Peringatan Keamanan

Oral LD50 (rat): 306 mg/kg; Oral LD50 (mice): 130 mg/kg; Oral LD50 (guinea pig): 198 mg/kg Registry of Toxic Effects of Chemical Substances. Ed. D. Sweet, US Dept. of Health & Human Services: Cincinatti, 2010.
Also a mild reproductive toxin to women of childbearing age.

Chlorpheniramine

DB01114

small molecule approved

Deskripsi

A histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma. It has also been used in veterinary applications. One of the most widely used of the classical antihistaminics, it generally causes less drowsiness and sedation than promethazine.

Struktur Molekul 2D

Berat 274.788
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 21-27 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Well absorbed in the gastrointestinal tract.

Metabolisme

Primarily hepatic via Cytochrome P450 (CYP450) enzymes.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food.

Interaksi Obat

1298 Data
Ivabradine Ivabradine may increase the QTc-prolonging activities of Chlorpheniramine.
Buprenorphine Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Magnesium sulfate The therapeutic efficacy of Chlorpheniramine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Chlorpheniramine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Orphenadrine Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Pramipexole Chlorpheniramine may increase the sedative activities of Pramipexole.
Ropinirole Chlorpheniramine may increase the sedative activities of Ropinirole.
Rotigotine Chlorpheniramine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Chlorpheniramine.
Sodium oxybate Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Thalidomide Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Benzylpenicilloyl polylysine Chlorpheniramine may decrease effectiveness of Benzylpenicilloyl polylysine as a diagnostic agent.
Betahistine The therapeutic efficacy of Betahistine can be decreased when used in combination with Chlorpheniramine.
Hyaluronidase (ovine) The therapeutic efficacy of Hyaluronidase (ovine) can be decreased when used in combination with Chlorpheniramine.
Hyaluronidase (human recombinant) The therapeutic efficacy of Hyaluronidase (human recombinant) can be decreased when used in combination with Chlorpheniramine.
Hyaluronidase The therapeutic efficacy of Hyaluronidase can be decreased when used in combination with Chlorpheniramine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Chlorpheniramine.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Chlorpheniramine.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Chlorpheniramine.
Dicoumarol The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Phenindione.
Coumarin The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Coumarin.
Tioclomarol The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Tioclomarol.
Warfarin The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with 4-hydroxycoumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Diphenadione.
(S)-Warfarin The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with (S)-Warfarin.
Mirabegron The serum concentration of Chlorpheniramine can be increased when it is combined with Mirabegron.
Tedizolid phosphate The risk or severity of serotonin syndrome can be increased when Tedizolid phosphate is combined with Chlorpheniramine.
Phenytoin The serum concentration of Phenytoin can be increased when it is combined with Chlorpheniramine.
Fosphenytoin The serum concentration of Fosphenytoin can be increased when it is combined with Chlorpheniramine.
Mirtazapine Chlorpheniramine may increase the serotonergic activities of Mirtazapine.
Ethanol Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Chlorpheniramine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Chlorpheniramine.
Sertraline The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Sibutramine.
Zimelidine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Milnacipran.
Desvenlafaxine The risk or severity of serotonin syndrome can be increased when Desvenlafaxine is combined with Chlorpheniramine.
Seproxetine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Seproxetine.
Levomilnacipran The risk or severity of serotonin syndrome can be increased when Chlorpheniramine is combined with Levomilnacipran.
Indalpine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Indalpine.
Alaproclate The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Alaproclate.
Amphetamine Amphetamine may decrease the sedative activities of Chlorpheniramine.
Phentermine Phentermine may decrease the sedative activities of Chlorpheniramine.
Benzphetamine Benzphetamine may decrease the sedative activities of Chlorpheniramine.
Diethylpropion Diethylpropion may decrease the sedative activities of Chlorpheniramine.
Lisdexamfetamine The risk or severity of serotonin syndrome can be increased when Chlorpheniramine is combined with Lisdexamfetamine.
Mephentermine Mephentermine may decrease the sedative activities of Chlorpheniramine.
MMDA MMDA may decrease the sedative activities of Chlorpheniramine.
Midomafetamine Midomafetamine may decrease the sedative activities of Chlorpheniramine.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the sedative activities of Chlorpheniramine.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the sedative activities of Chlorpheniramine.
Tenamfetamine Tenamfetamine may decrease the sedative activities of Chlorpheniramine.
Chlorphentermine Chlorphentermine may decrease the sedative activities of Chlorpheniramine.
Methylenedioxyethamphetamine Methylenedioxyethamphetamine may decrease the sedative activities of Chlorpheniramine.
Dextroamphetamine Dextroamphetamine may decrease the sedative activities of Chlorpheniramine.
Metamfetamine Metamfetamine may decrease the sedative activities of Chlorpheniramine.
Iofetamine I-123 Iofetamine I-123 may decrease the sedative activities of Chlorpheniramine.
Ritobegron Ritobegron may decrease the sedative activities of Chlorpheniramine.
Mephedrone Mephedrone may decrease the sedative activities of Chlorpheniramine.
Methoxyphenamine Methoxyphenamine may decrease the sedative activities of Chlorpheniramine.
Gepefrine Gepefrine may decrease the sedative activities of Chlorpheniramine.
2,5-Dimethoxy-4-ethylthioamphetamine 2,5-Dimethoxy-4-ethylthioamphetamine may decrease the sedative activities of Chlorpheniramine.
Phendimetrazine Phendimetrazine may decrease the sedative activities of Chlorpheniramine.
Methylene blue Chlorpheniramine may increase the serotonergic activities of Methylene blue.
Trospium The metabolism of Chlorpheniramine can be decreased when combined with Trospium.
Doxepin The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Doxepin.
Zopiclone The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Zopiclone.
Thiethylperazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Thiethylperazine.
Triflupromazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Triflupromazine.
Fluphenazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Fluphenazine.
Trifluoperazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Trifluoperazine.
Acetophenazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Acetophenazine.
Periciazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Periciazine.
Acepromazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Acepromazine.
Molindone The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Molindone.
Thioproperazine The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Thioproperazine.
Osanetant The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Osanetant.
Bifeprunox The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with Bifeprunox.
BL-1020 The risk or severity of adverse effects can be increased when Chlorpheniramine is combined with BL-1020.

