Peringatan Keamanan

Overdosage can lead to acute profound water loss, volume and electrolyte depletion, dehydration, reduction of blood volume and circulatory collapse with a possibility of vascular thrombosis and embolism. Electrolyte depletion may be manifested by weakness, dizziness, mental confusion, anorexia, lethargy, vomiting and cramps. Treatment consists of replacement of fluid and electrolyte losses by careful monitoring of the urine and electrolyte output and serum electrolyte levels.

Bumetanide

DB00887

small molecule approved

Deskripsi

Bumetanide is a sulfamyl diuretic.

Struktur Molekul 2D

Berat 364.416
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 60-90 minutes
Volume Distribusi -
Klirens (Clearance) * 0.2 - 1.1 mL/min/kg [preterm and full-term neonates with respiratory disorders] * 2.17 mL/min/kg [neonates receiving bumetanide for volume overload] * 1.8 +/- 0.3 mL/min/kg [geriatric subjects] * 2.9 +/- 0.2 mL/min/kg [younger subjects]

Absorpsi

Bumetanide is completely absorbed (80%), and the absorption is not altered when taken with food. Bioavailability is almost complete.

Metabolisme

45% is secreted unchanged. Urinary and biliary metabolites are formed by oxidation of the N-butyl side chain.

Rute Eliminasi

Oral administration of carbon-14 labeled Bumex to human volunteers revealed that 81% of the administered radioactivity was excreted in the urine, 45% of it as unchanged drug. Biliary excretion of Bumex amounted to only 2% of the administered dose.

