Peringatan Keamanan

Symptoms of overdose include stupor or coma, and children may have convulsive seizures. Signs of arousal may not occur for 48 hours. Oral LD50=318 mg/kg (rat); IPR LD50=64 mg/kg (mouse)

Perphenazine

DB00850

small molecule approved

Deskripsi

An antipsychotic phenothiazine derivative with actions and uses similar to those of chlorpromazine.

Struktur Molekul 2D

Berat 403.969
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 8-12 hours, but ranges up to 20 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Absolute bioavailability is 40% following oral administration.

Metabolisme

Hepatic.

Rute Eliminasi

Perphenazine is extensively metabolized in the liver to a number of metabolites by sulfoxidation, hydroxylation, dealkylation, and glucuronidation.

Interaksi Makanan

1 Data
  • 1. Avoid alcohol. Consuming alcohol may increase hypotension. Perphenazine may increase the effects of alcohol.

Interaksi Obat

1213 Data
Deferasirox The serum concentration of Perphenazine can be increased when it is combined with Deferasirox.
Peginterferon alfa-2b The serum concentration of Perphenazine can be increased when it is combined with Peginterferon alfa-2b.
Leflunomide The serum concentration of Perphenazine can be decreased when it is combined with Leflunomide.
Teriflunomide The serum concentration of Perphenazine can be decreased when it is combined with Teriflunomide.
Buprenorphine Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Hydrocodone Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Magnesium sulfate The therapeutic efficacy of Perphenazine can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Mirtazapine Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Orphenadrine Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Rotigotine Perphenazine may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Perphenazine.
Sodium oxybate Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Thalidomide Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Amisulpride Perphenazine may increase the antipsychotic activities of Amisulpride.
Methylphenidate The risk or severity of adverse effects can be increased when Perphenazine is combined with Methylphenidate.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Perphenazine is combined with Dexmethylphenidate.
Metoclopramide The risk or severity of adverse effects can be increased when Metoclopramide is combined with Perphenazine.
Quinagolide The therapeutic efficacy of Quinagolide can be decreased when used in combination with Perphenazine.
Sulpiride Perphenazine may increase the antipsychotic activities of Sulpiride.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Perphenazine.
Lithium citrate Lithium citrate may increase the neurotoxic activities of Perphenazine.
Lithium hydroxide Lithium hydroxide may increase the neurotoxic activities of Perphenazine.
Mequitazine Perphenazine may increase the arrhythmogenic activities of Mequitazine.
Thiopental The risk or severity of adverse effects can be increased when Perphenazine is combined with Thiopental.
Atomoxetine The metabolism of Atomoxetine can be decreased when combined with Perphenazine.
Metyrosine The risk or severity of extrapyramidal symptoms and CNS depression can be increased when Metyrosine is combined with Perphenazine.
Mirabegron The serum concentration of Perphenazine can be increased when it is combined with Mirabegron.
Abiraterone The serum concentration of Perphenazine can be increased when it is combined with Abiraterone.
Cyproterone acetate The metabolism of Perphenazine can be increased when combined with Cyproterone acetate.
Ethanol Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Perphenazine may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Perphenazine.
Zimelidine The risk or severity of adverse effects can be increased when Perphenazine is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Perphenazine is combined with Dapoxetine.
Seproxetine The risk or severity of adverse effects can be increased when Perphenazine is combined with Seproxetine.
Citalopram The risk or severity of adverse effects can be increased when Perphenazine is combined with Citalopram.
Trazodone The risk or severity of adverse effects can be increased when Perphenazine is combined with Trazodone.
Sertraline The risk or severity of adverse effects can be increased when Perphenazine is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Perphenazine is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Perphenazine is combined with Nefazodone.
Milnacipran The risk or severity of adverse effects can be increased when Perphenazine is combined with Milnacipran.
Desvenlafaxine The serum concentration of Perphenazine can be increased when it is combined with Desvenlafaxine.
Levomilnacipran The risk or severity of adverse effects can be increased when Levomilnacipran is combined with Perphenazine.
Indalpine The risk or severity of adverse effects can be increased when Perphenazine is combined with Indalpine.
Alaproclate The risk or severity of adverse effects can be increased when Perphenazine is combined with Alaproclate.
Esmolol The serum concentration of Esmolol can be increased when it is combined with Perphenazine.
Betaxolol The serum concentration of Betaxolol can be increased when it is combined with Perphenazine.
Atenolol The serum concentration of Atenolol can be increased when it is combined with Perphenazine.
Propranolol The serum concentration of Propranolol can be increased when it is combined with Perphenazine.
Labetalol The serum concentration of Labetalol can be increased when it is combined with Perphenazine.
Bisoprolol The serum concentration of Bisoprolol can be increased when it is combined with Perphenazine.
Alprenolol The serum concentration of Alprenolol can be increased when it is combined with Perphenazine.
Pindolol The serum concentration of Pindolol can be increased when it is combined with Perphenazine.
Carvedilol The serum concentration of Carvedilol can be increased when it is combined with Perphenazine.
Acebutolol The serum concentration of Acebutolol can be increased when it is combined with Perphenazine.
Nadolol The serum concentration of Nadolol can be increased when it is combined with Perphenazine.
Bevantolol The serum concentration of Bevantolol can be increased when it is combined with Perphenazine.
Practolol The serum concentration of Practolol can be increased when it is combined with Perphenazine.
Penbutolol The serum concentration of Penbutolol can be increased when it is combined with Perphenazine.
Oxprenolol The serum concentration of Oxprenolol can be increased when it is combined with Perphenazine.
Dexpropranolol The serum concentration of Dexpropranolol can be increased when it is combined with Perphenazine.
Celiprolol The serum concentration of Celiprolol can be increased when it is combined with Perphenazine.
Nebivolol The serum concentration of Nebivolol can be increased when it is combined with Perphenazine.
Bufuralol The serum concentration of Bufuralol can be increased when it is combined with Perphenazine.
Bopindolol The serum concentration of Bopindolol can be increased when it is combined with Perphenazine.
Bupranolol The serum concentration of Bupranolol can be increased when it is combined with Perphenazine.
Indenolol The serum concentration of Indenolol can be increased when it is combined with Perphenazine.
Arotinolol The serum concentration of Arotinolol can be increased when it is combined with Perphenazine.
Levobetaxolol The serum concentration of Levobetaxolol can be increased when it is combined with Perphenazine.
Talinolol The serum concentration of Talinolol can be increased when it is combined with Perphenazine.
Anisodamine The serum concentration of Anisodamine can be increased when it is combined with Perphenazine.
Bucindolol The serum concentration of Bucindolol can be increased when it is combined with Perphenazine.
Esatenolol The serum concentration of Esatenolol can be increased when it is combined with Perphenazine.
Cloranolol The serum concentration of Cloranolol can be increased when it is combined with Perphenazine.
Mepindolol The serum concentration of Mepindolol can be increased when it is combined with Perphenazine.
Epanolol The serum concentration of Epanolol can be increased when it is combined with Perphenazine.
Tertatolol The serum concentration of Tertatolol can be increased when it is combined with Perphenazine.
Morphine The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Morphine.
Codeine The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Codeine.
Hydromorphone The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Hydromorphone.
Oxycodone The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Oxycodone.
Butorphanol The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Butorphanol.
Dextropropoxyphene The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Dextropropoxyphene.
Pentazocine The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Pentazocine.
Naltrexone The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Naltrexone.
Sufentanil The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Sufentanil.
Nalbuphine The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Nalbuphine.
Levorphanol The risk or severity of hypotension and CNS depression can be increased when Perphenazine is combined with Levorphanol.

