Peringatan Keamanan

Severe allergic reactions and hemolytic anemia were observed during the first few months of use leading to fatalities and the drug's eventual withdrawal from the market.

Temafloxacin

DB01405

small molecule withdrawn

Deskripsi

Temafloxacin is an antibiotic agent belonging to the fluoroquinolone drug class. It was first approved for use in the U.S. market in 1992, but was withdrawn shortly due to the reports of serious adverse reactions, such as allergic reactions and hemolyric anemia, resulting in three deaths.

Struktur Molekul 2D

Berat 417.3811
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Approximately 8 hours in patients with normal renal function.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Studies in healthy volunteers indicate that the average bioavailability of temafloxacin exceeds 90%, with little intersubject variability.

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1023 Data
Deferasirox The serum concentration of Temafloxacin can be increased when it is combined with Deferasirox.
Peginterferon alfa-2b The serum concentration of Temafloxacin can be increased when it is combined with Peginterferon alfa-2b.
Leflunomide The serum concentration of Temafloxacin can be decreased when it is combined with Leflunomide.
Teriflunomide The serum concentration of Temafloxacin can be decreased when it is combined with Teriflunomide.
Didanosine Didanosine can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Probenecid Probenecid may decrease the excretion rate of Temafloxacin which could result in a higher serum level.
Quinapril Quinapril can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium acetate Calcium acetate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sevelamer Sevelamer can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Iron Dextran Iron Dextran can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium Calcium can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium carbonate Calcium carbonate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lanthanum carbonate Lanthanum carbonate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric carboxymaltose Ferric carboxymaltose can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Iron sucrose Iron sucrose can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric pyrophosphate Ferric pyrophosphate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium citrate Calcium citrate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium gluconate Calcium gluconate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric sulfate Ferric sulfate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric cation Ferric cation can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tetraferric tricitrate decahydrate Tetraferric tricitrate decahydrate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lanthanum III cation Lanthanum III cation can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium polycarbophil Calcium polycarbophil can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric oxyhydroxide Ferric oxyhydroxide can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sucralfate Sucralfate can cause a decrease in the absorption of Temafloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zolmitriptan The metabolism of Zolmitriptan can be decreased when combined with Temafloxacin.
Nitrofurantoin The therapeutic efficacy of Temafloxacin can be decreased when used in combination with Nitrofurantoin.
Abiraterone The serum concentration of Temafloxacin can be increased when it is combined with Abiraterone.
Mycophenolate mofetil The serum concentration of Mycophenolate mofetil can be decreased when it is combined with Temafloxacin.
Mycophenolic acid The serum concentration of Mycophenolic acid can be decreased when it is combined with Temafloxacin.
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Temafloxacin.
Insulin human The therapeutic efficacy of Insulin human can be increased when used in combination with Temafloxacin.
Insulin lispro The therapeutic efficacy of Insulin lispro can be increased when used in combination with Temafloxacin.
Insulin pork The therapeutic efficacy of Insulin pork can be increased when used in combination with Temafloxacin.
Troglitazone The therapeutic efficacy of Troglitazone can be increased when used in combination with Temafloxacin.
Glimepiride The therapeutic efficacy of Glimepiride can be increased when used in combination with Temafloxacin.
Acarbose The therapeutic efficacy of Acarbose can be increased when used in combination with Temafloxacin.
Metformin The therapeutic efficacy of Metformin can be increased when used in combination with Temafloxacin.
Sulfadiazine The therapeutic efficacy of Sulfadiazine can be increased when used in combination with Temafloxacin.
Rosiglitazone The therapeutic efficacy of Rosiglitazone can be increased when used in combination with Temafloxacin.
Acetohexamide The therapeutic efficacy of Acetohexamide can be increased when used in combination with Temafloxacin.
Miglitol The therapeutic efficacy of Miglitol can be increased when used in combination with Temafloxacin.
Chlorpropamide The therapeutic efficacy of Chlorpropamide can be increased when used in combination with Temafloxacin.
Nateglinide The therapeutic efficacy of Nateglinide can be increased when used in combination with Temafloxacin.
Tolazamide The therapeutic efficacy of Tolazamide can be increased when used in combination with Temafloxacin.
Repaglinide The therapeutic efficacy of Repaglinide can be increased when used in combination with Temafloxacin.
Phenformin The therapeutic efficacy of Phenformin can be increased when used in combination with Temafloxacin.
Glyburide The therapeutic efficacy of Glyburide can be increased when used in combination with Temafloxacin.
Glipizide The therapeutic efficacy of Glipizide can be increased when used in combination with Temafloxacin.
