metildigoxin Ajmaline may increase the arrhythmogenic activities of Metildigoxin.
Tiracizine Ajmaline may increase the arrhythmogenic activities of Tiracizine.
Ethacizine Ajmaline may increase the arrhythmogenic activities of Ethacizine.
Hydroquinine Ajmaline may increase the arrhythmogenic activities of Hydroquinine.
Bioallethrin Ajmaline may increase the arrhythmogenic activities of Bioallethrin.
Tertatolol Ajmaline may increase the arrhythmogenic activities of Tertatolol.
Caroverine Ajmaline may increase the arrhythmogenic activities of Caroverine.
Fosfructose Ajmaline may increase the arrhythmogenic activities of Fosfructose.
WIN 55212-2 Ajmaline may increase the arrhythmogenic activities of WIN 55212-2.
Fish oil Ajmaline may increase the arrhythmogenic activities of Fish oil.
Emopamil Ajmaline may increase the arrhythmogenic activities of Emopamil.
Lomerizine Ajmaline may increase the arrhythmogenic activities of Lomerizine.
Tetrandrine Ajmaline may increase the arrhythmogenic activities of Tetrandrine.
Dexniguldipine Ajmaline may increase the arrhythmogenic activities of Dexniguldipine.
Fosinoprilat Ajmaline may increase the arrhythmogenic activities of Fosinoprilat.
Hydroquinidine Ajmaline may increase the arrhythmogenic activities of Hydroquinidine.
SOR-C13 Ajmaline may increase the arrhythmogenic activities of SOR-C13.
Betaxolol Betaxolol may increase the arrhythmogenic activities of Ajmaline.
Diltiazem Diltiazem may increase the arrhythmogenic activities of Ajmaline.
Nimodipine Nimodipine may increase the arrhythmogenic activities of Ajmaline.
Cinnarizine Cinnarizine may increase the arrhythmogenic activities of Ajmaline.
Propranolol Propranolol may increase the arrhythmogenic activities of Ajmaline.
Atropine Atropine may increase the arrhythmogenic activities of Ajmaline.
Adenosine Adenosine may increase the arrhythmogenic activities of Ajmaline.
Loperamide Loperamide may increase the arrhythmogenic activities of Ajmaline.
Levosimendan Levosimendan may increase the arrhythmogenic activities of Ajmaline.
Nifedipine Nifedipine may increase the arrhythmogenic activities of Ajmaline.
Acebutolol Acebutolol may increase the arrhythmogenic activities of Ajmaline.
Flecainide Flecainide may increase the arrhythmogenic activities of Ajmaline.
Mibefradil Mibefradil may increase the arrhythmogenic activities of Ajmaline.
Oxprenolol Ajmaline may increase the arrhythmogenic activities of Oxprenolol.
Prenylamine Ajmaline may increase the arrhythmogenic activities of Prenylamine.
Fluspirilene Ajmaline may increase the arrhythmogenic activities of Fluspirilene.
Azimilide Ajmaline may increase the arrhythmogenic activities of Azimilide.
Tedisamil Ajmaline may increase the arrhythmogenic activities of Tedisamil.
Nilvadipine Ajmaline may increase the arrhythmogenic activities of Nilvadipine.
Indenolol Ajmaline may increase the arrhythmogenic activities of Indenolol.
Fendiline Ajmaline may increase the arrhythmogenic activities of Fendiline.
Eperisone Ajmaline may increase the arrhythmogenic activities of Eperisone.
Melperone Ajmaline may increase the arrhythmogenic activities of Melperone.
Benidipine Ajmaline may increase the arrhythmogenic activities of Benidipine.
Simendan Ajmaline may increase the arrhythmogenic activities of Simendan.
Otilonium Ajmaline may increase the arrhythmogenic activities of Otilonium.
Nizofenone Ajmaline may increase the arrhythmogenic activities of Nizofenone.
Bunaftine Ajmaline may increase the arrhythmogenic activities of Bunaftine.
Lorcainide Ajmaline may increase the arrhythmogenic activities of Lorcainide.
Penfluridol Ajmaline may increase the arrhythmogenic activities of Penfluridol.
Dexverapamil Ajmaline may increase the arrhythmogenic activities of Dexverapamil.
Dofetilide Dofetilide may increase the arrhythmogenic activities of Ajmaline.
Disopyramide Disopyramide may increase the arrhythmogenic activities of Ajmaline.
Ibutilide Ibutilide may increase the arrhythmogenic activities of Ajmaline.
Sotalol Sotalol may increase the arrhythmogenic activities of Ajmaline.

Target Protein

Sodium channel protein type 5 subunit alpha SCN5A

Referensi & Sumber

Synthesis reference: Ivan F. Makarevich, Yaroslav I. Khadzhai, Valeria V. Pavlova, Anastasia V. Nikolaeva, "Cardenolide and bufadienolide derivatives of ajmaline and process for producing same." U.S. Patent US4175078, issued May, 1975.
Artikel (PubMed)
  • PMID: 12804922
    Brugada J, Brugada P, Brugada R: The ajmaline challenge in Brugada syndrome: a useful tool or misleading information? Eur Heart J. 2003 Jun;24(12):1085-6.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Ajimalin

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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