Rabeprazole

DB01129

small molecule approved investigational

Deskripsi

Rabeprazole is an antiulcer drug in the class of proton pump inhibitors. It is a prodrug - in the acid environment of the parietal cells it turns into active sulphenamide form. Rabeprazole inhibits the H+, K+ATPase of the coating gastric cells and dose-dependent oppresses basal and stimulated gastric acid secretion.

Struktur Molekul 2D

Berat 359.443
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 1-2 hours (in plasma)
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Absolute bioavailability is approximately 52%.

Metabolisme

Hepatic

Rute Eliminasi

Following a single 20 mg oral dose of 14C-labeled rabeprazole, approximately 90% of the drug was eliminated in the urine, primarily as thioether carboxylic acid; its glucuronide, and mercapturic acid metabolites.

Interaksi Makanan

1 Data
  • 1. Take with or without food. Food delays drug absorption, but not to a clinically significant extent.

Interaksi Obat

1027 Data
Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Rabeprazole.
Dabrafenib The serum concentration of Rabeprazole can be decreased when it is combined with Dabrafenib.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Rabeprazole.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Rabeprazole.
Amphetamine Rabeprazole can cause an increase in the absorption of Amphetamine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Atazanavir Rabeprazole can cause a decrease in the absorption of Atazanavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Bosutinib Rabeprazole can cause a decrease in the absorption of Bosutinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefditoren The serum concentration of Cefditoren can be decreased when it is combined with Rabeprazole.
Dabigatran etexilate Rabeprazole can cause a decrease in the absorption of Dabigatran etexilate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dasatinib Rabeprazole can cause a decrease in the absorption of Dasatinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Delavirdine Rabeprazole can cause a decrease in the absorption of Delavirdine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dextroamphetamine Rabeprazole can cause an increase in the absorption of Dextroamphetamine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Erlotinib Rabeprazole can cause a decrease in the absorption of Erlotinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Fluconazole The metabolism of Rabeprazole can be decreased when combined with Fluconazole.
Gefitinib Rabeprazole can cause a decrease in the absorption of Gefitinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Indinavir Rabeprazole can cause a decrease in the absorption of Indinavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Itraconazole Rabeprazole can cause a decrease in the absorption of Itraconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ledipasvir Rabeprazole can cause a decrease in the absorption of Ledipasvir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Methotrexate The excretion of Methotrexate can be decreased when combined with Rabeprazole.
Methylphenidate Rabeprazole can cause an increase in the absorption of Methylphenidate resulting in an increased serum concentration and potentially a worsening of adverse effects.
Dexmethylphenidate Rabeprazole can cause an increase in the absorption of Dexmethylphenidate resulting in an increased serum concentration and potentially a worsening of adverse effects.
Nelfinavir The serum concentration of Nelfinavir can be decreased when it is combined with Rabeprazole.
Nilotinib The serum concentration of Nilotinib can be decreased when it is combined with Rabeprazole.
Pazopanib Rabeprazole can cause a decrease in the absorption of Pazopanib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Posaconazole Rabeprazole can cause a decrease in the absorption of Posaconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Raltegravir Rabeprazole can cause an increase in the absorption of Raltegravir resulting in an increased serum concentration and potentially a worsening of adverse effects.
Rilpivirine Rabeprazole can cause a decrease in the absorption of Rilpivirine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Riociguat Rabeprazole can cause a decrease in the absorption of Riociguat resulting in a reduced serum concentration and potentially a decrease in efficacy.
Risedronic acid Rabeprazole can cause an increase in the absorption of Risedronic acid resulting in an increased serum concentration and potentially a worsening of adverse effects.
Saquinavir The serum concentration of Saquinavir can be increased when it is combined with Rabeprazole.
Voriconazole The metabolism of Rabeprazole can be decreased when combined with Voriconazole.
Luliconazole The serum concentration of Rabeprazole can be increased when it is combined with Luliconazole.
Colchicine The metabolism of Colchicine can be decreased when combined with Rabeprazole.
Fentanyl Fentanyl may decrease the excretion rate of Rabeprazole which could result in a higher serum level.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Rabeprazole.
Retapamulin The metabolism of Retapamulin can be decreased when combined with Rabeprazole.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with Rabeprazole.
Vardenafil The metabolism of Vardenafil can be decreased when combined with Rabeprazole.
Eszopiclone The metabolism of Eszopiclone can be decreased when combined with Rabeprazole.
Zopiclone The metabolism of Zopiclone can be decreased when combined with Rabeprazole.
Lovastatin The metabolism of Lovastatin can be decreased when combined with Rabeprazole.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with Rabeprazole.
Alprazolam The metabolism of Alprazolam can be decreased when combined with Rabeprazole.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Rabeprazole.
Levothyroxine Rabeprazole can cause a decrease in the absorption of Levothyroxine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Warfarin The serum concentration of Warfarin can be increased when it is combined with Rabeprazole.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with Rabeprazole.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with Rabeprazole.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with Rabeprazole.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with Rabeprazole.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with Rabeprazole.
Midazolam The serum concentration of Midazolam can be increased when it is combined with Rabeprazole.
Clopidogrel The serum concentration of the active metabolites of Clopidogrel can be reduced when Clopidogrel is used in combination with Rabeprazole resulting in a loss in efficacy.
