Peringatan Keamanan

Death has followed ingestion of 10 to 30 g of salicylates in adults, but much larger amounts have been ingested without fatal outcome.

Salsalate

DB01399

small molecule approved

Deskripsi

Salsalate is a nonsteroidal anti-inflammatory agent for oral administration. Salsalate's mode of action as an anti-inflammatory and antirheumatic agent may be due to inhibition of synthesis and release of prostaglandins. The usefulness of salicylic acid, the active in vivo product of salsalate, in the treatment of arthritic disorders has been established. In contrast to aspirin, salsalate causes no greater fecal gastrointestinal blood loss than placebo. Salsalate is readily soluble in the small intestine where it is partially hydrolyzed to two molecules of salicylic acid. A significant portion of the parent compound is absorbed unchanged and undergoes rapid esterase hydrolysis in the body. The parent compound has an elimination half-life of about 1 hour. Salicylic acid (the active metabolite) biotransformation is saturated at anti-inflammatory doses of salsalate. Such capacity limited biotransformation results in an increase in the half-life of salicylic acid from 3.5 to 16 or more hours.

Struktur Molekul 2D

Berat 258.2262
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The parent compound has an elimination half-life of about 1 hour. Salicylic acid (the active metabolite) biotransformation is saturated at anti-inflammatory doses of salsalate. Such capacity limited biotransformation results in an increase in the half-life of salicylic acid from 3.5 to 16 or more hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Salsalate is insoluble in acid gastric fluids (< 0.1 mg/ml at pH 1.0), but readily soluble in the small intestine where it is partially hydrolyzed to two molecules of salicylic acid. A significant portion of the parent compound is absorbed unchanged. The amount of salicylic acid available from salsalate is about 15% less than from aspirin, when the two drugs are administered on a salicylic acid molar equivalent basis (3.6 g salsalate/5 g aspirin). Food slows the absorption of all salicylates including salsalate.

Metabolisme

Salsalate is readily soluble in the small intestine where it is partially hydrolyzed to two molecules of salicylic acid. A significant portion of the parent compound is absorbed unchanged and undergoes rapid esterase hydrolysis in the body.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid excessive or chronic alcohol consumption. Ingesting alcohol may increase the risk of developing a gastrointestinal bleed.
  • 2. Take with or without food. Taking salsalate with food may slow the absorption of salsalate but does not significantly impact the Cmax or AUC.

Interaksi Obat

1393 Data
Amlodipine Salsalate may decrease the antihypertensive activities of Amlodipine.
Phentermine The risk or severity of hypertension can be increased when Phentermine is combined with Salsalate.
Midodrine The risk or severity of hypertension can be increased when Midodrine is combined with Salsalate.
Eletriptan The risk or severity of hypertension can be increased when Eletriptan is combined with Salsalate.
Isoetharine The risk or severity of hypertension can be increased when Isoetharine is combined with Salsalate.
Ziprasidone The risk or severity of hypertension can be increased when Ziprasidone is combined with Salsalate.
Methysergide The risk or severity of hypertension can be increased when Methysergide is combined with Salsalate.
Cabergoline The risk or severity of hypertension can be increased when Cabergoline is combined with Salsalate.
Zolmitriptan The risk or severity of hypertension can be increased when Zolmitriptan is combined with Salsalate.
Dihydroergotamine The risk or severity of hypertension can be increased when Dihydroergotamine is combined with Salsalate.
Methylergometrine The risk or severity of hypertension can be increased when Methylergometrine is combined with Salsalate.
Norepinephrine The risk or severity of hypertension can be increased when Norepinephrine is combined with Salsalate.
Mirtazapine The risk or severity of hypertension can be increased when Mirtazapine is combined with Salsalate.
Phenylephrine The risk or severity of hypertension can be increased when Phenylephrine is combined with Salsalate.
Phenylpropanolamine The risk or severity of hypertension can be increased when Phenylpropanolamine is combined with Salsalate.
Promazine The risk or severity of hypertension can be increased when Promazine is combined with Salsalate.
Droperidol The risk or severity of hypertension can be increased when Droperidol is combined with Salsalate.
Doxapram The risk or severity of hypertension can be increased when Doxapram is combined with Salsalate.
Atropine The risk or severity of hypertension can be increased when Atropine is combined with Salsalate.
Lisuride The risk or severity of hypertension can be increased when Lisuride is combined with Salsalate.
Linezolid The risk or severity of hypertension can be increased when Linezolid is combined with Salsalate.
Metaraminol The risk or severity of hypertension can be increased when Metaraminol is combined with Salsalate.
Furazolidone The risk or severity of hypertension can be increased when Furazolidone is combined with Salsalate.
Epinephrine The risk or severity of hypertension can be increased when Epinephrine is combined with Salsalate.
Thioridazine The risk or severity of hypertension can be increased when Thioridazine is combined with Salsalate.
Ergotamine The risk or severity of hypertension can be increased when Ergotamine is combined with Salsalate.
Nicergoline The risk or severity of hypertension can be increased when Nicergoline is combined with Salsalate.
Sufentanil The risk or severity of hypertension can be increased when Sufentanil is combined with Salsalate.
Methoxamine The risk or severity of hypertension can be increased when Methoxamine is combined with Salsalate.
Risperidone The risk or severity of hypertension can be increased when Risperidone is combined with Salsalate.
Tranylcypromine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Salsalate.
Isoflurane The risk or severity of hypertension can be increased when Isoflurane is combined with Salsalate.
Propiomazine The risk or severity of hypertension can be increased when Propiomazine is combined with Salsalate.
Alfentanil The risk or severity of hypertension can be increased when Alfentanil is combined with Salsalate.
Minaprine The risk or severity of hypertension can be increased when Minaprine is combined with Salsalate.
Orciprenaline The risk or severity of hypertension can be increased when Orciprenaline is combined with Salsalate.
Propofol The risk or severity of hypertension can be increased when Propofol is combined with Salsalate.
Phenmetrazine The risk or severity of hypertension can be increased when Phenmetrazine is combined with Salsalate.
Trifluoperazine The risk or severity of hypertension can be increased when Trifluoperazine is combined with Salsalate.
Pseudoephedrine The risk or severity of hypertension can be increased when Pseudoephedrine is combined with Salsalate.
Benzphetamine The risk or severity of hypertension can be increased when Benzphetamine is combined with Salsalate.
Ritodrine The risk or severity of hypertension can be increased when Ritodrine is combined with Salsalate.
Flupentixol The risk or severity of hypertension can be increased when Flupentixol is combined with Salsalate.
Remifentanil The risk or severity of hypertension can be increased when Remifentanil is combined with Salsalate.
Bitolterol The risk or severity of hypertension can be increased when Bitolterol is combined with Salsalate.
Oxymetazoline The risk or severity of hypertension can be increased when Oxymetazoline is combined with Salsalate.
Diethylpropion The risk or severity of hypertension can be increased when Diethylpropion is combined with Salsalate.
Salmeterol The risk or severity of hypertension can be increased when Salmeterol is combined with Salsalate.
Naratriptan The risk or severity of hypertension can be increased when Naratriptan is combined with Salsalate.
Formoterol The risk or severity of hypertension can be increased when Formoterol is combined with Salsalate.
Frovatriptan The risk or severity of hypertension can be increased when Frovatriptan is combined with Salsalate.
Methoxyflurane The risk or severity of hypertension can be increased when Methoxyflurane is combined with Salsalate.
