Peringatan Keamanan

Symptoms of overdose: blurred vision (continuing) or changes in near vision, clumsiness or unsteadiness, confusion, convulsions, difficulty in breathing, muscle weakness (severe), or tiredness (severe), dizziness, drowsiness (severe), dryness of mouth, nose, or throat (severe), fast heartbeat, fever, hallucinations, slurred speech, unusual excitement, nervousness, restlessness, or irritability, unusual warmth, dryness, and flushing of skin.

Methantheline

DB00940

small molecule approved investigational

Deskripsi

Methantheline is a synthetic antispasmodic. Antispasmodics are used to relieve cramps or spasms of the stomach, intestines, and bladder. Methantheline is used to treat intestine or stomach ulcers (peptic ulcer disease), intestine problems (irritable bowel syndrome), pancreatitis, gastritis, biliary dyskinesia, pylorosplasm, or urinary problems (reflex neurogenic bladder in children).

Struktur Molekul 2D

Berat 340.436
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed.

Metabolisme

Hepatic, by enzymatic hydrolysis.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

608 Data
Aclidinium The risk or severity of adverse effects can be increased when Methantheline is combined with Aclidinium.
Mianserin Mianserin may increase the anticholinergic activities of Methantheline.
Mirabegron The risk or severity of urinary retention can be increased when Methantheline is combined with Mirabegron.
Pramlintide The risk or severity of reduced gastrointestinal motility can be increased when Pramlintide is combined with Methantheline.
Secretin porcine The therapeutic efficacy of Secretin porcine can be decreased when used in combination with Methantheline.
Tiotropium The risk or severity of adverse effects can be increased when Methantheline is combined with Tiotropium.
Topiramate The risk or severity of hyperthermia and oligohydrosis can be increased when Methantheline is combined with Topiramate.
Umeclidinium The risk or severity of adverse effects can be increased when Methantheline is combined with Umeclidinium.
Atazanavir Methantheline can cause a decrease in the absorption of Atazanavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefditoren The serum concentration of Cefditoren can be decreased when it is combined with Methantheline.
Dabigatran etexilate Methantheline can cause a decrease in the absorption of Dabigatran etexilate resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dabrafenib Methantheline can cause a decrease in the absorption of Dabrafenib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Erlotinib Methantheline can cause a decrease in the absorption of Erlotinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Pazopanib Methantheline can cause a decrease in the absorption of Pazopanib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Riociguat Methantheline can cause a decrease in the absorption of Riociguat resulting in a reduced serum concentration and potentially a decrease in efficacy.
Benzylpenicilloyl polylysine Methantheline may decrease effectiveness of Benzylpenicilloyl polylysine as a diagnostic agent.
Betahistine The therapeutic efficacy of Betahistine can be decreased when used in combination with Methantheline.
Hyaluronidase (ovine) The therapeutic efficacy of Hyaluronidase (ovine) can be decreased when used in combination with Methantheline.
Hyaluronidase (human recombinant) The therapeutic efficacy of Hyaluronidase (human recombinant) can be decreased when used in combination with Methantheline.
Hyaluronidase The therapeutic efficacy of Hyaluronidase can be decreased when used in combination with Methantheline.
Bosutinib Methantheline can cause a decrease in the absorption of Bosutinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefpodoxime Methantheline can cause a decrease in the absorption of Cefpodoxime resulting in a reduced serum concentration and potentially a decrease in efficacy.
Cefuroxime Methantheline can cause a decrease in the absorption of Cefuroxime resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dasatinib Methantheline can cause a decrease in the absorption of Dasatinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Delavirdine Methantheline can cause a decrease in the absorption of Delavirdine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Dexmethylphenidate The therapeutic efficacy of Dexmethylphenidate can be decreased when used in combination with Methantheline.
Amprenavir Methantheline can cause a decrease in the absorption of Amprenavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Fosamprenavir Methantheline can cause a decrease in the absorption of Fosamprenavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Gefitinib Methantheline can cause a decrease in the absorption of Gefitinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Indinavir Methantheline can cause a decrease in the absorption of Indinavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Itraconazole Methantheline can cause a decrease in the absorption of Itraconazole resulting in a reduced serum concentration and potentially a decrease in efficacy.
Ledipasvir Methantheline can cause a decrease in the absorption of Ledipasvir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Methylphenidate The therapeutic efficacy of Methylphenidate can be decreased when used in combination with Methantheline.
Nelfinavir Methantheline can cause a decrease in the absorption of Nelfinavir resulting in a reduced serum concentration and potentially a decrease in efficacy.
Nilotinib Methantheline can cause a decrease in the absorption of Nilotinib resulting in a reduced serum concentration and potentially a decrease in efficacy.
Rilpivirine Methantheline can cause a decrease in the absorption of Rilpivirine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Risedronic acid Methantheline can cause an increase in the absorption of Risedronic acid resulting in an increased serum concentration and potentially a worsening of adverse effects.
Saquinavir Methantheline can cause an increase in the absorption of Saquinavir resulting in an increased serum concentration and potentially a worsening of adverse effects.
Glycopyrronium The risk or severity of adverse effects can be increased when Methantheline is combined with Glycopyrronium.
Levothyroxine Methantheline can cause a decrease in the absorption of Levothyroxine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Bisacodyl The therapeutic efficacy of Bisacodyl can be decreased when used in combination with Methantheline.
Captopril Methantheline can cause a decrease in the absorption of Captopril resulting in a reduced serum concentration and potentially a decrease in efficacy.
Rifampin Methantheline can cause a decrease in the absorption of Rifampicin resulting in a reduced serum concentration and potentially a decrease in efficacy.
Memantine Methantheline may decrease the excretion rate of Memantine which could result in a higher serum level.
Botulinum toxin type A The risk or severity of adverse effects can be increased when Methantheline is combined with Botulinum toxin type A.
Glucagon Methantheline may increase the gastrointestinal motility reducing activities of Glucagon.
Sulpiride The therapeutic efficacy of Sulpiride can be increased when used in combination with Methantheline.
Botulinum toxin type B The risk or severity of adverse effects can be increased when Methantheline is combined with Botulinum toxin type B.
Mesalazine Methantheline can cause a decrease in the absorption of Mesalazine resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mycophenolate mofetil Methantheline can cause a decrease in the absorption of Mycophenolate mofetil resulting in a reduced serum concentration and potentially a decrease in efficacy.
Mycophenolic acid Methantheline can cause a decrease in the absorption of Mycophenolic acid resulting in a reduced serum concentration and potentially a decrease in efficacy.
Tolevamer The therapeutic efficacy of Tolevamer can be decreased when used in combination with Methantheline.
Eluxadoline The risk or severity of constipation can be increased when Methantheline is combined with Eluxadoline.
Ramosetron The risk or severity of constipation can be increased when Methantheline is combined with Ramosetron.
Amphetamine Amphetamine may decrease the sedative activities of Methantheline.
Phentermine Phentermine may decrease the sedative activities of Methantheline.
Pseudoephedrine Pseudoephedrine may decrease the sedative activities of Methantheline.
Benzphetamine Benzphetamine may decrease the sedative activities of Methantheline.
Diethylpropion Diethylpropion may decrease the sedative activities of Methantheline.
Lisdexamfetamine Lisdexamfetamine may decrease the sedative activities of Methantheline.
Mephentermine Mephentermine may decrease the sedative activities of Methantheline.
MMDA MMDA may decrease the sedative activities of Methantheline.