Atorvastatin The metabolism of Atorvastatin can be decreased when combined with Rabeprazole.
Bisacodyl The therapeutic efficacy of Bisacodyl can be decreased when used in combination with Rabeprazole.
Captopril Rabeprazole can cause a decrease in the absorption of Captopril resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefuroxime The serum concentration of Cefuroxime can be decreased when it is combined with Rabeprazole.
Rifampin Rabeprazole can cause a decrease in the absorption of Rifampicin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Memantine Rabeprazole may decrease the excretion rate of Memantine which could result in a higher serum level.
Sulpiride The therapeutic efficacy of Sulpiride can be increased when used in combination with Rabeprazole.
Mesalazine Rabeprazole can cause a decrease in the absorption of Mesalazine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tolevamer The therapeutic efficacy of Tolevamer can be decreased when used in combination with Rabeprazole.
Alendronic acid The therapeutic efficacy of Alendronic acid can be decreased when used in combination with Rabeprazole.
Ibandronate The therapeutic efficacy of Ibandronate can be decreased when used in combination with Rabeprazole.
Clodronic acid The therapeutic efficacy of Clodronic acid can be decreased when used in combination with Rabeprazole.
Etidronic acid The therapeutic efficacy of Etidronic acid can be decreased when used in combination with Rabeprazole.
Incadronic acid The therapeutic efficacy of Incadronic acid can be decreased when used in combination with Rabeprazole.
Cysteamine The bioavailability of Cysteamine can be decreased when combined with Rabeprazole.
Ketoconazole Rabeprazole can cause a decrease in the absorption of Ketoconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lumacaftor The serum concentration of Rabeprazole can be decreased when it is combined with Lumacaftor.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with Rabeprazole.
Methenamine The therapeutic efficacy of Methenamine can be decreased when used in combination with Rabeprazole.
Fluvoxamine The metabolism of Rabeprazole can be decreased when combined with Fluvoxamine.
Ticlopidine The metabolism of Rabeprazole can be decreased when combined with Ticlopidine.
Chloramphenicol The metabolism of Rabeprazole can be decreased when combined with Chloramphenicol.
Lansoprazole The metabolism of Rabeprazole can be decreased when combined with Lansoprazole.
Fluoxetine The metabolism of Rabeprazole can be decreased when combined with Fluoxetine.
Zafirlukast The metabolism of Rabeprazole can be decreased when combined with Zafirlukast.
Isoniazid The metabolism of Rabeprazole can be decreased when combined with Isoniazid.
Miconazole The metabolism of Rabeprazole can be decreased when combined with Miconazole.
Gemfibrozil The metabolism of Rabeprazole can be decreased when combined with Gemfibrozil.
Stiripentol The metabolism of Rabeprazole can be decreased when combined with Stiripentol.
Eslicarbazepine acetate The metabolism of Rabeprazole can be decreased when combined with Eslicarbazepine acetate.
Efavirenz The metabolism of Rabeprazole can be decreased when combined with Efavirenz.
Prussian blue Rabeprazole can cause a decrease in the absorption of Prussian blue resulting in a reduced serum concentration and potentially a decrease in efficacy.
Iron sucrose Rabeprazole can cause a decrease in the absorption of Iron sucrose resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric ammonium citrate Rabeprazole can cause a decrease in the absorption of Ferric ammonium citrate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferumoxsil Rabeprazole can cause a decrease in the absorption of Ferumoxsil resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferumoxides Rabeprazole can cause a decrease in the absorption of Ferumoxides resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric sulfate Rabeprazole can cause a decrease in the absorption of Ferric sulfate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferrous bisglycinate Rabeprazole can cause a decrease in the absorption of Ferrous bisglycinate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gleptoferron Rabeprazole can cause a decrease in the absorption of Gleptoferron resulting in a reduced serum concentration and potentially a decrease in efficacy.
Perflubutane Rabeprazole can cause a decrease in the absorption of Perflubutane resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sodium feredetate Rabeprazole can cause a decrease in the absorption of Sodium feredetate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric hydroxide Rabeprazole can cause a decrease in the absorption of Ferric hydroxide resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric cation Rabeprazole can cause a decrease in the absorption of Ferric cation resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferrous gluconate Rabeprazole can cause a decrease in the absorption of Ferrous gluconate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferrous succinate Rabeprazole can cause a decrease in the absorption of Ferrous succinate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferrous fumarate Rabeprazole can cause a decrease in the absorption of Ferrous fumarate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tetraferric tricitrate decahydrate Rabeprazole can cause a decrease in the absorption of Tetraferric tricitrate decahydrate resulting in a reduced serum concentration and potentially a decrease in efficacy.

Target Protein

Potassium-transporting ATPase alpha chain 1 ATP4A

Referensi & Sumber

Synthesis reference: Sundaram Venkatraman, "Crystalline form Z of rabeprazole sodium and process for preparation thereof." U.S. Patent US20040180935, issued September 16, 2004.

Contoh Produk & Brand

Produk: 129 • International brands: 1
Produk
  • Abbott-rabeprazole
    Tablet, delayed release • 10 mg • Oral • Canada • Generic • Approved
  • Abbott-rabeprazole
    Tablet, delayed release • 20 mg • Oral • Canada • Generic • Approved
  • Aciphex
    Tablet, delayed release • 20 mg/1 • Oral • US • Approved
  • AcipHex
    Tablet, delayed release • 20 mg/1 • Oral • US • Approved
  • AcipHex
    Tablet, delayed release • 20 mg/1 • Oral • US • Approved
  • AcipHex
    Tablet, delayed release • 20 mg/1 • Oral • US • Approved
  • AcipHex
    Tablet, delayed release • 20 mg/1 • Oral • US • Approved
  • AcipHex
    Tablet, delayed release • 20 mg/1 • Oral • US • Approved
Menampilkan 8 dari 129 produk.
International Brands
  • Pariet

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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