Quinupristin

DB01369

small molecule approved

Deskripsi

Quinupristin/dalfopristin is a combination of two antibiotics used to treat infections by staphylococci and by vancomycin-resistant Enterococcus faecium. Dalfopristin inhibits the early phase of protein synthesis in the bacterial ribosome and quinupristin inhibits the late phase of protein synthesis. The combination of the two components acts synergistically and is more effective in vitro than each component alone.

Struktur Molekul 2D

Berat 1022.23
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 3.1 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Quinupristin is converted to two conjugated active major metabolites, one with glutathione and one with cysteine.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

222 Data
Lomitapide The metabolism of Lomitapide can be decreased when combined with Quinupristin.
Cyclosporine The serum concentration of Cyclosporine can be increased when it is combined with Quinupristin.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Quinupristin.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Quinupristin.
Cilostazol The metabolism of Cilostazol can be decreased when combined with Quinupristin.
Colchicine The metabolism of Colchicine can be decreased when combined with Quinupristin.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Quinupristin.
Retapamulin The metabolism of Retapamulin can be decreased when combined with Quinupristin.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with Quinupristin.
Vardenafil The metabolism of Vardenafil can be decreased when combined with Quinupristin.
Eszopiclone The metabolism of Eszopiclone can be decreased when combined with Quinupristin.
Zopiclone The metabolism of Zopiclone can be decreased when combined with Quinupristin.
Lovastatin The metabolism of Lovastatin can be decreased when combined with Quinupristin.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with Quinupristin.
Alprazolam The metabolism of Alprazolam can be decreased when combined with Quinupristin.
Warfarin The serum concentration of Warfarin can be increased when it is combined with Quinupristin.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with Quinupristin.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with Quinupristin.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with Quinupristin.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with Quinupristin.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with Quinupristin.
Midazolam The serum concentration of Midazolam can be increased when it is combined with Quinupristin.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with Quinupristin.
Atorvastatin The metabolism of Atorvastatin can be decreased when combined with Quinupristin.
BCG vaccine The therapeutic efficacy of BCG vaccine can be decreased when used in combination with Quinupristin.
Typhoid vaccine The therapeutic efficacy of Typhoid vaccine can be decreased when used in combination with Quinupristin.
Aripiprazole The metabolism of Aripiprazole can be decreased when combined with Quinupristin.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be decreased when combined with Quinupristin.
Dicoumarol The risk or severity of bleeding can be increased when Quinupristin is combined with Dicoumarol.
Phenindione The risk or severity of bleeding can be increased when Quinupristin is combined with Phenindione.
Coumarin The risk or severity of bleeding can be increased when Quinupristin is combined with Coumarin.
Tioclomarol The risk or severity of bleeding can be increased when Quinupristin is combined with Tioclomarol.
Ethyl biscoumacetate The risk or severity of bleeding can be increased when Quinupristin is combined with Ethyl biscoumacetate.
Diphenadione The risk or severity of bleeding can be increased when Quinupristin is combined with Diphenadione.
4-hydroxycoumarin The risk or severity of bleeding can be increased when Quinupristin is combined with 4-hydroxycoumarin.
Fluindione The risk or severity of bleeding can be increased when Quinupristin is combined with Fluindione.
Clorindione The risk or severity of bleeding can be increased when Quinupristin is combined with Clorindione.
Azithromycin The metabolism of Azithromycin can be decreased when combined with Quinupristin.
Ziprasidone The metabolism of Ziprasidone can be decreased when combined with Quinupristin.
Chlorpromazine The metabolism of Chlorpromazine can be decreased when combined with Quinupristin.
Albendazole The metabolism of Albendazole can be decreased when combined with Quinupristin.
Cephalexin The metabolism of Cephalexin can be decreased when combined with Quinupristin.
Doxazosin The metabolism of Doxazosin can be decreased when combined with Quinupristin.
Norethisterone The metabolism of Norethisterone can be decreased when combined with Quinupristin.
Fenofibrate The metabolism of Fenofibrate can be decreased when combined with Quinupristin.
Atazanavir The metabolism of Atazanavir can be decreased when combined with Quinupristin.
Rosuvastatin The metabolism of Rosuvastatin can be decreased when combined with Quinupristin.
Drospirenone The metabolism of Drospirenone can be decreased when combined with Quinupristin.
Allylestrenol The metabolism of Allylestrenol can be decreased when combined with Quinupristin.
Zuclopenthixol The metabolism of Zuclopenthixol can be decreased when combined with Quinupristin.
Roflumilast The serum concentration of Roflumilast can be increased when it is combined with Quinupristin.
Lacosamide The metabolism of Lacosamide can be decreased when combined with Quinupristin.
Linagliptin The metabolism of Linagliptin can be decreased when combined with Quinupristin.
Vorapaxar The metabolism of Vorapaxar can be decreased when combined with Quinupristin.
Suvorexant The metabolism of Suvorexant can be decreased when combined with Quinupristin.
Netupitant The metabolism of Netupitant can be decreased when combined with Quinupristin.
Tasimelteon The metabolism of Tasimelteon can be decreased when combined with Quinupristin.
Nintedanib The metabolism of Nintedanib can be decreased when combined with Quinupristin.
Tenofovir alafenamide The metabolism of Tenofovir alafenamide can be decreased when combined with Quinupristin.
Dihydroergocornine The metabolism of Dihydroergocornine can be decreased when combined with Quinupristin.
Duvelisib The metabolism of Duvelisib can be decreased when combined with Quinupristin.
Gilteritinib The metabolism of Gilteritinib can be decreased when combined with Quinupristin.
9-aminocamptothecin The metabolism of 9-aminocamptothecin can be decreased when combined with Quinupristin.
Methylprednisone The metabolism of Methylprednisone can be decreased when combined with Quinupristin.
Dihydroergocristine The metabolism of Dihydroergocristine can be decreased when combined with Quinupristin.
Dihydroergocryptine The metabolism of Dihydroergocryptine can be decreased when combined with Quinupristin.
Medical Cannabis The metabolism of Medical Cannabis can be decreased when combined with Quinupristin.
Elexacaftor The metabolism of Elexacaftor can be decreased when combined with Quinupristin.
Fosaprepitant The metabolism of Fosaprepitant can be decreased when combined with Quinupristin.
Lefamulin The metabolism of Lefamulin can be decreased when combined with Quinupristin.
Tazemetostat The metabolism of Tazemetostat can be decreased when combined with Quinupristin.
Methysergide The metabolism of Methysergide can be decreased when combined with Quinupristin.
Meperidine The metabolism of Meperidine can be decreased when combined with Quinupristin.
Ebastine The metabolism of Ebastine can be decreased when combined with Quinupristin.
Terfenadine The metabolism of Terfenadine can be decreased when combined with Quinupristin.
Cisapride The metabolism of Cisapride can be decreased when combined with Quinupristin.
Isavuconazole The metabolism of Isavuconazole can be decreased when combined with Quinupristin.
Pretomanid The metabolism of Pretomanid can be decreased when combined with Quinupristin.
Pimavanserin The metabolism of Pimavanserin can be decreased when combined with Quinupristin.
Infigratinib The metabolism of Infigratinib can be decreased when combined with Quinupristin.
Dofetilide The metabolism of Dofetilide can be decreased when combined with Quinupristin.
Theophylline The metabolism of Theophylline can be decreased when combined with Quinupristin.
Carbamazepine The metabolism of Carbamazepine can be decreased when combined with Quinupristin.
Sirolimus The metabolism of Sirolimus can be decreased when combined with Quinupristin.
Quinidine The metabolism of Quinidine can be decreased when combined with Quinupristin.
Phenprocoumon The metabolism of Phenprocoumon can be decreased when combined with Quinupristin.
Busulfan The metabolism of Busulfan can be decreased when combined with Quinupristin.
Pimozide The metabolism of Pimozide can be decreased when combined with Quinupristin.
Amiodarone The metabolism of Amiodarone can be decreased when combined with Quinupristin.
Aminophylline The metabolism of Aminophylline can be decreased when combined with Quinupristin.
Paclitaxel The metabolism of Paclitaxel can be decreased when combined with Quinupristin.
Dasatinib The metabolism of Dasatinib can be decreased when combined with Quinupristin.
Fosphenytoin The metabolism of Fosphenytoin can be decreased when combined with Quinupristin.
Digitoxin The metabolism of Digitoxin can be decreased when combined with Quinupristin.
Everolimus The metabolism of Everolimus can be decreased when combined with Quinupristin.
Dronedarone The metabolism of Dronedarone can be decreased when combined with Quinupristin.
Cobimetinib The metabolism of Cobimetinib can be decreased when combined with Quinupristin.
Temsirolimus The metabolism of Temsirolimus can be decreased when combined with Quinupristin.
Idelalisib The metabolism of Idelalisib can be decreased when combined with Quinupristin.
Ceritinib The metabolism of Ceritinib can be decreased when combined with Quinupristin.

Target Protein

23S ribosomal RNA
50S ribosomal protein L10 rplJ
50S ribosomal protein L22 rplV

Referensi & Sumber

Artikel (PubMed)
  • PMID: 11219478
    Allington DR, Rivey MP: Quinupristin/dalfopristin: a therapeutic review. Clin Ther. 2001 Jan;23(1):24-44.
  • PMID: 10651391
    Lamb HM, Figgitt DP, Faulds D: Quinupristin/dalfopristin: a review of its use in the management of serious gram-positive infections. Drugs. 1999 Dec;58(6):1061-97.
  • PMID: 11764864
    Manzella JP: Quinupristin-dalfopristin: a new antibiotic for severe gram-positive infections. Am Fam Physician. 2001 Dec 1;64(11):1863-6.
  • PMID: 11190346
    Paradisi F, Corti G, Messeri D: Antistaphylococcal (MSSA, MRSA, MSSE, MRSE) antibiotics. Med Clin North Am. 2001 Jan;85(1):1-17.

Contoh Produk & Brand

Produk: 3 • International brands: 0
Produk
  • Synercid
    Injection • - • Intravenous • US • Approved
  • Synercid
    Injection, powder, lyophilized, for solution • - • Intravenous • US • Approved
  • Synercid
    Powder, for solution • - • Intravenous • Canada • Approved

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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