Rifapentine

DB01201

small molecule approved investigational

Deskripsi

Rifapentine is an antibiotic drug used in the treatment of tuberculosis. It inhibits DNA-dependent RNA polymerase activity in susceptible cells. Specifically, it interacts with bacterial RNA polymerase but does not inhibit the mammalian enzyme.

Struktur Molekul 2D

Berat 877.0307
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi * 70.2 ± 9.1 L
Klirens (Clearance) * Apparent Oral cl=2.51 +/- 0.14 L/h [Male tuberculosis patients who received 600 mg rifapentine in combination with isoniazid, pyrazinamide and ethambutol] * Apparent Oral cl=1.69 +/- 0.41 L/h [Female tuberculosis patients who received 600 mg rifapentine in combination with isoniazid, pyrazinamide and ethambutol]

Absorpsi

Rapidly and well absorbed from the gastrointestinal tract.

Metabolisme

Hepatic

Rute Eliminasi

Following a single 600 mg oral dose of radiolabeled rifapentine to healthy volunteers (n=4), 87% of the total 14C rifapentine was recovered in the urine (17%) and feces (70%).

Interaksi Makanan

1 Data
  • 1. Take with food. Taking rifapentine with food increases its bioavailability and reduces gastrointestinal upset. Rifapentine tablets can be crushed and mixed with semisolid food if necessary.