Interaksi Makanan

1 Data
  • 1. Take with food. Food reduces irritation.

Interaksi Obat

1370 Data
Duloxetine The risk or severity of orthostatic hypotension and syncope can be increased when Bumetanide is combined with Duloxetine.
Levodopa The risk or severity of hypotension and orthostatic hypotension can be increased when Bumetanide is combined with Levodopa.
Allopurinol The risk or severity of adverse effects can be increased when Bumetanide is combined with Allopurinol.
Canagliflozin The risk or severity of hypotension can be increased when Canagliflozin is combined with Bumetanide.
Cisplatin The risk or severity of ototoxicity and nephrotoxicity can be increased when Bumetanide is combined with Cisplatin.
Dofetilide The risk or severity of QTc prolongation, torsade de pointes, hypokalemia, hypomagnesemia, and cardiac arrest can be increased when Bumetanide is combined with Dofetilide.
Ivabradine The risk or severity of Cardiac Arrhythmia can be increased when Bumetanide is combined with Ivabradine.
Lithium citrate Bumetanide may decrease the excretion rate of Lithium citrate which could result in a higher serum level.
Lithium carbonate Bumetanide may decrease the excretion rate of Lithium carbonate which could result in a higher serum level.
Lithium hydroxide Bumetanide may decrease the excretion rate of Lithium hydroxide which could result in a higher serum level.
Nicotine The risk or severity of adverse effects can be increased when Bumetanide is combined with Nicotine.
Mecamylamine The risk or severity of adverse effects can be increased when Bumetanide is combined with Mecamylamine.
Pentolinium The risk or severity of adverse effects can be increased when Bumetanide is combined with Pentolinium.
Trimethaphan The risk or severity of adverse effects can be increased when Bumetanide is combined with Trimethaphan.
Hexamethonium The risk or severity of adverse effects can be increased when Bumetanide is combined with Hexamethonium.
Cyclopentamine The risk or severity of adverse effects can be increased when Bumetanide is combined with Cyclopentamine.
Probenecid The risk or severity of adverse effects can be increased when Probenecid is combined with Bumetanide.
Risperidone The risk or severity of hypotension can be increased when Bumetanide is combined with Risperidone.
Topiramate The risk or severity of hypokalemia can be increased when Bumetanide is combined with Topiramate.
Methotrexate The therapeutic efficacy of Bumetanide can be decreased when used in combination with Methotrexate.
Foscarnet Bumetanide may decrease the excretion rate of Foscarnet which could result in a higher serum level.
Mannitol The risk or severity of nephrotoxicity can be increased when Mannitol is combined with Bumetanide.
Tenofovir disoproxil Bumetanide may increase the nephrotoxic activities of Tenofovir disoproxil.
Tenofovir alafenamide The serum concentration of Tenofovir alafenamide can be increased when it is combined with Bumetanide.
Tenofovir Bumetanide may increase the nephrotoxic activities of Tenofovir.
Aspartame The excretion of Bumetanide can be decreased when combined with Aspartame.
Aminohippuric acid The excretion of Bumetanide can be decreased when combined with Aminohippuric acid.
Lansoprazole The excretion of Bumetanide can be decreased when combined with Lansoprazole.
Guanidine The excretion of Bumetanide can be decreased when combined with Guanidine.
Oxytetracycline The excretion of Bumetanide can be decreased when combined with Oxytetracycline.
Leucovorin The excretion of Bumetanide can be decreased when combined with Leucovorin.
Esomeprazole The excretion of Bumetanide can be decreased when combined with Esomeprazole.
Succinic acid The excretion of Succinic acid can be decreased when combined with Bumetanide.
Citrulline The excretion of Citrulline can be decreased when combined with Bumetanide.
Cefdinir The excretion of Cefdinir can be decreased when combined with Bumetanide.
Fluorescein The excretion of Fluorescein can be decreased when combined with Bumetanide.
Hydrocortisone The excretion of Hydrocortisone can be decreased when combined with Bumetanide.
Dinoprostone The excretion of Dinoprostone can be decreased when combined with Bumetanide.
Famotidine The excretion of Famotidine can be decreased when combined with Bumetanide.
Fexofenadine The excretion of Fexofenadine can be decreased when combined with Bumetanide.
Tazobactam The excretion of Tazobactam can be decreased when combined with Bumetanide.
Cyclic adenosine monophosphate The excretion of Cyclic adenosine monophosphate can be decreased when combined with Bumetanide.
Cholic Acid The excretion of Cholic Acid can be decreased when combined with Bumetanide.
Glutaric Acid The excretion of Glutaric Acid can be decreased when combined with Bumetanide.
Oxalic Acid The excretion of Oxalic Acid can be decreased when combined with Bumetanide.
Taurocholic acid The excretion of Taurocholic acid can be decreased when combined with Bumetanide.
Ellagic acid The excretion of Ellagic acid can be decreased when combined with Bumetanide.
Avibactam The excretion of Avibactam can be decreased when combined with Bumetanide.
Silibinin The excretion of Silibinin can be decreased when combined with Bumetanide.
Relebactam The excretion of Relebactam can be decreased when combined with Bumetanide.
Novobiocin The excretion of Bumetanide can be decreased when combined with Novobiocin.
Melatonin The excretion of Bumetanide can be decreased when combined with Melatonin.
Liotrix The excretion of Bumetanide can be decreased when combined with Liotrix.
Cilastatin The excretion of Bumetanide can be decreased when combined with Cilastatin.
trans-2-hydroxycinnamic acid The excretion of Bumetanide can be decreased when combined with trans-2-hydroxycinnamic acid.
Benzoic acid The excretion of Bumetanide can be decreased when combined with Benzoic acid.
Caprylic acid The excretion of Bumetanide can be decreased when combined with Caprylic acid.
Ataluren The excretion of Bumetanide can be decreased when combined with Ataluren.
Teriflunomide The excretion of Bumetanide can be decreased when combined with Teriflunomide.
Dabrafenib The excretion of Bumetanide can be decreased when combined with Dabrafenib.
Dolutegravir The excretion of Bumetanide can be decreased when combined with Dolutegravir.
Lenvatinib The excretion of Bumetanide can be decreased when combined with Lenvatinib.
Cabotegravir The excretion of Bumetanide can be decreased when combined with Cabotegravir.
Pradigastat The excretion of Bumetanide can be decreased when combined with Pradigastat.
Enasidenib The excretion of Bumetanide can be decreased when combined with Enasidenib.
Enalapril The excretion of Bumetanide can be decreased when combined with Enalapril.
Quinapril The excretion of Quinapril can be decreased when combined with Bumetanide.
Captopril The excretion of Captopril can be decreased when combined with Bumetanide.
Cefotiam The excretion of Bumetanide can be decreased when combined with Cefotiam.
Cefalotin The excretion of Bumetanide can be decreased when combined with Cefalotin.
Cefotaxime The excretion of Bumetanide can be decreased when combined with Cefotaxime.
Cephalexin The excretion of Bumetanide can be decreased when combined with Cephalexin.
Valaciclovir The excretion of Valaciclovir can be decreased when combined with Bumetanide.
Acyclovir The excretion of Bumetanide can be decreased when combined with Acyclovir.
Cefaclor The excretion of Bumetanide can be decreased when combined with Cefaclor.
Pantoprazole The excretion of Bumetanide can be decreased when combined with Pantoprazole.
Cefadroxil The excretion of Bumetanide can be decreased when combined with Cefadroxil.
Ceftriaxone The excretion of Bumetanide can be decreased when combined with Ceftriaxone.
Ceftibuten The excretion of Ceftibuten can be decreased when combined with Bumetanide.
Cefamandole The excretion of Bumetanide can be decreased when combined with Cefamandole.
Cefazolin The excretion of Cefazolin can be decreased when combined with Bumetanide.
Cefoperazone The excretion of Bumetanide can be decreased when combined with Cefoperazone.
Ceftizoxime The excretion of Ceftizoxime can be decreased when combined with Bumetanide.
Cefacetrile The excretion of Cefacetrile can be decreased when combined with Bumetanide.
Cefaloridine The excretion of Cefaloridine can be decreased when combined with Bumetanide.
Dronedarone The excretion of Bumetanide can be decreased when combined with Dronedarone.
Favipiravir The excretion of Bumetanide can be decreased when combined with Favipiravir.
Tafamidis The excretion of Bumetanide can be decreased when combined with Tafamidis.
Dexamethasone acetate The excretion of Dexamethasone acetate can be decreased when combined with Bumetanide.
Acamprosate The excretion of Acamprosate can be decreased when combined with Bumetanide.
Aripiprazole Aripiprazole may increase the hypotensive activities of Bumetanide.
Aripiprazole lauroxil Aripiprazole lauroxil may increase the hypotensive activities of Bumetanide.
Nicorandil Nicorandil may increase the hypotensive activities of Bumetanide.
Ouabain The risk or severity of adverse effects can be increased when Bumetanide is combined with Ouabain.
Acetyldigitoxin The risk or severity of adverse effects can be increased when Bumetanide is combined with Acetyldigitoxin.
Deslanoside The risk or severity of adverse effects can be increased when Bumetanide is combined with Deslanoside.
Digitoxin The risk or severity of adverse effects can be increased when Bumetanide is combined with Digitoxin.
Oleandrin The risk or severity of adverse effects can be increased when Bumetanide is combined with Oleandrin.
Cymarin The risk or severity of adverse effects can be increased when Bumetanide is combined with Cymarin.
Proscillaridin The risk or severity of adverse effects can be increased when Bumetanide is combined with Proscillaridin.

