Peringatan Keamanan

Oral, rat LD50: > 10 g/kg. Signs of overdose include those caused by electrolyte depletion (hypokalemia, hypochloremia, hyponatremia) and dehydration resulting from excessive diuresis. If digitalis has also been administered hypokalemia may accentuate cardiac arrhythmias.

Chlorothiazide

DB00880

small molecule approved vet_approved

Deskripsi

A thiazide diuretic with actions and uses similar to those of hydrochlorothiazide. (From Martindale, The Extra Pharmacopoeia, 30th ed, p812)

Struktur Molekul 2D

Berat 295.723
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 45-120 minutes
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly absorbed following oral administration.

Metabolisme

Chlorothiazide is not metabolized but is eliminated rapidly by the kidney.

Rute Eliminasi

Chlorothiazide is not metabolized but is eliminated rapidly by the kidney. After oral doses, 10 to 15 percent of the dose is excreted unchanged in the urine. Chlorothiazide crosses the placental but not the blood-brain barrier and is excreted in breast milk.

Interaksi Obat

1667 Data
Duloxetine The risk or severity of orthostatic hypotension and syncope can be increased when Chlorothiazide is combined with Duloxetine.
Levodopa The risk or severity of hypotension and orthostatic hypotension can be increased when Chlorothiazide is combined with Levodopa.
Risperidone Chlorothiazide may increase the hypotensive activities of Risperidone.
Alfuzosin Alfuzosin may increase the hypotensive activities of Chlorothiazide.
Amifostine Chlorothiazide may increase the hypotensive activities of Amifostine.
Diazoxide Diazoxide may increase the hypotensive activities of Chlorothiazide.
Forasartan Chlorothiazide may increase the hypotensive and Electrolyte Disturbance activities of Forasartan.
Tasosartan Chlorothiazide may increase the hypotensive and Electrolyte Disturbance activities of Tasosartan.
Saralasin Chlorothiazide may increase the hypotensive and Electrolyte Disturbance activities of Saralasin.
Fimasartan Chlorothiazide may increase the hypotensive and Electrolyte Disturbance activities of Fimasartan.
Methylphenidate Methylphenidate may decrease the antihypertensive activities of Chlorothiazide.
Dexmethylphenidate Dexmethylphenidate may decrease the antihypertensive activities of Chlorothiazide.
Obinutuzumab Chlorothiazide may increase the hypotensive activities of Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the hypotensive activities of Chlorothiazide.
Rituximab Chlorothiazide may increase the hypotensive activities of Rituximab.
Phentermine Phentermine may decrease the antihypertensive activities of Chlorothiazide.
Midodrine Midodrine may decrease the antihypertensive activities of Chlorothiazide.
Eletriptan Eletriptan may decrease the antihypertensive activities of Chlorothiazide.
Methysergide Methysergide may decrease the antihypertensive activities of Chlorothiazide.
Cabergoline Cabergoline may decrease the antihypertensive activities of Chlorothiazide.
Zolmitriptan Zolmitriptan may decrease the antihypertensive activities of Chlorothiazide.
Dihydroergotamine Dihydroergotamine may decrease the antihypertensive activities of Chlorothiazide.
Protriptyline Protriptyline may decrease the antihypertensive activities of Chlorothiazide.
Methylergometrine Methylergometrine may decrease the antihypertensive activities of Chlorothiazide.
Mirtazapine Mirtazapine may decrease the antihypertensive activities of Chlorothiazide.
Phenylephrine Phenylephrine may decrease the antihypertensive activities of Chlorothiazide.
Droperidol Droperidol may decrease the antihypertensive activities of Chlorothiazide.
Doxapram Doxapram may decrease the antihypertensive activities of Chlorothiazide.
Lisuride Lisuride may decrease the antihypertensive activities of Chlorothiazide.
Metaraminol Metaraminol may decrease the antihypertensive activities of Chlorothiazide.
Ergotamine Ergotamine may decrease the antihypertensive activities of Chlorothiazide.
Nicergoline Nicergoline may decrease the antihypertensive activities of Chlorothiazide.
Methoxamine Methoxamine may decrease the antihypertensive activities of Chlorothiazide.
Trimipramine Trimipramine may decrease the antihypertensive activities of Chlorothiazide.
Phenmetrazine Phenmetrazine may decrease the antihypertensive activities of Chlorothiazide.
Trifluoperazine Trifluoperazine may decrease the antihypertensive activities of Chlorothiazide.
Pseudoephedrine Pseudoephedrine may decrease the antihypertensive activities of Chlorothiazide.
Benzphetamine Benzphetamine may decrease the antihypertensive activities of Chlorothiazide.
Diethylpropion Diethylpropion may decrease the antihypertensive activities of Chlorothiazide.
Naratriptan Naratriptan may decrease the antihypertensive activities of Chlorothiazide.
Frovatriptan Frovatriptan may decrease the antihypertensive activities of Chlorothiazide.
Methoxyflurane Methoxyflurane may decrease the antihypertensive activities of Chlorothiazide.
Ergoloid mesylate Ergoloid mesylate may decrease the antihypertensive activities of Chlorothiazide.
Dutasteride Dutasteride may decrease the antihypertensive activities of Chlorothiazide.
Propafenone Propafenone may decrease the antihypertensive activities of Chlorothiazide.
Pergolide Pergolide may decrease the antihypertensive activities of Chlorothiazide.
Finasteride Finasteride may decrease the antihypertensive activities of Chlorothiazide.
Ergometrine Ergometrine may decrease the antihypertensive activities of Chlorothiazide.
Lisdexamfetamine Lisdexamfetamine may decrease the antihypertensive activities of Chlorothiazide.
Mephentermine Mephentermine may decrease the antihypertensive activities of Chlorothiazide.
Yohimbine Yohimbine may decrease the antihypertensive activities of Chlorothiazide.
MMDA MMDA may decrease the antihypertensive activities of Chlorothiazide.
Midomafetamine Midomafetamine may decrease the antihypertensive activities of Chlorothiazide.
2,5-Dimethoxy-4-ethylamphetamine 2,5-Dimethoxy-4-ethylamphetamine may decrease the antihypertensive activities of Chlorothiazide.
4-Methoxyamphetamine 4-Methoxyamphetamine may decrease the antihypertensive activities of Chlorothiazide.
4-Bromo-2,5-dimethoxyamphetamine 4-Bromo-2,5-dimethoxyamphetamine may decrease the antihypertensive activities of Chlorothiazide.
Tenamfetamine Tenamfetamine may decrease the antihypertensive activities of Chlorothiazide.
Chlorphentermine Chlorphentermine may decrease the antihypertensive activities of Chlorothiazide.
Dextroamphetamine Dextroamphetamine may decrease the antihypertensive activities of Chlorothiazide.
Phendimetrazine Phendimetrazine may decrease the antihypertensive activities of Chlorothiazide.
Periciazine Periciazine may decrease the antihypertensive activities of Chlorothiazide.
Acepromazine Acepromazine may decrease the antihypertensive activities of Chlorothiazide.
Thioproperazine Thioproperazine may decrease the antihypertensive activities of Chlorothiazide.
Zuclopenthixol Zuclopenthixol may decrease the antihypertensive activities of Chlorothiazide.
Epicaptopril Epicaptopril may decrease the antihypertensive activities of Chlorothiazide.
1-benzylimidazole 1-benzylimidazole may decrease the antihypertensive activities of Chlorothiazide.
Lysergic acid diethylamide Lysergic acid diethylamide may decrease the antihypertensive activities of Chlorothiazide.
Amineptine Amineptine may decrease the antihypertensive activities of Chlorothiazide.
Dronedarone Dronedarone may decrease the antihypertensive activities of Chlorothiazide.
Flibanserin Flibanserin may decrease the antihypertensive activities of Chlorothiazide.
