Peringatan Keamanan

Cases of life-threatening hepatic failure have been reported in patients treated with nefazodone.

Nefazodone

DB01149

small molecule approved withdrawn

Deskripsi

Nefazodone hydrochloride (trade name Serzone) is an antidepressant drug marketed by Bristol-Myers Squibb. Its sale was discontinued in 2003 in some countries, due to the small possibility of hepatic (liver) injury. Drug-induced hepatic injuries were associated with an risk of elevated need for a liver transplant, or even death, with the incidence of severe liver damage was shown to be approximately 1 in 250,000 to 300,000 patient-years. On May 20, 2004, Bristol-Myers Squibb discontinued the sale of Serzone in the United States.

Struktur Molekul 2D

Berat 470.007
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 2-4 hours
Volume Distribusi * 0.22 to 0.87 L/kg
Klirens (Clearance) -

Absorpsi

Nefazodone is rapidly and completely absorbed. Its absolute bioavailability is low (about 20%).

Metabolisme

Hepatic.

Rute Eliminasi

Nefazodone is extensively metabolized after oral administration by n-dealkylation and aliphatic and aromatic hydroxylation, and less than 1% of administered nefazodone is excreted unchanged in urine.

Interaksi Makanan

3 Data
  • 1. Avoid alcohol.
  • 2. Take at the same time every day.
  • 3. Take with or without food.

Interaksi Obat

2264 Data
Troglitazone Troglitazone may decrease the excretion rate of Nefazodone which could result in a higher serum level.
Ursodeoxycholic acid Ursodeoxycholic acid may decrease the excretion rate of Nefazodone which could result in a higher serum level.
Cholic Acid Cholic Acid may decrease the excretion rate of Nefazodone which could result in a higher serum level.
Letermovir The excretion of Letermovir can be decreased when combined with Nefazodone.
Valinomycin Valinomycin may decrease the excretion rate of Nefazodone which could result in a higher serum level.
Olmesartan Olmesartan may decrease the excretion rate of Nefazodone which could result in a higher serum level.
Lenvatinib Lenvatinib may decrease the excretion rate of Nefazodone which could result in a higher serum level.
Cyproheptadine The therapeutic efficacy of Nefazodone can be decreased when used in combination with Cyproheptadine.
Desmopressin The risk or severity of hyponatremia can be increased when Nefazodone is combined with Desmopressin.
Ioflupane I-123 Nefazodone may decrease effectiveness of Ioflupane I-123 as a diagnostic agent.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Nefazodone.
Metyrosine The risk or severity of extrapyramidal symptoms can be increased when Metyrosine is combined with Nefazodone.
Pimozide The risk or severity of QTc prolongation can be increased when Nefazodone is combined with Pimozide.
Ramipril Nefazodone may decrease the antihypertensive activities of Ramipril.
Remikiren Nefazodone may decrease the antihypertensive activities of Remikiren.
Guanadrel Nefazodone may decrease the antihypertensive activities of Guanadrel.
Minoxidil Nefazodone may decrease the antihypertensive activities of Minoxidil.
Treprostinil Nefazodone may decrease the antihypertensive activities of Treprostinil.
Trandolapril Nefazodone may decrease the antihypertensive activities of Trandolapril.
Benazepril Nefazodone may decrease the antihypertensive activities of Benazepril.
Candoxatril Nefazodone may decrease the antihypertensive activities of Candoxatril.
Moexipril Nefazodone may decrease the antihypertensive activities of Moexipril.
Nitroglycerin Nefazodone may decrease the antihypertensive activities of Nitroglycerin.
Cryptenamine Nefazodone may decrease the antihypertensive activities of Cryptenamine.
Candesartan cilexetil Nefazodone may decrease the antihypertensive activities of Candesartan cilexetil.
Eprosartan Nefazodone may decrease the antihypertensive activities of Eprosartan.
Quinapril Nefazodone may decrease the antihypertensive activities of Quinapril.
Deserpidine Nefazodone may decrease the antihypertensive activities of Deserpidine.
Pentolinium Nefazodone may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Nefazodone may decrease the antihypertensive activities of Trimethaphan.
Bretylium Nefazodone may decrease the antihypertensive activities of Bretylium.
Cilazapril Nefazodone may decrease the antihypertensive activities of Cilazapril.
Saprisartan Nefazodone may decrease the antihypertensive activities of Saprisartan.
Spirapril Nefazodone may decrease the antihypertensive activities of Spirapril.
Diethylnorspermine Nefazodone may decrease the antihypertensive activities of Diethylnorspermine.
Temocapril Nefazodone may decrease the antihypertensive activities of Temocapril.
Rauwolfia serpentina root Nefazodone may decrease the antihypertensive activities of Rauwolfia serpentina root.
Angiotensin 1-7 Nefazodone may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Nefazodone may decrease the antihypertensive activities of Imidapril.
BQ-123 Nefazodone may decrease the antihypertensive activities of BQ-123.
Dihydralazine Nefazodone may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Nefazodone may decrease the antihypertensive activities of Zofenopril.
Guanoxan Nefazodone may decrease the antihypertensive activities of Guanoxan.
Delapril Nefazodone may decrease the antihypertensive activities of Delapril.
Vincamine Nefazodone may decrease the antihypertensive activities of Vincamine.
Guanoxabenz Nefazodone may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Nefazodone may decrease the antihypertensive activities of Tolonidine.
Endralazine Nefazodone may decrease the antihypertensive activities of Endralazine.
Cadralazine Nefazodone may decrease the antihypertensive activities of Cadralazine.
Bietaserpine Nefazodone may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Nefazodone may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Nefazodone may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Nefazodone may decrease the antihypertensive activities of Guanoclor.
Candesartan Nefazodone may decrease the antihypertensive activities of Candesartan.
Benazeprilat Nefazodone may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Nefazodone may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Nefazodone may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Nefazodone may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Nefazodone may decrease the antihypertensive activities of Quinaprilat.
Enalapril Nefazodone may decrease the antihypertensive activities of Enalapril.
Captopril Nefazodone may decrease the antihypertensive activities of Captopril.
Irbesartan Nefazodone may decrease the antihypertensive activities of Irbesartan.
Sitaxentan Nefazodone may decrease the antihypertensive activities of Sitaxentan.
Azilsartan medoxomil Nefazodone may decrease the antihypertensive activities of Azilsartan medoxomil.
Diazoxide Nefazodone may decrease the antihypertensive activities of Diazoxide.
Buprenorphine Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Nefazodone.
Dronabinol The serum concentration of Dronabinol can be increased when it is combined with Nefazodone.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Nefazodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Nefazodone.
Magnesium sulfate The therapeutic efficacy of Nefazodone can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Nefazodone.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Nefazodone.
Orphenadrine Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Nefazodone.
Pramipexole Nefazodone may increase the sedative activities of Pramipexole.
Ropinirole Nefazodone may increase the sedative activities of Ropinirole.
Rotigotine Nefazodone may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Nefazodone.
Sodium oxybate Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Nefazodone.
Thalidomide Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Nefazodone may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Nefazodone.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Nefazodone.
Doxapram The risk or severity of hypertension can be increased when Doxapram is combined with Nefazodone.
Phenmetrazine The risk or severity of hypertension can be increased when Phenmetrazine is combined with Nefazodone.
Omapatrilat Nefazodone may decrease the antihypertensive activities of Omapatrilat.
Rescinnamine Nefazodone may decrease the antihypertensive activities of Rescinnamine.
Epicaptopril The risk or severity of hypertension can be increased when Nefazodone is combined with Epicaptopril.
1-benzylimidazole The risk or severity of hypertension can be increased when Nefazodone is combined with 1-benzylimidazole.
Saralasin The risk or severity of hypertension can be increased when Nefazodone is combined with Saralasin.
Tyramine The risk or severity of hypertension can be increased when Nefazodone is combined with Tyramine.
Atipamezole The risk or severity of hypertension can be increased when Nefazodone is combined with Atipamezole.
Idazoxan The risk or severity of hypertension can be increased when Nefazodone is combined with Idazoxan.
Tramazoline The risk or severity of hypertension can be increased when Nefazodone is combined with Tramazoline.
Fenozolone The risk or severity of hypertension can be increased when Nefazodone is combined with Fenozolone.

