Peringatan Keamanan

Oral, mouse LD50 = 100 mg/kg; oral, rat LD50 = 255 mg/kg

Orphenadrine

DB01173

small molecule approved

Deskripsi

A muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.

Struktur Molekul 2D

Berat 269.3813
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 13-20 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Orphenadrine is almost completely absorbed in the gastrointestinal tract.

Metabolisme

Biotransformation occurs mainly in the liver. Pharmacologically active metabolites are N-demethyl orphenadrine and N,N-didemethyl orphenadrine.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with or without food. Food does not significantly affect absorption.

Interaksi Obat

1521 Data
Lomitapide The metabolism of Lomitapide can be decreased when combined with Orphenadrine.
Buprenorphine Orphenadrine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Dronabinol The serum concentration of Dronabinol can be increased when it is combined with Orphenadrine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Hydrocodone Orphenadrine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Magnesium sulfate The therapeutic efficacy of Orphenadrine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Orphenadrine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Orphenadrine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Mirtazapine Orphenadrine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Botulinum toxin type B Botulinum toxin type B may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Tryptophan Tryptophan may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Fluvoxamine Fluvoxamine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Lorazepam Lorazepam may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Ethchlorvynol Ethchlorvynol may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Succinylcholine Succinylcholine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Reserpine Reserpine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Citalopram The risk or severity of QTc prolongation can be increased when Orphenadrine is combined with Citalopram.
Eletriptan Eletriptan may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Enflurane Enflurane may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Temazepam Temazepam may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Reboxetine Reboxetine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Butabarbital Butabarbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Butalbital Butalbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Methysergide Methysergide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Cabergoline Cabergoline may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Clemastine Clemastine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Venlafaxine Venlafaxine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Etomidate Etomidate may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Morphine Morphine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Talbutal Talbutal may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Pentobarbital Pentobarbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Valproic acid Valproic acid may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Codeine Codeine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Dihydroergotamine Dihydroergotamine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Tolcapone Tolcapone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Hydromorphone Hydromorphone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Olanzapine Olanzapine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Cetirizine Cetirizine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Protriptyline Protriptyline may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Trimethadione Trimethadione may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Clobazam The risk or severity of sedation, somnolence, and CNS depression can be increased when Clobazam is combined with Orphenadrine.
Chlorzoxazone Chlorzoxazone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Clozapine The serum concentration of Clozapine can be increased when it is combined with Orphenadrine.
Meprobamate Meprobamate may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Thiethylperazine Thiethylperazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Palonosetron Palonosetron may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Sulpiride Sulpiride may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Dexbrompheniramine Dexbrompheniramine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Loxapine Loxapine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Remoxipride Remoxipride may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Metocurine iodide Metocurine iodide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Secobarbital Secobarbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Promazine Promazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Methocarbamol Methocarbamol may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Triprolidine Triprolidine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Prochlorperazine Prochlorperazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Cyproheptadine Cyproheptadine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Meperidine Meperidine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Imipramine Imipramine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Metharbital Metharbital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Quinine Quinine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Methohexital Methohexital may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Chlordiazepoxide Chlordiazepoxide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Duloxetine Duloxetine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Chlorpromazine Chlorpromazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Gallamine triethiodide Gallamine triethiodide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Entacapone Entacapone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Oxycodone Oxycodone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Triflupromazine Triflupromazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Dextromethorphan Dextromethorphan may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Mephenytoin Mephenytoin may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Nortriptyline Nortriptyline may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Amoxapine Amoxapine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Adinazolam Adinazolam may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Lamotrigine Lamotrigine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Carbamazepine Carbamazepine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Cisatracurium Cisatracurium may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Fenfluramine Fenfluramine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Mazindol Mazindol may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Fluticasone propionate Fluticasone propionate may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Lisuride Lisuride may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Ethosuximide Ethosuximide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Thiopental Thiopental may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Cisapride Cisapride may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Butorphanol Butorphanol may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Furazolidone Furazolidone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paramethadione Paramethadione may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Fluphenazine Fluphenazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Efavirenz Efavirenz may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Clorazepic acid Clorazepic acid may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Dexmedetomidine Dexmedetomidine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Dyclonine Dyclonine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Dextropropoxyphene Dextropropoxyphene may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Pentazocine Pentazocine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Metaxalone Metaxalone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Trimethobenzamide Trimethobenzamide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.

Target Protein

Glutamate receptor ionotropic, NMDA 2D GRIN2D
Glutamate receptor ionotropic, NMDA 1 GRIN1
Glutamate receptor ionotropic, NMDA 3B GRIN3B
Glutamate receptor ionotropic, NMDA 3A GRIN3A
Histamine H1 receptor HRH1
Sodium-dependent noradrenaline transporter SLC6A2
Sodium channel protein type 10 subunit alpha SCN10A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 15662845
    Ji D, Sui ZY, Ma YY, Luo F, Cui CL, Han JS: NMDA receptor in nucleus accumbens is implicated in morphine withdrawal in rats. Neurochem Res. 2004 Nov;29(11):2113-20.

Contoh Produk & Brand

Produk: 83 • International brands: 8
Produk
  • Disipal Tab 50mg
    Tablet • 50 mg • Oral • Canada • Approved
  • Norflex
    Tablet, extended release • 100 mg/1 • Oral • US
  • Norflex
    Injection • 60 mg/2mL • Intramuscular; Intravenous • US • Approved
  • Norflex
    Tablet, extended release • 100000 ug/1 • Oral • US • Approved
  • Norflex
    Injection • 60 mg/2mL • Intramuscular; Intravenous • US • Approved
  • Norflex
    Liquid • 30 mg / mL • Intramuscular; Intravenous • Canada • Approved
  • Norflex
    Tablet, extended release • 100 mg • Oral • Canada • OTC • Approved
  • Norgesic
    Tablet, multilayer • - • Oral • US • Approved
Menampilkan 8 dari 83 produk.
International Brands
  • Antiflex
  • Banflex
  • Biorphen
  • Disipal
  • Flexoject
  • Mio-Rel
  • OrfenAce
  • Orfro

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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