Tubocurarine

DB01199

small molecule approved

Deskripsi

Tubocurarine is a non-depolarizing neuromuscular blocking agent and the first identified curare alkaloid.A216008 Curare is one of the names used to describe plant-derived poisons used by indigenous South Americans to coat the tips of hunting arrows and darts, which were typically derived from plants of the genera Chondrodendron and Strychnos.A216008 Tubocurarine is a benzylisoquinoline derivative and shares this structural backbone with a number of plant-derived alkaloids, including morphine and papaverine.A216028 It was first isolated by Harold King in 1935 and was used clinically to induce neuromuscular blockade during surgeries, particularly those involving the abdomen.A216038 Tubocurarine's clinical use was limited by its relatively long duration of action (30-60 minutes)A216038 and a number of significant side effects.A216048 Safer and more pharmacokinetically favorable non-depolarizing neuromuscular blockers, such as rocuronium, have largely replaced the use of tubocurarine in the clinical setting.A216048

Struktur Molekul 2D

Berat 609.7312
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 1-2 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1222 Data
Buprenorphine Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Hydrocodone Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Magnesium sulfate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Tubocurarine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Mirtazapine Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Orphenadrine Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Pramipexole Tubocurarine may increase the sedative activities of Pramipexole.
Ropinirole Tubocurarine may increase the sedative activities of Ropinirole.
Rotigotine Tubocurarine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Tubocurarine.
Sodium oxybate The risk or severity of CNS depression can be increased when Tubocurarine is combined with Sodium oxybate.
Suvorexant Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Tubocurarine.
Thalidomide Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Tubocurarine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Capreomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Capreomycin.
Quinidine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Quinidine.
Cyclosporine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Cyclosporine.
Doxycycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Doxycycline.
Lymecycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Lymecycline.
Piperacillin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Piperacillin.
Framycetin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Framycetin.
Clomocycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Clomocycline.
Quinine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Quinine.
Vancomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Vancomycin.
Tigecycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Tigecycline.
Oxytetracycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Oxytetracycline.
Chloroquine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Chloroquine.
Demeclocycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Demeclocycline.
Mecamylamine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Mecamylamine.
Tobramycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Tobramycin.
Tetracycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Tetracycline.
Gentamicin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Gentamicin.
Etacrynic acid The therapeutic efficacy of Tubocurarine can be increased when used in combination with Etacrynic acid.
Metacycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Metacycline.
Netilmicin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Netilmicin.
Neomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Neomycin.
Procainamide The therapeutic efficacy of Tubocurarine can be increased when used in combination with Procainamide.
Streptomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Streptomycin.
Colistimethate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Colistimethate.
Kanamycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Kanamycin.
Dantrolene The therapeutic efficacy of Tubocurarine can be increased when used in combination with Dantrolene.
Rolitetracycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Rolitetracycline.
Magnesium oxide The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium oxide.
Magnesium cation The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium cation.
Paromomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Paromomycin.
Lincomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Lincomycin.
Ribostamycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Ribostamycin.
Geneticin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Geneticin.
Apramycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Apramycin.
Gentamicin C1a The therapeutic efficacy of Tubocurarine can be increased when used in combination with Gentamicin C1a.
Neamine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Neamine.
Arbekacin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Arbekacin.
Viomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Viomycin.
Puromycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Puromycin.
Magnesium hydroxide The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium hydroxide.
Magnesium trisilicate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium trisilicate.
Magnesium chloride The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium chloride.
Magnesium acetate tetrahydrate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium acetate tetrahydrate.
Magnesium carbonate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium carbonate.
Magnesium citrate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium citrate.
Magnesium glycinate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium glycinate.
Magnesium Aluminum Silicate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium Aluminum Silicate.
Dihydrostreptomycin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Dihydrostreptomycin.
Hygromycin B The therapeutic efficacy of Tubocurarine can be increased when used in combination with Hygromycin B.
Sisomicin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Sisomicin.
Plazomicin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Plazomicin.
Magnesium silicate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium silicate.
Penimepicycline The therapeutic efficacy of Tubocurarine can be increased when used in combination with Penimepicycline.
Magnesium aspartate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium aspartate.
Isepamicin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Isepamicin.
Magnesium gluconate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium gluconate.
Magnesium orotate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium orotate.
Magnesium phosphate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium phosphate.
Magnesium acetate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium acetate.
Magnesium stearate The therapeutic efficacy of Tubocurarine can be increased when used in combination with Magnesium stearate.
Colistin The therapeutic efficacy of Tubocurarine can be increased when used in combination with Colistin.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Tubocurarine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Tubocurarine.
Dipyridamole The therapeutic efficacy of Tubocurarine can be decreased when used in combination with Dipyridamole.
Ephedrine Tubocurarine may increase the neuromuscular blocking activities of Ephedrine.
Sar9, Met (O2)11-Substance P Tubocurarine may increase the neuromuscular blocking activities of Sar9, Met (O2)11-Substance P.
Mirabegron Tubocurarine may increase the neuromuscular blocking activities of Mirabegron.
Moxisylyte Tubocurarine may increase the neuromuscular blocking activities of Moxisylyte.
Propacetamol Tubocurarine may increase the neuromuscular blocking activities of Propacetamol.
Pegvisomant Pegvisomant may increase the neuromuscular blocking activities of Tubocurarine.
Mefloquine Mefloquine may increase the neuromuscular blocking activities of Tubocurarine.
Tacrine Tacrine may increase the neuromuscular blocking activities of Tubocurarine.
Sulpiride Sulpiride may increase the neuromuscular blocking activities of Tubocurarine.
Profenamine Profenamine may increase the neuromuscular blocking activities of Tubocurarine.
Chlorpromazine Chlorpromazine may increase the neuromuscular blocking activities of Tubocurarine.

