Peringatan Keamanan

Oral, rat LD50: 15 mg/kg. Symptoms of overdose include nausea, vomiting, convulsions, decreased blood pressure, and CNS stimulation.

Pergolide

DB01186

small molecule approved investigational vet_approved withdrawn

Deskripsi

Pergolide is a long-acting dopamine agonist approved in 1982 for the treatment of Parkinson’s Disease. It is an ergot derivative that acts on the dopamine D2 and D3, alpha2- and alpha1-adrenergic, and 5-hydroxytryptamine (5-HT) receptors. It was indicated as adjunct therapy with levodopa/carbidopa in the symptomatic treatment of parkinsonian syndrome. It was later found that pergolide increased the risk of cardiac valvulopathy. The drug was withdrawn from the US market in March 2007 and from the Canadian market in August 2007. While the use of pergolide in humans is still approved in only some countries, pergolide is mainly used for veterinary purposes.

Struktur Molekul 2D

Berat 314.488
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 27 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Significant amount may be absorbed (evidence on bioavailability still lacking).

Metabolisme

Extensively hepatic.

Rute Eliminasi

The major route of excretion is the kidney.

Interaksi Makanan

1 Data
  • 1. Take with or without food.

Interaksi Obat

1257 Data
Valsartan Pergolide may decrease the antihypertensive activities of Valsartan.
Ramipril Pergolide may decrease the antihypertensive activities of Ramipril.
Remikiren Pergolide may decrease the antihypertensive activities of Remikiren.
Torasemide Pergolide may decrease the antihypertensive activities of Torasemide.
Olmesartan Pergolide may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Pergolide may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Pergolide may decrease the antihypertensive activities of Nitroprusside.
Minoxidil Pergolide may decrease the antihypertensive activities of Minoxidil.
Treprostinil Pergolide may decrease the antihypertensive activities of Treprostinil.
Bendroflumethiazide Pergolide may decrease the antihypertensive activities of Bendroflumethiazide.
Fosinopril Pergolide may decrease the antihypertensive activities of Fosinopril.
Trandolapril Pergolide may decrease the antihypertensive activities of Trandolapril.
Metolazone Pergolide may decrease the antihypertensive activities of Metolazone.
Benazepril Pergolide may decrease the antihypertensive activities of Benazepril.
Cyclothiazide Pergolide may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Pergolide may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Pergolide may decrease the antihypertensive activities of Mecamylamine.
Moexipril Pergolide may decrease the antihypertensive activities of Moexipril.
Lisinopril Pergolide may decrease the antihypertensive activities of Lisinopril.
Hydroflumethiazide Pergolide may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Pergolide may decrease the antihypertensive activities of Cryptenamine.
Perindopril Pergolide may decrease the antihypertensive activities of Perindopril.
Candesartan cilexetil Pergolide may decrease the antihypertensive activities of Candesartan cilexetil.
Eprosartan Pergolide may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Pergolide may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Pergolide may decrease the antihypertensive activities of Quinapril.
Telmisartan Pergolide may decrease the antihypertensive activities of Telmisartan.
Hydrochlorothiazide Pergolide may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Pergolide may decrease the antihypertensive activities of Trichlormethiazide.
Deserpidine Pergolide may decrease the antihypertensive activities of Deserpidine.
Pentolinium Pergolide may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Pergolide may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Pergolide may decrease the antihypertensive activities of Diazoxide.
Epoprostenol Pergolide may decrease the antihypertensive activities of Epoprostenol.
Polythiazide Pergolide may decrease the antihypertensive activities of Polythiazide.
Cilazapril Pergolide may decrease the antihypertensive activities of Cilazapril.
Saprisartan Pergolide may decrease the antihypertensive activities of Saprisartan.
Spirapril Pergolide may decrease the antihypertensive activities of Spirapril.
Tienilic acid Pergolide may decrease the antihypertensive activities of Tienilic acid.
Diethylnorspermine Pergolide may decrease the antihypertensive activities of Diethylnorspermine.
Temocapril Pergolide may decrease the antihypertensive activities of Temocapril.
Nicorandil Pergolide may decrease the antihypertensive activities of Nicorandil.
Rauwolfia serpentina root Pergolide may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Pergolide may decrease the antihypertensive activities of Enalaprilat.
Angiotensin 1-7 Pergolide may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Pergolide may decrease the antihypertensive activities of Imidapril.
BQ-123 Pergolide may decrease the antihypertensive activities of BQ-123.
Cicletanine Pergolide may decrease the antihypertensive activities of Cicletanine.
Dihydralazine Pergolide may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Pergolide may decrease the antihypertensive activities of Zofenopril.
Guanoxan Pergolide may decrease the antihypertensive activities of Guanoxan.
Delapril Pergolide may decrease the antihypertensive activities of Delapril.
Vincamine Pergolide may decrease the antihypertensive activities of Vincamine.
Linsidomine Pergolide may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Pergolide may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Pergolide may decrease the antihypertensive activities of Tolonidine.
Endralazine Pergolide may decrease the antihypertensive activities of Endralazine.
Cadralazine Pergolide may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Pergolide may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Pergolide may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Pergolide may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Pergolide may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Pergolide may decrease the antihypertensive activities of Guanoclor.
Muzolimine Pergolide may decrease the antihypertensive activities of Muzolimine.
Xipamide Pergolide may decrease the antihypertensive activities of Xipamide.
Candesartan Pergolide may decrease the antihypertensive activities of Candesartan.
Tocopherylquinone Pergolide may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Pergolide may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Pergolide may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Pergolide may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Pergolide may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Pergolide may decrease the antihypertensive activities of Quinaprilat.
Furosemide Pergolide may decrease the antihypertensive activities of Furosemide.
Enalapril Pergolide may decrease the antihypertensive activities of Enalapril.
Captopril Pergolide may decrease the antihypertensive activities of Captopril.
Isradipine Pergolide may decrease the antihypertensive activities of Isradipine.
Amlodipine Pergolide may decrease the antihypertensive activities of Amlodipine.
Nimodipine Pergolide may decrease the antihypertensive activities of Nimodipine.
Lercanidipine Pergolide may decrease the antihypertensive activities of Lercanidipine.
Bosentan Pergolide may decrease the antihypertensive activities of Bosentan.
Losartan Pergolide may decrease the antihypertensive activities of Losartan.
Indapamide Pergolide may decrease the antihypertensive activities of Indapamide.
Irbesartan Pergolide may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Pergolide may decrease the antihypertensive activities of Nitrendipine.
Hydralazine Pergolide may decrease the antihypertensive activities of Hydralazine.
Mibefradil Pergolide may decrease the antihypertensive activities of Mibefradil.
Sitaxentan Pergolide may decrease the antihypertensive activities of Sitaxentan.
Ambrisentan Pergolide may decrease the antihypertensive activities of Ambrisentan.
Nilvadipine Pergolide may decrease the antihypertensive activities of Nilvadipine.
Pinacidil Pergolide may decrease the antihypertensive activities of Pinacidil.
Riociguat Pergolide may decrease the antihypertensive activities of Riociguat.
Macitentan Pergolide may decrease the antihypertensive activities of Macitentan.
Aliskiren Pergolide may decrease the antihypertensive activities of Aliskiren.
Efonidipine Pergolide may decrease the antihypertensive activities of Efonidipine.
Lacidipine Pergolide may decrease the antihypertensive activities of Lacidipine.
Manidipine Pergolide may decrease the antihypertensive activities of Manidipine.
Selexipag Pergolide may decrease the antihypertensive activities of Selexipag.
Naftopidil Pergolide may decrease the antihypertensive activities of Naftopidil.
Dexniguldipine Pergolide may decrease the antihypertensive activities of Dexniguldipine.
Tadalafil Pergolide may decrease the antihypertensive activities of Tadalafil.