Gliclazide The therapeutic efficacy of Gliclazide can be increased when used in combination with Temafloxacin.
Tolbutamide The therapeutic efficacy of Tolbutamide can be increased when used in combination with Temafloxacin.
Pioglitazone The therapeutic efficacy of Pioglitazone can be increased when used in combination with Temafloxacin.
Bromocriptine The therapeutic efficacy of Bromocriptine can be increased when used in combination with Temafloxacin.
Gliquidone The therapeutic efficacy of Gliquidone can be increased when used in combination with Temafloxacin.
Mitiglinide The therapeutic efficacy of Mitiglinide can be increased when used in combination with Temafloxacin.
Sitagliptin The therapeutic efficacy of Sitagliptin can be increased when used in combination with Temafloxacin.
Exenatide The therapeutic efficacy of Exenatide can be increased when used in combination with Temafloxacin.
Mecasermin The therapeutic efficacy of Mecasermin can be increased when used in combination with Temafloxacin.
Pramlintide The therapeutic efficacy of Pramlintide can be increased when used in combination with Temafloxacin.
Glisoxepide The therapeutic efficacy of Glisoxepide can be increased when used in combination with Temafloxacin.
Insulin aspart The therapeutic efficacy of Insulin aspart can be increased when used in combination with Temafloxacin.
Insulin glulisine The therapeutic efficacy of Insulin glulisine can be increased when used in combination with Temafloxacin.
Glymidine The therapeutic efficacy of Glymidine can be increased when used in combination with Temafloxacin.
AICA ribonucleotide The therapeutic efficacy of AICA ribonucleotide can be increased when used in combination with Temafloxacin.
Buformin The therapeutic efficacy of Buformin can be increased when used in combination with Temafloxacin.
Vildagliptin The therapeutic efficacy of Vildagliptin can be increased when used in combination with Temafloxacin.
Voglibose The therapeutic efficacy of Voglibose can be increased when used in combination with Temafloxacin.
NN344 The therapeutic efficacy of NN344 can be increased when used in combination with Temafloxacin.
AMG-222 The therapeutic efficacy of AMG-222 can be increased when used in combination with Temafloxacin.
Bisegliptin The therapeutic efficacy of Bisegliptin can be increased when used in combination with Temafloxacin.
Alogliptin The therapeutic efficacy of Alogliptin can be increased when used in combination with Temafloxacin.
Dapagliflozin The therapeutic efficacy of Dapagliflozin can be increased when used in combination with Temafloxacin.
Saxagliptin The therapeutic efficacy of Saxagliptin can be increased when used in combination with Temafloxacin.
Liraglutide The therapeutic efficacy of Liraglutide can be increased when used in combination with Temafloxacin.
Gosogliptin The therapeutic efficacy of Gosogliptin can be increased when used in combination with Temafloxacin.
Linagliptin The therapeutic efficacy of Linagliptin can be increased when used in combination with Temafloxacin.
Canagliflozin The therapeutic efficacy of Canagliflozin can be increased when used in combination with Temafloxacin.
Glibornuride The therapeutic efficacy of Glibornuride can be increased when used in combination with Temafloxacin.
Benfluorex The therapeutic efficacy of Benfluorex can be increased when used in combination with Temafloxacin.
Empagliflozin The therapeutic efficacy of Empagliflozin can be increased when used in combination with Temafloxacin.
Albiglutide The therapeutic efficacy of Albiglutide can be increased when used in combination with Temafloxacin.
Dulaglutide The therapeutic efficacy of Dulaglutide can be increased when used in combination with Temafloxacin.
Lobeglitazone The therapeutic efficacy of Lobeglitazone can be increased when used in combination with Temafloxacin.
Netoglitazone The therapeutic efficacy of Netoglitazone can be increased when used in combination with Temafloxacin.
Rivoglitazone The therapeutic efficacy of Rivoglitazone can be increased when used in combination with Temafloxacin.
Ciglitazone The therapeutic efficacy of Ciglitazone can be increased when used in combination with Temafloxacin.
Lixisenatide The therapeutic efficacy of Lixisenatide can be increased when used in combination with Temafloxacin.
Insulin beef The therapeutic efficacy of Insulin beef can be increased when used in combination with Temafloxacin.
Insulin degludec The therapeutic efficacy of Insulin degludec can be increased when used in combination with Temafloxacin.
Insulin peglispro The therapeutic efficacy of Insulin peglispro can be increased when used in combination with Temafloxacin.
Insulin tregopil The therapeutic efficacy of Insulin tregopil can be increased when used in combination with Temafloxacin.
Ipragliflozin The therapeutic efficacy of Ipragliflozin can be increased when used in combination with Temafloxacin.
Dutogliptin The therapeutic efficacy of Dutogliptin can be increased when used in combination with Temafloxacin.
Allicin The therapeutic efficacy of Allicin can be increased when used in combination with Temafloxacin.
Tofogliflozin The therapeutic efficacy of Tofogliflozin can be increased when used in combination with Temafloxacin.
Ertugliflozin The therapeutic efficacy of Ertugliflozin can be increased when used in combination with Temafloxacin.
2,4-thiazolidinedione The therapeutic efficacy of 2,4-thiazolidinedione can be increased when used in combination with Temafloxacin.
Teneligliptin The therapeutic efficacy of Teneligliptin can be increased when used in combination with Temafloxacin.
Omarigliptin The therapeutic efficacy of Omarigliptin can be increased when used in combination with Temafloxacin.
Carmegliptin The therapeutic efficacy of Carmegliptin can be increased when used in combination with Temafloxacin.

Target Protein

DNA gyrase subunit A gyrA
DNA gyrase subunit B gyrB
DNA gyrase subunit A gyrA
DNA topoisomerase 4 subunit A parC

Referensi & Sumber

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