Peringatan Keamanan

Oral, rat: LD50 = 70 mg/kg. Pulmonary toxicity has been reported at cumulative doses usually greater than 1,100 mg/m2. There is one report of pulmonary toxicity at a cumulative dose of only 600 mg. The onset of toxicity has varied from 6 months after initiation of therapy, to as late as 15 years after.

Lomustine

DB01206

small molecule approved investigational

Deskripsi

An alkylating agent of value against both hematologic malignancies and solid tumors.

Struktur Molekul 2D

Berat 233.695
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Approximately 94 minutes, however the metabolites have a serum half-life of 16 to 48 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Well and rapidly absorbed from the gastrointestinal tract.

Metabolisme

Hepatic. Rapid and complete, with active metabolites.

Rute Eliminasi

Following oral administration of radioactive CeeNU at doses ranging from 30 mg/m2 to 100 mg/m2, about half of the radioactivity given was excreted in the urine in the form of degradation products within 24 hours.

Interaksi Obat

526 Data
Denosumab The risk or severity of adverse effects can be increased when Denosumab is combined with Lomustine.
Etanercept The risk or severity of adverse effects can be increased when Etanercept is combined with Lomustine.
Peginterferon alfa-2a The risk or severity of adverse effects can be increased when Peginterferon alfa-2a is combined with Lomustine.
Interferon alfa-n1 The risk or severity of adverse effects can be increased when Interferon alfa-n1 is combined with Lomustine.
Interferon alfa-n3 The risk or severity of adverse effects can be increased when Interferon alfa-n3 is combined with Lomustine.
Peginterferon alfa-2b The risk or severity of adverse effects can be increased when Peginterferon alfa-2b is combined with Lomustine.
Anakinra The risk or severity of adverse effects can be increased when Anakinra is combined with Lomustine.
Interferon gamma-1b The risk or severity of adverse effects can be increased when Interferon gamma-1b is combined with Lomustine.
Interferon alfa-2a The risk or severity of adverse effects can be increased when Interferon alfa-2a is combined with Lomustine.
Aldesleukin The risk or severity of adverse effects can be increased when Aldesleukin is combined with Lomustine.
Adalimumab The risk or severity of adverse effects can be increased when Adalimumab is combined with Lomustine.
Gemtuzumab ozogamicin The risk or severity of adverse effects can be increased when Gemtuzumab ozogamicin is combined with Lomustine.
Pegaspargase The risk or severity of adverse effects can be increased when Pegaspargase is combined with Lomustine.
Infliximab The risk or severity of adverse effects can be increased when Infliximab is combined with Lomustine.
Interferon beta-1b The risk or severity of adverse effects can be increased when Interferon beta-1b is combined with Lomustine.
Interferon alfacon-1 The risk or severity of adverse effects can be increased when Interferon alfacon-1 is combined with Lomustine.
Rituximab The risk or severity of adverse effects can be increased when Rituximab is combined with Lomustine.
Basiliximab The risk or severity of adverse effects can be increased when Basiliximab is combined with Lomustine.
Muromonab The risk or severity of adverse effects can be increased when Muromonab is combined with Lomustine.
Ibritumomab tiuxetan The risk or severity of adverse effects can be increased when Ibritumomab tiuxetan is combined with Lomustine.
Tositumomab The risk or severity of adverse effects can be increased when Tositumomab is combined with Lomustine.
Alemtuzumab The risk or severity of adverse effects can be increased when Alemtuzumab is combined with Lomustine.
Alefacept The risk or severity of adverse effects can be increased when Alefacept is combined with Lomustine.
Efalizumab The risk or severity of adverse effects can be increased when Efalizumab is combined with Lomustine.
Antithymocyte immunoglobulin (rabbit) The risk or severity of adverse effects can be increased when Antithymocyte immunoglobulin (rabbit) is combined with Lomustine.
Interferon alfa-2b The risk or severity of adverse effects can be increased when Interferon alfa-2b is combined with Lomustine.
Daclizumab The risk or severity of adverse effects can be increased when Daclizumab is combined with Lomustine.
Phenylalanine The risk or severity of adverse effects can be increased when Phenylalanine is combined with Lomustine.
Flunisolide The risk or severity of adverse effects can be increased when Flunisolide is combined with Lomustine.
Bortezomib The risk or severity of adverse effects can be increased when Bortezomib is combined with Lomustine.
Cladribine Lomustine may increase the immunosuppressive activities of Cladribine.
Carmustine The risk or severity of adverse effects can be increased when Carmustine is combined with Lomustine.
Amsacrine The risk or severity of adverse effects can be increased when Amsacrine is combined with Lomustine.
Bleomycin The risk or severity of adverse effects can be increased when Bleomycin is combined with Lomustine.
Chlorambucil The risk or severity of adverse effects can be increased when Chlorambucil is combined with Lomustine.
Raltitrexed The risk or severity of adverse effects can be increased when Raltitrexed is combined with Lomustine.
Mitomycin The risk or severity of adverse effects can be increased when Mitomycin is combined with Lomustine.
Bexarotene The risk or severity of adverse effects can be increased when Bexarotene is combined with Lomustine.
Vindesine The risk or severity of adverse effects can be increased when Vindesine is combined with Lomustine.
Floxuridine The risk or severity of adverse effects can be increased when Floxuridine is combined with Lomustine.
Indomethacin The risk or severity of adverse effects can be increased when Indomethacin is combined with Lomustine.
Tioguanine The risk or severity of adverse effects can be increased when Tioguanine is combined with Lomustine.
Vinorelbine The risk or severity of adverse effects can be increased when Vinorelbine is combined with Lomustine.
Dexrazoxane The risk or severity of adverse effects can be increased when Dexrazoxane is combined with Lomustine.
Beclomethasone dipropionate The risk or severity of adverse effects can be increased when Beclomethasone dipropionate is combined with Lomustine.
Sorafenib The risk or severity of adverse effects can be increased when Sorafenib is combined with Lomustine.
Streptozocin The risk or severity of adverse effects can be increased when Streptozocin is combined with Lomustine.
Trifluridine The risk or severity of adverse effects can be increased when Trifluridine is combined with Lomustine.
Gemcitabine The risk or severity of adverse effects can be increased when Gemcitabine is combined with Lomustine.
Betamethasone The risk or severity of adverse effects can be increased when Betamethasone is combined with Lomustine.
Teniposide The risk or severity of adverse effects can be increased when Teniposide is combined with Lomustine.
Epirubicin The risk or severity of adverse effects can be increased when Epirubicin is combined with Lomustine.
Chloramphenicol The risk or severity of adverse effects can be increased when Chloramphenicol is combined with Lomustine.
Lenalidomide The risk or severity of adverse effects can be increased when Lenalidomide is combined with Lomustine.
Altretamine The risk or severity of adverse effects can be increased when Altretamine is combined with Lomustine.
Zidovudine The risk or severity of adverse effects can be increased when Zidovudine is combined with Lomustine.
Cisplatin The risk or severity of adverse effects can be increased when Cisplatin is combined with Lomustine.
Oxaliplatin The risk or severity of adverse effects can be increased when Oxaliplatin is combined with Lomustine.
Cyclophosphamide The risk or severity of adverse effects can be increased when Cyclophosphamide is combined with Lomustine.
Vincristine The risk or severity of adverse effects can be increased when Vincristine is combined with Lomustine.
Fluorouracil The risk or severity of adverse effects can be increased when Fluorouracil is combined with Lomustine.
Propylthiouracil The risk or severity of adverse effects can be increased when Propylthiouracil is combined with Lomustine.
Pentostatin The risk or severity of adverse effects can be increased when Pentostatin is combined with Lomustine.
Methotrexate The risk or severity of adverse effects can be increased when Methotrexate is combined with Lomustine.
Vinblastine The risk or severity of adverse effects can be increased when Vinblastine is combined with Lomustine.
Fluticasone propionate The risk or severity of adverse effects can be increased when Fluticasone propionate is combined with Lomustine.
Fluocinolone acetonide The risk or severity of adverse effects can be increased when Fluocinolone acetonide is combined with Lomustine.
Linezolid The risk or severity of adverse effects can be increased when Linezolid is combined with Lomustine.
Imatinib The risk or severity of adverse effects can be increased when Imatinib is combined with Lomustine.
Triamcinolone The risk or severity of adverse effects can be increased when Triamcinolone is combined with Lomustine.
Clofarabine The risk or severity of adverse effects can be increased when Clofarabine is combined with Lomustine.
Prednisone The risk or severity of adverse effects can be increased when Prednisone is combined with Lomustine.
Pemetrexed The risk or severity of adverse effects can be increased when Pemetrexed is combined with Lomustine.
Fludrocortisone The risk or severity of adverse effects can be increased when Fludrocortisone is combined with Lomustine.
Mycophenolate mofetil The risk or severity of adverse effects can be increased when Mycophenolate mofetil is combined with Lomustine.
Daunorubicin The risk or severity of adverse effects can be increased when Daunorubicin is combined with Lomustine.
Irinotecan The risk or severity of adverse effects can be increased when Irinotecan is combined with Lomustine.
Methimazole The risk or severity of adverse effects can be increased when Methimazole is combined with Lomustine.
Etoposide The risk or severity of adverse effects can be increased when Etoposide is combined with Lomustine.
Sulfasalazine The risk or severity of adverse effects can be increased when Sulfasalazine is combined with Lomustine.
Dacarbazine The risk or severity of adverse effects can be increased when Dacarbazine is combined with Lomustine.
Temozolomide The risk or severity of adverse effects can be increased when Temozolomide is combined with Lomustine.
Penicillamine The risk or severity of adverse effects can be increased when Penicillamine is combined with Lomustine.
Prednisolone The risk or severity of adverse effects can be increased when Prednisolone is combined with Lomustine.
Mechlorethamine The risk or severity of adverse effects can be increased when Mechlorethamine is combined with Lomustine.
Azacitidine The risk or severity of adverse effects can be increased when Azacitidine is combined with Lomustine.
Carboplatin The risk or severity of adverse effects can be increased when Carboplatin is combined with Lomustine.
Methylprednisolone The risk or severity of adverse effects can be increased when Methylprednisolone is combined with Lomustine.
Dactinomycin The risk or severity of adverse effects can be increased when Dactinomycin is combined with Lomustine.
Cytarabine The risk or severity of adverse effects can be increased when Cytarabine is combined with Lomustine.
Azathioprine The risk or severity of adverse effects can be increased when Azathioprine is combined with Lomustine.
Doxorubicin The risk or severity of adverse effects can be increased when Doxorubicin is combined with Lomustine.
Hydroxyurea The risk or severity of adverse effects can be increased when Hydroxyurea is combined with Lomustine.
Mycophenolic acid The risk or severity of adverse effects can be increased when Mycophenolic acid is combined with Lomustine.
Topotecan The risk or severity of adverse effects can be increased when Topotecan is combined with Lomustine.
Mercaptopurine The risk or severity of adverse effects can be increased when Mercaptopurine is combined with Lomustine.
Thalidomide The risk or severity of adverse effects can be increased when Thalidomide is combined with Lomustine.
Melphalan The risk or severity of adverse effects can be increased when Melphalan is combined with Lomustine.
Fludarabine The risk or severity of adverse effects can be increased when Fludarabine is combined with Lomustine.
Flucytosine The risk or severity of adverse effects can be increased when Flucytosine is combined with Lomustine.

Target Protein

DNA
Stathmin-4 STMN4

Contoh Produk & Brand

Produk: 16 • International brands: 3
Produk
  • Ceenu
    Capsule, gelatin coated • 100 mg/1 • Oral • US • Approved
  • Ceenu
    Capsule, gelatin coated • 40 mg/1 • Oral • US • Approved
  • Ceenu
    Capsule, gelatin coated • 10 mg/1 • Oral • US • Approved
  • Ceenu
    Kit • - • Oral • US • Approved
  • Ceenu
    Kit • - • Oral • US • Approved
  • Ceenu
    Kit • - • Oral • US • Approved
  • Ceenu
    Capsule • 100 mg • Oral • Canada • Approved
  • Ceenu
    Capsule • 40 mg • Oral • Canada • Approved
Menampilkan 8 dari 16 produk.
International Brands
  • Belustine
  • CCNU
  • Cecenu

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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