Oxybuprocaine

DB00892

small molecule approved investigational

Deskripsi

Oxybuprocaine (also known as Benoxinate) is a local anesthetic, which is used especially in ophthalmology and otolaryngology. Oxybuprocaine binds to sodium channels and reversibly stabilizes the neuronal membrane which decreases its permeability to sodium ions.

Struktur Molekul 2D

Berat 308.4158
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) -
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1642 Data
Buprenorphine Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Hydrocodone Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Magnesium sulfate The therapeutic efficacy of Oxybuprocaine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Oxybuprocaine may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Mirtazapine Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Orphenadrine Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Pramipexole Oxybuprocaine may increase the sedative activities of Pramipexole.
Ropinirole Oxybuprocaine may increase the sedative activities of Ropinirole.
Rotigotine Oxybuprocaine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Oxybuprocaine.
Sodium oxybate Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Thalidomide Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Hyaluronidase (ovine) Hyaluronidase (ovine) can cause an increase in the absorption of Oxybuprocaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase (human recombinant) Hyaluronidase (human recombinant) can cause an increase in the absorption of Oxybuprocaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Hyaluronidase Hyaluronidase can cause an increase in the absorption of Oxybuprocaine resulting in an increased serum concentration and potentially a worsening of adverse effects.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Oxybuprocaine.
Pegvisomant Pegvisomant may increase the neuromuscular blocking activities of Oxybuprocaine.
Mefloquine The risk or severity of methemoglobinemia can be increased when Mefloquine is combined with Oxybuprocaine.
Tacrine Tacrine may increase the neuromuscular blocking activities of Oxybuprocaine.
Sulpiride Sulpiride may increase the neuromuscular blocking activities of Oxybuprocaine.
Profenamine Profenamine may increase the neuromuscular blocking activities of Oxybuprocaine.
Chlorpromazine Chlorpromazine may increase the neuromuscular blocking activities of Oxybuprocaine.
Gallamine triethiodide Gallamine triethiodide may increase the neuromuscular blocking activities of Oxybuprocaine.
Triflupromazine Triflupromazine may increase the neuromuscular blocking activities of Oxybuprocaine.
Cisplatin The risk or severity of methemoglobinemia can be increased when Cisplatin is combined with Oxybuprocaine.
Cinchocaine The risk or severity of methemoglobinemia can be increased when Cinchocaine is combined with Oxybuprocaine.
Pyridostigmine Pyridostigmine may increase the neuromuscular blocking activities of Oxybuprocaine.
Nizatidine Nizatidine may increase the neuromuscular blocking activities of Oxybuprocaine.
Galantamine Galantamine may increase the neuromuscular blocking activities of Oxybuprocaine.
Isoflurophate Isoflurophate may increase the neuromuscular blocking activities of Oxybuprocaine.
Diethylcarbamazine Diethylcarbamazine may increase the neuromuscular blocking activities of Oxybuprocaine.
Procaine The risk or severity of methemoglobinemia can be increased when Procaine is combined with Oxybuprocaine.
Minaprine Minaprine may increase the neuromuscular blocking activities of Oxybuprocaine.
Donepezil Donepezil may increase the neuromuscular blocking activities of Oxybuprocaine.
Terbutaline Terbutaline may increase the neuromuscular blocking activities of Oxybuprocaine.
Mechlorethamine The risk or severity of methemoglobinemia can be increased when Mechlorethamine is combined with Oxybuprocaine.
Hexafluronium Hexafluronium may increase the neuromuscular blocking activities of Oxybuprocaine.
Demecarium Demecarium may increase the neuromuscular blocking activities of Oxybuprocaine.
Physostigmine Physostigmine may increase the neuromuscular blocking activities of Oxybuprocaine.
Rivastigmine Rivastigmine may increase the neuromuscular blocking activities of Oxybuprocaine.
Edrophonium Edrophonium may increase the neuromuscular blocking activities of Oxybuprocaine.
Procainamide Procainamide may increase the neuromuscular blocking activities of Oxybuprocaine.
Memantine Memantine may increase the neuromuscular blocking activities of Oxybuprocaine.
Ambenonium Ambenonium may increase the neuromuscular blocking activities of Oxybuprocaine.
Tubocurarine Tubocurarine may increase the neuromuscular blocking activities of Oxybuprocaine.
Ketamine Ketamine may increase the neuromuscular blocking activities of Oxybuprocaine.
Decamethonium Decamethonium may increase the neuromuscular blocking activities of Oxybuprocaine.
Pancuronium Pancuronium may increase the neuromuscular blocking activities of Oxybuprocaine.
Pipecuronium Pipecuronium may increase the neuromuscular blocking activities of Oxybuprocaine.
Ginkgo biloba Ginkgo biloba may increase the neuromuscular blocking activities of Oxybuprocaine.
Neostigmine Neostigmine may increase the neuromuscular blocking activities of Oxybuprocaine.
Bambuterol Bambuterol may increase the neuromuscular blocking activities of Oxybuprocaine.
1,10-Phenanthroline 1,10-Phenanthroline may increase the neuromuscular blocking activities of Oxybuprocaine.
Methylphosphinic Acid Methylphosphinic Acid may increase the neuromuscular blocking activities of Oxybuprocaine.
Thiotepa The risk or severity of methemoglobinemia can be increased when Thiotepa is combined with Oxybuprocaine.
Huperzine A Huperzine A may increase the neuromuscular blocking activities of Oxybuprocaine.
Phenserine Phenserine may increase the neuromuscular blocking activities of Oxybuprocaine.
Regramostim Regramostim may increase the neuromuscular blocking activities of Oxybuprocaine.
Aprotinin Aprotinin may increase the neuromuscular blocking activities of Oxybuprocaine.
Betaine Betaine may increase the neuromuscular blocking activities of Oxybuprocaine.
Capsaicin The risk or severity of methemoglobinemia can be increased when Oxybuprocaine is combined with Capsaicin.
Coumaphos Coumaphos may increase the neuromuscular blocking activities of Oxybuprocaine.
Dichlorvos Dichlorvos may increase the neuromuscular blocking activities of Oxybuprocaine.
Fenthion Fenthion may increase the neuromuscular blocking activities of Oxybuprocaine.
Metrifonate Metrifonate may increase the neuromuscular blocking activities of Oxybuprocaine.
Acotiamide Acotiamide may increase the neuromuscular blocking activities of Oxybuprocaine.
Methanesulfonyl Fluoride Methanesulfonyl Fluoride may increase the neuromuscular blocking activities of Oxybuprocaine.
Paraoxon Paraoxon may increase the neuromuscular blocking activities of Oxybuprocaine.
Tyrothricin The risk or severity of methemoglobinemia can be increased when Tyrothricin is combined with Oxybuprocaine.
Ipidacrine Ipidacrine may increase the neuromuscular blocking activities of Oxybuprocaine.
Distigmine Distigmine may increase the neuromuscular blocking activities of Oxybuprocaine.
Tretamine The risk or severity of methemoglobinemia can be increased when Tretamine is combined with Oxybuprocaine.
Posiphen Posiphen may increase the neuromuscular blocking activities of Oxybuprocaine.
Ethanol Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Oxybuprocaine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Oxybuprocaine.
Fluvoxamine The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Oxybuprocaine is combined with Milnacipran.

Target Protein

Sodium channel protein type 10 subunit alpha SCN10A

Referensi & Sumber

Synthesis reference: Katsuyuki Inoo, Mitsuhiro Kawada, Kenjiro Mori, "Oxybuprocaine-Containing Analgesic/Antipruritic External Preparation." U.S. Patent US20110124727, issued May 26, 2011.

Contoh Produk & Brand

Produk: 14 • International brands: 8
Produk
  • Altafluor
    Solution • - • Ophthalmic • US • Approved
  • Altafluor
    Solution • - • Ophthalmic • US • Approved
  • Fluorescein Sodium & Benoxinate Hydrochloride Ophthalmic Solution, USP
    Solution • - • Ophthalmic • Canada • Approved
  • Fluorescein Sodium and Benoxinate Hydrochloride
    Solution / drops • - • Ophthalmic • US • Approved
  • Fluorescein Sodium and Benoxinate Hydrochloride
    Solution / drops • - • Ophthalmic • US
  • Fluorescein Sodium and Benoxinate Hydrochloride
    Solution / drops • - • Ophthalmic • US • Generic • Approved
  • Fluorescein Sodium and Benoxinate Hydrochloride
    Solution / drops • - • Ophthalmic • US • Generic • Approved
  • Fluorox
    Solution • - • Ophthalmic • Canada • Approved
Menampilkan 8 dari 14 produk.
International Brands
  • Benoxil — Santen
  • Cebesine — Chauvin Bausch & Lomb
  • Conjuncain
  • Dorsacaine
  • Lacrimin — Santen
  • Novesin — Novartis
  • Novesine — Novartis
  • Prescaina — Llorens

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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