Peringatan Keamanan

The oral LD50 of tocainide was calculated to be about 800 mg/kg in mice, 1000 mg/kg in rats, and 230 mg/kg in guinea pigs; deaths were usually preceded by convulsions.

Tocainide

DB01056

small molecule approved

Deskripsi

An antiarrhythmic agent which exerts a potential- and frequency-dependent block of sodium channels.

Struktur Molekul 2D

Berat 192.2575
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The average plasma half-life in patients is approximately 15 hours. May be prolonged up to 35 hours in patients with severe renal function impairment (creatinine clearance less than 30 mL per min per 1.73 square meters of body surface area.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Following oral administration, the bioavailability approaches 100 percent, and is unaffected by food.

Metabolisme

Negligible first pass hepatic degradation. No active metabolites have been found.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

448 Data
Tizanidine The serum concentration of Tizanidine can be increased when it is combined with Tocainide.
Deferasirox The serum concentration of Tocainide can be increased when it is combined with Deferasirox.
Peginterferon alfa-2b The serum concentration of Tocainide can be increased when it is combined with Peginterferon alfa-2b.
Leflunomide The serum concentration of Tocainide can be decreased when it is combined with Leflunomide.
Teriflunomide The serum concentration of Tocainide can be decreased when it is combined with Teriflunomide.
Zolmitriptan The metabolism of Zolmitriptan can be decreased when combined with Tocainide.
Abiraterone The serum concentration of Tocainide can be increased when it is combined with Abiraterone.
Cyproterone acetate The metabolism of Tocainide can be increased when combined with Cyproterone acetate.
Esmolol Esmolol may increase the arrhythmogenic activities of Tocainide.
Dofetilide Dofetilide may increase the arrhythmogenic activities of Tocainide.
Metoprolol Metoprolol may increase the arrhythmogenic activities of Tocainide.
Isradipine Isradipine may increase the arrhythmogenic activities of Tocainide.
Ibutilide Ibutilide may increase the arrhythmogenic activities of Tocainide.
Atenolol Atenolol may increase the arrhythmogenic activities of Tocainide.
Diltiazem Diltiazem may increase the arrhythmogenic activities of Tocainide.
Trimethadione Trimethadione may increase the arrhythmogenic activities of Tocainide.
Timolol Timolol may increase the arrhythmogenic activities of Tocainide.
Amlodipine Amlodipine may increase the arrhythmogenic activities of Tocainide.
Digoxin Digoxin may increase the arrhythmogenic activities of Tocainide.
Nimodipine Nimodipine may increase the arrhythmogenic activities of Tocainide.
Nisoldipine Nisoldipine may increase the arrhythmogenic activities of Tocainide.
Hyoscyamine Hyoscyamine may increase the arrhythmogenic activities of Tocainide.
Sotalol Sotalol may increase the arrhythmogenic activities of Tocainide.
Acetyldigitoxin Acetyldigitoxin may increase the arrhythmogenic activities of Tocainide.
Lercanidipine Lercanidipine may increase the arrhythmogenic activities of Tocainide.
Lamotrigine Lamotrigine may increase the arrhythmogenic activities of Tocainide.
Atropine Atropine may increase the arrhythmogenic activities of Tocainide.
Ethosuximide Ethosuximide may increase the arrhythmogenic activities of Tocainide.
Nicardipine Nicardipine may increase the arrhythmogenic activities of Tocainide.
Adenosine Adenosine may increase the arrhythmogenic activities of Tocainide.
Magnesium sulfate Magnesium sulfate may increase the arrhythmogenic activities of Tocainide.
Losartan Losartan may increase the arrhythmogenic activities of Tocainide.
Moricizine Moricizine may increase the arrhythmogenic activities of Tocainide.
Levomenthol Levomenthol may increase the arrhythmogenic activities of Tocainide.
Loperamide Loperamide may increase the arrhythmogenic activities of Tocainide.
Alprenolol Alprenolol may increase the arrhythmogenic activities of Tocainide.
Zonisamide Zonisamide may increase the arrhythmogenic activities of Tocainide.
Levosimendan Levosimendan may increase the arrhythmogenic activities of Tocainide.
Felodipine Felodipine may increase the arrhythmogenic activities of Tocainide.
Procainamide Procainamide may increase the arrhythmogenic activities of Tocainide.
Nitrendipine Nitrendipine may increase the arrhythmogenic activities of Tocainide.
Carteolol Tocainide may increase the arrhythmogenic activities of Carteolol.
Perhexiline Tocainide may increase the arrhythmogenic activities of Perhexiline.
Deslanoside Tocainide may increase the arrhythmogenic activities of Deslanoside.
Bretylium Tocainide may increase the arrhythmogenic activities of Bretylium.
