Saprisartan

DB01347

small molecule experimental

Deskripsi

Saprisartan is an AT1 receptor antagonist. It is based on medications of losartan's prototypical chemical structure. The mode of (functional) AT1 receptor antagonism has been characterized as insurmountable/noncompetitive for saprisartan. It is very likely that slow dissociation kinetics from the AT1 receptor underlie insurmountable antagonism A14009.

Struktur Molekul 2D

Berat 611.431
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

784 Data
Alfuzosin Alfuzosin may increase the hypotensive activities of Saprisartan.
Aliskiren The risk or severity of hyperkalemia can be increased when Aliskiren is combined with Saprisartan.
Amifostine Saprisartan may increase the hypotensive activities of Amifostine.
Canagliflozin The risk or severity of hypotension, hyperkalemia, and reduced intravascular volume can be increased when Canagliflozin is combined with Saprisartan.
Diazoxide Diazoxide may increase the hypotensive activities of Saprisartan.
Drospirenone The risk or severity of hyperkalemia can be increased when Saprisartan is combined with Drospirenone.
Eplerenone The risk or severity of hyperkalemia can be increased when Eplerenone is combined with Saprisartan.
Semuloparin The risk or severity of hyperkalemia can be increased when Semuloparin is combined with Saprisartan.
Lithium citrate The serum concentration of Lithium citrate can be increased when it is combined with Saprisartan.
Lithium carbonate The serum concentration of Lithium carbonate can be increased when it is combined with Saprisartan.
Lithium hydroxide The serum concentration of Lithium hydroxide can be increased when it is combined with Saprisartan.
Methylphenidate Methylphenidate may decrease the antihypertensive activities of Saprisartan.
Dexmethylphenidate Dexmethylphenidate may decrease the antihypertensive activities of Saprisartan.
Obinutuzumab Saprisartan may increase the hypotensive activities of Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the hypotensive activities of Saprisartan.
Rituximab Saprisartan may increase the hypotensive activities of Rituximab.
Tolvaptan The risk or severity of hyperkalemia can be increased when Tolvaptan is combined with Saprisartan.
Trimethoprim The risk or severity of hyperkalemia can be increased when Trimethoprim is combined with Saprisartan.
Desmopressin Desmopressin may decrease the antihypertensive activities of Saprisartan.
Phentermine Phentermine may decrease the antihypertensive activities of Saprisartan.
Midodrine Midodrine may decrease the antihypertensive activities of Saprisartan.
Eletriptan Eletriptan may decrease the antihypertensive activities of Saprisartan.
Isoetharine Isoetharine may decrease the antihypertensive activities of Saprisartan.
Methysergide Methysergide may decrease the antihypertensive activities of Saprisartan.
Cabergoline Cabergoline may decrease the antihypertensive activities of Saprisartan.
Atomoxetine Atomoxetine may decrease the antihypertensive activities of Saprisartan.
Etomidate Etomidate may decrease the antihypertensive activities of Saprisartan.
Zolmitriptan Zolmitriptan may decrease the antihypertensive activities of Saprisartan.
Dihydroergotamine Dihydroergotamine may decrease the antihypertensive activities of Saprisartan.
Amitriptyline Amitriptyline may decrease the antihypertensive activities of Saprisartan.
Protriptyline Protriptyline may decrease the antihypertensive activities of Saprisartan.
Methylergometrine Methylergometrine may decrease the antihypertensive activities of Saprisartan.
Norepinephrine Norepinephrine may decrease the antihypertensive activities of Saprisartan.
Mirtazapine Mirtazapine may decrease the antihypertensive activities of Saprisartan.
Phenylephrine Phenylephrine may decrease the antihypertensive activities of Saprisartan.
Phenylpropanolamine Phenylpropanolamine may decrease the antihypertensive activities of Saprisartan.
Promazine Promazine may decrease the antihypertensive activities of Saprisartan.
Droperidol Droperidol may decrease the antihypertensive activities of Saprisartan.
Buspirone Buspirone may decrease the antihypertensive activities of Saprisartan.
Nortriptyline Nortriptyline may decrease the antihypertensive activities of Saprisartan.
Amoxapine Amoxapine may decrease the antihypertensive activities of Saprisartan.
Doxapram Doxapram may decrease the antihypertensive activities of Saprisartan.
Atropine Atropine may decrease the antihypertensive activities of Saprisartan.
Lisuride Lisuride may decrease the antihypertensive activities of Saprisartan.
Metaraminol Metaraminol may decrease the antihypertensive activities of Saprisartan.
Trazodone Trazodone may decrease the antihypertensive activities of Saprisartan.
Epinephrine Epinephrine may decrease the antihypertensive activities of Saprisartan.
Sumatriptan Sumatriptan may decrease the antihypertensive activities of Saprisartan.
Ergotamine Ergotamine may decrease the antihypertensive activities of Saprisartan.
Nicergoline Nicergoline may decrease the antihypertensive activities of Saprisartan.
Methoxamine Methoxamine may decrease the antihypertensive activities of Saprisartan.
Trimipramine Trimipramine may decrease the antihypertensive activities of Saprisartan.
Risperidone Risperidone may decrease the antihypertensive activities of Saprisartan.
Propiomazine Propiomazine may decrease the antihypertensive activities of Saprisartan.
Alfentanil Alfentanil may decrease the antihypertensive activities of Saprisartan.
Fentanyl Fentanyl may decrease the antihypertensive activities of Saprisartan.
Orciprenaline Orciprenaline may decrease the antihypertensive activities of Saprisartan.
Phenmetrazine Phenmetrazine may decrease the antihypertensive activities of Saprisartan.
Trifluoperazine Trifluoperazine may decrease the antihypertensive activities of Saprisartan.
Dobutamine Dobutamine may decrease the antihypertensive activities of Saprisartan.
Pseudoephedrine Pseudoephedrine may decrease the antihypertensive activities of Saprisartan.
Benzphetamine Benzphetamine may decrease the antihypertensive activities of Saprisartan.
Ritodrine Ritodrine may decrease the antihypertensive activities of Saprisartan.
Terbutaline Terbutaline may decrease the antihypertensive activities of Saprisartan.
Flupentixol Flupentixol may decrease the antihypertensive activities of Saprisartan.
Bitolterol Bitolterol may decrease the antihypertensive activities of Saprisartan.
Quinidine Quinidine may decrease the antihypertensive activities of Saprisartan.
Almotriptan Almotriptan may decrease the antihypertensive activities of Saprisartan.
Diethylpropion Diethylpropion may decrease the antihypertensive activities of Saprisartan.
Salmeterol Salmeterol may decrease the antihypertensive activities of Saprisartan.
Naratriptan Naratriptan may decrease the antihypertensive activities of Saprisartan.
Rizatriptan Rizatriptan may decrease the antihypertensive activities of Saprisartan.
Formoterol Formoterol may decrease the antihypertensive activities of Saprisartan.
Dopamine Dopamine may decrease the antihypertensive activities of Saprisartan.
Frovatriptan Frovatriptan may decrease the antihypertensive activities of Saprisartan.
Albuterol Salbutamol may decrease the antihypertensive activities of Saprisartan.
Methoxyflurane Methoxyflurane may decrease the antihypertensive activities of Saprisartan.
Ergoloid mesylate Ergoloid mesylate may decrease the antihypertensive activities of Saprisartan.
Isoprenaline Isoprenaline may decrease the antihypertensive activities of Saprisartan.
Arbutamine Arbutamine may decrease the antihypertensive activities of Saprisartan.
Dutasteride Dutasteride may decrease the antihypertensive activities of Saprisartan.
Doxepin Doxepin may decrease the antihypertensive activities of Saprisartan.
Nefazodone Nefazodone may decrease the antihypertensive activities of Saprisartan.
Desipramine Desipramine may decrease the antihypertensive activities of Saprisartan.
Pergolide Pergolide may decrease the antihypertensive activities of Saprisartan.
Finasteride Finasteride may decrease the antihypertensive activities of Saprisartan.
Ergometrine Ergometrine may decrease the antihypertensive activities of Saprisartan.
Lisdexamfetamine Lisdexamfetamine may decrease the antihypertensive activities of Saprisartan.
Paliperidone Paliperidone may decrease the antihypertensive activities of Saprisartan.
Arformoterol Arformoterol may decrease the antihypertensive activities of Saprisartan.
Fenoterol Fenoterol may decrease the antihypertensive activities of Saprisartan.
Pirbuterol Pirbuterol may decrease the antihypertensive activities of Saprisartan.
Ephedra sinica root Ephedra sinica root may decrease the antihypertensive activities of Saprisartan.
Ephedrine Ephedrine may decrease the antihypertensive activities of Saprisartan.
Mephentermine Mephentermine may decrease the antihypertensive activities of Saprisartan.
Procaterol Procaterol may decrease the antihypertensive activities of Saprisartan.
Yohimbine Yohimbine may decrease the antihypertensive activities of Saprisartan.
Methotrimeprazine Methotrimeprazine may decrease the antihypertensive activities of Saprisartan.
Clenbuterol Clenbuterol may decrease the antihypertensive activities of Saprisartan.
Bambuterol Bambuterol may decrease the antihypertensive activities of Saprisartan.

Target Protein

Type-1 angiotensin II receptor AGTR1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 10579749
    Timmermans PB: Pharmacological properties of angiotensin II receptor antagonists. Can J Cardiol. 1999 Nov;15 Suppl F:26F-8F.

Contoh Produk & Brand

Produk: 0 • International brands: 0
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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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