Peringatan Keamanan

Oral LD50 in rats is 5450 mg/kg. Overdosage with colistimethate can cause neuromuscular blockade characterized by paresthesia, lethargy, confusion, dizziness, ataxia, nystagmus, disorders of speech and apnea. Respiratory muscle paralysis may lead to apnea, respiratory arrest and death.

Colistimethate

DB01111

small molecule approved vet_approved

Deskripsi

Colistimethate is an antibiotic that has been shown to have bactericidal activity against aerobic gram-negative microorganisms. Colistimethate is particularly indicated when the infection is caused by sensitive strains of Pseudomonas aeruginosa.

Struktur Molekul 2D

Berat 1634.87
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 2-3 hours following either intravenous or intramuscular administration in adults and in the pediatric population, including premature infants.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Very poor absorption from gastrointestinal tract.

Metabolisme

As 80% of the dose can be recovered unchanged in the urine, and there is no biliary excretion, it can be assumed that the remaining drug is inactivated in the tissues, however the mechanism is unknown.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

740 Data
Succinylcholine The therapeutic efficacy of Succinylcholine can be increased when used in combination with Colistimethate.
Metocurine iodide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Colistimethate.
Gallamine triethiodide The therapeutic efficacy of Gallamine triethiodide can be increased when used in combination with Colistimethate.
Cisatracurium The therapeutic efficacy of Cisatracurium can be increased when used in combination with Colistimethate.
Rocuronium The therapeutic efficacy of Rocuronium can be increased when used in combination with Colistimethate.
Atracurium besylate The therapeutic efficacy of Atracurium besylate can be increased when used in combination with Colistimethate.
Doxacurium The therapeutic efficacy of Doxacurium can be increased when used in combination with Colistimethate.
Mivacurium The therapeutic efficacy of Mivacurium can be increased when used in combination with Colistimethate.
Decamethonium The therapeutic efficacy of Decamethonium can be increased when used in combination with Colistimethate.
Metocurine The therapeutic efficacy of Metocurine can be increased when used in combination with Colistimethate.
Pancuronium The therapeutic efficacy of Pancuronium can be increased when used in combination with Colistimethate.
Pipecuronium The therapeutic efficacy of Pipecuronium can be increased when used in combination with Colistimethate.
Vecuronium The therapeutic efficacy of Vecuronium can be increased when used in combination with Colistimethate.
Rapacuronium The therapeutic efficacy of Rapacuronium can be increased when used in combination with Colistimethate.
Pyrantel The therapeutic efficacy of Pyrantel can be increased when used in combination with Colistimethate.
Neosaxitoxin The therapeutic efficacy of Neosaxitoxin can be increased when used in combination with Colistimethate.
Atracurium The therapeutic efficacy of Atracurium can be increased when used in combination with Colistimethate.
Gallamine The therapeutic efficacy of Gallamine can be increased when used in combination with Colistimethate.
Alcuronium The therapeutic efficacy of Alcuronium can be increased when used in combination with Colistimethate.
Tubocurarine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Colistimethate.
Foscarnet The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Foscarnet.
Mannitol The risk or severity of nephrotoxicity can be increased when Mannitol is combined with Colistimethate.
Tenofovir disoproxil Colistimethate may increase the nephrotoxic activities of Tenofovir disoproxil.
Tenofovir alafenamide Colistimethate may increase the nephrotoxic activities of Tenofovir alafenamide.
Tenofovir Colistimethate may increase the nephrotoxic activities of Tenofovir.
Amphotericin B Amphotericin B may increase the nephrotoxic activities of Colistimethate.
Polymyxin B Polymyxin B may increase the nephrotoxic and neuromuscular blocking activities of Colistimethate.
Cyclosporine The risk or severity of nephrotoxicity can be increased when Cyclosporine is combined with Colistimethate.
Icosapent The risk or severity of nephrotoxicity can be increased when Icosapent is combined with Colistimethate.
Cefotiam The risk or severity of nephrotoxicity can be increased when Cefotiam is combined with Colistimethate.
Mesalazine The risk or severity of nephrotoxicity can be increased when Mesalazine is combined with Colistimethate.
Cefmenoxime The risk or severity of nephrotoxicity can be increased when Cefmenoxime is combined with Colistimethate.
Cefmetazole The risk or severity of nephrotoxicity can be increased when Cefmetazole is combined with Colistimethate.
Indomethacin The risk or severity of nephrotoxicity can be increased when Indomethacin is combined with Colistimethate.
Triamterene The risk or severity of nephrotoxicity can be increased when Triamterene is combined with Colistimethate.
Cefpiramide The risk or severity of nephrotoxicity can be increased when Cefpiramide is combined with Colistimethate.
Loracarbef The risk or severity of nephrotoxicity can be increased when Loracarbef is combined with Colistimethate.
Cefalotin The risk or severity of nephrotoxicity can be increased when Cefalotin is combined with Colistimethate.
Nabumetone The risk or severity of nephrotoxicity can be increased when Nabumetone is combined with Colistimethate.
Ketorolac The risk or severity of nephrotoxicity can be increased when Ketorolac is combined with Colistimethate.
Tenoxicam The risk or severity of nephrotoxicity can be increased when Tenoxicam is combined with Colistimethate.
Celecoxib The risk or severity of nephrotoxicity can be increased when Celecoxib is combined with Colistimethate.
Cefotaxime The risk or severity of nephrotoxicity can be increased when Cefotaxime is combined with Colistimethate.
Tolmetin The risk or severity of nephrotoxicity can be increased when Tolmetin is combined with Colistimethate.
Rofecoxib The risk or severity of nephrotoxicity can be increased when Rofecoxib is combined with Colistimethate.
Fenoprofen The risk or severity of nephrotoxicity can be increased when Fenoprofen is combined with Colistimethate.
Valdecoxib The risk or severity of nephrotoxicity can be increased when Valdecoxib is combined with Colistimethate.
Diclofenac The risk or severity of nephrotoxicity can be increased when Diclofenac is combined with Colistimethate.
Sulindac The risk or severity of nephrotoxicity can be increased when Sulindac is combined with Colistimethate.
Bacitracin The risk or severity of nephrotoxicity can be increased when Bacitracin is combined with Colistimethate.
Cephaloglycin The risk or severity of nephrotoxicity can be increased when Cephaloglycin is combined with Colistimethate.
Adefovir dipivoxil The risk or severity of nephrotoxicity can be increased when Adefovir dipivoxil is combined with Colistimethate.
Pentamidine The risk or severity of nephrotoxicity can be increased when Pentamidine is combined with Colistimethate.
Mefenamic acid The risk or severity of nephrotoxicity can be increased when Mefenamic acid is combined with Colistimethate.
Naproxen The risk or severity of nephrotoxicity can be increased when Naproxen is combined with Colistimethate.
Sulfasalazine The risk or severity of nephrotoxicity can be increased when Sulfasalazine is combined with Colistimethate.
Phenylbutazone The risk or severity of nephrotoxicity can be increased when Phenylbutazone is combined with Colistimethate.
Meloxicam The risk or severity of nephrotoxicity can be increased when Meloxicam is combined with Colistimethate.
Carprofen The risk or severity of nephrotoxicity can be increased when Carprofen is combined with Colistimethate.
Tacrolimus The risk or severity of nephrotoxicity can be increased when Tacrolimus is combined with Colistimethate.
Etacrynic acid The risk or severity of nephrotoxicity can be increased when Etacrynic acid is combined with Colistimethate.
Ceforanide The risk or severity of nephrotoxicity can be increased when Ceforanide is combined with Colistimethate.
Salicylic acid The risk or severity of nephrotoxicity can be increased when Salicylic acid is combined with Colistimethate.
Acetylsalicylic acid The risk or severity of nephrotoxicity can be increased when Acetylsalicylic acid is combined with Colistimethate.
Hydrochlorothiazide The risk or severity of nephrotoxicity can be increased when Hydrochlorothiazide is combined with Colistimethate.
Balsalazide The risk or severity of nephrotoxicity can be increased when Balsalazide is combined with Colistimethate.
Cefditoren The risk or severity of nephrotoxicity can be increased when Cefditoren is combined with Colistimethate.
Atazanavir The risk or severity of nephrotoxicity can be increased when Atazanavir is combined with Colistimethate.
Cefuroxime The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefuroxime.
Cefapirin The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefapirin.
Cefprozil The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefprozil.
Olsalazine The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Olsalazine.
Lumiracoxib The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Lumiracoxib.
Cefamandole The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefamandole.
Cefazolin The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefazolin.
Cefonicid The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefonicid.
Cefoperazone The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefoperazone.
Cefoxitin The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefoxitin.
Ceftizoxime The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Ceftizoxime.
Magnesium salicylate The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Magnesium salicylate.
Salsalate The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Salsalate.
Choline magnesium trisalicylate The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Choline magnesium trisalicylate.
Cefepime The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefepime.
Cefacetrile The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefacetrile.
Cefpodoxime The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cefpodoxime.
Antrafenine The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Antrafenine.
Aminophenazone The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Aminophenazone.
Antipyrine The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Antipyrine.
Tiaprofenic acid The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Tiaprofenic acid.
Lopinavir The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Lopinavir.
Etoricoxib The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Etoricoxib.
Hydrolyzed Cephalothin The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Hydrolyzed Cephalothin.
Cephalothin Group The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Cephalothin Group.
Oxyphenbutazone The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Oxyphenbutazone.
Latamoxef The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Latamoxef.
Nimesulide The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Nimesulide.
Benoxaprofen The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Benoxaprofen.
Metamizole The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Metamizole.
Zomepirac The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Zomepirac.
Ceftobiprole The risk or severity of nephrotoxicity can be increased when Colistimethate is combined with Ceftobiprole.

Target Protein

Dihydropteroate synthase folP
Bacterial outer membrane

Contoh Produk & Brand

Produk: 19 • International brands: 0
Produk
  • Colistimethate
    Injection, powder, lyophilized, for solution • 150 mg/2mL • Intramuscular; Intravenous • US • Generic • Approved
  • Colistimethate
    Injection • 150 mg/2mL • Intramuscular; Intravenous • US • Generic • Approved
  • Colistimethate
    Injection, powder, lyophilized, for solution • 150 mg/2mL • Intramuscular; Intravenous • US • Generic • Approved
  • Colistimethate
    Injection • 150 mg/2mL • Intramuscular; Intravenous • US • Generic • Approved
  • Colistimethate
    Injection, powder, for solution • 150 mg/1 • Intramuscular; Intravenous • US • Generic • Approved
  • Colistimethate
    Injection, powder, lyophilized, for solution • 150 mg/2mL • Intramuscular; Intravenous • US • Generic • Approved
  • Colistimethate
    Injection, powder, lyophilized, for solution • 150 mg/2mL • Intramuscular; Intravenous • US • Generic • Approved
  • Colistimethate
    Injection • 150 mg/2mL • Intramuscular; Intravenous • US • Generic • Approved
Menampilkan 8 dari 19 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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