Phenformin

DB00914

small molecule approved investigational withdrawn

Deskripsi

A biguanide hypoglycemic agent with actions and uses similar to those of metformin. Although it is generally considered to be associated with an unacceptably high incidence of lactic acidosis, often fatal, it is still available in some countries. (From Martindale, The Extra Pharmacopoeia, 30th ed, p290)

Struktur Molekul 2D

Berat 205.2596
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

895 Data
Pegvisomant The risk or severity of hypoglycemia can be increased when Pegvisomant is combined with Phenformin.
Mirabegron The serum concentration of Phenformin can be increased when it is combined with Mirabegron.
Lipoic acid The risk or severity of hypoglycemia can be increased when Lipoic acid is combined with Phenformin.
Moxifloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Moxifloxacin.
Grepafloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Grepafloxacin.
Enoxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Enoxacin.
Pefloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Pefloxacin.
Ciprofloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Ciprofloxacin.
Trovafloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Trovafloxacin.
Nalidixic acid The therapeutic efficacy of Phenformin can be increased when used in combination with Nalidixic acid.
Rosoxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Rosoxacin.
Cinoxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Cinoxacin.
Lomefloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Lomefloxacin.
Gatifloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Gatifloxacin.
Norfloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Norfloxacin.
Levofloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Levofloxacin.
Gemifloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Gemifloxacin.
Ofloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Ofloxacin.
Sparfloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Sparfloxacin.
Temafloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Temafloxacin.
Fleroxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Fleroxacin.
Technetium Tc-99m ciprofloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Technetium Tc-99m ciprofloxacin.
Garenoxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Garenoxacin.
Nemonoxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Nemonoxacin.
Flumequine The therapeutic efficacy of Phenformin can be increased when used in combination with Flumequine.
Enrofloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Enrofloxacin.
Orbifloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Orbifloxacin.
Sarafloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Sarafloxacin.
Difloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Difloxacin.
Pazufloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Pazufloxacin.
Prulifloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Prulifloxacin.
Delafloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Delafloxacin.
Sitafloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Sitafloxacin.
Oxolinic acid The therapeutic efficacy of Phenformin can be increased when used in combination with Oxolinic acid.
Rufloxacin The therapeutic efficacy of Phenformin can be increased when used in combination with Rufloxacin.
Pipemidic acid The therapeutic efficacy of Phenformin can be increased when used in combination with Pipemidic acid.
Methyclothiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Methyclothiazide.
Chlorthalidone The therapeutic efficacy of Phenformin can be decreased when used in combination with Chlorthalidone.
Bendroflumethiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Bendroflumethiazide.
Metolazone The therapeutic efficacy of Phenformin can be decreased when used in combination with Metolazone.
Benzthiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Benzthiazide.
Hydroflumethiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Hydroflumethiazide.
Indapamide The therapeutic efficacy of Phenformin can be decreased when used in combination with Indapamide.
Chlorothiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Chlorothiazide.
Hydrochlorothiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Hydrochlorothiazide.
Trichlormethiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Trichlormethiazide.
Polythiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Polythiazide.
Quinethazone The therapeutic efficacy of Phenformin can be decreased when used in combination with Quinethazone.
Cyclopenthiazide The therapeutic efficacy of Phenformin can be decreased when used in combination with Cyclopenthiazide.
Epitizide The therapeutic efficacy of Phenformin can be decreased when used in combination with Epitizide.
Amineptine Amineptine may decrease the hypoglycemic activities of Phenformin.
Dimetacrine Dimetacrine may decrease the hypoglycemic activities of Phenformin.
Butriptyline Butriptyline may decrease the hypoglycemic activities of Phenformin.
Tianeptine Tianeptine may decrease the hypoglycemic activities of Phenformin.
Oxaprotiline Oxaprotiline may decrease the hypoglycemic activities of Phenformin.
Amitriptylinoxide Amitriptylinoxide may decrease the hypoglycemic activities of Phenformin.
Dibenzepin Dibenzepin may decrease the hypoglycemic activities of Phenformin.
Quinupramine Quinupramine may decrease the hypoglycemic activities of Phenformin.
Melitracen Melitracen may decrease the hypoglycemic activities of Phenformin.
Lofepramine Lofepramine may decrease the hypoglycemic activities of Phenformin.
Iprindole Iprindole may decrease the hypoglycemic activities of Phenformin.
Imipramine oxide Imipramine oxide may decrease the hypoglycemic activities of Phenformin.
Protriptyline Protriptyline may decrease the hypoglycemic activities of Phenformin.
Opipramol Opipramol may decrease the hypoglycemic activities of Phenformin.
Doxepin Doxepin may decrease the hypoglycemic activities of Phenformin.
Dapagliflozin Dapagliflozin may increase the hypoglycemic activities of Phenformin.
Canagliflozin Canagliflozin may increase the hypoglycemic activities of Phenformin.
Leuprolide The therapeutic efficacy of Phenformin can be decreased when used in combination with Leuprolide.
Goserelin The therapeutic efficacy of Phenformin can be decreased when used in combination with Goserelin.
Indinavir The therapeutic efficacy of Phenformin can be decreased when used in combination with Indinavir.
Ziprasidone The therapeutic efficacy of Phenformin can be decreased when used in combination with Ziprasidone.
Etonogestrel The therapeutic efficacy of Phenformin can be decreased when used in combination with Etonogestrel.
Desogestrel The therapeutic efficacy of Phenformin can be decreased when used in combination with Desogestrel.
Olanzapine The therapeutic efficacy of Phenformin can be decreased when used in combination with Olanzapine.
Megestrol acetate The therapeutic efficacy of Phenformin can be decreased when used in combination with Megestrol acetate.
Levonorgestrel The therapeutic efficacy of Phenformin can be decreased when used in combination with Levonorgestrel.
Progesterone The therapeutic efficacy of Phenformin can be decreased when used in combination with Progesterone.
Piperazine The therapeutic efficacy of Phenformin can be decreased when used in combination with Piperazine.
Medroxyprogesterone acetate The therapeutic efficacy of Phenformin can be decreased when used in combination with Medroxyprogesterone acetate.
Niacin The therapeutic efficacy of Phenformin can be decreased when used in combination with Niacin.
Norethisterone The therapeutic efficacy of Phenformin can be decreased when used in combination with Norethisterone.
Risperidone The therapeutic efficacy of Phenformin can be decreased when used in combination with Risperidone.
Pentamidine The therapeutic efficacy of Phenformin can be decreased when used in combination with Pentamidine.
Ethynodiol diacetate The therapeutic efficacy of Phenformin can be decreased when used in combination with Ethynodiol diacetate.
Pseudoephedrine The therapeutic efficacy of Phenformin can be decreased when used in combination with Pseudoephedrine.
Tacrolimus The therapeutic efficacy of Phenformin can be decreased when used in combination with Tacrolimus.
Sirolimus The therapeutic efficacy of Phenformin can be decreased when used in combination with Sirolimus.
Etacrynic acid The therapeutic efficacy of Phenformin can be decreased when used in combination with Etacrynic acid.
Norgestimate The therapeutic efficacy of Phenformin can be decreased when used in combination with Norgestimate.
Ethinylestradiol The therapeutic efficacy of Phenformin can be decreased when used in combination with Ethinylestradiol.
Atazanavir The therapeutic efficacy of Phenformin can be decreased when used in combination with Atazanavir.
Arsenic trioxide The therapeutic efficacy of Phenformin can be decreased when used in combination with Arsenic trioxide.
Quetiapine The therapeutic efficacy of Phenformin can be decreased when used in combination with Quetiapine.
Saquinavir The therapeutic efficacy of Phenformin can be decreased when used in combination with Saquinavir.
Aripiprazole The therapeutic efficacy of Phenformin can be decreased when used in combination with Aripiprazole.
Paliperidone The therapeutic efficacy of Phenformin can be decreased when used in combination with Paliperidone.
Fosamprenavir The therapeutic efficacy of Phenformin can be decreased when used in combination with Fosamprenavir.
St. John's Wort The therapeutic efficacy of Phenformin can be decreased when used in combination with St. John's Wort.
Mestranol The therapeutic efficacy of Phenformin can be decreased when used in combination with Mestranol.
Ephedra sinica root The therapeutic efficacy of Phenformin can be decreased when used in combination with Ephedra sinica root.

Target Protein

5'-AMP-activated protein kinase catalytic subunit alpha-1 PRKAA1
5'-AMP-activated protein kinase subunit gamma-1 PRKAG1
5'-AMP-activated protein kinase subunit beta-1 PRKAB1
ATP-sensitive inward rectifier potassium channel 8 KCNJ8

Referensi & Sumber

Artikel (PubMed)
  • PMID: 9418116
    Enia G, Garozzo M, Zoccali C: Lactic acidosis induced by phenformin is still a public health problem in Italy. BMJ. 1997 Nov 29;315(7120):1466-7.
  • PMID: 9230023
    Rosand J, Friedberg JW, Yang JM: Fatal phenformin-associated lactic acidosis. Ann Intern Med. 1997 Jul 15;127(2):170.

Contoh Produk & Brand

Produk: 0 • International brands: 1
International Brands
  • DBI — Ciba-Geigy

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul