Peringatan Keamanan

50=500 mg/kg. Symptoms of overdose includes suspected or overt abnormal bleeding (e.g., appearance of blood in stools or urine, hematuria, excessive menstrual bleeding, melena, petechiae, excessive bruising or persistent oozing from superficial injuries).

Phenprocoumon

DB00946

small molecule approved investigational

Deskripsi

Coumarin derivative that acts as a long-acting oral anticoagulant.

Struktur Molekul 2D

Berat 280.3178
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 5-6 days
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Bioavailability is close to 100%

Metabolisme

Phenprocoumon is stereoselectively metabolized by hepatic microsomal enzymes (cytochrome P-450) to inactive hydroxylated metabolites (predominant route) and by reductases to reduced metabolites. Cytochrome P450 2C9 is the principal form of human liver P-450 responsible for metabolism.

Rute Eliminasi

Data eliminasi belum tersedia.

Farmakogenomik

3 Varian
CYP2C9 (rs1799853)

The presence of this polymorphism in CYP2C9 is associated with reduction in phenprocoumon metabolism.

CYP2C9 (rs1057910)

The presence of this polymorphism in CYP2C9 is associated with reduction in phenprocoumon metabolism.

VKORC1 (rs9934438)

The presence of this polymorphism in VKORC1 is associated with reduction in phenprocoumon metabolism.

Interaksi Makanan

4 Data
  • 1. Avoid herbs and supplements with anticoagulant/antiplatelet activity. Examples include garlic, ginger, bilberry, danshen, piracetam, and ginkgo biloba.
  • 2. Ensure consistent Vitamin K intake. Changes in vitamin K intake may impact coagulation.
  • 3. Exercise caution with grapefruit products.
  • 4. Exercise caution with St. John's Wort.

