Spirapril

DB01348

small molecule approved

Deskripsi

Spirapril is an ACE inhibitor antihypertensive drug used to treat hypertension. Spirapril is converted to the active spiraprilat after administration. ACE inhibitors are used primarily in treatment of hypertension and congestive heart failure.

Struktur Molekul 2D

Berat 466.614
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 30 to 35 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Bioavailability is 50% following oral administration.

Metabolisme

Hepatic. Converted to spiraprilat following oral administration.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

3 Data
  • 1. Avoid hypertensive herbs (e.g. bayberry, blue cohosh, cayenne, ephedra, and licorice).
  • 2. Avoid potassium-containing products. Potassium products increase the risk of hyperkalemia.
  • 3. Limit salt intake. Salt may attenuate the antihypertensive effect.

Interaksi Obat

834 Data
Alfuzosin Alfuzosin may increase the hypotensive activities of Spirapril.
Amifostine Spirapril may increase the hypotensive activities of Amifostine.
Diazoxide Diazoxide may increase the hypotensive activities of Spirapril.
Methylphenidate Methylphenidate may decrease the antihypertensive activities of Spirapril.
Dexmethylphenidate Dexmethylphenidate may decrease the antihypertensive activities of Spirapril.
Obinutuzumab Spirapril may increase the hypotensive activities of Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the hypotensive activities of Spirapril.
Rituximab Spirapril may increase the hypotensive activities of Rituximab.
Desmopressin Desmopressin may decrease the antihypertensive activities of Spirapril.
Phentermine Phentermine may decrease the antihypertensive activities of Spirapril.
Midodrine Midodrine may decrease the antihypertensive activities of Spirapril.
Eletriptan Eletriptan may decrease the antihypertensive activities of Spirapril.
Isoetharine Isoetharine may decrease the antihypertensive activities of Spirapril.
Methysergide Methysergide may decrease the antihypertensive activities of Spirapril.
Cabergoline Cabergoline may decrease the antihypertensive activities of Spirapril.
Atomoxetine Atomoxetine may decrease the antihypertensive activities of Spirapril.
Etomidate Etomidate may decrease the antihypertensive activities of Spirapril.
Zolmitriptan Zolmitriptan may decrease the antihypertensive activities of Spirapril.
Dihydroergotamine Dihydroergotamine may decrease the antihypertensive activities of Spirapril.
Amitriptyline Amitriptyline may decrease the antihypertensive activities of Spirapril.
Protriptyline Protriptyline may decrease the antihypertensive activities of Spirapril.
Methylergometrine Methylergometrine may decrease the antihypertensive activities of Spirapril.
Norepinephrine Norepinephrine may decrease the antihypertensive activities of Spirapril.
Mirtazapine Mirtazapine may decrease the antihypertensive activities of Spirapril.
Phenylephrine Phenylephrine may decrease the antihypertensive activities of Spirapril.
Phenylpropanolamine Phenylpropanolamine may decrease the antihypertensive activities of Spirapril.
Promazine Promazine may decrease the antihypertensive activities of Spirapril.
Droperidol Droperidol may decrease the antihypertensive activities of Spirapril.
Buspirone Buspirone may decrease the antihypertensive activities of Spirapril.
Nortriptyline Nortriptyline may decrease the antihypertensive activities of Spirapril.
Amoxapine Amoxapine may decrease the antihypertensive activities of Spirapril.
Doxapram Doxapram may decrease the antihypertensive activities of Spirapril.
Atropine Atropine may decrease the antihypertensive activities of Spirapril.
Lisuride Lisuride may decrease the antihypertensive activities of Spirapril.
Metaraminol Metaraminol may decrease the antihypertensive activities of Spirapril.
Trazodone Trazodone may decrease the antihypertensive activities of Spirapril.
Epinephrine Epinephrine may decrease the antihypertensive activities of Spirapril.
Sumatriptan Sumatriptan may decrease the antihypertensive activities of Spirapril.
Ergotamine Ergotamine may decrease the antihypertensive activities of Spirapril.
Nicergoline Nicergoline may decrease the antihypertensive activities of Spirapril.
Methoxamine Methoxamine may decrease the antihypertensive activities of Spirapril.
Trimipramine Trimipramine may decrease the antihypertensive activities of Spirapril.
Risperidone Risperidone may decrease the antihypertensive activities of Spirapril.
Propiomazine Propiomazine may decrease the antihypertensive activities of Spirapril.
Alfentanil Alfentanil may decrease the antihypertensive activities of Spirapril.
Fentanyl Fentanyl may decrease the antihypertensive activities of Spirapril.
Orciprenaline Orciprenaline may decrease the antihypertensive activities of Spirapril.
Phenmetrazine Phenmetrazine may decrease the antihypertensive activities of Spirapril.
Trifluoperazine Trifluoperazine may decrease the antihypertensive activities of Spirapril.
Dobutamine Dobutamine may decrease the antihypertensive activities of Spirapril.
Pseudoephedrine Pseudoephedrine may decrease the antihypertensive activities of Spirapril.
Benzphetamine Benzphetamine may decrease the antihypertensive activities of Spirapril.
Ritodrine Ritodrine may decrease the antihypertensive activities of Spirapril.
Terbutaline Terbutaline may decrease the antihypertensive activities of Spirapril.
Flupentixol Flupentixol may decrease the antihypertensive activities of Spirapril.
Bitolterol Bitolterol may decrease the antihypertensive activities of Spirapril.
Quinidine Quinidine may decrease the antihypertensive activities of Spirapril.
Almotriptan Almotriptan may decrease the antihypertensive activities of Spirapril.
Diethylpropion Diethylpropion may decrease the antihypertensive activities of Spirapril.
Salmeterol Salmeterol may decrease the antihypertensive activities of Spirapril.
Naratriptan Naratriptan may decrease the antihypertensive activities of Spirapril.
Rizatriptan Rizatriptan may decrease the antihypertensive activities of Spirapril.
Formoterol Formoterol may decrease the antihypertensive activities of Spirapril.
Dopamine Dopamine may decrease the antihypertensive activities of Spirapril.
Frovatriptan Frovatriptan may decrease the antihypertensive activities of Spirapril.
Albuterol Salbutamol may decrease the antihypertensive activities of Spirapril.
Methoxyflurane Methoxyflurane may decrease the antihypertensive activities of Spirapril.
Ergoloid mesylate Ergoloid mesylate may decrease the antihypertensive activities of Spirapril.
Isoprenaline Isoprenaline may decrease the antihypertensive activities of Spirapril.
Arbutamine Arbutamine may decrease the antihypertensive activities of Spirapril.
Dutasteride Dutasteride may decrease the antihypertensive activities of Spirapril.
Doxepin Doxepin may decrease the antihypertensive activities of Spirapril.
Nefazodone Nefazodone may decrease the antihypertensive activities of Spirapril.
Desipramine Desipramine may decrease the antihypertensive activities of Spirapril.
Pergolide Pergolide may decrease the antihypertensive activities of Spirapril.
Finasteride Finasteride may decrease the antihypertensive activities of Spirapril.
Ergometrine Ergometrine may decrease the antihypertensive activities of Spirapril.
Lisdexamfetamine Lisdexamfetamine may decrease the antihypertensive activities of Spirapril.
Paliperidone Paliperidone may decrease the antihypertensive activities of Spirapril.
Arformoterol Arformoterol may decrease the antihypertensive activities of Spirapril.
Fenoterol Fenoterol may decrease the antihypertensive activities of Spirapril.
Pirbuterol Pirbuterol may decrease the antihypertensive activities of Spirapril.
Ephedra sinica root Ephedra sinica root may decrease the antihypertensive activities of Spirapril.
Ephedrine Ephedrine may decrease the antihypertensive activities of Spirapril.
Mephentermine Mephentermine may decrease the antihypertensive activities of Spirapril.
Procaterol Procaterol may decrease the antihypertensive activities of Spirapril.
Yohimbine Yohimbine may decrease the antihypertensive activities of Spirapril.
Methotrimeprazine Methotrimeprazine may decrease the antihypertensive activities of Spirapril.
Clenbuterol Clenbuterol may decrease the antihypertensive activities of Spirapril.
Bambuterol Bambuterol may decrease the antihypertensive activities of Spirapril.
MMDA MMDA may decrease the antihypertensive activities of Spirapril.
Midomafetamine Midomafetamine may decrease the antihypertensive activities of Spirapril.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the antihypertensive activities of Spirapril.
4-Methoxyamphetamine 4-Methoxyamphetamine may decrease the antihypertensive activities of Spirapril.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the antihypertensive activities of Spirapril.
Tenamfetamine Tenamfetamine may decrease the antihypertensive activities of Spirapril.
Chlorphentermine Chlorphentermine may decrease the antihypertensive activities of Spirapril.
Dextroamphetamine Dextroamphetamine may decrease the antihypertensive activities of Spirapril.
Metamfetamine Metamfetamine may decrease the antihypertensive activities of Spirapril.
Phendimetrazine Phendimetrazine may decrease the antihypertensive activities of Spirapril.

Target Protein

Angiotensin-converting enzyme ACE

Referensi & Sumber

Artikel (PubMed)
  • PMID: 1382161
    Hannedouche T, Ikeni A, Marques LP, Natov S, Dechaux M, Schmitt F, Lacour B, Grunfeld JP: Renal effects of angiotensin II in normotensive subjects on short-term cilazapril treatment. J Cardiovasc Pharmacol. 1992;19 Suppl 6:S25-7.
  • PMID: 7601014
    Noble S, Sorkin EM: Spirapril. A preliminary review of its pharmacology and therapeutic efficacy in the treatment of hypertension. Drugs. 1995 May;49(5):750-66.
  • PMID: 1382157
    Rosendorff C, Patton J, Radford HM, Kalliatakis B: Alpha-adrenergic and angiotensin II pressor sensitivity in hypertensive patients treated with an angiotensin-converting enzyme inhibitor. J Cardiovasc Pharmacol. 1992;19 Suppl 6:S105-9.
  • PMID: 10100366
    Shohat J, Wittenberg C, Erman A, Rosenfeld J, Boner G: Acute and chronic effects of spirapril, alone or in combination with isradipine on kidney function and blood pressure in patients with reduced kidney function and hypertension. Scand J Urol Nephrol. 1999 Feb;33(1):57-62.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Renormax

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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