Target Protein

D(2) dopamine receptor DRD2
D(1A) dopamine receptor DRD1
Calmodulin CALM1

Referensi & Sumber

Belum ada data referensi/link/attachment untuk obat ini pada database. Jalankan import DrugBank untuk mengisi field referensi.

Contoh Produk & Brand

Produk: 204 • International brands: 7
Produk
  • Apo Peram Tab 2-25
    Tablet • - • Oral • Canada • Generic • Approved
  • Apo Peram Tab 3-15
    Tablet • - • Oral • Canada • Generic • Approved
  • Elavil Plus Tab
    Tablet • - • Oral • Canada • Approved
  • Etrafon 2 10
    Tablet • - • Oral • Canada • Approved
  • Etrafon A Tab
    Tablet • - • Oral • Canada • Approved
  • Etrafon D Tab
    Tablet • - • Oral • Canada • Approved
  • Etrafon F Tab
    Tablet • - • Oral • Canada • Approved
  • Perphenazine
    Tablet, sugar coated • 2 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 204 produk.
International Brands
  • Decentan — Merck
  • Emesinal
  • Fentazin — Mercury
  • Perphenan — Taro
  • PZC — Tanabe Mitsubishi Pharma
  • Trilafon — Schering-Plough
  • Trilifan

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
© 2025 Digital Pharmacy Research - Universitas Esa Unggul