Target Protein

Histamine H1 receptor HRH1
Sodium-dependent serotonin transporter SLC6A4
Sodium-dependent noradrenaline transporter SLC6A2
Sodium-dependent dopamine transporter SLC6A3

Referensi & Sumber

Synthesis reference: Anil M. Salpekar, John Johnson, "Acetaminophen compositions containing low doses of chlorpheniramine maleate, method for preparing same and tablets formed therefrom." U.S. Patent US4631284, issued April, 1975.

Contoh Produk & Brand

Produk: 1304 • International brands: 4
Produk
  • 4 Hour Allergy Relief
    Tablet • 4 mg/1 • Oral • US • OTC
  • 999 Cold Remedy
    Capsule • - • Oral • US • OTC
  • 999 Cold Remedy Granular
    Granule • - • Oral • US • OTC
  • 999 Cold Remedy Granular
    Capsule • - • Oral • US • OTC
  • 999 GANMAOLING Cold
    Capsule • - • Oral • US • OTC
  • AccuHist
    Solution • - • Oral • US • OTC
  • AccuHist PDX
    Solution • - • Oral • US • OTC
  • Acetaminophen, Ascorbic acid, Chlorpheniramine Maleate
    Powder, for solution • - • Oral • US • OTC
Menampilkan 8 dari 1304 produk.
International Brands
  • Chlo-Amine
  • Chlor-Trimeton — Schering-Plough
  • Haynon
  • Piriton — GlaxoSmithKline

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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