Peringatan Keamanan

Single oral doses in mice and rats resulted in mortality and/or moribundity at doses of 600 mg/kg and 500 mg/kg, respectively. Single intraperitoneal doses in mice and rats results in mortality/moribundity at 750 mg/kg and 1000 mg/kg, respectively. The maximum non-lethal single oral and intraperitoneal dose in mouse was 300 mg/kg and 250 mg/kg, respectively. In the rat it was 150 mg/kg and 250 mg/kg, respectively.

Lumiracoxib

DB01283

small molecule approved investigational

Deskripsi

Lumiracoxib is a COX-2 selective non-steroidal anti-inflammatory drug (NSAID). On August 11, 2007, Australia's Therapeutic Goods Administration (TGA, the Australian equivalent of the FDA) cancelled the registration of lumiracoxib in Australia due to concerns that it may cause liver failure. New Zealand and Canada have also followed suit in recalling the drug.

Struktur Molekul 2D

Berat 293.721
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Terminal half-life is approximately 4 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed following oral administration, with an absolute oral bioavailablity of 74%.

Metabolisme

Hepatic oxidation and hydroxylation via CYP2C9. Three major metabolites have been identified in plasma: 4'-hydroxy-lumiracoxib, 5-carboxy-lumiracoxib, and 4'-hydroxy-5-carboxy-lumiracoxib.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

