Peringatan Keamanan

LD50=5000 mg/kg (Orally in rats)

Felbamate

DB00949

small molecule approved

Deskripsi

Felbamate is an anticonvulsant drug used in the treatment of epilepsy. In particular, in the adult patient population, it can be employed to treat partial seizures (with and without generalization). Alternatively, it is used to treat partial and generalized seizures associated with Lennox-Gastaut syndrome in children. It has a weak inhibitory effect on GABA receptor binding sites.

Struktur Molekul 2D

Berat 238.2399
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 20-23 hours
Volume Distribusi * 756±82 mL/kg
Klirens (Clearance) * 26 +/- 3 mL/hr/kg [single 1200 mg dose] * 30 +/- 8 mL/hr/kg [multiple daily doses of 3600 mg]

Absorpsi

>90%

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Avoid alcohol.

Interaksi Obat

1370 Data
Aripiprazole The metabolism of Aripiprazole can be increased when combined with Felbamate.
Aripiprazole lauroxil The metabolism of Aripiprazole lauroxil can be increased when combined with Felbamate.
Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Felbamate.
Buprenorphine Felbamate may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Felbamate.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Felbamate.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Felbamate.
Hydrocodone Felbamate may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Magnesium sulfate The therapeutic efficacy of Felbamate can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Felbamate may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Felbamate may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Felbamate.
Mirtazapine Felbamate may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Felbamate.
Orphenadrine Felbamate may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Felbamate may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Pramipexole Felbamate may increase the sedative activities of Pramipexole.
Ropinirole Felbamate may increase the sedative activities of Ropinirole.
Rotigotine Felbamate may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Felbamate.
Sodium oxybate Felbamate may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Felbamate may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Felbamate.
Thalidomide Felbamate may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Felbamate may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Mefloquine The therapeutic efficacy of Felbamate can be decreased when used in combination with Mefloquine.
Mianserin The therapeutic efficacy of Felbamate can be decreased when used in combination with Mianserin.
Orlistat Orlistat can cause a decrease in the absorption of Felbamate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Butalbital The serum concentration of Butalbital can be increased when it is combined with Felbamate.
Pentobarbital The serum concentration of Pentobarbital can be increased when it is combined with Felbamate.
Secobarbital The serum concentration of Secobarbital can be increased when it is combined with Felbamate.
Methohexital The serum concentration of Methohexital can be increased when it is combined with Felbamate.
Thiopental The serum concentration of Thiopental can be increased when it is combined with Felbamate.
Thiamylal The serum concentration of Thiamylal can be increased when it is combined with Felbamate.
Amobarbital The serum concentration of Amobarbital can be increased when it is combined with Felbamate.
Hexobarbital The serum concentration of Hexobarbital can be increased when it is combined with Felbamate.
Barbital The serum concentration of Barbital can be increased when it is combined with Felbamate.
Barbexaclone The serum concentration of Barbexaclone can be increased when it is combined with Felbamate.
Butabarbital The serum concentration of Butabarbital can be increased when it is combined with Felbamate.
Phenytoin The serum concentration of Phenytoin can be increased when it is combined with Felbamate.
Fosphenytoin The serum concentration of Fosphenytoin can be increased when it is combined with Felbamate.
Topotecan Felbamate may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Valproic acid The serum concentration of Valproic acid can be increased when it is combined with Felbamate.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Felbamate.
Memantine The risk or severity of adverse effects can be increased when Felbamate is combined with Memantine.
Carbamazepine The serum concentration of Felbamate can be decreased when it is combined with Carbamazepine.
Ifosfamide The metabolism of Ifosfamide can be increased when combined with Felbamate.
Perampanel The metabolism of Perampanel can be increased when combined with Felbamate.
Warfarin The metabolism of Warfarin can be increased when combined with Felbamate.
Acenocoumarol The metabolism of Acenocoumarol can be increased when combined with Felbamate.
(R)-warfarin The metabolism of (R)-warfarin can be increased when combined with Felbamate.
R,S-Warfarin alcohol The metabolism of R,S-Warfarin alcohol can be increased when combined with Felbamate.
S,R-Warfarin alcohol The metabolism of S,R-Warfarin alcohol can be increased when combined with Felbamate.
(S)-Warfarin The metabolism of (S)-Warfarin can be increased when combined with Felbamate.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Felbamate.
Primidone The serum concentration of Phenobarbital, an active metabolite of Primidone, can be increased when used in combination with Felbamate.
Methylphenobarbital The serum concentration of Phenobarbital, an active metabolite of Methylphenobarbital, can be increased when used in combination with Felbamate.
Phenobarbital The serum concentration of Phenobarbital, an active metabolite of Phenobarbital, can be increased when used in combination with Felbamate.
Ethanol Felbamate may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Felbamate may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Felbamate.
Fluvoxamine The risk or severity of adverse effects can be increased when Felbamate is combined with Fluvoxamine.
Duloxetine The risk or severity of adverse effects can be increased when Felbamate is combined with Duloxetine.
Paroxetine The risk or severity of adverse effects can be increased when Felbamate is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Felbamate is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Felbamate is combined with Sibutramine.
Zimelidine The risk or severity of adverse effects can be increased when Felbamate is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Felbamate is combined with Dapoxetine.
Desvenlafaxine The risk or severity of adverse effects can be increased when Felbamate is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Felbamate is combined with Seproxetine.
Indalpine The risk or severity of adverse effects can be increased when Felbamate is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Felbamate is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Felbamate is combined with Alaproclate.
Escitalopram The risk or severity of adverse effects can be increased when Felbamate is combined with Escitalopram.
Erlotinib The serum concentration of Erlotinib can be decreased when it is combined with Felbamate.
Benzatropine The risk or severity of QTc prolongation can be increased when Benzatropine is combined with Felbamate.
Buclizine The risk or severity of QTc prolongation can be increased when Buclizine is combined with Felbamate.
Hyoscyamine The risk or severity of QTc prolongation can be increased when Hyoscyamine is combined with Felbamate.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Felbamate.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Felbamate.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Felbamate.
Maprotiline The risk or severity of CNS depression can be increased when Maprotiline is combined with Felbamate.
Desipramine The risk or severity of CNS depression can be increased when Felbamate is combined with Desipramine.
Solifenacin The risk or severity of QTc prolongation can be increased when Felbamate is combined with Solifenacin.
Pizotifen The risk or severity of CNS depression can be increased when Felbamate is combined with Pizotifen.
Trimebutine The risk or severity of QTc prolongation can be increased when Felbamate is combined with Trimebutine.
Dosulepin The risk or severity of CNS depression can be increased when Felbamate is combined with Dosulepin.
Nicardipine The metabolism of Felbamate can be decreased when combined with Nicardipine.
Clozapine The risk or severity of QTc prolongation can be increased when Felbamate is combined with Clozapine.
Zopiclone The risk or severity of adverse effects can be increased when Felbamate is combined with Zopiclone.
Leuprolide The risk or severity of QTc prolongation can be increased when Felbamate is combined with Leuprolide.
Goserelin The risk or severity of QTc prolongation can be increased when Felbamate is combined with Goserelin.
Erythromycin The serum concentration of Felbamate can be increased when it is combined with Erythromycin.
Azithromycin The metabolism of Azithromycin can be increased when combined with Felbamate.
Moxifloxacin The risk or severity of QTc prolongation can be increased when Felbamate is combined with Moxifloxacin.
Sulfisoxazole The risk or severity of QTc prolongation can be increased when Felbamate is combined with Sulfisoxazole.
Diltiazem The metabolism of Felbamate can be decreased when combined with Diltiazem.
Nimodipine The risk or severity of QTc prolongation can be increased when Felbamate is combined with Nimodipine.
Oxaliplatin The risk or severity of QTc prolongation can be increased when Oxaliplatin is combined with Felbamate.
Ciprofloxacin The metabolism of Felbamate can be decreased when combined with Ciprofloxacin.

Target Protein

Glutamate receptor ionotropic, NMDA 2B GRIN2B
Glutamate receptor ionotropic, NMDA 2A GRIN2A

Referensi & Sumber

Artikel (PubMed)
  • PMID: 1944909
    Leppik IE, Dreifuss FE, Pledger GW, Graves NM, Santilli N, Drury I, Tsay JY, Jacobs MP, Bertram E, Cereghino JJ, et al.: Felbamate for partial seizures: results of a controlled clinical trial. Neurology. 1991 Nov;41(11):1785-9.

Contoh Produk & Brand

Produk: 43 • International brands: 2
Produk
  • Felbamate
    Tablet • 400 mg/1 • Oral • US • Generic • Approved
  • Felbamate
    Tablet • 600 mg/1 • Oral • US • Generic • Approved
  • Felbamate
    Tablet • 400 mg/1 • Oral • US • Generic • Approved
  • Felbamate
    Tablet • 600 mg/1 • Oral • US • Generic • Approved
  • Felbamate
    Tablet • 600 mg/1 • Oral • US • Generic • Approved
  • Felbamate
    Tablet • 400 mg/1 • Oral • US • Generic • Approved
  • Felbamate
    Tablet • 600 mg/1 • Oral • US • Generic • Approved
  • Felbamate
    Suspension • 600 mg/5mL • Oral • US • Generic • Approved
Menampilkan 8 dari 43 produk.
International Brands
  • Felbamyl
  • Taloxa

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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