Peringatan Keamanan

Side effects include drowsiness, dizziness, tiredness or confusion. LD50=1000 mg/kg (mouse, oral)

Guanethidine

DB01170

small molecule approved

Deskripsi

An antihypertensive agent that acts by inhibiting selectively transmission in post-ganglionic adrenergic nerves. It is believed to act mainly by preventing the release of norepinephrine at nerve endings and causes depletion of norepinephrine in peripheral sympathetic nerve terminals as well as in tissues. PubChem

Struktur Molekul 2D

Berat 198.3085
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 1.5 days
Volume Distribusi -
Klirens (Clearance) * Renal cl=56 ml/min

Absorpsi

3-30% of oral dose (poor and highly variable)

Metabolisme

Guanethidine is converted by the liver to three metabolites, which are excreted in the urine. The metabolites are pharmacologically less active than the parent compound.

Rute Eliminasi

Ismelin is converted by the liver to three metabolites, which are excreted in the urine.

Interaksi Makanan

1 Data
  • 1. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

1147 Data
Alfuzosin Alfuzosin may increase the hypotensive activities of Guanethidine.
Amifostine Guanethidine may increase the hypotensive activities of Amifostine.
Diazoxide Diazoxide may increase the hypotensive activities of Guanethidine.
Methylphenidate Methylphenidate may decrease the antihypertensive activities of Guanethidine.
Dexmethylphenidate Dexmethylphenidate may decrease the antihypertensive activities of Guanethidine.
Obinutuzumab Guanethidine may increase the hypotensive activities of Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the hypotensive activities of Guanethidine.
Rituximab Guanethidine may increase the hypotensive activities of Rituximab.
Zolmitriptan Zolmitriptan may decrease the antihypertensive activities of Guanethidine.
Protriptyline Protriptyline may decrease the antihypertensive activities of Guanethidine.
Droperidol Droperidol may decrease the antihypertensive activities of Guanethidine.
Amoxapine Amoxapine may decrease the antihypertensive activities of Guanethidine.
Doxapram Doxapram may decrease the antihypertensive activities of Guanethidine.
Atropine Atropine may decrease the antihypertensive activities of Guanethidine.
Nicergoline Nicergoline may decrease the antihypertensive activities of Guanethidine.
Propiomazine Propiomazine may decrease the antihypertensive activities of Guanethidine.
Phenmetrazine Phenmetrazine may decrease the antihypertensive activities of Guanethidine.
Trifluoperazine Trifluoperazine may decrease the antihypertensive activities of Guanethidine.
Naratriptan Naratriptan may decrease the antihypertensive activities of Guanethidine.
Frovatriptan Frovatriptan may decrease the antihypertensive activities of Guanethidine.
Methotrimeprazine Methotrimeprazine may decrease the antihypertensive activities of Guanethidine.
Periciazine Periciazine may decrease the antihypertensive activities of Guanethidine.
Acepromazine Acepromazine may decrease the antihypertensive activities of Guanethidine.
Thioproperazine Thioproperazine may decrease the antihypertensive activities of Guanethidine.
Epicaptopril Epicaptopril may decrease the antihypertensive activities of Guanethidine.
1-benzylimidazole 1-benzylimidazole may decrease the antihypertensive activities of Guanethidine.
Amineptine Amineptine may decrease the antihypertensive activities of Guanethidine.
Naluzotan Naluzotan may decrease the antihypertensive activities of Guanethidine.
Pizotifen Pizotifen may decrease the antihypertensive activities of Guanethidine.
Esmirtazapine Esmirtazapine may decrease the antihypertensive activities of Guanethidine.
Nitrous oxide Nitrous oxide may decrease the antihypertensive activities of Guanethidine.
Saralasin Saralasin may decrease the antihypertensive activities of Guanethidine.
Cinitapride Cinitapride may decrease the antihypertensive activities of Guanethidine.
Tyramine Tyramine may decrease the antihypertensive activities of Guanethidine.
Ifenprodil Ifenprodil may decrease the antihypertensive activities of Guanethidine.
Butriptyline Butriptyline may decrease the antihypertensive activities of Guanethidine.
Dosulepin Dosulepin may decrease the antihypertensive activities of Guanethidine.
Oxaprotiline Oxaprotiline may decrease the antihypertensive activities of Guanethidine.
Atipamezole Atipamezole may decrease the antihypertensive activities of Guanethidine.
Tetrahydrocannabivarin Tetrahydrocannabivarin may decrease the antihypertensive activities of Guanethidine.
Piclozotan Piclozotan may decrease the antihypertensive activities of Guanethidine.
Idazoxan Idazoxan may decrease the antihypertensive activities of Guanethidine.
Theodrenaline Theodrenaline may decrease the antihypertensive activities of Guanethidine.
Opipramol Opipramol may decrease the antihypertensive activities of Guanethidine.
Tramazoline Tramazoline may decrease the antihypertensive activities of Guanethidine.
Amitriptylinoxide Amitriptylinoxide may decrease the antihypertensive activities of Guanethidine.
Dibenzepin Dibenzepin may decrease the antihypertensive activities of Guanethidine.
Quinupramine Quinupramine may decrease the antihypertensive activities of Guanethidine.
Trichloroethylene Trichloroethylene may decrease the antihypertensive activities of Guanethidine.