Target Protein

5-hydroxytryptamine receptor 2A HTR2A
5-hydroxytryptamine receptor 2C HTR2C
Sodium-dependent serotonin transporter SLC6A4
5-hydroxytryptamine receptor 1A HTR1A
Sodium-dependent noradrenaline transporter SLC6A2
Sodium-dependent dopamine transporter SLC6A3
Alpha-1B adrenergic receptor ADRA1B
Alpha-2A adrenergic receptor ADRA2A
Alpha-1A adrenergic receptor ADRA1A
Voltage-gated inwardly rectifying potassium channel KCNH2 KCNH2

Referensi & Sumber

Artikel (PubMed)
  • PMID: 9098663
    Davis R, Whittington R, Bryson HM: Nefazodone. A review of its pharmacology and clinical efficacy in the management of major depression. Drugs. 1997 Apr;53(4):608-36.

Contoh Produk & Brand

Produk: 41 • International brands: 1
Produk
  • Lin-nefazodone
    Tablet • 50 mg / tab • Oral • Canada • Generic • Approved
  • Lin-nefazodone
    Tablet • 100 mg / tab • Oral • Canada • Generic • Approved
  • Lin-nefazodone
    Tablet • 150 mg / tab • Oral • Canada • Generic • Approved
  • Lin-nefazodone
    Tablet • 200 mg / tab • Oral • Canada • Generic • Approved
  • Nefazodone hydrochloride
    Tablet • 50 mg/1 • Oral • US • Approved
  • Nefazodone hydrochloride
    Tablet • 100 mg/1 • Oral • US • Approved
  • Nefazodone hydrochloride
    Tablet • 150 mg/1 • Oral • US • Approved
  • Nefazodone hydrochloride
    Tablet • 200 mg/1 • Oral • US • Approved
Menampilkan 8 dari 41 produk.
International Brands
  • Dutonin

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul