Peringatan Keamanan

Rats exposed via the oral route to cephapirin displayed low acute toxicity (LD50 = 14000 mg/kg). The most common adverse reactions are hypersensitivity reactions and alterations to liver function. Evidence of white blood cell disorders and anaemia were noted in some subjects.

Cefapirin

DB01139

small molecule approved vet_approved

Deskripsi

Cefapirin (INN, also spelled cephapirin), commonly marketed under the trade name Cefadyl, is a first-generation cephalosporin antibiotic that is available in injectable formulations. Production for use in humans has been discontinued in the United States. Cefapirin is partly plasma-bound and is effective against gram-negative and gram-positive organisms.

Struktur Molekul 2D

Berat 423.463
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Major metabolite detected is desacetylcephapirin.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

796 Data
Probenecid The serum concentration of Cefapirin can be increased when it is combined with Probenecid.
Foscarnet The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Foscarnet.
Mannitol The risk or severity of nephrotoxicity can be increased when Mannitol is combined with Cefapirin.
Tenofovir disoproxil Cefapirin may increase the nephrotoxic activities of Tenofovir disoproxil.
Tenofovir alafenamide Cefapirin may increase the nephrotoxic activities of Tenofovir alafenamide.
Tenofovir Cefapirin may increase the nephrotoxic activities of Tenofovir.
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Cefapirin.
Cyclosporine The risk or severity of nephrotoxicity can be increased when Cyclosporine is combined with Cefapirin.
Icosapent The risk or severity of nephrotoxicity can be increased when Icosapent is combined with Cefapirin.
Cefotiam The risk or severity of nephrotoxicity can be increased when Cefotiam is combined with Cefapirin.
Mesalazine The risk or severity of nephrotoxicity can be increased when Mesalazine is combined with Cefapirin.
Cefmenoxime The risk or severity of nephrotoxicity can be increased when Cefmenoxime is combined with Cefapirin.
Cefmetazole The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Cefapirin.
Indomethacin The risk or severity of nephrotoxicity can be increased when Indomethacin is combined with Cefapirin.
Triamterene The risk or severity of nephrotoxicity can be increased when Triamterene is combined with Cefapirin.
Cefpiramide The risk or severity of nephrotoxicity can be increased when Cefpiramide is combined with Cefapirin.
Loracarbef The risk or severity of nephrotoxicity can be increased when Loracarbef is combined with Cefapirin.
Cefalotin The risk or severity of nephrotoxicity can be increased when Cefalotin is combined with Cefapirin.
Nabumetone The risk or severity of nephrotoxicity can be increased when Nabumetone is combined with Cefapirin.
Ketorolac The risk or severity of nephrotoxicity can be increased when Ketorolac is combined with Cefapirin.
Tenoxicam The risk or severity of nephrotoxicity can be increased when Tenoxicam is combined with Cefapirin.
Celecoxib The risk or severity of nephrotoxicity can be increased when Celecoxib is combined with Cefapirin.
Cefotaxime The risk or severity of nephrotoxicity can be increased when Cefotaxime is combined with Cefapirin.
Tolmetin The risk or severity of nephrotoxicity can be increased when Tolmetin is combined with Cefapirin.
Rofecoxib The risk or severity of nephrotoxicity can be increased when Rofecoxib is combined with Cefapirin.
Fenoprofen The risk or severity of nephrotoxicity can be increased when Fenoprofen is combined with Cefapirin.
Valdecoxib The risk or severity of nephrotoxicity can be increased when Valdecoxib is combined with Cefapirin.
Diclofenac The risk or severity of nephrotoxicity can be increased when Diclofenac is combined with Cefapirin.
Sulindac The risk or severity of nephrotoxicity can be increased when Sulindac is combined with Cefapirin.
Bacitracin The risk or severity of nephrotoxicity can be increased when Bacitracin is combined with Cefapirin.
Amphotericin B The risk or severity of nephrotoxicity can be increased when Amphotericin B is combined with Cefapirin.
Cephaloglycin The risk or severity of nephrotoxicity can be increased when Cephaloglycin is combined with Cefapirin.
Adefovir dipivoxil The risk or severity of nephrotoxicity can be increased when Adefovir dipivoxil is combined with Cefapirin.
Pentamidine The risk or severity of nephrotoxicity can be increased when Pentamidine is combined with Cefapirin.
Mefenamic acid The risk or severity of nephrotoxicity can be increased when Mefenamic acid is combined with Cefapirin.
Naproxen The risk or severity of nephrotoxicity can be increased when Naproxen is combined with Cefapirin.
Sulfasalazine The risk or severity of nephrotoxicity can be increased when Sulfasalazine is combined with Cefapirin.
Phenylbutazone The risk or severity of nephrotoxicity can be increased when Phenylbutazone is combined with Cefapirin.
Meloxicam The risk or severity of methemoglobinemia can be increased when Cefapirin is combined with Meloxicam.
Carprofen The risk or severity of nephrotoxicity can be increased when Carprofen is combined with Cefapirin.
Tacrolimus The risk or severity of nephrotoxicity can be increased when Tacrolimus is combined with Cefapirin.
Etacrynic acid The risk or severity of nephrotoxicity can be increased when Etacrynic acid is combined with Cefapirin.
Ceforanide The risk or severity of nephrotoxicity can be increased when Ceforanide is combined with Cefapirin.
Salicylic acid The risk or severity of nephrotoxicity can be increased when Salicylic acid is combined with Cefapirin.
Acetylsalicylic acid The risk or severity of nephrotoxicity can be increased when Acetylsalicylic acid is combined with Cefapirin.
Hydrochlorothiazide The risk or severity of nephrotoxicity can be increased when Hydrochlorothiazide is combined with Cefapirin.
Balsalazide The risk or severity of nephrotoxicity can be increased when Balsalazide is combined with Cefapirin.
Cefditoren The risk or severity of nephrotoxicity can be increased when Cefditoren is combined with Cefapirin.
Atazanavir The risk or severity of nephrotoxicity can be increased when Atazanavir is combined with Cefapirin.
Colistimethate The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefapirin.
Cefuroxime The risk or severity of nephrotoxicity can be increased when Cefuroxime is combined with Cefapirin.
Cefprozil The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefprozil.
Olsalazine The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Olsalazine.
Lumiracoxib The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Lumiracoxib.
Cefamandole The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefamandole.
Cefazolin The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefazolin.
Cefonicid The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefonicid.
Cefoperazone The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefoperazone.
Cefoxitin The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefoxitin.
Ceftizoxime The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Ceftizoxime.
Magnesium salicylate The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Magnesium salicylate.
Salsalate The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Salsalate.
Choline magnesium trisalicylate The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Choline magnesium trisalicylate.
Cefepime The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefepime.
Cefacetrile The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefacetrile.
Cefpodoxime The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefpodoxime.
Antrafenine The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Antrafenine.
Aminophenazone The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Aminophenazone.
Antipyrine The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Antipyrine.
Tiaprofenic acid The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Tiaprofenic acid.
Lopinavir The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Lopinavir.
Etoricoxib The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Etoricoxib.
Hydrolyzed Cephalothin The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Hydrolyzed Cephalothin.
Cephalothin Group The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cephalothin Group.
Oxyphenbutazone The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Oxyphenbutazone.
Latamoxef The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Latamoxef.
Nimesulide The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Nimesulide.
Benoxaprofen The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Benoxaprofen.
Metamizole The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Metamizole.
Zomepirac The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Zomepirac.
Ceftobiprole The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Ceftobiprole.
Cimicoxib The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cimicoxib.
Ceftaroline fosamil The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Ceftaroline fosamil.
Lornoxicam The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Lornoxicam.
Zaltoprofen The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Zaltoprofen.
Azapropazone The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Azapropazone.
Parecoxib The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Parecoxib.
Salicylamide The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Salicylamide.
Kebuzone The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Kebuzone.
Isoxicam The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Isoxicam.
Indoprofen The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Indoprofen.
Ibuproxam The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Ibuproxam.
Floctafenine The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Floctafenine.
Fenbufen The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Fenbufen.
Etofenamate The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Etofenamate.
Epirizole The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Epirizole.
Cefaloridine The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefaloridine.
Cefminox The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Cefminox.
Dexibuprofen The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Dexibuprofen.
Droxicam The risk or severity of nephrotoxicity can be increased when Cefapirin is combined with Droxicam.

Target Protein

Penicillin-binding protein 1A pbpA

Referensi & Sumber

Synthesis reference: Crast, L.B. Jr.; U.S. Patent 3,422,100; January 14, 1969; assigned to Bristol-Myers Company Silvestri, H.H.and Johnson, D.A.; US. Patent 3,503,967; March 31,1970; assigned to Bristol-Myers Company. Havranek, R.E. and Crast, L.B. Jr.; U.S. Patent 3,578,661; May 11, 1971; assigned to Bristol- Myers Company.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • Cefadyl

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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