Interaksi Obat

944 Data
Aripiprazole The metabolism of Aripiprazole can be increased when combined with Rifapentine.
Aripiprazole lauroxil The serum concentration of aripiprazole, an active metabolite of Rifapentine, can be decreased when used in combination with Aripiprazole lauroxil.
Clopidogrel The therapeutic efficacy of Clopidogrel can be increased when used in combination with Rifapentine.
Ifosfamide The metabolism of Ifosfamide can be increased when combined with Rifapentine.
Isoniazid Rifapentine may increase the hepatotoxic activities of Isoniazid.
Perampanel The metabolism of Perampanel can be increased when combined with Rifapentine.
Warfarin The metabolism of Warfarin can be increased when combined with Rifapentine.
Acenocoumarol The metabolism of Acenocoumarol can be increased when combined with Rifapentine.
(R)-warfarin The metabolism of (R)-warfarin can be increased when combined with Rifapentine.
R,S-Warfarin alcohol The metabolism of R,S-Warfarin alcohol can be increased when combined with Rifapentine.
S,R-Warfarin alcohol The metabolism of S,R-Warfarin alcohol can be increased when combined with Rifapentine.
(S)-Warfarin The metabolism of (S)-Warfarin can be increased when combined with Rifapentine.
Mycophenolate mofetil The serum concentration of Mycophenolate mofetil can be decreased when it is combined with Rifapentine.
Mycophenolic acid The serum concentration of Mycophenolic acid can be decreased when it is combined with Rifapentine.
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Rifapentine.
Erlotinib The metabolism of Erlotinib can be increased when combined with Rifapentine.
BCG vaccine The therapeutic efficacy of BCG vaccine can be decreased when used in combination with Rifapentine.
Typhoid vaccine The therapeutic efficacy of Typhoid vaccine can be decreased when used in combination with Rifapentine.
Esmolol The metabolism of Esmolol can be increased when combined with Rifapentine.
Betaxolol The metabolism of Betaxolol can be increased when combined with Rifapentine.
Metoprolol The metabolism of Metoprolol can be increased when combined with Rifapentine.
Atenolol The metabolism of Atenolol can be increased when combined with Rifapentine.
Timolol The metabolism of Timolol can be increased when combined with Rifapentine.
Sotalol The metabolism of Sotalol can be increased when combined with Rifapentine.
Labetalol The metabolism of Labetalol can be increased when combined with Rifapentine.
Bisoprolol The metabolism of Bisoprolol can be increased when combined with Rifapentine.
Alprenolol The metabolism of Alprenolol can be increased when combined with Rifapentine.
Pindolol The metabolism of Pindolol can be increased when combined with Rifapentine.
Carvedilol The metabolism of Carvedilol can be increased when combined with Rifapentine.
Propafenone The metabolism of Propafenone can be increased when combined with Rifapentine.
Acebutolol The metabolism of Acebutolol can be increased when combined with Rifapentine.
Nadolol The metabolism of Nadolol can be increased when combined with Rifapentine.
Bevantolol The metabolism of Bevantolol can be increased when combined with Rifapentine.
Practolol The metabolism of Practolol can be increased when combined with Rifapentine.
Penbutolol The metabolism of Penbutolol can be increased when combined with Rifapentine.
Oxprenolol The metabolism of Oxprenolol can be increased when combined with Rifapentine.
Dexpropranolol The metabolism of Dexpropranolol can be increased when combined with Rifapentine.
Celiprolol The metabolism of Celiprolol can be increased when combined with Rifapentine.
Nebivolol The metabolism of Nebivolol can be increased when combined with Rifapentine.
Bufuralol The metabolism of Bufuralol can be increased when combined with Rifapentine.
Bopindolol The metabolism of Bopindolol can be increased when combined with Rifapentine.
Bupranolol The metabolism of Bupranolol can be increased when combined with Rifapentine.
Indenolol The metabolism of Indenolol can be increased when combined with Rifapentine.
Arotinolol The metabolism of Arotinolol can be increased when combined with Rifapentine.
Levobetaxolol The metabolism of Levobetaxolol can be increased when combined with Rifapentine.
Talinolol The metabolism of Talinolol can be increased when combined with Rifapentine.
Anisodamine The metabolism of Anisodamine can be increased when combined with Rifapentine.
Bucindolol The metabolism of Bucindolol can be increased when combined with Rifapentine.
Esatenolol The metabolism of Esatenolol can be increased when combined with Rifapentine.
Cloranolol The metabolism of Cloranolol can be increased when combined with Rifapentine.
Mepindolol The metabolism of Mepindolol can be increased when combined with Rifapentine.
Epanolol The metabolism of Epanolol can be increased when combined with Rifapentine.
Tertatolol The metabolism of Tertatolol can be increased when combined with Rifapentine.
Landiolol The metabolism of Landiolol can be increased when combined with Rifapentine.
Pitolisant The metabolism of Pitolisant can be increased when combined with Rifapentine.
Segesterone acetate The metabolism of Segesterone acetate can be increased when combined with Rifapentine.
Metreleptin The metabolism of Rifapentine can be increased when combined with Metreleptin.
Diethylstilbestrol The metabolism of Diethylstilbestrol can be increased when combined with Rifapentine.
Etonogestrel The metabolism of Etonogestrel can be increased when combined with Rifapentine.
Megestrol acetate The metabolism of Megestrol acetate can be increased when combined with Rifapentine.
Levonorgestrel The metabolism of Levonorgestrel can be increased when combined with Rifapentine.
Medroxyprogesterone acetate The metabolism of Medroxyprogesterone acetate can be increased when combined with Rifapentine.
Norethisterone The metabolism of Norethisterone can be increased when combined with Rifapentine.
Ethynodiol diacetate The metabolism of Ethynodiol diacetate can be increased when combined with Rifapentine.
Mifepristone The metabolism of Mifepristone can be increased when combined with Rifapentine.
Norgestimate The metabolism of Norgestimate can be increased when combined with Rifapentine.
Ethinylestradiol The metabolism of Ethinylestradiol can be increased when combined with Rifapentine.
Drospirenone The metabolism of Drospirenone can be increased when combined with Rifapentine.
Octylphenoxy polyethoxyethanol The metabolism of Octylphenoxy polyethoxyethanol can be increased when combined with Rifapentine.
Cyproterone acetate The metabolism of Cyproterone acetate can be increased when combined with Rifapentine.
Trestolone The metabolism of Trestolone can be increased when combined with Rifapentine.
Norelgestromin The metabolism of Norelgestromin can be increased when combined with Rifapentine.
Gestodene The metabolism of Gestodene can be increased when combined with Rifapentine.
Hydroxyprogesterone caproate The metabolism of Hydroxyprogesterone caproate can be increased when combined with Rifapentine.
Dienogest The metabolism of Dienogest can be increased when combined with Rifapentine.
Norethynodrel The metabolism of Norethynodrel can be increased when combined with Rifapentine.
Norgestrel The metabolism of Norgestrel can be increased when combined with Rifapentine.
Cloprostenol The metabolism of Cloprostenol can be increased when combined with Rifapentine.
Gestrinone The metabolism of Gestrinone can be increased when combined with Rifapentine.
Nomegestrol The metabolism of Nomegestrol can be increased when combined with Rifapentine.
Gossypol The metabolism of Gossypol can be increased when combined with Rifapentine.
Ormeloxifene The metabolism of Ormeloxifene can be increased when combined with Rifapentine.
Chlormadinone The metabolism of Chlormadinone can be increased when combined with Rifapentine.
Norgestrienone The metabolism of Norgestrienone can be increased when combined with Rifapentine.
Quingestanol The metabolism of Quingestanol can be increased when combined with Rifapentine.
Demegestone The metabolism of Demegestone can be increased when combined with Rifapentine.
Etynodiol The metabolism of Etynodiol can be increased when combined with Rifapentine.
Nomegestrol acetate The metabolism of Nomegestrol acetate can be increased when combined with Rifapentine.
Norethindrone enanthate The metabolism of Norethindrone enanthate can be increased when combined with Rifapentine.
Desogestrel The metabolism of Desogestrel can be increased when combined with Rifapentine.
Mestranol The metabolism of Mestranol can be increased when combined with Rifapentine.
Estrone sulfate The metabolism of Estrone sulfate can be increased when combined with Rifapentine.
Ulipristal The metabolism of Ulipristal can be increased when combined with Rifapentine.
Testosterone enanthate The metabolism of Testosterone enanthate can be increased when combined with Rifapentine.
Estradiol benzoate The metabolism of Estradiol benzoate can be increased when combined with Rifapentine.
Estradiol cypionate The metabolism of Estradiol cypionate can be increased when combined with Rifapentine.
Estradiol valerate The metabolism of Estradiol valerate can be increased when combined with Rifapentine.
Phenindione The risk or severity of bleeding can be increased when Rifapentine is combined with Phenindione.
Coumarin The risk or severity of bleeding can be increased when Rifapentine is combined with Coumarin.
Tioclomarol The risk or severity of bleeding can be increased when Rifapentine is combined with Tioclomarol.

Target Protein

DNA-directed RNA polymerase subunit beta' rpoC

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

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Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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