Peringatan Keamanan

Overdosage may lead to excessive diuresis with electrolyte depletion.

Etacrynic acid

DB00903

small molecule approved investigational

Deskripsi

A compound that inhibits symport of sodium, potassium, and chloride primarily in the ascending limb of Henle, but also in the proximal and distal tubules. This pharmacological action results in excretion of these ions, increased urinary output, and reduction in extracellular fluid. This compound has been classified as a loop or high ceiling diuretic.

Struktur Molekul 2D

Berat 303.138
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Onset of action is rapid, usually within 30 minutes after an oral dose of ethacrynic acid or within 5 minutes after an intravenous injection of ethacrynic acid.

Metabolisme

Hepatic.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

1 Data
  • 1. Take with food. Food reduces irritation.

Interaksi Obat

1284 Data
Duloxetine The risk or severity of orthostatic hypotension and syncope can be increased when Etacrynic acid is combined with Duloxetine.
Levodopa The risk or severity of hypotension and orthostatic hypotension can be increased when Etacrynic acid is combined with Levodopa.
Succinylcholine The therapeutic efficacy of Succinylcholine can be increased when used in combination with Etacrynic acid.
Metocurine iodide The therapeutic efficacy of Metocurine iodide can be increased when used in combination with Etacrynic acid.
Gallamine triethiodide The therapeutic efficacy of Gallamine triethiodide can be increased when used in combination with Etacrynic acid.
Cisatracurium The therapeutic efficacy of Cisatracurium can be increased when used in combination with Etacrynic acid.
Rocuronium The therapeutic efficacy of Rocuronium can be increased when used in combination with Etacrynic acid.
Atracurium besylate The therapeutic efficacy of Atracurium besylate can be increased when used in combination with Etacrynic acid.
Doxacurium The therapeutic efficacy of Doxacurium can be increased when used in combination with Etacrynic acid.
Mivacurium The therapeutic efficacy of Mivacurium can be increased when used in combination with Etacrynic acid.
Decamethonium The therapeutic efficacy of Decamethonium can be increased when used in combination with Etacrynic acid.
Metocurine The therapeutic efficacy of Metocurine can be increased when used in combination with Etacrynic acid.
Pancuronium The therapeutic efficacy of Pancuronium can be increased when used in combination with Etacrynic acid.
Pipecuronium The therapeutic efficacy of Pipecuronium can be increased when used in combination with Etacrynic acid.
Vecuronium The therapeutic efficacy of Vecuronium can be increased when used in combination with Etacrynic acid.
Rapacuronium The therapeutic efficacy of Rapacuronium can be increased when used in combination with Etacrynic acid.
Pyrantel The therapeutic efficacy of Pyrantel can be increased when used in combination with Etacrynic acid.
Neosaxitoxin The therapeutic efficacy of Neosaxitoxin can be increased when used in combination with Etacrynic acid.
Atracurium The therapeutic efficacy of Atracurium can be increased when used in combination with Etacrynic acid.
Gallamine The therapeutic efficacy of Gallamine can be increased when used in combination with Etacrynic acid.
Alcuronium The therapeutic efficacy of Alcuronium can be increased when used in combination with Etacrynic acid.
Tubocurarine The therapeutic efficacy of Tubocurarine can be increased when used in combination with Etacrynic acid.
Allopurinol The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Allopurinol.
Canagliflozin The risk or severity of hypotension can be increased when Canagliflozin is combined with Etacrynic acid.
Cisplatin The risk or severity of ototoxicity and nephrotoxicity can be increased when Etacrynic acid is combined with Cisplatin.
Dofetilide The risk or severity of QTc prolongation, torsade de pointes, hypokalemia, hypomagnesemia, and cardiac arrest can be increased when Etacrynic acid is combined with Dofetilide.
Ivabradine The risk or severity of Cardiac Arrhythmia can be increased when Etacrynic acid is combined with Ivabradine.
Lithium citrate Etacrynic acid may decrease the excretion rate of Lithium citrate which could result in a higher serum level.
Lithium carbonate Etacrynic acid may decrease the excretion rate of Lithium carbonate which could result in a higher serum level.
Lithium hydroxide Etacrynic acid may decrease the excretion rate of Lithium hydroxide which could result in a higher serum level.
Methotrexate The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Methotrexate.
Probenecid The risk or severity of adverse effects can be increased when Probenecid is combined with Etacrynic acid.
Risperidone The risk or severity of hypotension can be increased when Etacrynic acid is combined with Risperidone.
Topiramate The risk or severity of hypokalemia can be increased when Etacrynic acid is combined with Topiramate.
Foscarnet Etacrynic acid may decrease the excretion rate of Foscarnet which could result in a higher serum level.
Mannitol The risk or severity of nephrotoxicity can be increased when Mannitol is combined with Etacrynic acid.
Tenofovir disoproxil Etacrynic acid may increase the nephrotoxic activities of Tenofovir disoproxil.
Tenofovir alafenamide Etacrynic acid may increase the nephrotoxic activities of Tenofovir alafenamide.
Tenofovir Etacrynic acid may increase the nephrotoxic activities of Tenofovir.
Dicoumarol The protein binding of Dicoumarol can be decreased when combined with Etacrynic acid.
Phenindione The protein binding of Phenindione can be decreased when combined with Etacrynic acid.
Warfarin The protein binding of Warfarin can be decreased when combined with Etacrynic acid.
Phenprocoumon The protein binding of Phenprocoumon can be decreased when combined with Etacrynic acid.
Acenocoumarol The protein binding of Acenocoumarol can be decreased when combined with Etacrynic acid.
4-hydroxycoumarin The protein binding of 4-hydroxycoumarin can be decreased when combined with Etacrynic acid.
Coumarin The protein binding of Coumarin can be decreased when combined with Etacrynic acid.
(R)-warfarin The protein binding of (R)-warfarin can be decreased when combined with Etacrynic acid.
Ethyl biscoumacetate The protein binding of Ethyl biscoumacetate can be decreased when combined with Etacrynic acid.
Fluindione The protein binding of Fluindione can be decreased when combined with Etacrynic acid.
Clorindione The protein binding of Clorindione can be decreased when combined with Etacrynic acid.
Diphenadione The protein binding of Diphenadione can be decreased when combined with Etacrynic acid.
Tioclomarol The protein binding of Tioclomarol can be decreased when combined with Etacrynic acid.
(S)-Warfarin The protein binding of (S)-Warfarin can be decreased when combined with Etacrynic acid.
Aripiprazole Aripiprazole may increase the hypotensive activities of Etacrynic acid.
Aripiprazole lauroxil Aripiprazole lauroxil may increase the hypotensive activities of Etacrynic acid.
Nicorandil Nicorandil may increase the hypotensive activities of Etacrynic acid.
Acetyldigitoxin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Acetyldigitoxin.
Deslanoside The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Deslanoside.
Ouabain The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Ouabain.
Digitoxin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Digitoxin.
Oleandrin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Oleandrin.
Cymarin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Cymarin.
Proscillaridin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Proscillaridin.
Metildigoxin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Metildigoxin.
Lanatoside C The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Lanatoside C.
Gitoformate The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Gitoformate.
Acetyldigoxin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Acetyldigoxin.
Peruvoside The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Peruvoside.
Digoxin The risk or severity of adverse effects can be increased when Etacrynic acid is combined with Digoxin.
Cyclosporine The risk or severity of adverse effects can be increased when Cyclosporine is combined with Etacrynic acid.
Icosapent The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Icosapent.
Mesalazine The risk or severity of nephrotoxicity can be increased when Mesalazine is combined with Etacrynic acid.
Nabumetone The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Nabumetone.
Ketorolac The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Ketorolac.
Tenoxicam The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Tenoxicam.
Celecoxib The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Celecoxib.
Tolmetin The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Tolmetin.
Rofecoxib The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Rofecoxib.
Piroxicam The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Piroxicam.
Fenoprofen The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Fenoprofen.
Valdecoxib The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Valdecoxib.
Diclofenac The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Diclofenac.
Sulindac The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Sulindac.
Flurbiprofen The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Flurbiprofen.
Etodolac The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Etodolac.
Mefenamic acid The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Mefenamic acid.
Naproxen The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Naproxen.
Sulfasalazine The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Sulfasalazine.
Phenylbutazone The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Phenylbutazone.
Carprofen The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Carprofen.
Diflunisal The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Diflunisal.
Salicylic acid The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Salicylic acid.
Meclofenamic acid The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Meclofenamic acid.
Oxaprozin The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Oxaprozin.
Ketoprofen The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Ketoprofen.
Balsalazide The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Balsalazide.
Ibuprofen The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Ibuprofen.
Olsalazine The risk or severity of nephrotoxicity can be increased when Etacrynic acid is combined with Olsalazine.
Lumiracoxib The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Lumiracoxib.
Magnesium salicylate The therapeutic efficacy of Etacrynic acid can be decreased when used in combination with Magnesium salicylate.

Target Protein

Solute carrier family 12 member 1 SLC12A1
Sodium/potassium-transporting ATPase subunit alpha-1 ATP1A1
Lymphoid enhancer-binding factor 1 LEF1
Glutathione S-transferase P GSTP1

Referensi & Sumber

Synthesis reference: Schultz, E.M. and Sprague, J.M.; U.S. Patent 3,255,241; June 7, 1966; assigned to Merck & co., Inc.

Contoh Produk & Brand

Produk: 35 • International brands: 11
Produk
  • Edecrin
    Tablet • 25 mg/1 • Oral • US • Approved
  • Edecrin
    Tablet • 25 mg/1 • Oral • US • Approved
  • Edecrin
    Tablet • 25 mg/1 • Oral • US • Approved
  • Edecrin
    Tablet • 25 mg/1 • Oral • US • Approved
  • Edecrin
    Tablet • 25 mg/1 • Oral • US • Approved
  • Edecrin
    Tablet • 25 mg • Oral • Canada • Approved
  • Edecrin Sodium
    Injection, powder, lyophilized, for solution • 50 mg/50mL • Intravenous • US • Approved
  • Edecrin Tab 50mg
    Tablet • 50 mg • Oral • Canada • Approved
Menampilkan 8 dari 35 produk.
International Brands
  • Crinuryl — Assia
  • Edecril — Merck
  • Edecrina
  • Endecril
  • Hidromedin
  • Hydromedin — Merck
  • Mingit
  • Otacril
  • Reomax — Bioindustria
  • Taladren — Malesci

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul