Peringatan Keamanan

A single oral dose of balsalazide disodium at 5 grams/kg or 4-aminobenzoyl-(beta)-alanine, a metabolite of balsalazide disodium, at 1 gram/kg was non-lethal in mice and rats. No symptoms of acute toxicity were seen at these doses.

Balsalazide

DB01014

small molecule approved investigational

Deskripsi

Balsalazide is an anti-inflammatory drug used in the treatment of Inflammatory Bowel Disease. It is sold under the name "Colazal" in the US and "Colazide" in the UK.

The chemical name is (E)-5-[-4-(2-carboxyethyl) aminocarbonyl phenyl]azo] -2-hydroxybenzoic acid. It is usually administered as the disodium salt.

Balsalazide works by deliverying mesalazine to the large intestine to act directly on ulcerative colitis. Mesalazine is also known as 5-aminosalicylic acid, or 5-ASA.

Struktur Molekul 2D

Berat 357.3175
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) Half-life could not be determined.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Low and variable, intact balsalazide is poorly absorbed systemically.

Metabolisme

Cleaved in the colon via bacterial azoreduction to 5–aminosalicylic acid (5–ASA) and 4–aminobenzoyl-beta-alanine, the inactive carrier moiety.

Rute Eliminasi

The products of the azoreduction of this compound, 5-ASA and 4-aminobenzoyl-ß-alanine, and their N-acetylated metabolites have been identified in plasma, urine and feces. Following single-dose administration of 2.25 g COLAZAL (three 750 mg capsules) under fasting conditions in healthy subjects, mean urinary recovery of balsalazide, 5-ASA, and N-Ac-5-ASA was 0.20%, 0.22% and 10.2%, respectively.

Interaksi Makanan

1 Data
  • 1. Take with or without food.

Interaksi Obat

1492 Data
Amlodipine Balsalazide may decrease the antihypertensive activities of Amlodipine.
Phentermine The risk or severity of hypertension can be increased when Phentermine is combined with Balsalazide.
Midodrine The risk or severity of hypertension can be increased when Midodrine is combined with Balsalazide.
Eletriptan The risk or severity of hypertension can be increased when Eletriptan is combined with Balsalazide.
Isoetharine The risk or severity of hypertension can be increased when Isoetharine is combined with Balsalazide.
Ziprasidone The risk or severity of hypertension can be increased when Ziprasidone is combined with Balsalazide.
Methysergide The risk or severity of hypertension can be increased when Methysergide is combined with Balsalazide.
Cabergoline The risk or severity of hypertension can be increased when Cabergoline is combined with Balsalazide.
Zolmitriptan The risk or severity of hypertension can be increased when Zolmitriptan is combined with Balsalazide.
Dihydroergotamine The risk or severity of hypertension can be increased when Dihydroergotamine is combined with Balsalazide.
Methylergometrine The risk or severity of hypertension can be increased when Methylergometrine is combined with Balsalazide.
Norepinephrine The risk or severity of hypertension can be increased when Norepinephrine is combined with Balsalazide.
Mirtazapine The risk or severity of hypertension can be increased when Mirtazapine is combined with Balsalazide.
Phenylephrine The risk or severity of hypertension can be increased when Phenylephrine is combined with Balsalazide.
Phenylpropanolamine The risk or severity of hypertension can be increased when Phenylpropanolamine is combined with Balsalazide.
Promazine The risk or severity of hypertension can be increased when Promazine is combined with Balsalazide.
Droperidol The risk or severity of hypertension can be increased when Droperidol is combined with Balsalazide.
Doxapram The risk or severity of hypertension can be increased when Doxapram is combined with Balsalazide.
Atropine The risk or severity of hypertension can be increased when Atropine is combined with Balsalazide.
Lisuride The risk or severity of hypertension can be increased when Lisuride is combined with Balsalazide.
Linezolid The risk or severity of hypertension can be increased when Linezolid is combined with Balsalazide.
Metaraminol The risk or severity of hypertension can be increased when Metaraminol is combined with Balsalazide.
Furazolidone The risk or severity of hypertension can be increased when Furazolidone is combined with Balsalazide.
Epinephrine The risk or severity of hypertension can be increased when Epinephrine is combined with Balsalazide.
Thioridazine The risk or severity of hypertension can be increased when Thioridazine is combined with Balsalazide.
Ergotamine The risk or severity of hypertension can be increased when Ergotamine is combined with Balsalazide.
Nicergoline The risk or severity of hypertension can be increased when Nicergoline is combined with Balsalazide.
Sufentanil The risk or severity of hypertension can be increased when Sufentanil is combined with Balsalazide.
Methoxamine The risk or severity of hypertension can be increased when Methoxamine is combined with Balsalazide.
Risperidone The risk or severity of hypertension can be increased when Risperidone is combined with Balsalazide.
Tranylcypromine The risk or severity of hypertension can be increased when Tranylcypromine is combined with Balsalazide.
Isoflurane The risk or severity of hypertension can be increased when Isoflurane is combined with Balsalazide.
Propiomazine The risk or severity of hypertension can be increased when Propiomazine is combined with Balsalazide.
Alfentanil The risk or severity of hypertension can be increased when Alfentanil is combined with Balsalazide.
Minaprine The risk or severity of hypertension can be increased when Minaprine is combined with Balsalazide.
Orciprenaline The risk or severity of hypertension can be increased when Orciprenaline is combined with Balsalazide.
Propofol The risk or severity of hypertension can be increased when Propofol is combined with Balsalazide.
Phenmetrazine The risk or severity of hypertension can be increased when Phenmetrazine is combined with Balsalazide.
Trifluoperazine The risk or severity of hypertension can be increased when Trifluoperazine is combined with Balsalazide.
Pseudoephedrine The risk or severity of hypertension can be increased when Pseudoephedrine is combined with Balsalazide.
Benzphetamine The risk or severity of hypertension can be increased when Benzphetamine is combined with Balsalazide.
Ritodrine The risk or severity of hypertension can be increased when Ritodrine is combined with Balsalazide.
Flupentixol The risk or severity of hypertension can be increased when Flupentixol is combined with Balsalazide.
Remifentanil The risk or severity of hypertension can be increased when Remifentanil is combined with Balsalazide.
Bitolterol The risk or severity of hypertension can be increased when Bitolterol is combined with Balsalazide.
Oxymetazoline The risk or severity of hypertension can be increased when Oxymetazoline is combined with Balsalazide.
Diethylpropion The risk or severity of hypertension can be increased when Diethylpropion is combined with Balsalazide.
Salmeterol The risk or severity of hypertension can be increased when Salmeterol is combined with Balsalazide.
Naratriptan The risk or severity of hypertension can be increased when Naratriptan is combined with Balsalazide.
Formoterol The risk or severity of hypertension can be increased when Formoterol is combined with Balsalazide.
Frovatriptan The risk or severity of hypertension can be increased when Frovatriptan is combined with Balsalazide.
Methoxyflurane The risk or severity of hypertension can be increased when Balsalazide is combined with Methoxyflurane.
Selegiline The risk or severity of hypertension can be increased when Balsalazide is combined with Selegiline.
Ergoloid mesylate The risk or severity of hypertension can be increased when Balsalazide is combined with Ergoloid mesylate.
Isoprenaline The risk or severity of hypertension can be increased when Balsalazide is combined with Isoprenaline.
Arbutamine The risk or severity of hypertension can be increased when Balsalazide is combined with Arbutamine.
Dutasteride The risk or severity of hypertension can be increased when Balsalazide is combined with Dutasteride.
Halothane The risk or severity of hypertension can be increased when Balsalazide is combined with Halothane.
Moclobemide The risk or severity of hypertension can be increased when Balsalazide is combined with Moclobemide.
Pergolide The risk or severity of hypertension can be increased when Balsalazide is combined with Pergolide.
Desflurane The risk or severity of hypertension can be increased when Balsalazide is combined with Desflurane.
Finasteride The risk or severity of hypertension can be increased when Balsalazide is combined with Finasteride.
Aripiprazole The risk or severity of hypertension can be increased when Balsalazide is combined with Aripiprazole.
Isocarboxazid The risk or severity of hypertension can be increased when Balsalazide is combined with Isocarboxazid.
Ergometrine The risk or severity of hypertension can be increased when Balsalazide is combined with Ergometrine.
Lisdexamfetamine The risk or severity of hypertension can be increased when Balsalazide is combined with Lisdexamfetamine.
Fenoterol The risk or severity of hypertension can be increased when Balsalazide is combined with Fenoterol.
Pirbuterol The risk or severity of hypertension can be increased when Balsalazide is combined with Pirbuterol.
Ephedra sinica root The risk or severity of hypertension can be increased when Balsalazide is combined with Ephedra sinica root.
Ephedrine The risk or severity of hypertension can be increased when Balsalazide is combined with Ephedrine.
Mephentermine The risk or severity of hypertension can be increased when Balsalazide is combined with Mephentermine.
Procaterol The risk or severity of hypertension can be increased when Balsalazide is combined with Procaterol.
Yohimbine The risk or severity of hypertension can be increased when Balsalazide is combined with Yohimbine.
Methotrimeprazine The risk or severity of hypertension can be increased when Balsalazide is combined with Methotrimeprazine.
Clenbuterol The risk or severity of hypertension can be increased when Balsalazide is combined with Clenbuterol.
Bambuterol The risk or severity of hypertension can be increased when Balsalazide is combined with Bambuterol.
MMDA The risk or severity of hypertension can be increased when Balsalazide is combined with MMDA.
Midomafetamine The risk or severity of hypertension can be increased when Balsalazide is combined with Midomafetamine.
2,5-Dimethoxy-4-ethylamphetamine The risk or severity of hypertension can be increased when Balsalazide is combined with 2,5-Dimethoxy-4-ethylamphetamine.
4-Methoxyamphetamine The risk or severity of hypertension can be increased when Balsalazide is combined with 4-Methoxyamphetamine.
4-Bromo-2,5-dimethoxyamphetamine The risk or severity of hypertension can be increased when Balsalazide is combined with 4-Bromo-2,5-dimethoxyamphetamine.
Tenamfetamine The risk or severity of hypertension can be increased when Balsalazide is combined with Tenamfetamine.
Chlorphentermine The risk or severity of hypertension can be increased when Balsalazide is combined with Chlorphentermine.
Dextroamphetamine The risk or severity of hypertension can be increased when Balsalazide is combined with Dextroamphetamine.
Phendimetrazine The risk or severity of hypertension can be increased when Balsalazide is combined with Phendimetrazine.
Solifenacin The risk or severity of hypertension can be increased when Balsalazide is combined with Solifenacin.
Periciazine The risk or severity of hypertension can be increased when Balsalazide is combined with Periciazine.
Acepromazine The risk or severity of hypertension can be increased when Balsalazide is combined with Acepromazine.
Thioproperazine The risk or severity of hypertension can be increased when Balsalazide is combined with Thioproperazine.
Zuclopenthixol The risk or severity of hypertension can be increased when Balsalazide is combined with Zuclopenthixol.
Epicaptopril The risk or severity of hypertension can be increased when Balsalazide is combined with Epicaptopril.
Clorgiline The risk or severity of hypertension can be increased when Balsalazide is combined with Clorgiline.
1-benzylimidazole The risk or severity of hypertension can be increased when Balsalazide is combined with 1-benzylimidazole.
Iproniazid The risk or severity of hypertension can be increased when Balsalazide is combined with Iproniazid.
Nialamide The risk or severity of hypertension can be increased when Balsalazide is combined with Nialamide.
Lysergic acid diethylamide The risk or severity of hypertension can be increased when Balsalazide is combined with Lysergic acid diethylamide.
Dronedarone The risk or severity of hypertension can be increased when Balsalazide is combined with Dronedarone.
Flibanserin The risk or severity of hypertension can be increased when Balsalazide is combined with Flibanserin.
Iloperidone The risk or severity of hypertension can be increased when Balsalazide is combined with Iloperidone.
Indacaterol The risk or severity of hypertension can be increased when Balsalazide is combined with Indacaterol.

Target Protein

Peroxisome proliferator-activated receptor gamma PPARG
Prostaglandin G/H synthase 2 PTGS2
Prostaglandin G/H synthase 1 PTGS1
Polyunsaturated fatty acid 5-lipoxygenase ALOX5

Referensi & Sumber

Synthesis reference: Eckardt C. G. Wolf, Nageib Mohamed, Bhaskar Reddy Guntoori, "Safe process for the preparation of balsalazide." U.S. Patent US07271253, issued September 18, 2007.
Artikel (PubMed)
  • PMID: 19743890
    Wiggins JB, Rajapakse R: Balsalazide: a novel 5-aminosalicylate prodrug for the treatment of active ulcerative colitis. Expert Opin Drug Metab Toxicol. 2009 Oct;5(10):1279-84. doi: 10.1517/17425250903206996.
  • PMID: 11563993
    Ragunath K, Williams JG: Review article: balsalazide therapy in ulcerative colitis. Aliment Pharmacol Ther. 2001 Oct;15(10):1549-54.

Contoh Produk & Brand

Produk: 22 • International brands: 1
Produk
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
  • Balsalazide Disodium
    Capsule • 750 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 22 produk.
International Brands
  • Colazide

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