Nitrendipine

DB01054

small molecule approved investigational

Deskripsi

Nitrendipine is a calcium channel blocker with marked vasodilator action. It is an effective antihypertensive agent and differs from other calcium channel blockers in that it does not reduce glomerular filtration rate and is mildly natriuretic, rather than sodium retentive.

Struktur Molekul 2D

Berat 360.3612
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Take with or without food.

Interaksi Obat

1457 Data
Duloxetine The risk or severity of orthostatic hypotension and syncope can be increased when Nitrendipine is combined with Duloxetine.
Levodopa The risk or severity of hypotension and orthostatic hypotension can be increased when Nitrendipine is combined with Levodopa.
Risperidone Nitrendipine may increase the hypotensive activities of Risperidone.
Troglitazone Troglitazone may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Reserpine Reserpine may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Progesterone Progesterone may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Chlorpromazine Chlorpromazine may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Bosentan Bosentan may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Ethinylestradiol Ethinylestradiol may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Glyburide Glyburide may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Cholic Acid Cholic Acid may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Fusidic acid Fusidic acid may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Simeprevir Simeprevir may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Lenvatinib Lenvatinib may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Letermovir The metabolism of Nitrendipine can be decreased when combined with Letermovir.
Valinomycin Valinomycin may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Olmesartan Olmesartan may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Pralsetinib Pralsetinib may decrease the excretion rate of Nitrendipine which could result in a higher serum level.
Ceritinib Nitrendipine may increase the bradycardic activities of Ceritinib.
Ivabradine Nitrendipine may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of Nitrendipine.
Alfuzosin Alfuzosin may increase the hypotensive activities of Nitrendipine.
Amifostine Nitrendipine may increase the hypotensive activities of Amifostine.
Diazoxide Diazoxide may increase the hypotensive activities of Nitrendipine.
Methylphenidate Methylphenidate may decrease the antihypertensive activities of Nitrendipine.
Dexmethylphenidate Dexmethylphenidate may decrease the antihypertensive activities of Nitrendipine.
Obinutuzumab Nitrendipine may increase the hypotensive activities of Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the hypotensive activities of Nitrendipine.
Rituximab Nitrendipine may increase the hypotensive activities of Rituximab.
Desmopressin Desmopressin may decrease the antihypertensive activities of Nitrendipine.
Isoetharine Isoetharine may decrease the antihypertensive activities of Nitrendipine.
Etomidate Etomidate may decrease the antihypertensive activities of Nitrendipine.
Zolmitriptan Zolmitriptan may decrease the antihypertensive activities of Nitrendipine.
Norepinephrine Norepinephrine may decrease the antihypertensive activities of Nitrendipine.
Phenylpropanolamine Phenylpropanolamine may decrease the antihypertensive activities of Nitrendipine.
Doxapram Doxapram may decrease the antihypertensive activities of Nitrendipine.
Metaraminol Metaraminol may decrease the antihypertensive activities of Nitrendipine.
Methoxamine Methoxamine may decrease the antihypertensive activities of Nitrendipine.
Orciprenaline Orciprenaline may decrease the antihypertensive activities of Nitrendipine.
Phenmetrazine Phenmetrazine may decrease the antihypertensive activities of Nitrendipine.
Dobutamine Dobutamine may decrease the antihypertensive activities of Nitrendipine.
Pseudoephedrine Pseudoephedrine may decrease the antihypertensive activities of Nitrendipine.
Ritodrine Ritodrine may decrease the antihypertensive activities of Nitrendipine.
Bitolterol Bitolterol may decrease the antihypertensive activities of Nitrendipine.
Diethylpropion Diethylpropion may decrease the antihypertensive activities of Nitrendipine.
Naratriptan Naratriptan may decrease the antihypertensive activities of Nitrendipine.
Rizatriptan Rizatriptan may decrease the antihypertensive activities of Nitrendipine.
Dopamine Dopamine may decrease the antihypertensive activities of Nitrendipine.
Frovatriptan Frovatriptan may decrease the antihypertensive activities of Nitrendipine.
Isoprenaline Isoprenaline may decrease the antihypertensive activities of Nitrendipine.
Arbutamine Arbutamine may decrease the antihypertensive activities of Nitrendipine.
Lisdexamfetamine Lisdexamfetamine may decrease the antihypertensive activities of Nitrendipine.
Fenoterol Fenoterol may decrease the antihypertensive activities of Nitrendipine.
Pirbuterol Pirbuterol may decrease the antihypertensive activities of Nitrendipine.
Ephedra sinica root Ephedra sinica root may decrease the antihypertensive activities of Nitrendipine.
Ephedrine Ephedrine may decrease the antihypertensive activities of Nitrendipine.
Mephentermine Mephentermine may decrease the antihypertensive activities of Nitrendipine.
Procaterol Procaterol may decrease the antihypertensive activities of Nitrendipine.
Clenbuterol Clenbuterol may decrease the antihypertensive activities of Nitrendipine.
Bambuterol Bambuterol may decrease the antihypertensive activities of Nitrendipine.
MMDA MMDA may decrease the antihypertensive activities of Nitrendipine.
Midomafetamine Midomafetamine may decrease the antihypertensive activities of Nitrendipine.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the antihypertensive activities of Nitrendipine.
4-Methoxyamphetamine 4-Methoxyamphetamine may decrease the antihypertensive activities of Nitrendipine.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the antihypertensive activities of Nitrendipine.
Tenamfetamine Tenamfetamine may decrease the antihypertensive activities of Nitrendipine.
Chlorphentermine Chlorphentermine may decrease the antihypertensive activities of Nitrendipine.
Dextroamphetamine Dextroamphetamine may decrease the antihypertensive activities of Nitrendipine.
Metamfetamine Metamfetamine may decrease the antihypertensive activities of Nitrendipine.
Phendimetrazine Phendimetrazine may decrease the antihypertensive activities of Nitrendipine.
Epicaptopril Epicaptopril may decrease the antihypertensive activities of Nitrendipine.
1-benzylimidazole 1-benzylimidazole may decrease the antihypertensive activities of Nitrendipine.
Amineptine Amineptine may decrease the antihypertensive activities of Nitrendipine.
Amibegron Amibegron may decrease the antihypertensive activities of Nitrendipine.
Naluzotan Naluzotan may decrease the antihypertensive activities of Nitrendipine.
Solabegron Solabegron may decrease the antihypertensive activities of Nitrendipine.
Droxidopa Droxidopa may decrease the antihypertensive activities of Nitrendipine.
Esmirtazapine Esmirtazapine may decrease the antihypertensive activities of Nitrendipine.
Nitrous oxide Nitrous oxide may decrease the antihypertensive activities of Nitrendipine.
Isometheptene Isometheptene may decrease the antihypertensive activities of Nitrendipine.
Levonordefrin Levonordefrin may decrease the antihypertensive activities of Nitrendipine.
Naphazoline Naphazoline may decrease the antihypertensive activities of Nitrendipine.
Tetryzoline Tetryzoline may decrease the antihypertensive activities of Nitrendipine.
Cinitapride Cinitapride may decrease the antihypertensive activities of Nitrendipine.
Tyramine Tyramine may decrease the antihypertensive activities of Nitrendipine.
Adrafinil Adrafinil may decrease the antihypertensive activities of Nitrendipine.
Ifenprodil Ifenprodil may decrease the antihypertensive activities of Nitrendipine.
Hexoprenaline Hexoprenaline may decrease the antihypertensive activities of Nitrendipine.
Etilefrine Etilefrine may decrease the antihypertensive activities of Nitrendipine.
Dimetacrine Dimetacrine may decrease the antihypertensive activities of Nitrendipine.
Cirazoline Cirazoline may decrease the antihypertensive activities of Nitrendipine.
Synephrine Synephrine may decrease the antihypertensive activities of Nitrendipine.
Moxisylyte Moxisylyte may decrease the antihypertensive activities of Nitrendipine.
Oxaprotiline Oxaprotiline may decrease the antihypertensive activities of Nitrendipine.
Iofetamine I-123 Iofetamine I-123 may decrease the antihypertensive activities of Nitrendipine.
Racepinephrine Racepinephrine may decrease the antihypertensive activities of Nitrendipine.
DL-Methylephedrine DL-Methylephedrine may decrease the antihypertensive activities of Nitrendipine.
Amitraz Amitraz may decrease the antihypertensive activities of Nitrendipine.
Medetomidine Medetomidine may decrease the antihypertensive activities of Nitrendipine.
Xylazine Xylazine may decrease the antihypertensive activities of Nitrendipine.

Target Protein

Voltage-dependent L-type calcium channel subunit alpha-1C CACNA1C
Voltage-dependent calcium channel subunit alpha-2/delta-1 CACNA2D1
Voltage-dependent L-type calcium channel subunit beta-2 CACNB2
Voltage-dependent L-type calcium channel subunit alpha-1D CACNA1D
Voltage-dependent L-type calcium channel subunit alpha-1S CACNA1S
Voltage-dependent calcium channel subunit alpha-2/delta-2 CACNA2D2
Voltage-dependent T-type calcium channel subunit alpha-1H CACNA1H
Voltage-dependent L-type calcium channel CACNA1C
Calcium-activated potassium channel KCNMA1

Referensi & Sumber

Synthesis reference: Wolfgang Schmidt, Bernhard Streuff, Manfred Winter, "Preparation of solid medicament formulation containing nitrendipine." U.S. Patent US4724141, issued April, 1980.

Contoh Produk & Brand

Produk: 0 • International brands: 7
International Brands
  • Bayotensin
  • Baypress
  • Bylotensin
  • Deiten
  • Nidrel
  • Nitrepin
  • Nitrezic

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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