Interaksi Obat

1659 Data
Apixaban Apixaban may increase the anticoagulant activities of Phenprocoumon.
Dabigatran etexilate Dabigatran etexilate may increase the anticoagulant activities of Phenprocoumon.
Dasatinib The risk or severity of bleeding and hemorrhage can be increased when Dasatinib is combined with Phenprocoumon.
Deferasirox The risk or severity of gastrointestinal bleeding can be increased when Phenprocoumon is combined with Deferasirox.
Ursodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Ursodeoxycholic acid.
Glycochenodeoxycholic Acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Glycochenodeoxycholic Acid.
Cholic Acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Cholic Acid.
Glycocholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Glycocholic acid.
Deoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Deoxycholic acid.
Taurocholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Taurocholic acid.
Obeticholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Obeticholic acid.
Chenodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Chenodeoxycholic acid.
Taurochenodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Taurochenodeoxycholic acid.
Tauroursodeoxycholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Tauroursodeoxycholic acid.
Bamet-UD2 The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Bamet-UD2.
Dehydrocholic acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Dehydrocholic acid.
Hyodeoxycholic Acid The risk or severity of bleeding and bruising can be increased when Phenprocoumon is combined with Hyodeoxycholic Acid.
Edoxaban The risk or severity of bleeding can be increased when Edoxaban is combined with Phenprocoumon.
Ibrutinib The risk or severity of bleeding and hemorrhage can be increased when Ibrutinib is combined with Phenprocoumon.
Obinutuzumab The risk or severity of bleeding and hemorrhage can be increased when Phenprocoumon is combined with Obinutuzumab.
Rivaroxaban Phenprocoumon may increase the anticoagulant activities of Rivaroxaban.
Sugammadex The risk or severity of bleeding and hemorrhage can be increased when Phenprocoumon is combined with Sugammadex.
Tibolone Tibolone may increase the anticoagulant activities of Phenprocoumon.
Tipranavir The risk or severity of bleeding and hemorrhage can be increased when Tipranavir is combined with Phenprocoumon.
Urokinase Urokinase may increase the anticoagulant activities of Phenprocoumon.
Vitamin E Vitamin E may increase the anticoagulant activities of Phenprocoumon.
Vorapaxar The risk or severity of bleeding and hemorrhage can be increased when Vorapaxar is combined with Phenprocoumon.
Modafinil The metabolism of Phenprocoumon can be increased when combined with Modafinil.
Armodafinil The metabolism of Phenprocoumon can be increased when combined with Armodafinil.
Metreleptin The metabolism of Phenprocoumon can be increased when combined with Metreleptin.
Mifepristone The serum concentration of Phenprocoumon can be increased when it is combined with Mifepristone.
Gemcitabine The therapeutic efficacy of Phenprocoumon can be increased when used in combination with Gemcitabine.
Flunisolide Flunisolide may increase the anticoagulant activities of Phenprocoumon.
Beclomethasone dipropionate Beclomethasone dipropionate may increase the anticoagulant activities of Phenprocoumon.
Betamethasone Betamethasone may increase the anticoagulant activities of Phenprocoumon.
Fluticasone propionate Fluticasone propionate may increase the anticoagulant activities of Phenprocoumon.
Fluocinolone acetonide Fluocinolone acetonide may increase the anticoagulant activities of Phenprocoumon.
Prednisone Prednisone may increase the anticoagulant activities of Phenprocoumon.
Fludrocortisone Fludrocortisone may increase the anticoagulant activities of Phenprocoumon.
Hydrocortisone Hydrocortisone may increase the anticoagulant activities of Phenprocoumon.
Prednisolone Prednisolone may increase the anticoagulant activities of Phenprocoumon.
Methylprednisolone Methylprednisolone may increase the anticoagulant activities of Phenprocoumon.
Trilostane Trilostane may increase the anticoagulant activities of Phenprocoumon.
Budesonide Budesonide may increase the anticoagulant activities of Phenprocoumon.
Dexamethasone Dexamethasone may increase the anticoagulant activities of Phenprocoumon.
Corticotropin Corticotropin may increase the anticoagulant activities of Phenprocoumon.
Cortisone acetate Cortisone acetate may increase the anticoagulant activities of Phenprocoumon.
Paramethasone Paramethasone may increase the anticoagulant activities of Phenprocoumon.
Ciclesonide Ciclesonide may increase the anticoagulant activities of Phenprocoumon.
Aldosterone Aldosterone may increase the anticoagulant activities of Phenprocoumon.
Fluticasone furoate Fluticasone furoate may increase the anticoagulant activities of Phenprocoumon.
Fluprednidene Fluprednidene may increase the anticoagulant activities of Phenprocoumon.
Tixocortol Tixocortol may increase the anticoagulant activities of Phenprocoumon.
Fluprednisolone Fluprednisolone may increase the anticoagulant activities of Phenprocoumon.
Meprednisone Meprednisone may increase the anticoagulant activities of Phenprocoumon.
Dexamethasone isonicotinate Dexamethasone isonicotinate may increase the anticoagulant activities of Phenprocoumon.
Melengestrol Melengestrol may increase the anticoagulant activities of Phenprocoumon.
Deflazacort Deflazacort may increase the anticoagulant activities of Phenprocoumon.
Cortivazol Cortivazol may increase the anticoagulant activities of Phenprocoumon.
Prednylidene Prednylidene may increase the anticoagulant activities of Phenprocoumon.
Fluocortin Fluocortin may increase the anticoagulant activities of Phenprocoumon.
Fluperolone Fluperolone may increase the anticoagulant activities of Phenprocoumon.
Cloprednol Cloprednol may increase the anticoagulant activities of Phenprocoumon.
Fluclorolone Fluclorolone may increase the anticoagulant activities of Phenprocoumon.
Fluticasone Fluticasone may increase the anticoagulant activities of Phenprocoumon.
Mometasone furoate Mometasone furoate may increase the anticoagulant activities of Phenprocoumon.
Hydrocortisone acetate Hydrocortisone acetate may increase the anticoagulant activities of Phenprocoumon.
Hydrocortisone cypionate Hydrocortisone cypionate may increase the anticoagulant activities of Phenprocoumon.
Hydrocortisone succinate Hydrocortisone succinate may increase the anticoagulant activities of Phenprocoumon.
Prednisolone phosphate Prednisolone phosphate may increase the anticoagulant activities of Phenprocoumon.
Prednisolone hemisuccinate Prednisolone hemisuccinate may increase the anticoagulant activities of Phenprocoumon.
Methylprednisolone hemisuccinate Methylprednisolone hemisuccinate may increase the anticoagulant activities of Phenprocoumon.
Prednisone acetate Prednisone acetate may increase the anticoagulant activities of Phenprocoumon.
Clocortolone acetate Clocortolone acetate may increase the anticoagulant activities of Phenprocoumon.
Melengestrol acetate Melengestrol acetate may increase the anticoagulant activities of Phenprocoumon.
Betamethasone phosphate Betamethasone phosphate may increase the anticoagulant activities of Phenprocoumon.
Cortisone Cortisone may increase the anticoagulant activities of Phenprocoumon.
Clobetasol propionate Clobetasol propionate may increase the anticoagulant activities of Phenprocoumon.
Fluocinonide Fluocinonide may increase the anticoagulant activities of Phenprocoumon.
Hydrocortisone butyrate Hydrocortisone butyrate may increase the anticoagulant activities of Phenprocoumon.
Desoximetasone Desoximetasone may increase the anticoagulant activities of Phenprocoumon.
Mometasone Mometasone may increase the anticoagulant activities of Phenprocoumon.
Fluocortolone Fluocortolone may increase the anticoagulant activities of Phenprocoumon.
Prednisolone acetate Prednisolone acetate may increase the anticoagulant activities of Phenprocoumon.
Fluorometholone Fluorometholone may increase the anticoagulant activities of Phenprocoumon.
Difluocortolone Difluocortolone may increase the anticoagulant activities of Phenprocoumon.
Flumethasone Flumethasone may increase the anticoagulant activities of Phenprocoumon.
Methylprednisolone aceponate Methylprednisolone aceponate may increase the anticoagulant activities of Phenprocoumon.
Erlotinib The serum concentration of Phenprocoumon can be increased when it is combined with Erlotinib.
Allopurinol The risk or severity of bleeding can be increased when Allopurinol is combined with Phenprocoumon.
Azathioprine The therapeutic efficacy of Phenprocoumon can be decreased when used in combination with Azathioprine.
Chloral hydrate The protein binding of Phenprocoumon can be decreased when combined with Chloral hydrate.
Methylphenidate The metabolism of Phenprocoumon can be decreased when combined with Methylphenidate.
Disulfiram Disulfiram may increase the anticoagulant activities of Phenprocoumon.
Etacrynic acid The protein binding of Phenprocoumon can be decreased when combined with Etacrynic acid.
Ethotoin The therapeutic efficacy of Phenprocoumon can be increased when used in combination with Ethotoin.
Etoposide The therapeutic efficacy of Phenprocoumon can be increased when used in combination with Etoposide.
Exenatide Exenatide can cause an increase in the absorption of Phenprocoumon resulting in an increased serum concentration and potentially a worsening of adverse effects.
Gefitinib Gefitinib may increase the anticoagulant activities of Phenprocoumon.
Ginkgo biloba Ginkgo biloba may increase the anticoagulant activities of Phenprocoumon.

Target Protein

Vitamin K epoxide reductase complex subunit 1 VKORC1

Referensi & Sumber

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Contoh Produk & Brand

Produk: 0 • International brands: 4
International Brands
  • Falithrom
  • Liquamar
  • Marcoumar
  • Marcumar

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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