Target Protein

Solute carrier family 12 member 1 SLC12A1
Solute carrier family 12 member 2 SLC12A2
Solute carrier family 12 member 4 SLC12A4
Solute carrier family 12 member 5 SLC12A5
Cystic fibrosis transmembrane conductance regulator CFTR

Referensi & Sumber

Synthesis reference: Felt, P.W.; US. Patent 3,634,583; January 11, 1972; assigned to Lovens Kemiske Fabrik Produktionsaktieselskab, Denmark.

Contoh Produk & Brand

Produk: 167 • International brands: 3
Produk
  • Bumetanide
    Tablet • 0.5 mg/1 • Oral • US • Generic • Approved
  • Bumetanide
    Tablet • 1 mg/1 • Oral • US • Generic • Approved
  • Bumetanide
    Tablet • 2 mg/1 • Oral • US • Generic • Approved
  • Bumetanide
    Tablet • .5 mg/1 • Oral • US • Generic • Approved
  • Bumetanide
    Tablet • 1 mg/1 • Oral • US • Generic • Approved
  • Bumetanide
    Tablet • 2 mg/1 • Oral • US • Generic • Approved
  • Bumetanide
    Tablet • 0.5 mg/1 • Oral • US • Generic • Approved
  • Bumetanide
    Tablet • 1 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 167 produk.
International Brands
  • Burinex — F. Hoffmann-La Roche Ltd.
  • Fordiuran — LEO Pharma A/S
  • Lunetoron — Daiichi Sankyo

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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