Gatifloxacin

DB01044

small molecule approved investigational withdrawn

Deskripsi

Gatifloxacin is an antibiotic agent and a member of the fourth-generation fluoroquinolone family. It works by inhibiting the bacterial enzymes DNA gyrase and topoisomerase IV. It was first introduced by Bristol-Myers Squibb in 1999 under the brand name Tequin® for the treatment of respiratory tract infections. Gatifloxacin is available as tablets and in various aqueous solutions for intravenous therapy. It is also available as eye drops under the brand name Zymar® marketed by Allergan.

The FDA withdrew its approval for the use of non-ophthalmic drug products containing gatifloxacin due to the high prevalence of gatifloxacin-associated dysglycemia adverse event reports and the high incidence of hyperglycemic and hypoglycemic episodes in patients taking gatifloxacin compared to those on macrolide antibiotics.L43942,L44037

Struktur Molekul 2D

Berat 375.3941
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 7-14 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Well absorbed from the gastrointestinal tract after oral administration with absolute bioavailability of gatifloxacin is 96%

Metabolisme

Gatifloxacin undergoes limited biotransformation in humans with less than 1% of the dose excreted in the urine as ethylenediamine and methylethylenediamine metabolites

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Drink plenty of fluids.
  • 2. Take with or without food. The absorption is unaffected by food.

Interaksi Obat

952 Data
Didanosine Didanosine can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Probenecid Probenecid may decrease the excretion rate of Gatifloxacin which could result in a higher serum level.
Quinapril Quinapril can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium acetate Calcium acetate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sevelamer Sevelamer can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Iron Dextran Iron Dextran can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium Calcium can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium carbonate Calcium carbonate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lanthanum carbonate Lanthanum carbonate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric carboxymaltose Ferric carboxymaltose can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Iron sucrose Iron sucrose can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric pyrophosphate Ferric pyrophosphate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium citrate Calcium citrate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium gluconate Calcium gluconate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric sulfate Ferric sulfate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric cation Ferric cation can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tetraferric tricitrate decahydrate Tetraferric tricitrate decahydrate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Lanthanum III cation Lanthanum III cation can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Calcium polycarbophil Calcium polycarbophil can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ferric oxyhydroxide Ferric oxyhydroxide can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Sucralfate Sucralfate can cause a decrease in the absorption of Gatifloxacin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Zolmitriptan The metabolism of Zolmitriptan can be decreased when combined with Gatifloxacin.
Nitrofurantoin The therapeutic efficacy of Gatifloxacin can be decreased when used in combination with Nitrofurantoin.
Agomelatine The serum concentration of Agomelatine can be increased when it is combined with Gatifloxacin.
Pirfenidone The metabolism of Pirfenidone can be decreased when combined with Gatifloxacin.
Tizanidine The serum concentration of Tizanidine can be increased when it is combined with Gatifloxacin.
Mycophenolate mofetil The serum concentration of Mycophenolate mofetil can be decreased when it is combined with Gatifloxacin.
Mycophenolic acid The serum concentration of Mycophenolic acid can be decreased when it is combined with Gatifloxacin.
Picosulfuric acid The therapeutic efficacy of Picosulfuric acid can be decreased when used in combination with Gatifloxacin.
Insulin human The therapeutic efficacy of Insulin human can be increased when used in combination with Gatifloxacin.
Insulin lispro The therapeutic efficacy of Insulin lispro can be increased when used in combination with Gatifloxacin.
Insulin pork The therapeutic efficacy of Insulin pork can be increased when used in combination with Gatifloxacin.
Troglitazone The therapeutic efficacy of Troglitazone can be increased when used in combination with Gatifloxacin.
Glimepiride The therapeutic efficacy of Glimepiride can be increased when used in combination with Gatifloxacin.
Sulfisoxazole The therapeutic efficacy of Sulfisoxazole can be increased when used in combination with Gatifloxacin.
Acarbose The therapeutic efficacy of Acarbose can be increased when used in combination with Gatifloxacin.
Metformin The therapeutic efficacy of Metformin can be increased when used in combination with Gatifloxacin.
Sulfadiazine The therapeutic efficacy of Sulfadiazine can be increased when used in combination with Gatifloxacin.
Rosiglitazone The therapeutic efficacy of Rosiglitazone can be increased when used in combination with Gatifloxacin.
Acetohexamide The therapeutic efficacy of Acetohexamide can be increased when used in combination with Gatifloxacin.
Miglitol The therapeutic efficacy of Miglitol can be increased when used in combination with Gatifloxacin.
Chlorpropamide The therapeutic efficacy of Chlorpropamide can be increased when used in combination with Gatifloxacin.
Nateglinide The therapeutic efficacy of Nateglinide can be increased when used in combination with Gatifloxacin.
Pentamidine The therapeutic efficacy of Pentamidine can be increased when used in combination with Gatifloxacin.
Tolazamide The therapeutic efficacy of Tolazamide can be increased when used in combination with Gatifloxacin.
Repaglinide The therapeutic efficacy of Repaglinide can be increased when used in combination with Gatifloxacin.
Phenformin The therapeutic efficacy of Phenformin can be increased when used in combination with Gatifloxacin.
Sulfamethoxazole The therapeutic efficacy of Sulfamethoxazole can be increased when used in combination with Gatifloxacin.
Glyburide The therapeutic efficacy of Glyburide can be increased when used in combination with Gatifloxacin.
Glipizide The therapeutic efficacy of Glipizide can be increased when used in combination with Gatifloxacin.
Gliclazide The therapeutic efficacy of Gliclazide can be increased when used in combination with Gatifloxacin.
Tolbutamide The therapeutic efficacy of Tolbutamide can be increased when used in combination with Gatifloxacin.
Pioglitazone The therapeutic efficacy of Pioglitazone can be increased when used in combination with Gatifloxacin.
Bromocriptine The therapeutic efficacy of Bromocriptine can be increased when used in combination with Gatifloxacin.
Gliquidone The therapeutic efficacy of Gliquidone can be increased when used in combination with Gatifloxacin.
Mitiglinide The therapeutic efficacy of Mitiglinide can be increased when used in combination with Gatifloxacin.
Sitagliptin The therapeutic efficacy of Sitagliptin can be increased when used in combination with Gatifloxacin.
Sunitinib The therapeutic efficacy of Sunitinib can be increased when used in combination with Gatifloxacin.
Exenatide The therapeutic efficacy of Exenatide can be increased when used in combination with Gatifloxacin.
Mecasermin The therapeutic efficacy of Mecasermin can be increased when used in combination with Gatifloxacin.
Pramlintide The therapeutic efficacy of Pramlintide can be increased when used in combination with Gatifloxacin.
Glisoxepide The therapeutic efficacy of Glisoxepide can be increased when used in combination with Gatifloxacin.
Insulin aspart The therapeutic efficacy of Insulin aspart can be increased when used in combination with Gatifloxacin.
Insulin glulisine The therapeutic efficacy of Insulin glulisine can be increased when used in combination with Gatifloxacin.
Glymidine The therapeutic efficacy of Glymidine can be increased when used in combination with Gatifloxacin.
AICA ribonucleotide The therapeutic efficacy of AICA ribonucleotide can be increased when used in combination with Gatifloxacin.
Buformin The therapeutic efficacy of Buformin can be increased when used in combination with Gatifloxacin.
Vildagliptin The therapeutic efficacy of Vildagliptin can be increased when used in combination with Gatifloxacin.
Voglibose The therapeutic efficacy of Voglibose can be increased when used in combination with Gatifloxacin.
NN344 The therapeutic efficacy of NN344 can be increased when used in combination with Gatifloxacin.
AMG-222 The therapeutic efficacy of AMG-222 can be increased when used in combination with Gatifloxacin.
Bisegliptin The therapeutic efficacy of Bisegliptin can be increased when used in combination with Gatifloxacin.
Alogliptin The therapeutic efficacy of Alogliptin can be increased when used in combination with Gatifloxacin.
Dapagliflozin The therapeutic efficacy of Dapagliflozin can be increased when used in combination with Gatifloxacin.
Saxagliptin The therapeutic efficacy of Saxagliptin can be increased when used in combination with Gatifloxacin.
Liraglutide The therapeutic efficacy of Liraglutide can be increased when used in combination with Gatifloxacin.
Gosogliptin The therapeutic efficacy of Gosogliptin can be increased when used in combination with Gatifloxacin.
Linagliptin The therapeutic efficacy of Linagliptin can be increased when used in combination with Gatifloxacin.
Canagliflozin The therapeutic efficacy of Canagliflozin can be increased when used in combination with Gatifloxacin.
Glibornuride The therapeutic efficacy of Glibornuride can be increased when used in combination with Gatifloxacin.
Benfluorex The therapeutic efficacy of Benfluorex can be increased when used in combination with Gatifloxacin.
Empagliflozin The therapeutic efficacy of Empagliflozin can be increased when used in combination with Gatifloxacin.
Albiglutide The therapeutic efficacy of Albiglutide can be increased when used in combination with Gatifloxacin.
Dulaglutide The therapeutic efficacy of Dulaglutide can be increased when used in combination with Gatifloxacin.
Lobeglitazone The therapeutic efficacy of Lobeglitazone can be increased when used in combination with Gatifloxacin.
Netoglitazone The therapeutic efficacy of Netoglitazone can be increased when used in combination with Gatifloxacin.
Rivoglitazone The therapeutic efficacy of Rivoglitazone can be increased when used in combination with Gatifloxacin.
Ciglitazone The therapeutic efficacy of Ciglitazone can be increased when used in combination with Gatifloxacin.
Lixisenatide The therapeutic efficacy of Lixisenatide can be increased when used in combination with Gatifloxacin.
Insulin beef The therapeutic efficacy of Insulin beef can be increased when used in combination with Gatifloxacin.
Insulin degludec The therapeutic efficacy of Insulin degludec can be increased when used in combination with Gatifloxacin.
Insulin peglispro The therapeutic efficacy of Insulin peglispro can be increased when used in combination with Gatifloxacin.
Insulin tregopil The therapeutic efficacy of Insulin tregopil can be increased when used in combination with Gatifloxacin.
Ipragliflozin The therapeutic efficacy of Ipragliflozin can be increased when used in combination with Gatifloxacin.
Dutogliptin The therapeutic efficacy of Dutogliptin can be increased when used in combination with Gatifloxacin.
Allicin The therapeutic efficacy of Allicin can be increased when used in combination with Gatifloxacin.
Tofogliflozin The therapeutic efficacy of Tofogliflozin can be increased when used in combination with Gatifloxacin.
Ertugliflozin The therapeutic efficacy of Ertugliflozin can be increased when used in combination with Gatifloxacin.
2,4-thiazolidinedione The therapeutic efficacy of 2,4-thiazolidinedione can be increased when used in combination with Gatifloxacin.
Teneligliptin The therapeutic efficacy of Teneligliptin can be increased when used in combination with Gatifloxacin.

Target Protein

DNA gyrase subunit A gyrA
DNA gyrase subunit B gyrB
DNA gyrase subunit A gyrA
DNA gyrase subunit B gyrB
DNA topoisomerase 4 subunit A parC
DNA topoisomerase 4 subunit B parE

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16510739
    Park-Wyllie LY, Juurlink DN, Kopp A, Shah BR, Stukel TA, Stumpo C, Dresser L, Low DE, Mamdani MM: Outpatient gatifloxacin therapy and dysglycemia in older adults. N Engl J Med. 2006 Mar 30;354(13):1352-61. Epub 2006 Mar 1.
  • PMID: 16510740
    Gurwitz JH: Serious adverse drug effects--seeing the trees through the forest. N Engl J Med. 2006 Mar 30;354(13):1413-5. Epub 2006 Mar 1.

Contoh Produk & Brand

Produk: 28 • International brands: 0
Produk
  • Apo-gatifloxacin
    Solution • 0.3 % • Ophthalmic • Canada • Generic • Approved
  • Gati-Dex
    Solution / drops • - • Ophthalmic • US
  • Gatifloxacin
    Solution / drops • 5 mg/1mL • Ophthalmic • US • Generic • Approved
  • Gatifloxacin
    Solution • 3 mg/1mL • Ophthalmic • US • Generic • Approved
  • Gatifloxacin
    Solution / drops • 5 mg/1mL • Ophthalmic • US • Generic • Approved
  • Gatifloxacin
    Solution / drops • 5 mg/1mL • Ophthalmic • US • Generic • Approved
  • Gatifloxacin
    Solution / drops • 5 mg/1mL • Ophthalmic • US • Generic • Approved
  • Gatifloxacin
    Solution / drops • 5 mg/1mL • Ophthalmic • US • Generic • Approved
Menampilkan 8 dari 28 produk.

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