Midomafetamine Midomafetamine may decrease the sedative activities of Methantheline.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the sedative activities of Methantheline.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the sedative activities of Methantheline.
Tenamfetamine Tenamfetamine may decrease the sedative activities of Methantheline.
Chlorphentermine Chlorphentermine may decrease the sedative activities of Methantheline.
Methylenedioxyethamphetamine Methylenedioxyethamphetamine may decrease the sedative activities of Methantheline.
Dextroamphetamine Dextroamphetamine may decrease the sedative activities of Methantheline.
Metamfetamine Metamfetamine may decrease the sedative activities of Methantheline.
Iofetamine I-123 Iofetamine I-123 may decrease the sedative activities of Methantheline.
Ritobegron Ritobegron may decrease the sedative activities of Methantheline.
Mephedrone Mephedrone may decrease the sedative activities of Methantheline.
Methoxyphenamine Methoxyphenamine may decrease the sedative activities of Methantheline.
Gepefrine Gepefrine may decrease the sedative activities of Methantheline.
2,5-Dimethoxy-4-ethylthioamphetamine 2,5-Dimethoxy-4-ethylthioamphetamine may decrease the sedative activities of Methantheline.
Phendimetrazine Phendimetrazine may decrease the sedative activities of Methantheline.
Naltrexone The risk or severity of adverse effects can be increased when Methantheline is combined with Naltrexone.
Bezitramide The risk or severity of adverse effects can be increased when Methantheline is combined with Bezitramide.
Tramadol The risk or severity of adverse effects can be increased when Methantheline is combined with Tramadol.
Morphine The risk or severity of adverse effects can be increased when Methantheline is combined with Morphine.
Codeine The risk or severity of adverse effects can be increased when Methantheline is combined with Codeine.
Hydromorphone The risk or severity of adverse effects can be increased when Methantheline is combined with Hydromorphone.
Methadone The risk or severity of adverse effects can be increased when Methantheline is combined with Methadone.
Meperidine The risk or severity of adverse effects can be increased when Methantheline is combined with Meperidine.
Oxycodone The risk or severity of adverse effects can be increased when Methantheline is combined with Oxycodone.
Butorphanol The risk or severity of adverse effects can be increased when Methantheline is combined with Butorphanol.
Dextropropoxyphene The risk or severity of adverse effects can be increased when Methantheline is combined with Dextropropoxyphene.
Pentazocine The risk or severity of adverse effects can be increased when Methantheline is combined with Pentazocine.
Sufentanil The risk or severity of adverse effects can be increased when Methantheline is combined with Sufentanil.
Alfentanil The risk or severity of adverse effects can be increased when Methantheline is combined with Alfentanil.
Fentanyl The risk or severity of adverse effects can be increased when Methantheline is combined with Fentanyl.
Nalbuphine The risk or severity of adverse effects can be increased when Methantheline is combined with Nalbuphine.
Levorphanol The risk or severity of adverse effects can be increased when Methantheline is combined with Levorphanol.
Remifentanil The risk or severity of adverse effects can be increased when Methantheline is combined with Remifentanil.
Buprenorphine The risk or severity of adverse effects can be increased when Methantheline is combined with Buprenorphine.
Hydrocodone The risk or severity of adverse effects can be increased when Methantheline is combined with Hydrocodone.
Diphenoxylate The risk or severity of adverse effects can be increased when Methantheline is combined with Diphenoxylate.
Oxymorphone The risk or severity of adverse effects can be increased when Methantheline is combined with Oxymorphone.
Dezocine The risk or severity of adverse effects can be increased when Methantheline is combined with Dezocine.

Target Protein

Histamine H2 receptor HRH2
Muscarinic acetylcholine receptor M5 CHRM5
Muscarinic acetylcholine receptor M2 CHRM2
Muscarinic acetylcholine receptor M3 CHRM3
Muscarinic acetylcholine receptor M4 CHRM4
Muscarinic acetylcholine receptor M1 CHRM1

Referensi & Sumber

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Contoh Produk & Brand

Produk: 0 • International brands: 2
International Brands
  • Banthine
  • Vagantin

Sekuens Gen/Protein (FASTA)

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