Peringatan Keamanan

Coma, dry skin and mucous membranes, enlarged pupils of the eyes, extremely high body temperature, flushing, involuntary eyeball movement, lower than normal muscle tone, pinpoint pupils, rapid heartbeat, restlessness, sluggishness, suppressed breathing

Diphenoxylate

DB01081

small molecule approved illicit

Deskripsi

A meperidine congener used as an antidiarrheal, usually in combination with atropine. At high doses, it acts like morphine. Its unesterified metabolite difenoxin has similar properties and is used similarly. It has little or no analgesic activity. This medication is classified as a Schedule V under the Controlled Substances Act by the Food and Drug Administration (FDA) and the DEA in the United States when used in preparations. When diphenoxylate is used alone, it is classified as a Schedule II.

Struktur Molekul 2D

Berat 452.5873
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 12-14 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

90%

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Avoid alcohol.
  • 2. Take with food.

Interaksi Obat

917 Data
Buprenorphine Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Hydrocodone Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Magnesium sulfate The therapeutic efficacy of Diphenoxylate can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Diphenoxylate may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Orphenadrine Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Pramipexole Diphenoxylate may increase the sedative activities of Pramipexole.
Ropinirole Diphenoxylate may increase the sedative activities of Ropinirole.
Rotigotine Diphenoxylate may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Diphenoxylate.
Sodium oxybate Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Thalidomide Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Alvimopan The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Alvimopan.
Desmopressin The risk or severity of hyponatremia can be increased when Diphenoxylate is combined with Desmopressin.
Morphine The risk or severity of adverse effects can be increased when Morphine is combined with Diphenoxylate.
Codeine The risk or severity of adverse effects can be increased when Codeine is combined with Diphenoxylate.
Hydromorphone The risk or severity of adverse effects can be increased when Hydromorphone is combined with Diphenoxylate.
Meperidine The risk or severity of adverse effects can be increased when Meperidine is combined with Diphenoxylate.
Oxycodone The risk or severity of adverse effects can be increased when Oxycodone is combined with Diphenoxylate.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Dextropropoxyphene is combined with Diphenoxylate.
Naltrexone The therapeutic efficacy of Diphenoxylate can be decreased when used in combination with Naltrexone.
Sufentanil The risk or severity of adverse effects can be increased when Sufentanil is combined with Diphenoxylate.
Alfentanil The risk or severity of adverse effects can be increased when Alfentanil is combined with Diphenoxylate.
Fentanyl The risk or severity of adverse effects can be increased when Fentanyl is combined with Diphenoxylate.
Levorphanol The risk or severity of adverse effects can be increased when Levorphanol is combined with Diphenoxylate.
Remifentanil The risk or severity of adverse effects can be increased when Remifentanil is combined with Diphenoxylate.
Oxymorphone The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Oxymorphone.
Dezocine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Dezocine.
Methadyl acetate The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Methadyl acetate.
Dihydroetorphine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Dihydroetorphine.
Diamorphine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Diamorphine.
Bezitramide The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Bezitramide.
Ethylmorphine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Ethylmorphine.
Etorphine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Etorphine.
Dextromoramide The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Dextromoramide.
Desomorphine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Desomorphine.
Carfentanil The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Carfentanil.
Dihydrocodeine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Dihydrocodeine.
Alphacetylmethadol The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Alphacetylmethadol.
Dihydromorphine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Dihydromorphine.
Ketobemidone The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Ketobemidone.
DPDPE The risk or severity of adverse effects can be increased when Diphenoxylate is combined with DPDPE.
Lofentanil The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Lofentanil.
Opium The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Opium.
Normethadone The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Normethadone.
Piritramide The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Piritramide.
Alphaprodine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Alphaprodine.
Nicomorphine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Nicomorphine.
Meptazinol The therapeutic efficacy of Diphenoxylate can be decreased when used in combination with Meptazinol.
Phenoperidine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Phenoperidine.
Phenazocine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Phenazocine.
Tilidine The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Tilidine.
Carfentanil, C-11 The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Carfentanil, C-11.
Naloxegol The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Naloxegol.
Benzhydrocodone The risk or severity of adverse effects can be increased when Diphenoxylate is combined with Benzhydrocodone.
Pegvisomant The therapeutic efficacy of Pegvisomant can be decreased when used in combination with Diphenoxylate.
Succinylcholine The risk or severity of bradycardia can be increased when Succinylcholine is combined with Diphenoxylate.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Diphenoxylate.
Linezolid The risk or severity of serotonin syndrome can be increased when Linezolid is combined with Diphenoxylate.
Mirtazapine Diphenoxylate may increase the serotonergic activities of Mirtazapine.
Fluvoxamine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Fluvoxamine.
Citalopram The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Citalopram.
Duloxetine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Duloxetine.
Paroxetine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Paroxetine.
Sertraline The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Sertraline.
Sibutramine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Sibutramine.
Nefazodone The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Nefazodone.
Zimelidine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Zimelidine.
Dapoxetine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Dapoxetine.
Milnacipran The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Milnacipran.
Desvenlafaxine The risk or severity of serotonin syndrome can be increased when Desvenlafaxine is combined with Diphenoxylate.
Seproxetine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Seproxetine.
Levomilnacipran The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Levomilnacipran.
Indalpine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Indalpine.
Ritanserin The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Ritanserin.
Alaproclate The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Alaproclate.
Ethanol Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Diphenoxylate may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Diphenoxylate.
Amphetamine Amphetamine may increase the analgesic activities of Diphenoxylate.
Phentermine Phentermine may increase the analgesic activities of Diphenoxylate.
Pseudoephedrine Pseudoephedrine may increase the analgesic activities of Diphenoxylate.
Benzphetamine Benzphetamine may increase the analgesic activities of Diphenoxylate.
Diethylpropion Diethylpropion may increase the analgesic activities of Diphenoxylate.
Lisdexamfetamine The risk or severity of serotonin syndrome can be increased when Diphenoxylate is combined with Lisdexamfetamine.
Mephentermine Mephentermine may increase the analgesic activities of Diphenoxylate.
MMDA MMDA may increase the analgesic activities of Diphenoxylate.
Midomafetamine Midomafetamine may increase the analgesic activities of Diphenoxylate.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may increase the analgesic activities of Diphenoxylate.

Target Protein

Mu-type opioid receptor OPRM1
Delta-type opioid receptor OPRD1

Referensi & Sumber

Synthesis reference: Janssen, P.A.J.; U.S.Patent 2,898,340; August 4,1959. Dryden, H.L. Jr. and Erickson, R.A.; U.S. Patent 4,086,234; April 25,1978; assigned to G.D.Searle & Co.

Contoh Produk & Brand

Produk: 97 • International brands: 0
Produk
  • Diphenoxylate Hcl and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
  • Diphenoxylate Hydrochloride and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
  • Diphenoxylate Hydrochloride and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
  • Diphenoxylate Hydrochloride and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
  • Diphenoxylate Hydrochloride and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
  • Diphenoxylate Hydrochloride and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
  • Diphenoxylate Hydrochloride and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
  • Diphenoxylate Hydrochloride and Atropine Sulfate
    Tablet • - • Oral • US • Generic • Approved
Menampilkan 8 dari 97 produk.

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