Selegiline The risk or severity of hypertension can be increased when Selegiline is combined with Salsalate.
Ergoloid mesylate The risk or severity of hypertension can be increased when Ergoloid mesylate is combined with Salsalate.
Isoprenaline The risk or severity of hypertension can be increased when Isoprenaline is combined with Salsalate.
Arbutamine The risk or severity of hypertension can be increased when Arbutamine is combined with Salsalate.
Dutasteride The risk or severity of hypertension can be increased when Dutasteride is combined with Salsalate.
Halothane The risk or severity of hypertension can be increased when Halothane is combined with Salsalate.
Moclobemide The risk or severity of hypertension can be increased when Moclobemide is combined with Salsalate.
Pergolide The risk or severity of hypertension can be increased when Pergolide is combined with Salsalate.
Desflurane The risk or severity of hypertension can be increased when Desflurane is combined with Salsalate.
Bromocriptine The risk or severity of hypertension can be increased when Bromocriptine is combined with Salsalate.
Finasteride The risk or severity of hypertension can be increased when Finasteride is combined with Salsalate.
Aripiprazole The risk or severity of hypertension can be increased when Aripiprazole is combined with Salsalate.
Isocarboxazid The risk or severity of hypertension can be increased when Isocarboxazid is combined with Salsalate.
Ergometrine The risk or severity of hypertension can be increased when Ergometrine is combined with Salsalate.
Lisdexamfetamine The risk or severity of hypertension can be increased when Lisdexamfetamine is combined with Salsalate.
Fenoterol The risk or severity of hypertension can be increased when Fenoterol is combined with Salsalate.
Pirbuterol The risk or severity of hypertension can be increased when Pirbuterol is combined with Salsalate.
Ephedra sinica root The risk or severity of hypertension can be increased when Ephedra sinica root is combined with Salsalate.
Ephedrine The risk or severity of hypertension can be increased when Ephedrine is combined with Salsalate.
Mephentermine The risk or severity of hypertension can be increased when Mephentermine is combined with Salsalate.
Procaterol The risk or severity of hypertension can be increased when Procaterol is combined with Salsalate.
Yohimbine The risk or severity of hypertension can be increased when Yohimbine is combined with Salsalate.
Methotrimeprazine The risk or severity of hypertension can be increased when Salsalate is combined with Methotrimeprazine.
Clenbuterol The risk or severity of hypertension can be increased when Salsalate is combined with Clenbuterol.
Bambuterol The risk or severity of hypertension can be increased when Salsalate is combined with Bambuterol.
MMDA The risk or severity of hypertension can be increased when Salsalate is combined with MMDA.
Midomafetamine The risk or severity of hypertension can be increased when Salsalate is combined with Midomafetamine.
2,5-Dimethoxy-4-ethylamphetamine The risk or severity of hypertension can be increased when Salsalate is combined with 2,5-Dimethoxy-4-ethylamphetamine.
4-Methoxyamphetamine The risk or severity of hypertension can be increased when Salsalate is combined with 4-Methoxyamphetamine.
4-Bromo-2,5-dimethoxyamphetamine The risk or severity of hypertension can be increased when Salsalate is combined with 4-Bromo-2,5-dimethoxyamphetamine.
Tenamfetamine The risk or severity of hypertension can be increased when Salsalate is combined with Tenamfetamine.
Chlorphentermine The risk or severity of hypertension can be increased when Salsalate is combined with Chlorphentermine.
Dextroamphetamine The risk or severity of hypertension can be increased when Salsalate is combined with Dextroamphetamine.
Phendimetrazine The risk or severity of hypertension can be increased when Salsalate is combined with Phendimetrazine.
Solifenacin The risk or severity of hypertension can be increased when Salsalate is combined with Solifenacin.
Periciazine The risk or severity of hypertension can be increased when Salsalate is combined with Periciazine.
Acepromazine The risk or severity of hypertension can be increased when Salsalate is combined with Acepromazine.
Thioproperazine The risk or severity of hypertension can be increased when Salsalate is combined with Thioproperazine.
Zuclopenthixol The risk or severity of hypertension can be increased when Salsalate is combined with Zuclopenthixol.
Epicaptopril The risk or severity of hypertension can be increased when Salsalate is combined with Epicaptopril.
Clorgiline The risk or severity of hypertension can be increased when Salsalate is combined with Clorgiline.
1-benzylimidazole The risk or severity of hypertension can be increased when Salsalate is combined with 1-benzylimidazole.
Iproniazid The risk or severity of hypertension can be increased when Salsalate is combined with Iproniazid.
Nialamide The risk or severity of hypertension can be increased when Salsalate is combined with Nialamide.
Lysergic acid diethylamide The risk or severity of hypertension can be increased when Salsalate is combined with Lysergic acid diethylamide.
Dronedarone The risk or severity of hypertension can be increased when Salsalate is combined with Dronedarone.
Flibanserin The risk or severity of hypertension can be increased when Salsalate is combined with Flibanserin.
Iloperidone The risk or severity of hypertension can be increased when Salsalate is combined with Iloperidone.

Target Protein

Prostaglandin G/H synthase 2 PTGS2
Prostaglandin G/H synthase 1 PTGS1

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 72 • International brands: 0
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