Peringatan Keamanan

Overdosage of sulfonylureas can produce hypoglycemia. Severe hypoglycemic reactions with coma, seizure, or other neurological impairment occur infrequently, but constitute medical emergencies requiring immediate hospitalization.

Tolazamide

DB00839

small molecule approved investigational

Deskripsi

A sulphonylurea hypoglycemic agent with actions and uses similar to those of chlorpropamide.

Struktur Molekul 2D

Berat 311.4
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) The average biological half-life of the drug is 7 hours.
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Rapidly and well absorbed from the gastrointestinal tract.

Metabolisme

Tolazamide is metabolized to five major metabolites ranging in hypoglycemic activity from 0 to 70%.

Rute Eliminasi

Tolazamide is metabolized to five major metabolites ranging in hypoglycemic activity from 0% to 70%. They are excreted principally in the urine.

Interaksi Makanan

2 Data
  • 1. Avoid excessive or chronic alcohol consumption. Ingesting alcohol may increase the risk of hypoglycemia.
  • 2. Take with food. Taking tolazamide with breakfast may help reduce the risk of hypoglycemia.

Interaksi Obat

1501 Data
Pegvisomant The risk or severity of hypoglycemia can be increased when Pegvisomant is combined with Tolazamide.
Carbocisteine The risk or severity of adverse effects can be increased when Tolazamide is combined with Carbocisteine.
Chloramphenicol The metabolism of Tolazamide can be decreased when combined with Chloramphenicol.
Cimetidine The serum concentration of Tolazamide can be increased when it is combined with Cimetidine.
Fluconazole The serum concentration of Tolazamide can be increased when it is combined with Fluconazole.
Metreleptin Metreleptin may increase the hypoglycemic activities of Tolazamide.
Probenecid The protein binding of Tolazamide can be decreased when combined with Probenecid.
Ranitidine The serum concentration of Tolazamide can be increased when it is combined with Ranitidine.
Voriconazole The serum concentration of Tolazamide can be increased when it is combined with Voriconazole.
Clarithromycin The serum concentration of Tolazamide can be increased when it is combined with Clarithromycin.
Lipoic acid The risk or severity of hypoglycemia can be increased when Lipoic acid is combined with Tolazamide.
Rifampin The serum concentration of Tolazamide can be decreased when it is combined with Rifampicin.
Moxifloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Moxifloxacin.
Grepafloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Grepafloxacin.
Enoxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Enoxacin.
Pefloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Pefloxacin.
Ciprofloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Ciprofloxacin.
Trovafloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Trovafloxacin.
Nalidixic acid The therapeutic efficacy of Tolazamide can be increased when used in combination with Nalidixic acid.
Rosoxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Rosoxacin.
Cinoxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Cinoxacin.
Lomefloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Lomefloxacin.
Gatifloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Gatifloxacin.
Norfloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Norfloxacin.
Levofloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Levofloxacin.
Gemifloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Gemifloxacin.
Ofloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Ofloxacin.
Sparfloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Sparfloxacin.
Temafloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Temafloxacin.
Fleroxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Fleroxacin.
Technetium Tc-99m ciprofloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Technetium Tc-99m ciprofloxacin.
Garenoxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Garenoxacin.
Nemonoxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Nemonoxacin.
Flumequine The therapeutic efficacy of Tolazamide can be increased when used in combination with Flumequine.
Enrofloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Enrofloxacin.
Orbifloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Orbifloxacin.
Sarafloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Sarafloxacin.
Difloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Difloxacin.
Pazufloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Pazufloxacin.
Prulifloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Prulifloxacin.
Delafloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Delafloxacin.
Sitafloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Sitafloxacin.
Oxolinic acid The therapeutic efficacy of Tolazamide can be increased when used in combination with Oxolinic acid.
Rufloxacin The therapeutic efficacy of Tolazamide can be increased when used in combination with Rufloxacin.
Pipemidic acid The therapeutic efficacy of Tolazamide can be increased when used in combination with Pipemidic acid.
Methyclothiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Methyclothiazide.
Chlorthalidone The therapeutic efficacy of Tolazamide can be decreased when used in combination with Chlorthalidone.
Bendroflumethiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Bendroflumethiazide.
Metolazone The therapeutic efficacy of Tolazamide can be decreased when used in combination with Metolazone.
Benzthiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Benzthiazide.
Hydroflumethiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Hydroflumethiazide.
Indapamide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Indapamide.
Chlorothiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Chlorothiazide.
Hydrochlorothiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Hydrochlorothiazide.
Trichlormethiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Trichlormethiazide.
Polythiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Polythiazide.
Quinethazone The therapeutic efficacy of Tolazamide can be decreased when used in combination with Quinethazone.
Cyclopenthiazide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Cyclopenthiazide.
Epitizide The therapeutic efficacy of Tolazamide can be decreased when used in combination with Epitizide.
Esmolol Esmolol may increase the hypoglycemic activities of Tolazamide.
Landiolol Landiolol may increase the hypoglycemic activities of Tolazamide.
Ethanol The risk or severity of adverse effects can be increased when Tolazamide is combined with Ethanol.
Protriptyline Protriptyline may decrease the hypoglycemic activities of Tolazamide.
Nortriptyline Nortriptyline may decrease the hypoglycemic activities of Tolazamide.
Amoxapine Amoxapine may decrease the hypoglycemic activities of Tolazamide.
Amineptine Amineptine may decrease the hypoglycemic activities of Tolazamide.
Butriptyline Butriptyline may decrease the hypoglycemic activities of Tolazamide.
Dosulepin Dosulepin may decrease the hypoglycemic activities of Tolazamide.
Tianeptine Tianeptine may decrease the hypoglycemic activities of Tolazamide.
Oxaprotiline Oxaprotiline may decrease the hypoglycemic activities of Tolazamide.
Opipramol Opipramol may decrease the hypoglycemic activities of Tolazamide.
Amitriptylinoxide Amitriptylinoxide may decrease the hypoglycemic activities of Tolazamide.
Dibenzepin Dibenzepin may decrease the hypoglycemic activities of Tolazamide.
Quinupramine Quinupramine may decrease the hypoglycemic activities of Tolazamide.
Melitracen Melitracen may decrease the hypoglycemic activities of Tolazamide.
Lofepramine Lofepramine may decrease the hypoglycemic activities of Tolazamide.
Iprindole Iprindole may decrease the hypoglycemic activities of Tolazamide.
Imipramine oxide Imipramine oxide may decrease the hypoglycemic activities of Tolazamide.
Amitriptyline Amitriptyline may decrease the hypoglycemic activities of Tolazamide.
Doxepin Doxepin may decrease the hypoglycemic activities of Tolazamide.
Imipramine Imipramine may decrease the hypoglycemic activities of Tolazamide.
Desipramine Desipramine may decrease the hypoglycemic activities of Tolazamide.
Clomipramine Clomipramine may decrease the hypoglycemic activities of Tolazamide.
Dimetacrine Dimetacrine may decrease the hypoglycemic activities of Tolazamide.
Clofibrate The risk or severity of hypoglycemia can be increased when Clofibrate is combined with Tolazamide.
Fenofibrate The risk or severity of hypoglycemia can be increased when Fenofibrate is combined with Tolazamide.
Bezafibrate The risk or severity of hypoglycemia can be increased when Bezafibrate is combined with Tolazamide.
Etofibrate The risk or severity of hypoglycemia can be increased when Etofibrate is combined with Tolazamide.
Ciprofibrate The risk or severity of hypoglycemia can be increased when Ciprofibrate is combined with Tolazamide.
Simfibrate The risk or severity of hypoglycemia can be increased when Simfibrate is combined with Tolazamide.
Ronifibrate The risk or severity of hypoglycemia can be increased when Ronifibrate is combined with Tolazamide.
Aluminium clofibrate The risk or severity of hypoglycemia can be increased when Aluminium clofibrate is combined with Tolazamide.
Clofibride The risk or severity of hypoglycemia can be increased when Clofibride is combined with Tolazamide.
Fenofibric acid The risk or severity of hypoglycemia can be increased when Fenofibric acid is combined with Tolazamide.
Miconazole The serum concentration of Tolazamide can be increased when it is combined with Miconazole.
Phenindione Tolazamide may increase the anticoagulant activities of Phenindione.
Coumarin Tolazamide may increase the anticoagulant activities of Coumarin.
(R)-warfarin Tolazamide may increase the anticoagulant activities of (R)-warfarin.
Clorindione Tolazamide may increase the anticoagulant activities of Clorindione.
Diphenadione Tolazamide may increase the anticoagulant activities of Diphenadione.

