Peringatan Keamanan

LD50=3600 mg/kg (Orally in rats). Symptoms of overexposure include eye irritation, CNS depression, analgesia, anesthesia, seizures, respiratory depression, and liver and kidney damage.

Methoxyflurane

DB01028

small molecule approved investigational vet_approved withdrawn

Deskripsi

An inhalation anesthetic. Currently, methoxyflurane is rarely used for surgical, obstetric, or dental anesthesia. If so employed, it should be administered with nitrous oxide to achieve a relatively light level of anesthesia, and a neuromuscular blocking agent given concurrently to obtain the desired degree of muscular relaxation. (From AMA Drug Evaluations Annual, 1994, p180)

In the US, methoxyflurane is one of the products that have been withdrawn or removed from the market for reasons of safety or effectiveness.L43942

Struktur Molekul 2D

Berat 164.966
Wujud liquid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Avoid alcohol. Ingesting alcohol may increase the CNS depressant effects of methoxyflurane.

Interaksi Obat

1464 Data
Ramipril Methoxyflurane may decrease the antihypertensive activities of Ramipril.
Remikiren Methoxyflurane may decrease the antihypertensive activities of Remikiren.
Guanadrel Methoxyflurane may decrease the antihypertensive activities of Guanadrel.
Olmesartan Methoxyflurane may decrease the antihypertensive activities of Olmesartan.
Chlorthalidone Methoxyflurane may decrease the antihypertensive activities of Chlorthalidone.
Nitroprusside Methoxyflurane may decrease the antihypertensive activities of Nitroprusside.
Minoxidil Methoxyflurane may decrease the antihypertensive activities of Minoxidil.
Bendroflumethiazide Methoxyflurane may decrease the antihypertensive activities of Bendroflumethiazide.
Prazosin Methoxyflurane may decrease the antihypertensive activities of Prazosin.
Fosinopril Methoxyflurane may decrease the antihypertensive activities of Fosinopril.
Trandolapril Methoxyflurane may decrease the antihypertensive activities of Trandolapril.
Metolazone Methoxyflurane may decrease the antihypertensive activities of Metolazone.
Benazepril Methoxyflurane may decrease the antihypertensive activities of Benazepril.
Cyclothiazide Methoxyflurane may decrease the antihypertensive activities of Cyclothiazide.
Candoxatril Methoxyflurane may decrease the antihypertensive activities of Candoxatril.
Mecamylamine Methoxyflurane may decrease the antihypertensive activities of Mecamylamine.
Moexipril Methoxyflurane may decrease the antihypertensive activities of Moexipril.
Lisinopril Methoxyflurane may decrease the antihypertensive activities of Lisinopril.
Nitroglycerin Methoxyflurane may decrease the antihypertensive activities of Nitroglycerin.
Hydroflumethiazide Methoxyflurane may decrease the antihypertensive activities of Hydroflumethiazide.
Cryptenamine Methoxyflurane may decrease the antihypertensive activities of Cryptenamine.
Perindopril Methoxyflurane may decrease the antihypertensive activities of Perindopril.
Fenoldopam Methoxyflurane may decrease the antihypertensive activities of Fenoldopam.
Eprosartan Methoxyflurane may decrease the antihypertensive activities of Eprosartan.
Chlorothiazide Methoxyflurane may decrease the antihypertensive activities of Chlorothiazide.
Quinapril Methoxyflurane may decrease the antihypertensive activities of Quinapril.
Telmisartan Methoxyflurane may decrease the antihypertensive activities of Telmisartan.
Methyldopa Methoxyflurane may decrease the antihypertensive activities of Methyldopa.
Hydrochlorothiazide Methoxyflurane may decrease the antihypertensive activities of Hydrochlorothiazide.
Trichlormethiazide Methoxyflurane may decrease the antihypertensive activities of Trichlormethiazide.
Deserpidine Methoxyflurane may decrease the antihypertensive activities of Deserpidine.
Pentolinium Methoxyflurane may decrease the antihypertensive activities of Pentolinium.
Trimethaphan Methoxyflurane may decrease the antihypertensive activities of Trimethaphan.
Diazoxide Methoxyflurane may decrease the antihypertensive activities of Diazoxide.
Bretylium Methoxyflurane may decrease the antihypertensive activities of Bretylium.
Terazosin Methoxyflurane may decrease the antihypertensive activities of Terazosin.
Epoprostenol Methoxyflurane may decrease the antihypertensive activities of Epoprostenol.
Polythiazide Methoxyflurane may decrease the antihypertensive activities of Polythiazide.
Cilazapril Methoxyflurane may decrease the antihypertensive activities of Cilazapril.
Saprisartan Methoxyflurane may decrease the antihypertensive activities of Saprisartan.
Spirapril Methoxyflurane may decrease the antihypertensive activities of Spirapril.
Dexpropranolol Methoxyflurane may decrease the antihypertensive activities of Dexpropranolol.
Diethylnorspermine Methoxyflurane may decrease the antihypertensive activities of Diethylnorspermine.
Temocapril Methoxyflurane may decrease the antihypertensive activities of Temocapril.
Trimazosin Methoxyflurane may decrease the antihypertensive activities of Trimazosin.
Nicorandil Methoxyflurane may decrease the antihypertensive activities of Nicorandil.
Rauwolfia serpentina root Methoxyflurane may decrease the antihypertensive activities of Rauwolfia serpentina root.