Target Protein

Neuronal acetylcholine receptor subunit alpha-2 CHRNA2
5-hydroxytryptamine receptor 3A HTR3A
Acetylcholinesterase ACHE
Neuronal acetylcholine receptor subunit alpha-7 CHRNA7

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16402115
    Bowman WC: Neuromuscular block. Br J Pharmacol. 2006 Jan;147 Suppl 1:S277-86. doi: 10.1038/sj.bjp.0706404.
  • PMID: 20205728
    Singla D, Sharma A, Kaur J, Panwar B, Raghava GP: BIAdb: a curated database of benzylisoquinoline alkaloids. BMC Pharmacol. 2010 Mar 5;10:4. doi: 10.1186/1471-2210-10-4.
  • PMID: 6465573
    Matteo RS, Lieberman IG, Salanitre E, McDaniel DD, Diaz J: Distribution, elimination, and action of d-tubocurarine in neonates, infants, children, and adults. Anesth Analg. 1984 Sep;63(9):799-804.
  • PMID: 31570201
    Huang L, Sang CN, Desai MS: A Chronology for the Identification and Disclosure of Adverse Effects of Succinylcholine. J Anesth Hist. 2019 Jul;5(3):65-84. doi: 10.1016/j.janh.2018.07.003. Epub 2018 Jul 29.
  • PMID: 16119481
    Ball C, Westhorpe R: Muscle relaxants--d-tubocurarine. Anaesth Intensive Care. 2005 Aug;33(4):431. doi: 10.1177/0310057X0503300401.
  • PMID: 8159634
    Bevan DR: Newer neuromuscular blocking agents. Pharmacol Toxicol. 1994 Jan;74(1):3-9. doi: 10.1111/j.1600-0773.1994.tb01065.x.

Contoh Produk & Brand

Produk: 2 • International brands: 1
Produk
  • Tubocurarine Chloride Inj 3mg/ml
    Solution • 3 mg / mL • Intravenous • Canada • Approved
  • Tubocurarine Chloride Inj 3mg/ml USP
    Solution • 3 mg / mL • Intramuscular; Intravenous • Canada • Approved
International Brands
  • Tubarine

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul