Probenecid

DB01032

small molecule approved investigational

Deskripsi

The prototypical uricosuric agent. It inhibits the renal excretion of organic anions and reduces tubular reabsorption of urate. Probenecid has also been used to treat patients with renal impairment, and, because it reduces the renal tubular excretion of other drugs, has been used as an adjunct to antibacterial therapy.

Struktur Molekul 2D

Berat 285.359
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 6-12 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Excreted principally in the urine as monoacyl glucuronide and unchanged drug. Alkalinization of urine increases renal probenecid excretion.

Interaksi Makanan

3 Data
  • 1. Avoid alcohol.
  • 2. Drink plenty of fluids.
  • 3. Take with food. Food reduces irritation.

Interaksi Obat

1328 Data
Aripiprazole The metabolism of Aripiprazole can be increased when combined with Probenecid.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be increased when combined with Probenecid.
Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Probenecid.
Lorazepam The serum concentration of Lorazepam can be increased when it is combined with Probenecid.
Oseltamivir The serum concentration of the active metabolites of Oseltamivir can be increased when Oseltamivir is used in combination with Probenecid.
Nicotine The risk or severity of adverse effects can be increased when Probenecid is combined with Nicotine.
Mecamylamine The risk or severity of adverse effects can be increased when Probenecid is combined with Mecamylamine.
Pentolinium The risk or severity of adverse effects can be increased when Probenecid is combined with Pentolinium.
Trimethaphan The risk or severity of adverse effects can be increased when Probenecid is combined with Trimethaphan.
Hexamethonium The risk or severity of adverse effects can be increased when Probenecid is combined with Hexamethonium.
Cyclopentamine The risk or severity of adverse effects can be increased when Probenecid is combined with Cyclopentamine.
Torasemide The risk or severity of adverse effects can be increased when Probenecid is combined with Torasemide.
Furosemide The risk or severity of adverse effects can be increased when Probenecid is combined with Furosemide.
Bumetanide The risk or severity of adverse effects can be increased when Probenecid is combined with Bumetanide.
Etacrynic acid The risk or severity of adverse effects can be increased when Probenecid is combined with Etacrynic acid.
Piretanide The risk or severity of adverse effects can be increased when Probenecid is combined with Piretanide.
Azosemide The risk or severity of adverse effects can be increased when Probenecid is combined with Azosemide.
Tripamide The risk or severity of adverse effects can be increased when Probenecid is combined with Tripamide.
Moxifloxacin Probenecid may decrease the excretion rate of Moxifloxacin which could result in a higher serum level.
Grepafloxacin Probenecid may decrease the excretion rate of Grepafloxacin which could result in a higher serum level.
Enoxacin Probenecid may decrease the excretion rate of Enoxacin which could result in a higher serum level.
Pefloxacin Probenecid may decrease the excretion rate of Pefloxacin which could result in a higher serum level.
Ciprofloxacin Probenecid may decrease the excretion rate of Ciprofloxacin which could result in a higher serum level.
Trovafloxacin Probenecid may decrease the excretion rate of Trovafloxacin which could result in a higher serum level.
Nalidixic acid Probenecid may decrease the excretion rate of Nalidixic acid which could result in a higher serum level.
Rosoxacin Probenecid may decrease the excretion rate of Rosoxacin which could result in a higher serum level.
Cinoxacin Probenecid may decrease the excretion rate of Cinoxacin which could result in a higher serum level.
Lomefloxacin Probenecid may decrease the excretion rate of Lomefloxacin which could result in a higher serum level.
Gatifloxacin Probenecid may decrease the excretion rate of Gatifloxacin which could result in a higher serum level.
Norfloxacin Probenecid may decrease the excretion rate of Norfloxacin which could result in a higher serum level.
Ofloxacin Probenecid may decrease the excretion rate of Ofloxacin which could result in a higher serum level.
Sparfloxacin Probenecid may decrease the excretion rate of Sparfloxacin which could result in a higher serum level.
Temafloxacin Probenecid may decrease the excretion rate of Temafloxacin which could result in a higher serum level.
Fleroxacin Probenecid may decrease the excretion rate of Fleroxacin which could result in a higher serum level.
Technetium Tc-99m ciprofloxacin Probenecid may decrease the excretion rate of Technetium Tc-99m ciprofloxacin which could result in a higher serum level.
Garenoxacin Probenecid may decrease the excretion rate of Garenoxacin which could result in a higher serum level.
Nemonoxacin Probenecid may decrease the excretion rate of Nemonoxacin which could result in a higher serum level.
Flumequine Probenecid may decrease the excretion rate of Flumequine which could result in a higher serum level.
Enrofloxacin Probenecid may decrease the excretion rate of Enrofloxacin which could result in a higher serum level.
Orbifloxacin Probenecid may decrease the excretion rate of Orbifloxacin which could result in a higher serum level.
Sarafloxacin Probenecid may decrease the excretion rate of Sarafloxacin which could result in a higher serum level.
Difloxacin Probenecid may decrease the excretion rate of Difloxacin which could result in a higher serum level.
Pazufloxacin Probenecid may decrease the excretion rate of Pazufloxacin which could result in a higher serum level.
Prulifloxacin Probenecid may decrease the excretion rate of Prulifloxacin which could result in a higher serum level.
Delafloxacin Probenecid may decrease the excretion rate of Delafloxacin which could result in a higher serum level.
Sitafloxacin Probenecid may decrease the excretion rate of Sitafloxacin which could result in a higher serum level.
Oxolinic acid Probenecid may decrease the excretion rate of Oxolinic acid which could result in a higher serum level.
Rufloxacin Probenecid may decrease the excretion rate of Rufloxacin which could result in a higher serum level.
Pipemidic acid Probenecid may decrease the excretion rate of Pipemidic acid which could result in a higher serum level.
Glimepiride The protein binding of Glimepiride can be decreased when combined with Probenecid.
Acetohexamide The protein binding of Acetohexamide can be decreased when combined with Probenecid.
Chlorpropamide The protein binding of Chlorpropamide can be decreased when combined with Probenecid.
Tolazamide The protein binding of Tolazamide can be decreased when combined with Probenecid.
Glyburide The protein binding of Glyburide can be decreased when combined with Probenecid.
Glipizide The protein binding of Glipizide can be decreased when combined with Probenecid.
Gliclazide The protein binding of Gliclazide can be decreased when combined with Probenecid.
Tolbutamide The protein binding of Tolbutamide can be decreased when combined with Probenecid.
Gliquidone The protein binding of Gliquidone can be decreased when combined with Probenecid.
Glisoxepide The protein binding of Glisoxepide can be decreased when combined with Probenecid.
Glibornuride The protein binding of Glibornuride can be decreased when combined with Probenecid.
Carbutamide The protein binding of Carbutamide can be decreased when combined with Probenecid.
Metahexamide The protein binding of Metahexamide can be decreased when combined with Probenecid.
Irinotecan The risk or severity of neutropenia can be increased when Probenecid is combined with Irinotecan.
Aminosalicylic acid The therapeutic efficacy of Probenecid can be decreased when used in combination with Aminosalicylic acid.
Bismuth subsalicylate The therapeutic efficacy of Probenecid can be decreased when used in combination with Bismuth subsalicylate.
Dersalazine The therapeutic efficacy of Probenecid can be decreased when used in combination with Dersalazine.
Phenyl aminosalicylate The therapeutic efficacy of Probenecid can be decreased when used in combination with Phenyl aminosalicylate.
Methyl salicylate The therapeutic efficacy of Probenecid can be decreased when used in combination with Methyl salicylate.
Aloxiprin The therapeutic efficacy of Probenecid can be decreased when used in combination with Aloxiprin.
Choline salicylate The therapeutic efficacy of Probenecid can be decreased when used in combination with Choline salicylate.
Thiosalicylic acid The therapeutic efficacy of Probenecid can be decreased when used in combination with Thiosalicylic acid.
Dapsone Probenecid may decrease the excretion rate of Dapsone which could result in a higher serum level.
Ertapenem Probenecid may decrease the excretion rate of Ertapenem which could result in a higher serum level.
Flucloxacillin The excretion of Flucloxacillin can be decreased when combined with Probenecid.
Piperacillin The excretion of Piperacillin can be decreased when combined with Probenecid.
Phenoxymethylpenicillin The excretion of Phenoxymethylpenicillin can be decreased when combined with Probenecid.
Dicloxacillin The excretion of Dicloxacillin can be decreased when combined with Probenecid.
Carbenicillin The excretion of Carbenicillin can be decreased when combined with Probenecid.
Nafcillin The excretion of Nafcillin can be decreased when combined with Probenecid.
Oxacillin The excretion of Oxacillin can be decreased when combined with Probenecid.
Hetacillin The excretion of Hetacillin can be decreased when combined with Probenecid.
Benzylpenicilloyl polylysine The excretion of Benzylpenicilloyl polylysine can be decreased when combined with Probenecid.
Mezlocillin The excretion of Mezlocillin can be decreased when combined with Probenecid.
Cyclacillin The excretion of Cyclacillin can be decreased when combined with Probenecid.
Benzylpenicillin The excretion of Benzylpenicillin can be decreased when combined with Probenecid.
Amoxicillin The excretion of Amoxicillin can be decreased when combined with Probenecid.
Azlocillin The excretion of Azlocillin can be decreased when combined with Probenecid.
Cloxacillin The excretion of Cloxacillin can be decreased when combined with Probenecid.
Amdinocillin The excretion of Amdinocillin can be decreased when combined with Probenecid.
Bacampicillin The excretion of Bacampicillin can be decreased when combined with Probenecid.
Meticillin The excretion of Meticillin can be decreased when combined with Probenecid.
Pivampicillin The excretion of Pivampicillin can be decreased when combined with Probenecid.
Pivmecillinam The excretion of Pivmecillinam can be decreased when combined with Probenecid.
Ticarcillin The excretion of Ticarcillin can be decreased when combined with Probenecid.
Azidocillin The excretion of Azidocillin can be decreased when combined with Probenecid.
Carindacillin The excretion of Carindacillin can be decreased when combined with Probenecid.
Procaine benzylpenicillin The excretion of Procaine benzylpenicillin can be decreased when combined with Probenecid.
Sultamicillin The excretion of Sultamicillin can be decreased when combined with Probenecid.
Temocillin The excretion of Temocillin can be decreased when combined with Probenecid.
Epicillin The excretion of Epicillin can be decreased when combined with Probenecid.

