Peringatan Keamanan

LD50=597.0 mg/kg (Orally in rats)

Alprenolol

DB00866

small molecule experimental withdrawn

Deskripsi

One of the adrenergic beta-antagonists used as an antihypertensive, anti-anginal, and anti-arrhythmic agent. Alprenolol is no longer marketed by AstraZeneca, but may still be available in generic varieties.

Struktur Molekul 2D

Berat 249.3486
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 2-3 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Hepatic. One of the active metabolites, 4-OH-alprenolol, is an active beta-blocker.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

1673 Data
Ceritinib Alprenolol may increase the bradycardic activities of Ceritinib.
Ivabradine Alprenolol may increase the bradycardic activities of Ivabradine.
Ruxolitinib Ruxolitinib may increase the bradycardic activities of Alprenolol.
Alfuzosin Alfuzosin may increase the hypotensive activities of Alprenolol.
Amifostine Alprenolol may increase the hypotensive activities of Amifostine.
Diazoxide Diazoxide may increase the hypotensive activities of Alprenolol.
Methylphenidate Methylphenidate may decrease the antihypertensive activities of Alprenolol.
Dexmethylphenidate Dexmethylphenidate may decrease the antihypertensive activities of Alprenolol.
Obinutuzumab Alprenolol may increase the hypotensive activities of Obinutuzumab.
Pentoxifylline Pentoxifylline may increase the hypotensive activities of Alprenolol.
Rituximab Alprenolol may increase the hypotensive activities of Rituximab.
Desmopressin Desmopressin may decrease the antihypertensive activities of Alprenolol.
Doxapram Doxapram may decrease the antihypertensive activities of Alprenolol.
Phenmetrazine Phenmetrazine may decrease the antihypertensive activities of Alprenolol.
Dopamine Dopamine may decrease the antihypertensive activities of Alprenolol.
Dutasteride Dutasteride may decrease the antihypertensive activities of Alprenolol.
Finasteride Finasteride may decrease the antihypertensive activities of Alprenolol.
Epicaptopril Epicaptopril may decrease the antihypertensive activities of Alprenolol.
1-benzylimidazole 1-benzylimidazole may decrease the antihypertensive activities of Alprenolol.
Tyramine Tyramine may decrease the antihypertensive activities of Alprenolol.
Moxisylyte Moxisylyte may decrease the antihypertensive activities of Alprenolol.
Atipamezole Atipamezole may decrease the antihypertensive activities of Alprenolol.
Siponimod Siponimod may decrease the antihypertensive activities of Alprenolol.
Idazoxan Idazoxan may decrease the antihypertensive activities of Alprenolol.
Tramazoline Tramazoline may decrease the antihypertensive activities of Alprenolol.
Fenozolone Fenozolone may decrease the antihypertensive activities of Alprenolol.
Xenon Xenon may decrease the antihypertensive activities of Alprenolol.
Buflomedil Buflomedil may decrease the antihypertensive activities of Alprenolol.
Mefenorex Mefenorex may decrease the antihypertensive activities of Alprenolol.
Quinoline Yellow WS Quinoline Yellow WS may decrease the antihypertensive activities of Alprenolol.
Selpercatinib Selpercatinib may decrease the antihypertensive activities of Alprenolol.
Naxitamab Naxitamab may decrease the antihypertensive activities of Alprenolol.
Buprenorphine Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Hydrocodone Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Magnesium sulfate The therapeutic efficacy of Alprenolol can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Alprenolol may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Mirtazapine Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Orphenadrine Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Pramipexole Alprenolol may increase the sedative activities of Pramipexole.
Ropinirole Alprenolol may increase the sedative activities of Ropinirole.
Rotigotine Alprenolol may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Alprenolol.
Sodium oxybate Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Alprenolol.
Thalidomide Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Alprenolol may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Amiodarone The therapeutic efficacy of Alprenolol can be increased when used in combination with Amiodarone.
Bupivacaine The serum concentration of Bupivacaine can be increased when it is combined with Alprenolol.
Dipyridamole Dipyridamole may increase the bradycardic activities of Alprenolol.
Disopyramide Disopyramide may increase the bradycardic activities of Alprenolol.
Dronedarone Dronedarone may increase the bradycardic activities of Alprenolol.
Fingolimod Alprenolol may increase the bradycardic activities of Fingolimod.
Floctafenine The risk or severity of adverse effects can be increased when Alprenolol is combined with Floctafenine.
Mepivacaine The serum concentration of Mepivacaine can be increased when it is combined with Alprenolol.
Methacholine Alprenolol may increase the bronchoconstrictory activities of Methacholine.
Midodrine The therapeutic efficacy of Midodrine can be decreased when used in combination with Alprenolol.
Nifedipine The risk or severity of congestive heart failure and hypotension can be increased when Nifedipine is combined with Alprenolol.
Propafenone The risk or severity of adverse effects can be increased when Propafenone is combined with Alprenolol.
Regorafenib Regorafenib may increase the bradycardic activities of Alprenolol.
Reserpine Reserpine may increase the hypotensive activities of Alprenolol.
Deserpidine Deserpidine may increase the hypotensive activities of Alprenolol.
Guanethidine Guanethidine may increase the hypotensive activities of Alprenolol.
Rivastigmine Alprenolol may increase the bradycardic activities of Rivastigmine.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Alprenolol.
Dicoumarol The risk or severity of adverse effects can be increased when Alprenolol is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Alprenolol is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when Alprenolol is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Alprenolol is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Alprenolol is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Alprenolol is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when Alprenolol is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Alprenolol is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Alprenolol is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Alprenolol is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Alprenolol is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Alprenolol is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when Alprenolol is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when Alprenolol is combined with (S)-Warfarin.
Mirabegron The serum concentration of Alprenolol can be increased when it is combined with Mirabegron.
Molsidomine Molsidomine may increase the hypotensive activities of Alprenolol.
Insulin argine Alprenolol may increase the hypoglycemic activities of Insulin argine.
Remikiren Remikiren may increase the hypotensive activities of Alprenolol.
Guanadrel Guanadrel may increase the hypotensive activities of Alprenolol.
Bosentan Bosentan may increase the hypotensive activities of Alprenolol.
Candoxatril Candoxatril may increase the hypotensive activities of Alprenolol.
Cryptenamine Cryptenamine may increase the hypotensive activities of Alprenolol.
Dorzolamide Alprenolol may increase the hypotensive activities of Dorzolamide.
Bimatoprost Alprenolol may increase the hypotensive activities of Bimatoprost.
Pentolinium Alprenolol may increase the hypotensive activities of Pentolinium.
Trimethaphan Alprenolol may increase the hypotensive activities of Trimethaphan.

Target Protein

Beta-1 adrenergic receptor ADRB1
Beta-2 adrenergic receptor ADRB2
5-hydroxytryptamine receptor 1A HTR1A
Beta-3 adrenergic receptor ADRB3

Referensi & Sumber

Synthesis reference: http://www.google.com.mx/patents/US3466376
Artikel (PubMed)
  • PMID: 8586675
    Hold KM, de Boer D, Bos KL, van Ooijen RD, Zuidema J, Maes RA: Enantioselective quantitation of (R)- and (S)-alprenolol by gas chromatography-mass spectrometry in human saliva an plasma. J Chromatogr Sci. 1996 Jan;34(1):13-9.
  • PMID: 15525
    Himori N, Ishimori T, Izumi A, Hiramatsu Y: Effects of beta-adrenoceptor blocking agents, pindolol, alprenolol and practolol on blood pressure and heart rate in conscious renal hypertensive dogs. Arch Int Pharmacodyn Ther. 1977 Jan;225(1):152-65.

Contoh Produk & Brand

Produk: 0 • International brands: 10
International Brands
  • Apllobal — AstraZeneca
  • Aptin — AstraZeneca
  • Aptine
  • Aptol Duriles
  • Atenenol — Tsuruhara Seiyaku
  • Elp — Shyh Dar
  • Gubernal
  • Regletin
  • Skajilol — Kotobuki Seiyaku
  • Yobir

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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