Fenozolone Fenozolone may decrease the antihypertensive activities of Guanethidine.
Melitracen Melitracen may decrease the antihypertensive activities of Guanethidine.
Lofepramine Lofepramine may decrease the antihypertensive activities of Guanethidine.
Xenon Xenon may decrease the antihypertensive activities of Guanethidine.
Iprindole Iprindole may decrease the antihypertensive activities of Guanethidine.
Buflomedil Buflomedil may decrease the antihypertensive activities of Guanethidine.
Metergoline Metergoline may decrease the antihypertensive activities of Guanethidine.
Diethyl ether Diethyl ether may decrease the antihypertensive activities of Guanethidine.
Imipramine oxide Imipramine oxide may decrease the antihypertensive activities of Guanethidine.
Mefenorex Mefenorex may decrease the antihypertensive activities of Guanethidine.
Deoxyepinephrine Deoxyepinephrine may decrease the antihypertensive activities of Guanethidine.
5-methoxy-N,N-dimethyltryptamine 5-methoxy-N,N-dimethyltryptamine may decrease the antihypertensive activities of Guanethidine.
Quinoline Yellow WS Quinoline Yellow WS may decrease the antihypertensive activities of Guanethidine.
Thioridazine Thioridazine may decrease the antihypertensive activities of Guanethidine.
Isoflurane Isoflurane may decrease the antihypertensive activities of Guanethidine.
Tolazoline Tolazoline may decrease the antihypertensive activities of Guanethidine.
Propofol Propofol may decrease the antihypertensive activities of Guanethidine.
Remifentanil Remifentanil may decrease the antihypertensive activities of Guanethidine.
Phenoxybenzamine Phenoxybenzamine may decrease the antihypertensive activities of Guanethidine.
Desflurane Desflurane may decrease the antihypertensive activities of Guanethidine.
Isoxsuprine Isoxsuprine may decrease the antihypertensive activities of Guanethidine.
Indoramin Indoramin may decrease the antihypertensive activities of Guanethidine.
Moxonidine Moxonidine may decrease the antihypertensive activities of Guanethidine.
Trimipramine Trimipramine may decrease the antihypertensive activities of Guanethidine.
Dutasteride Dutasteride may decrease the antihypertensive activities of Guanethidine.
Sufentanil Sufentanil may decrease the antihypertensive activities of Guanethidine.
Halothane Halothane may decrease the antihypertensive activities of Guanethidine.
Bromocriptine Bromocriptine may decrease the antihypertensive activities of Guanethidine.
Sevoflurane Sevoflurane may decrease the antihypertensive activities of Guanethidine.
Rotigotine Rotigotine may decrease the antihypertensive activities of Guanethidine.
Eletriptan Eletriptan may decrease the antihypertensive activities of Guanethidine.
Methysergide Methysergide may decrease the antihypertensive activities of Guanethidine.
Cabergoline Cabergoline may decrease the antihypertensive activities of Guanethidine.
Dihydroergotamine Dihydroergotamine may decrease the antihypertensive activities of Guanethidine.
Methylergometrine Methylergometrine may decrease the antihypertensive activities of Guanethidine.
Mirtazapine Mirtazapine may decrease the antihypertensive activities of Guanethidine.
Promazine Promazine may decrease the antihypertensive activities of Guanethidine.
Nortriptyline Nortriptyline may decrease the antihypertensive activities of Guanethidine.
Lisuride Lisuride may decrease the antihypertensive activities of Guanethidine.
Trazodone Trazodone may decrease the antihypertensive activities of Guanethidine.
Ergotamine Ergotamine may decrease the antihypertensive activities of Guanethidine.
Risperidone Risperidone may decrease the antihypertensive activities of Guanethidine.
Alfentanil Alfentanil may decrease the antihypertensive activities of Guanethidine.
Methoxyflurane Methoxyflurane may decrease the antihypertensive activities of Guanethidine.
Ergoloid mesylate Ergoloid mesylate may decrease the antihypertensive activities of Guanethidine.
Finasteride Finasteride may decrease the antihypertensive activities of Guanethidine.
Yohimbine Yohimbine may decrease the antihypertensive activities of Guanethidine.
Solifenacin Solifenacin may decrease the antihypertensive activities of Guanethidine.
Zuclopenthixol Zuclopenthixol may decrease the antihypertensive activities of Guanethidine.
Lysergic acid diethylamide Lysergic acid diethylamide may decrease the antihypertensive activities of Guanethidine.
Dronedarone Dronedarone may decrease the antihypertensive activities of Guanethidine.

Target Protein

Sodium-dependent noradrenaline transporter SLC6A2

Referensi & Sumber

Synthesis reference: U.S. Patent 2,928,829 U.S. Patent 3,006,913 U.S. Patent 3,055,882

Contoh Produk & Brand

Produk: 6 • International brands: 1
Produk
  • Apo Guanethidine Sulfate Tab 10mg
    Tablet • 10 mg • Oral • Canada • Generic • Approved
  • Apo Guanethidine Sulfate Tab 25mg
    Tablet • 25 mg • Oral • Canada • Generic • Approved
  • Guanethidine 10 Tab 10mg
    Tablet • 10 mg / tab • Oral • Canada • Approved
  • Ismelin
    Tablet • 10 mg/1 • Oral • US • Approved
  • Ismelin
    Tablet • 25 mg/1 • Oral • US • Approved
  • Ismelin 25mg
    Tablet • 25 mg / tab • Oral • Canada • Approved
International Brands
  • Ismedine — Chen Ho

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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