Target Protein

D(2) dopamine receptor DRD2
D(3) dopamine receptor DRD3
D(4) dopamine receptor DRD4
D(1B) dopamine receptor DRD5
D(1A) dopamine receptor DRD1
5-hydroxytryptamine receptor 1A HTR1A
5-hydroxytryptamine receptor 2B HTR2B
5-hydroxytryptamine receptor 2A HTR2A
5-hydroxytryptamine receptor 1D HTR1D
Alpha-2 adrenergic receptors ADRA2A
5-hydroxytryptamine receptor 1B HTR1B
5-hydroxytryptamine receptor 2C HTR2C
Alpha-1A adrenergic receptor ADRA1A
Alpha-1B adrenergic receptor ADRA1B
Alpha-1D adrenergic receptor ADRA1D

Referensi & Sumber

Artikel (PubMed)
  • PMID: 17202453
    Schade R, Andersohn F, Suissa S, Haverkamp W, Garbe E: Dopamine agonists and the risk of cardiac-valve regurgitation. N Engl J Med. 2007 Jan 4;356(1):29-38.
  • PMID: 16880771
    Breitenstein C, Korsukewitz C, Floel A, Kretzschmar T, Diederich K, Knecht S: Tonic dopaminergic stimulation impairs associative learning in healthy subjects. Neuropsychopharmacology. 2006 Nov;31(11):2552-64. Epub 2006 Jul 26.

Contoh Produk & Brand

Produk: 12 • International brands: 0
Produk
  • Pergolide Mesylate
    Tablet • 0.25 mg/1 • Oral • US • Generic • Approved
  • Pergolide Mesylate
    Tablet • 0.05 mg/1 • Oral • US • Generic • Approved
  • Pergolide Mesylate
    Tablet • 1 mg/1 • Oral • US • Generic • Approved
  • Pergolide Mesylate
    Tablet • 0.05 mg/1 • Oral • US • Generic • Approved
  • Pergolide Mesylate
    Tablet • 0.25 mg/1 • Oral • US • Generic • Approved
  • Pergolide Mesylate
    Tablet • 1 mg/1 • Oral • US • Generic • Approved
  • Permax
    Tablet • 0.05 mg/1 • Oral • US • Approved
  • Permax
    Tablet • 0.25 mg/1 • Oral • US • Approved
Menampilkan 8 dari 12 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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