Target Protein

Solute carrier family 22 member 6 SLC22A6
Solute carrier family 22 member 11 SLC22A11
Organic anion transporter 3 SLC22A8
Pannexin-1 PANX1
Taste receptor type 2 member 16 TAS2R16

Referensi & Sumber

Artikel (PubMed)
  • PMID: 16267514
    Butler D: Wartime tactic doubles power of scarce bird-flu drug. Nature. 2005 Nov 3;438(7064):6.

Contoh Produk & Brand

Produk: 28 • International brands: 5
Produk
  • Benemid Tab 500mg
    Tablet • 500 mg / tab • Oral • Canada • Approved
  • Benuryl
    Tablet • 500 mg • Oral • Canada • Approved
  • Pro Biosan Kit
    Capsule; Tablet • - • Oral • Canada • Approved
  • Probenecid
    Tablet, film coated • 500 mg/1 • Oral • US • Generic • Approved
  • Probenecid
    Tablet, film coated • 500 mg/1 • Oral • US • Generic • Approved
  • Probenecid
    Tablet, film coated • 500 mg/1 • Oral • US • Generic • Approved
  • Probenecid
    Tablet, film coated • 500 mg/1 • Oral • US • Generic • Approved
  • Probenecid
    Tablet • 500 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 28 produk.
International Brands
  • Benecid
  • Benemid
  • Probalan
  • Probecid
  • Proben

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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