1568 Data
Amlodipine The metabolism of Lumiracoxib can be decreased when combined with Amlodipine.
Phentermine The risk or severity of hypertension can be increased when Phentermine is combined with Lumiracoxib.
Midodrine The risk or severity of hypertension can be increased when Midodrine is combined with Lumiracoxib.
Isoetharine The risk or severity of hypertension can be increased when Isoetharine is combined with Lumiracoxib.
Ziprasidone The risk or severity of hypertension can be increased when Ziprasidone is combined with Lumiracoxib.
Methysergide The risk or severity of hypertension can be increased when Methysergide is combined with Lumiracoxib.
Cabergoline The risk or severity of hypertension can be increased when Cabergoline is combined with Lumiracoxib.
Zolmitriptan The risk or severity of hypertension can be increased when Zolmitriptan is combined with Lumiracoxib.
Dihydroergotamine The risk or severity of hypertension can be increased when Dihydroergotamine is combined with Lumiracoxib.
Methylergometrine The risk or severity of hypertension can be increased when Methylergometrine is combined with Lumiracoxib.
Norepinephrine The risk or severity of hypertension can be increased when Norepinephrine is combined with Lumiracoxib.
Mirtazapine The risk or severity of hypertension can be increased when Mirtazapine is combined with Lumiracoxib.
Phenylephrine The risk or severity of hypertension can be increased when Phenylephrine is combined with Lumiracoxib.
Phenylpropanolamine The risk or severity of hypertension can be increased when Phenylpropanolamine is combined with Lumiracoxib.
Droperidol The risk or severity of hypertension can be increased when Droperidol is combined with Lumiracoxib.
Doxapram The risk or severity of hypertension can be increased when Doxapram is combined with Lumiracoxib.
Atropine The risk or severity of hypertension can be increased when Atropine is combined with Lumiracoxib.
Lisuride The risk or severity of hypertension can be increased when Lisuride is combined with Lumiracoxib.
Linezolid The risk or severity of hypertension can be increased when Linezolid is combined with Lumiracoxib.
Metaraminol The risk or severity of hypertension can be increased when Metaraminol is combined with Lumiracoxib.
Furazolidone The risk or severity of hypertension can be increased when Furazolidone is combined with Lumiracoxib.
Thioridazine The risk or severity of hypertension can be increased when Thioridazine is combined with Lumiracoxib.
Ergotamine The risk or severity of hypertension can be increased when Ergotamine is combined with Lumiracoxib.
Nicergoline The risk or severity of hypertension can be increased when Nicergoline is combined with Lumiracoxib.
Sufentanil The risk or severity of hypertension can be increased when Sufentanil is combined with Lumiracoxib.
Methoxamine The risk or severity of hypertension can be increased when Methoxamine is combined with Lumiracoxib.
Risperidone The risk or severity of hypertension can be increased when Risperidone is combined with Lumiracoxib.
Isoflurane The risk or severity of hypertension can be increased when Isoflurane is combined with Lumiracoxib.
Propiomazine The risk or severity of hypertension can be increased when Propiomazine is combined with Lumiracoxib.
Alfentanil The risk or severity of hypertension can be increased when Alfentanil is combined with Lumiracoxib.
Minaprine The risk or severity of hypertension can be increased when Minaprine is combined with Lumiracoxib.
Orciprenaline The risk or severity of hypertension can be increased when Orciprenaline is combined with Lumiracoxib.
Phenmetrazine The risk or severity of hypertension can be increased when Phenmetrazine is combined with Lumiracoxib.
Trifluoperazine The risk or severity of hypertension can be increased when Trifluoperazine is combined with Lumiracoxib.
Pseudoephedrine The risk or severity of hypertension can be increased when Pseudoephedrine is combined with Lumiracoxib.
Benzphetamine The risk or severity of hypertension can be increased when Benzphetamine is combined with Lumiracoxib.
Ritodrine The risk or severity of hypertension can be increased when Ritodrine is combined with Lumiracoxib.
Flupentixol The risk or severity of hypertension can be increased when Flupentixol is combined with Lumiracoxib.
Remifentanil The risk or severity of hypertension can be increased when Remifentanil is combined with Lumiracoxib.
Bitolterol The risk or severity of hypertension can be increased when Bitolterol is combined with Lumiracoxib.
Oxymetazoline The risk or severity of hypertension can be increased when Oxymetazoline is combined with Lumiracoxib.
Diethylpropion The risk or severity of hypertension can be increased when Diethylpropion is combined with Lumiracoxib.
Salmeterol The risk or severity of hypertension can be increased when Salmeterol is combined with Lumiracoxib.
Naratriptan The risk or severity of hypertension can be increased when Naratriptan is combined with Lumiracoxib.
Frovatriptan The risk or severity of hypertension can be increased when Frovatriptan is combined with Lumiracoxib.
Ergoloid mesylate The risk or severity of hypertension can be increased when Ergoloid mesylate is combined with Lumiracoxib.
Isoprenaline The risk or severity of hypertension can be increased when Isoprenaline is combined with Lumiracoxib.
Arbutamine The risk or severity of hypertension can be increased when Arbutamine is combined with Lumiracoxib.
Dutasteride The risk or severity of hypertension can be increased when Dutasteride is combined with Lumiracoxib.
Pergolide The risk or severity of hypertension can be increased when Pergolide is combined with Lumiracoxib.
Desflurane The risk or severity of hypertension can be increased when Desflurane is combined with Lumiracoxib.
Bromocriptine The risk or severity of hypertension can be increased when Bromocriptine is combined with Lumiracoxib.
Finasteride The risk or severity of hypertension can be increased when Finasteride is combined with Lumiracoxib.
Aripiprazole The risk or severity of hypertension can be increased when Aripiprazole is combined with Lumiracoxib.
Isocarboxazid The risk or severity of hypertension can be increased when Isocarboxazid is combined with Lumiracoxib.
Ergometrine The risk or severity of hypertension can be increased when Ergometrine is combined with Lumiracoxib.
Lisdexamfetamine The risk or severity of hypertension can be increased when Lisdexamfetamine is combined with Lumiracoxib.
Fenoterol The risk or severity of hypertension can be increased when Lumiracoxib is combined with Fenoterol.
Pirbuterol The risk or severity of hypertension can be increased when Lumiracoxib is combined with Pirbuterol.
Ephedra sinica root The risk or severity of hypertension can be increased when Lumiracoxib is combined with Ephedra sinica root.
Ephedrine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Ephedrine.
Mephentermine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Mephentermine.
Procaterol The risk or severity of hypertension can be increased when Lumiracoxib is combined with Procaterol.
Yohimbine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Yohimbine.
Methotrimeprazine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Methotrimeprazine.
Clenbuterol The risk or severity of hypertension can be increased when Lumiracoxib is combined with Clenbuterol.
Bambuterol The risk or severity of hypertension can be increased when Lumiracoxib is combined with Bambuterol.
MMDA The risk or severity of hypertension can be increased when Lumiracoxib is combined with MMDA.
Midomafetamine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Midomafetamine.
2,5-Dimethoxy-4-ethylamphetamine The risk or severity of hypertension can be increased when Lumiracoxib is combined with 2,5-Dimethoxy-4-ethylamphetamine.
4-Methoxyamphetamine The risk or severity of hypertension can be increased when Lumiracoxib is combined with 4-Methoxyamphetamine.
4-Bromo-2,5-dimethoxyamphetamine The risk or severity of hypertension can be increased when Lumiracoxib is combined with 4-Bromo-2,5-dimethoxyamphetamine.
Tenamfetamine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Tenamfetamine.
Chlorphentermine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Chlorphentermine.
Dextroamphetamine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Dextroamphetamine.
Phendimetrazine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Phendimetrazine.
Solifenacin The risk or severity of hypertension can be increased when Lumiracoxib is combined with Solifenacin.
Periciazine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Periciazine.
Acepromazine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Acepromazine.
Thioproperazine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Thioproperazine.
Zuclopenthixol The risk or severity of hypertension can be increased when Lumiracoxib is combined with Zuclopenthixol.
Epicaptopril The risk or severity of hypertension can be increased when Lumiracoxib is combined with Epicaptopril.
Clorgiline The risk or severity of hypertension can be increased when Lumiracoxib is combined with Clorgiline.
1-benzylimidazole The risk or severity of hypertension can be increased when Lumiracoxib is combined with 1-benzylimidazole.
Nialamide The risk or severity of hypertension can be increased when Lumiracoxib is combined with Nialamide.
Lysergic acid diethylamide The risk or severity of hypertension can be increased when Lumiracoxib is combined with Lysergic acid diethylamide.
Dronedarone The risk or severity of hypertension can be increased when Lumiracoxib is combined with Dronedarone.
Flibanserin The risk or severity of hypertension can be increased when Lumiracoxib is combined with Flibanserin.
Iloperidone The risk or severity of hypertension can be increased when Lumiracoxib is combined with Iloperidone.
Indacaterol The risk or severity of hypertension can be increased when Lumiracoxib is combined with Indacaterol.
Rotigotine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Rotigotine.
Amibegron The risk or severity of hypertension can be increased when Lumiracoxib is combined with Amibegron.
Naluzotan The risk or severity of hypertension can be increased when Lumiracoxib is combined with Naluzotan.
Cariprazine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Cariprazine.
Mianserin The risk or severity of hypertension can be increased when Lumiracoxib is combined with Mianserin.
Pizotifen The risk or severity of hypertension can be increased when Lumiracoxib is combined with Pizotifen.
Solabegron The risk or severity of hypertension can be increased when Lumiracoxib is combined with Solabegron.
Asenapine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Asenapine.
Esmirtazapine The risk or severity of hypertension can be increased when Lumiracoxib is combined with Esmirtazapine.
Vilazodone The risk or severity of hypertension can be increased when Lumiracoxib is combined with Vilazodone.

Target Protein

Prostaglandin G/H synthase 2 PTGS2
Prostaglandin G/H synthase 1 PTGS1

Referensi & Sumber

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Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Prexige — Novartis

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