Acebutolol Tocainide may increase the arrhythmogenic activities of Acebutolol.
Flecainide Tocainide may increase the arrhythmogenic activities of Flecainide.
Nadolol Tocainide may increase the arrhythmogenic activities of Nadolol.
Metipranolol Tocainide may increase the arrhythmogenic activities of Metipranolol.
Encainide Tocainide may increase the arrhythmogenic activities of Encainide.
Bepridil Tocainide may increase the arrhythmogenic activities of Bepridil.
Practolol Tocainide may increase the arrhythmogenic activities of Practolol.
Digitoxin Tocainide may increase the arrhythmogenic activities of Digitoxin.
Ajmaline Tocainide may increase the arrhythmogenic activities of Ajmaline.
Aprindine Tocainide may increase the arrhythmogenic activities of Aprindine.
Oxprenolol Tocainide may increase the arrhythmogenic activities of Oxprenolol.
Dexpropranolol Tocainide may increase the arrhythmogenic activities of Dexpropranolol.
Nimesulide Tocainide may increase the arrhythmogenic activities of Nimesulide.
Prenylamine Tocainide may increase the arrhythmogenic activities of Prenylamine.
Cyclandelate Tocainide may increase the arrhythmogenic activities of Cyclandelate.
Fluspirilene Tocainide may increase the arrhythmogenic activities of Fluspirilene.
Celiprolol Tocainide may increase the arrhythmogenic activities of Celiprolol.
Dronedarone Tocainide may increase the arrhythmogenic activities of Dronedarone.
Nebivolol Tocainide may increase the arrhythmogenic activities of Nebivolol.
Clevidipine Tocainide may increase the arrhythmogenic activities of Clevidipine.
Azimilide Tocainide may increase the arrhythmogenic activities of Azimilide.
Methsuximide Tocainide may increase the arrhythmogenic activities of Methsuximide.
Seletracetam Tocainide may increase the arrhythmogenic activities of Seletracetam.
Nylidrin Tocainide may increase the arrhythmogenic activities of Nylidrin.
Tedisamil Tocainide may increase the arrhythmogenic activities of Tedisamil.
Vernakalant Tocainide may increase the arrhythmogenic activities of Vernakalant.
Ziconotide Tocainide may increase the arrhythmogenic activities of Ziconotide.
Dotarizine Tocainide may increase the arrhythmogenic activities of Dotarizine.
Cariporide Tocainide may increase the arrhythmogenic activities of Cariporide.
Xylometazoline Tocainide may increase the arrhythmogenic activities of Xylometazoline.
Nilvadipine Tocainide may increase the arrhythmogenic activities of Nilvadipine.
Sparteine Tocainide may increase the arrhythmogenic activities of Sparteine.
Tranilast Tocainide may increase the arrhythmogenic activities of Tranilast.
Fasudil Tocainide may increase the arrhythmogenic activities of Fasudil.
Bupranolol Tocainide may increase the arrhythmogenic activities of Bupranolol.
Agmatine Tocainide may increase the arrhythmogenic activities of Agmatine.
Indenolol Tocainide may increase the arrhythmogenic activities of Indenolol.
Fendiline Tocainide may increase the arrhythmogenic activities of Fendiline.
Eperisone Tocainide may increase the arrhythmogenic activities of Eperisone.
Trimebutine Tocainide may increase the arrhythmogenic activities of Trimebutine.
Pinaverium Tocainide may increase the arrhythmogenic activities of Pinaverium.
Nicorandil Tocainide may increase the arrhythmogenic activities of Nicorandil.
Melperone Tocainide may increase the arrhythmogenic activities of Melperone.
Barnidipine Tocainide may increase the arrhythmogenic activities of Barnidipine.
Aranidipine Tocainide may increase the arrhythmogenic activities of Aranidipine.
Azelnidipine Tocainide may increase the arrhythmogenic activities of Azelnidipine.
Benidipine Tocainide may increase the arrhythmogenic activities of Benidipine.
Cilnidipine Tocainide may increase the arrhythmogenic activities of Cilnidipine.
Darodipine Tocainide may increase the arrhythmogenic activities of Darodipine.
Efonidipine Tocainide may increase the arrhythmogenic activities of Efonidipine.
Lacidipine Tocainide may increase the arrhythmogenic activities of Lacidipine.
Manidipine Tocainide may increase the arrhythmogenic activities of Manidipine.
Niguldipine Tocainide may increase the arrhythmogenic activities of Niguldipine.
Niludipine Tocainide may increase the arrhythmogenic activities of Niludipine.
Tropisetron Tocainide may increase the arrhythmogenic activities of Tropisetron.

Target Protein

Sodium channel protein type 5 subunit alpha SCN5A

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 1 • International brands: 1
Produk
  • Tonocard Tab 400 mg
    Tablet • 400 mg • Oral • Canada • Approved
International Brands
  • Tonocard

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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