Enalaprilat Methoxyflurane may decrease the antihypertensive activities of Enalaprilat.
Angiotensin 1-7 Methoxyflurane may decrease the antihypertensive activities of Angiotensin 1-7.
Imidapril Methoxyflurane may decrease the antihypertensive activities of Imidapril.
BQ-123 Methoxyflurane may decrease the antihypertensive activities of BQ-123.
Cicletanine Methoxyflurane may decrease the antihypertensive activities of Cicletanine.
Dihydralazine Methoxyflurane may decrease the antihypertensive activities of Dihydralazine.
Zofenopril Methoxyflurane may decrease the antihypertensive activities of Zofenopril.
Guanoxan Methoxyflurane may decrease the antihypertensive activities of Guanoxan.
Delapril Methoxyflurane may decrease the antihypertensive activities of Delapril.
Vincamine Methoxyflurane may decrease the antihypertensive activities of Vincamine.
Linsidomine Methoxyflurane may decrease the antihypertensive activities of Linsidomine.
Guanoxabenz Methoxyflurane may decrease the antihypertensive activities of Guanoxabenz.
Tolonidine Methoxyflurane may decrease the antihypertensive activities of Tolonidine.
Endralazine Methoxyflurane may decrease the antihypertensive activities of Endralazine.
Cadralazine Methoxyflurane may decrease the antihypertensive activities of Cadralazine.
Cyclopenthiazide Methoxyflurane may decrease the antihypertensive activities of Cyclopenthiazide.
Bietaserpine Methoxyflurane may decrease the antihypertensive activities of Bietaserpine.
Guanazodine Methoxyflurane may decrease the antihypertensive activities of Guanazodine.
Methoserpidine Methoxyflurane may decrease the antihypertensive activities of Methoserpidine.
Guanoclor Methoxyflurane may decrease the antihypertensive activities of Guanoclor.
Muzolimine Methoxyflurane may decrease the antihypertensive activities of Muzolimine.
Xipamide Methoxyflurane may decrease the antihypertensive activities of Xipamide.
Tocopherylquinone Methoxyflurane may decrease the antihypertensive activities of Tocopherylquinone.
Benazeprilat Methoxyflurane may decrease the antihypertensive activities of Benazeprilat.
Fosinoprilat Methoxyflurane may decrease the antihypertensive activities of Fosinoprilat.
Ramiprilat Methoxyflurane may decrease the antihypertensive activities of Ramiprilat.
Perindoprilat Methoxyflurane may decrease the antihypertensive activities of Perindoprilat.
Quinaprilat Methoxyflurane may decrease the antihypertensive activities of Quinaprilat.
Furosemide Methoxyflurane may decrease the antihypertensive activities of Furosemide.
Enalapril Methoxyflurane may decrease the antihypertensive activities of Enalapril.
Captopril Methoxyflurane may decrease the antihypertensive activities of Captopril.
Isradipine The metabolism of Methoxyflurane can be decreased when combined with Isradipine.
Diltiazem The metabolism of Methoxyflurane can be decreased when combined with Diltiazem.
Nimodipine Methoxyflurane may decrease the antihypertensive activities of Nimodipine.
Nisoldipine Methoxyflurane may decrease the antihypertensive activities of Nisoldipine.
Propranolol Methoxyflurane may decrease the antihypertensive activities of Propranolol.
Doxazosin Methoxyflurane may decrease the antihypertensive activities of Doxazosin.
Bisoprolol Methoxyflurane may decrease the antihypertensive activities of Bisoprolol.
Losartan Methoxyflurane may decrease the antihypertensive activities of Losartan.
Eplerenone Methoxyflurane may decrease the antihypertensive activities of Eplerenone.
Indapamide Methoxyflurane may decrease the antihypertensive activities of Indapamide.
Tadalafil Methoxyflurane may decrease the antihypertensive activities of Tadalafil.
Irbesartan Methoxyflurane may decrease the antihypertensive activities of Irbesartan.
Nitrendipine Methoxyflurane may decrease the antihypertensive activities of Nitrendipine.
Guanethidine Methoxyflurane may decrease the antihypertensive activities of Guanethidine.
Hydralazine Methoxyflurane may decrease the antihypertensive activities of Hydralazine.
Nebivolol Methoxyflurane may decrease the antihypertensive activities of Nebivolol.
Ambrisentan Methoxyflurane may decrease the antihypertensive activities of Ambrisentan.
Pinacidil Methoxyflurane may decrease the antihypertensive activities of Pinacidil.
Riociguat Methoxyflurane may decrease the antihypertensive activities of Riociguat.
Macitentan Methoxyflurane may decrease the antihypertensive activities of Macitentan.
Aliskiren Methoxyflurane may decrease the antihypertensive activities of Aliskiren.
Efonidipine Methoxyflurane may decrease the antihypertensive activities of Efonidipine.

Target Protein

Gamma-aminobutyric acid receptor subunit alpha-1 GABRA1
Glutamate receptor 1 GRIA1
Glycine receptor subunit alpha-1 GLRA1
Potassium voltage-gated channel subfamily A member 1 KCNA1
GABA(A) Receptor GABRA1
Calcium-transporting ATPase type 2C member 1 ATP2C1
NADH-ubiquinone oxidoreductase chain 1 MT-ND1

Contoh Produk & Brand

Produk: 2 • International brands: 1
Produk
  • Penthrox
    Solution • 99.9 % • Respiratory (inhalation) • Canada • Approved
  • Penthrox
    Kit; Solution • 99.9 % • Respiratory (inhalation) • Canada • Approved
International Brands
  • Penthrane — Abbott Laboratories

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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