Peringatan Keamanan

Can cause life-threatening agranulocytosis.

Aminophenazone

DB01424

small molecule approved withdrawn

Deskripsi

Aminophenazone is a pyrazolone with analgesic, anti-inflammatory, and antipyretic properties that carries a risk of agranulocytosis. In biomedical applications, radiolabelled (13C-labeled) aminophenazone has been used in breath tests to measure the cytochrome P-450 metabolic activity in liver function tests. The FDA suspended the use of aminophenazone due to its association with agranulocytosis, a life-threatening side effect.A254242,L43942

Struktur Molekul 2D

Berat 231.2936
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1834 Data
Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Aminophenazone.
Peginterferon alfa-2b The serum concentration of Aminophenazone can be increased when it is combined with Peginterferon alfa-2b.
Leflunomide The serum concentration of Aminophenazone can be decreased when it is combined with Leflunomide.
Teriflunomide The serum concentration of Aminophenazone can be decreased when it is combined with Teriflunomide.
Amlodipine The metabolism of Aminophenazone can be decreased when combined with Amlodipine.
Isoetharine The risk or severity of hypertension can be increased when Isoetharine is combined with Aminophenazone.
Norepinephrine The risk or severity of hypertension can be increased when Norepinephrine is combined with Aminophenazone.
Phenylpropanolamine The risk or severity of hypertension can be increased when Phenylpropanolamine is combined with Aminophenazone.
Droperidol The risk or severity of hypertension can be increased when Droperidol is combined with Aminophenazone.
Doxapram The risk or severity of hypertension can be increased when Doxapram is combined with Aminophenazone.
Atropine The risk or severity of hypertension can be increased when Atropine is combined with Aminophenazone.
Linezolid The risk or severity of hypertension can be increased when Linezolid is combined with Aminophenazone.
Metaraminol The risk or severity of hypertension can be increased when Metaraminol is combined with Aminophenazone.
Furazolidone The risk or severity of hypertension can be increased when Furazolidone is combined with Aminophenazone.
Methoxamine The risk or severity of hypertension can be increased when Methoxamine is combined with Aminophenazone.
Isoflurane The risk or severity of hypertension can be increased when Isoflurane is combined with Aminophenazone.
Propiomazine The risk or severity of hypertension can be increased when Propiomazine is combined with Aminophenazone.
Orciprenaline The risk or severity of hypertension can be increased when Orciprenaline is combined with Aminophenazone.
Phenmetrazine The risk or severity of hypertension can be increased when Phenmetrazine is combined with Aminophenazone.
Pseudoephedrine The risk or severity of hypertension can be increased when Pseudoephedrine is combined with Aminophenazone.
Ritodrine The risk or severity of hypertension can be increased when Ritodrine is combined with Aminophenazone.
Flupentixol The risk or severity of hypertension can be increased when Flupentixol is combined with Aminophenazone.
Remifentanil The risk or severity of hypertension can be increased when Remifentanil is combined with Aminophenazone.
Bitolterol The risk or severity of hypertension can be increased when Bitolterol is combined with Aminophenazone.
Oxymetazoline The risk or severity of hypertension can be increased when Oxymetazoline is combined with Aminophenazone.
Diethylpropion The risk or severity of hypertension can be increased when Diethylpropion is combined with Aminophenazone.
Naratriptan The risk or severity of hypertension can be increased when Naratriptan is combined with Aminophenazone.
Isoprenaline The risk or severity of hypertension can be increased when Isoprenaline is combined with Aminophenazone.
Arbutamine The risk or severity of hypertension can be increased when Arbutamine is combined with Aminophenazone.
Desflurane The risk or severity of hypertension can be increased when Desflurane is combined with Aminophenazone.
Isocarboxazid The risk or severity of hypertension can be increased when Isocarboxazid is combined with Aminophenazone.
Lisdexamfetamine The risk or severity of hypertension can be increased when Lisdexamfetamine is combined with Aminophenazone.
Fenoterol The risk or severity of hypertension can be increased when Fenoterol is combined with Aminophenazone.
Pirbuterol The risk or severity of hypertension can be increased when Pirbuterol is combined with Aminophenazone.
Ephedra sinica root The risk or severity of hypertension can be increased when Ephedra sinica root is combined with Aminophenazone.
Ephedrine The risk or severity of hypertension can be increased when Ephedrine is combined with Aminophenazone.
Mephentermine The risk or severity of hypertension can be increased when Mephentermine is combined with Aminophenazone.
Procaterol The risk or severity of hypertension can be increased when Procaterol is combined with Aminophenazone.
Clenbuterol The risk or severity of hypertension can be increased when Clenbuterol is combined with Aminophenazone.
Bambuterol The risk or severity of hypertension can be increased when Bambuterol is combined with Aminophenazone.
MMDA The risk or severity of hypertension can be increased when Aminophenazone is combined with MMDA.
2,5-Dimethoxy-4-ethylamphetamine The risk or severity of hypertension can be increased when Aminophenazone is combined with 2,5-Dimethoxy-4-ethylamphetamine.
4-Bromo-2,5-dimethoxyamphetamine The risk or severity of hypertension can be increased when Aminophenazone is combined with 4-Bromo-2,5-dimethoxyamphetamine.
Tenamfetamine The risk or severity of hypertension can be increased when Aminophenazone is combined with Tenamfetamine.
Chlorphentermine The risk or severity of hypertension can be increased when Aminophenazone is combined with Chlorphentermine.
Dextroamphetamine The risk or severity of hypertension can be increased when Aminophenazone is combined with Dextroamphetamine.
Phendimetrazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Phendimetrazine.
Periciazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Periciazine.
Acepromazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Acepromazine.
Thioproperazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Thioproperazine.
Epicaptopril The risk or severity of hypertension can be increased when Aminophenazone is combined with Epicaptopril.
Clorgiline The risk or severity of hypertension can be increased when Aminophenazone is combined with Clorgiline.
1-benzylimidazole The risk or severity of hypertension can be increased when Aminophenazone is combined with 1-benzylimidazole.
Nialamide The risk or severity of hypertension can be increased when Aminophenazone is combined with Nialamide.
Amibegron The risk or severity of hypertension can be increased when Aminophenazone is combined with Amibegron.
Naluzotan The risk or severity of hypertension can be increased when Aminophenazone is combined with Naluzotan.
Pizotifen The risk or severity of hypertension can be increased when Aminophenazone is combined with Pizotifen.
Solabegron The risk or severity of hypertension can be increased when Aminophenazone is combined with Solabegron.
Nitrous oxide The risk or severity of hypertension can be increased when Aminophenazone is combined with Nitrous oxide.
Xylometazoline The risk or severity of hypertension can be increased when Aminophenazone is combined with Xylometazoline.
Dexmethylphenidate The risk or severity of hypertension can be increased when Aminophenazone is combined with Dexmethylphenidate.
Isometheptene The risk or severity of hypertension can be increased when Aminophenazone is combined with Isometheptene.
Levonordefrin The risk or severity of hypertension can be increased when Aminophenazone is combined with Levonordefrin.
Naphazoline The risk or severity of hypertension can be increased when Aminophenazone is combined with Naphazoline.
Tetryzoline The risk or severity of hypertension can be increased when Aminophenazone is combined with Tetryzoline.
Cinitapride The risk or severity of hypertension can be increased when Aminophenazone is combined with Cinitapride.
Tyramine The risk or severity of hypertension can be increased when Aminophenazone is combined with Tyramine.
Adrafinil The risk or severity of hypertension can be increased when Aminophenazone is combined with Adrafinil.
Isoxsuprine The risk or severity of hypertension can be increased when Aminophenazone is combined with Isoxsuprine.
Ifenprodil The risk or severity of hypertension can be increased when Aminophenazone is combined with Ifenprodil.
Hexoprenaline The risk or severity of hypertension can be increased when Aminophenazone is combined with Hexoprenaline.
Etilefrine The risk or severity of hypertension can be increased when Aminophenazone is combined with Etilefrine.
Cirazoline The risk or severity of hypertension can be increased when Aminophenazone is combined with Cirazoline.
Synephrine The risk or severity of hypertension can be increased when Aminophenazone is combined with Synephrine.
Hydracarbazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Hydracarbazine.
Benmoxin The risk or severity of hypertension can be increased when Aminophenazone is combined with Benmoxin.
Mebanazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Mebanazine.
Octamoxin The risk or severity of hypertension can be increased when Aminophenazone is combined with Octamoxin.
Pheniprazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Pheniprazine.
Phenoxypropazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Phenoxypropazine.
Pivhydrazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Pivhydrazine.
Safrazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Safrazine.
Caroxazone The risk or severity of hypertension can be increased when Aminophenazone is combined with Caroxazone.
Iofetamine I-123 The risk or severity of hypertension can be increased when Aminophenazone is combined with Iofetamine I-123.
Racepinephrine The risk or severity of hypertension can be increased when Aminophenazone is combined with Racepinephrine.
Amitraz The risk or severity of hypertension can be increased when Aminophenazone is combined with Amitraz.
Medetomidine The risk or severity of hypertension can be increased when Aminophenazone is combined with Medetomidine.
Xylazine The risk or severity of hypertension can be increased when Aminophenazone is combined with Xylazine.
Atipamezole The risk or severity of hypertension can be increased when Aminophenazone is combined with Atipamezole.
Ractopamine The risk or severity of hypertension can be increased when Aminophenazone is combined with Ractopamine.
Romifidine The risk or severity of hypertension can be increased when Aminophenazone is combined with Romifidine.
Detomidine The risk or severity of hypertension can be increased when Aminophenazone is combined with Detomidine.
Tetrahydrocannabivarin The risk or severity of hypertension can be increased when Aminophenazone is combined with Tetrahydrocannabivarin.
PF-00610355 The risk or severity of hypertension can be increased when Aminophenazone is combined with PF-00610355.
Ritobegron The risk or severity of hypertension can be increased when Aminophenazone is combined with Ritobegron.
Abediterol The risk or severity of hypertension can be increased when Aminophenazone is combined with Abediterol.
Tulobuterol The risk or severity of hypertension can be increased when Aminophenazone is combined with Tulobuterol.
Dopexamine The risk or severity of hypertension can be increased when Aminophenazone is combined with Dopexamine.
Piclozotan The risk or severity of hypertension can be increased when Aminophenazone is combined with Piclozotan.
Idazoxan The risk or severity of hypertension can be increased when Aminophenazone is combined with Idazoxan.

Referensi & Sumber

Artikel (PubMed)
  • PMID: 9266210
    Rating D, Langhans CD: Breath tests: concepts, applications and limitations. Eur J Pediatr. 1997 Aug;156 Suppl 1:S18-23.
  • PMID: 15073823
    Chan TY, Chan AW: Aminopyrine-induced blood dyscrasias--still a problem in many parts of the world. Pharmacoepidemiol Drug Saf. 1996 Jul;5(4):215-9. doi: 10.1002/(SICI)1099-1557(199607)5:4<215::AID-PDS208>3.0.CO;2-5.

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