Target Protein

Sulfonylurea receptor 1, Kir6.2 ABCC8
ATP-sensitive inward rectifier potassium channel 10 KCNJ10

Referensi & Sumber

Artikel (PubMed)
  • PMID: 8237731
    Tal A: Oral hypoglycemic agents in the treatment of type II diabetes. Am Fam Physician. 1993 Nov 1;48(6):1089-95.
  • PMID: 15901207
    Granberry MC, Fonseca VA: Cardiovascular risk factors associated with insulin resistance: effects of oral antidiabetic agents. Am J Cardiovasc Drugs. 2005;5(3):201-9.

Contoh Produk & Brand

Produk: 11 • International brands: 5
Produk
  • Tolazamide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Tolazamide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Tolazamide
    Tablet • 100 mg/1 • Oral • US • Approved
  • Tolazamide
    Tablet • 250 mg/1 • Oral • US • Approved
  • Tolazamide
    Tablet • 500 mg/1 • Oral • US • Approved
  • Tolazamide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Tolazamide
    Tablet • 500 mg/1 • Oral • US • Generic • Approved
  • Tolazamide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 11 produk.
International Brands
  • Desumide — Hua Shin
  • Diabewas
  • Esulin — Chung Mei
  • Norglycin — Pfizer
  • Tolanase — Upjohn

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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