Iloperidone Iloperidone may decrease the antihypertensive activities of Chlorothiazide.
Amibegron Amibegron may decrease the antihypertensive activities of Chlorothiazide.
Naluzotan Naluzotan may decrease the antihypertensive activities of Chlorothiazide.
Cariprazine Cariprazine may decrease the antihypertensive activities of Chlorothiazide.
Mianserin Mianserin may decrease the antihypertensive activities of Chlorothiazide.
Nylidrin Nylidrin may decrease the antihypertensive activities of Chlorothiazide.
Solabegron Solabegron may decrease the antihypertensive activities of Chlorothiazide.
Asenapine Asenapine may decrease the antihypertensive activities of Chlorothiazide.
Esmirtazapine Esmirtazapine may decrease the antihypertensive activities of Chlorothiazide.
Vilazodone Vilazodone may decrease the antihypertensive activities of Chlorothiazide.
Nitrous oxide Nitrous oxide may decrease the antihypertensive activities of Chlorothiazide.
Xylometazoline Xylometazoline may decrease the antihypertensive activities of Chlorothiazide.
Isometheptene Isometheptene may decrease the antihypertensive activities of Chlorothiazide.
Naphazoline Naphazoline may decrease the antihypertensive activities of Chlorothiazide.
Tetryzoline Tetryzoline may decrease the antihypertensive activities of Chlorothiazide.
Cinitapride Cinitapride may decrease the antihypertensive activities of Chlorothiazide.
Lurasidone Lurasidone may decrease the antihypertensive activities of Chlorothiazide.
Tyramine Tyramine may decrease the antihypertensive activities of Chlorothiazide.
Adrafinil Adrafinil may decrease the antihypertensive activities of Chlorothiazide.
Ifenprodil Ifenprodil may decrease the antihypertensive activities of Chlorothiazide.
Etilefrine Etilefrine may decrease the antihypertensive activities of Chlorothiazide.
Butriptyline Butriptyline may decrease the antihypertensive activities of Chlorothiazide.
Cannabidiol Cannabidiol may decrease the antihypertensive activities of Chlorothiazide.
Brexpiprazole Brexpiprazole may decrease the antihypertensive activities of Chlorothiazide.
Cirazoline Cirazoline may decrease the antihypertensive activities of Chlorothiazide.
Synephrine Synephrine may decrease the antihypertensive activities of Chlorothiazide.
Tianeptine Tianeptine may decrease the antihypertensive activities of Chlorothiazide.
Oxaprotiline Oxaprotiline may decrease the antihypertensive activities of Chlorothiazide.
Iofetamine I-123 Iofetamine I-123 may decrease the antihypertensive activities of Chlorothiazide.
Dihydroergocornine Dihydroergocornine may decrease the antihypertensive activities of Chlorothiazide.

Target Protein

Solute carrier family 12 member 3 SLC12A3
Carbonic anhydrase 1 CA1
Carbonic anhydrase 2 CA2

Referensi & Sumber

Synthesis reference: Eugene S. Barabas, "Water soluble complex of a poly (vinyl lactam) and chlorothiazide and process for producing same." U.S. Patent US4713238, issued December, 1985.

Contoh Produk & Brand

Produk: 24 • International brands: 0
Produk
  • Chlorothiazide
    Tablet • 500 mg/1 • Oral • US • Generic • Approved
  • Chlorothiazide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Chlorothiazide
    Tablet • 500 mg/1 • Oral • US • Generic • Approved
  • Chlorothiazide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Chlorothiazide
    Tablet • 500 mg/1 • Oral • US • Generic • Approved
  • Chlorothiazide
    Injection, powder, lyophilized, for solution • 500 mg/18mL • Intravenous • US • Generic • Approved
  • Chlorothiazide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Chlorothiazide
    Tablet • 500 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 24 produk.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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