Progabide

DB00837

small molecule experimental

Deskripsi

Progabide is an analog and prodrug of gamma-aminobutyric acid. It is commonly used in the treatment of epilepsy. It has agonistic activity for both the GABAA and GABAB receptors. In clinical trials, progabide has been investigated for Parkinson's disease, schizophrenia, clinical depression and anxiety disorder; its therapeutic effectiveness in these conditions is not fully elucidated.

Struktur Molekul 2D

Berat 334.78
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 4 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Well absorbed with a bioavailability of 60%

Metabolisme

Hepatic

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Obat

824 Data
Buprenorphine Progabide may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Dronabinol Dronabinol may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Hydrocodone Progabide may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Magnesium sulfate The therapeutic efficacy of Progabide can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Progabide may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Progabide may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Mirtazapine Progabide may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Orphenadrine Progabide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Progabide may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Pramipexole Progabide may increase the sedative activities of Pramipexole.
Ropinirole Progabide may increase the sedative activities of Ropinirole.
Rotigotine Progabide may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Progabide.
Sodium oxybate Progabide may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Progabide may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Thalidomide Progabide may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Progabide may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Mefloquine The therapeutic efficacy of Progabide can be decreased when used in combination with Mefloquine.
Mianserin The therapeutic efficacy of Progabide can be decreased when used in combination with Mianserin.
Orlistat Orlistat can cause a decrease in the absorption of Progabide resulting in a reduced serum concentration and potentially a decrease in efficacy.
Topotecan Progabide may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Methylphenidate The risk or severity of adverse effects can be increased when Methylphenidate is combined with Progabide.
Dexmethylphenidate The risk or severity of adverse effects can be increased when Dexmethylphenidate is combined with Progabide.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Progabide.
Dicoumarol The risk or severity of adverse effects can be increased when Progabide is combined with Dicoumarol.
Phenindione The risk or severity of adverse effects can be increased when Progabide is combined with Phenindione.
Warfarin The risk or severity of adverse effects can be increased when Progabide is combined with Warfarin.
Phenprocoumon The risk or severity of adverse effects can be increased when Progabide is combined with Phenprocoumon.
Acenocoumarol The risk or severity of adverse effects can be increased when Progabide is combined with Acenocoumarol.
4-hydroxycoumarin The risk or severity of adverse effects can be increased when Progabide is combined with 4-hydroxycoumarin.
Coumarin The risk or severity of adverse effects can be increased when Progabide is combined with Coumarin.
(R)-warfarin The risk or severity of adverse effects can be increased when Progabide is combined with (R)-warfarin.
Ethyl biscoumacetate The risk or severity of adverse effects can be increased when Progabide is combined with Ethyl biscoumacetate.
Fluindione The risk or severity of adverse effects can be increased when Progabide is combined with Fluindione.
Clorindione The risk or severity of adverse effects can be increased when Progabide is combined with Clorindione.
Diphenadione The risk or severity of adverse effects can be increased when Progabide is combined with Diphenadione.
Tioclomarol The risk or severity of adverse effects can be increased when Progabide is combined with Tioclomarol.
(S)-Warfarin The risk or severity of adverse effects can be increased when Progabide is combined with (S)-Warfarin.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Progabide.
Ethanol Progabide may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Progabide may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Zimelidine The risk or severity of adverse effects can be increased when Progabide is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Progabide is combined with Dapoxetine.
Seproxetine The risk or severity of adverse effects can be increased when Progabide is combined with Seproxetine.
Fluvoxamine The risk or severity of adverse effects can be increased when Progabide is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Progabide is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Progabide is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Progabide is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Progabide is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Progabide is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Progabide is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Progabide is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Progabide is combined with Escitalopram.
Milnacipran The risk or severity of adverse effects can be increased when Progabide is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Progabide is combined with Desvenlafaxine.
Levomilnacipran The risk or severity of adverse effects can be increased when Progabide is combined with Levomilnacipran.
Indalpine The risk or severity of adverse effects can be increased when Progabide is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Progabide is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Progabide is combined with Alaproclate.
Bifeprunox The therapeutic efficacy of Progabide can be decreased when used in combination with Bifeprunox.
Lumateperone The therapeutic efficacy of Progabide can be decreased when used in combination with Lumateperone.
Brexpiprazole The therapeutic efficacy of Progabide can be decreased when used in combination with Brexpiprazole.
Blonanserin The therapeutic efficacy of Progabide can be decreased when used in combination with Blonanserin.
Periciazine The therapeutic efficacy of Progabide can be decreased when used in combination with Periciazine.
Thioproperazine The therapeutic efficacy of Progabide can be decreased when used in combination with Thioproperazine.
Loxapine The therapeutic efficacy of Progabide can be decreased when used in combination with Loxapine.
Promazine The therapeutic efficacy of Progabide can be decreased when used in combination with Promazine.
Prochlorperazine The therapeutic efficacy of Progabide can be decreased when used in combination with Prochlorperazine.
Chlorpromazine The therapeutic efficacy of Progabide can be decreased when used in combination with Chlorpromazine.
Fluphenazine The therapeutic efficacy of Progabide can be decreased when used in combination with Fluphenazine.
Thioridazine The therapeutic efficacy of Progabide can be decreased when used in combination with Thioridazine.
Trifluoperazine The therapeutic efficacy of Progabide can be decreased when used in combination with Trifluoperazine.
Perphenazine The therapeutic efficacy of Progabide can be decreased when used in combination with Perphenazine.
Mesoridazine The therapeutic efficacy of Progabide can be decreased when used in combination with Mesoridazine.
Pimozide The therapeutic efficacy of Progabide can be decreased when used in combination with Pimozide.
Chlorprothixene The therapeutic efficacy of Progabide can be decreased when used in combination with Chlorprothixene.
Molindone The therapeutic efficacy of Progabide can be decreased when used in combination with Molindone.
Thiothixene The therapeutic efficacy of Progabide can be decreased when used in combination with Thiothixene.
Zuclopenthixol The therapeutic efficacy of Progabide can be decreased when used in combination with Zuclopenthixol.
Azaperone The therapeutic efficacy of Progabide can be decreased when used in combination with Azaperone.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Progabide.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Progabide.
Cocaine The risk or severity of methemoglobinemia can be increased when Progabide is combined with Cocaine.
Quinidine The therapeutic efficacy of Progabide can be decreased when used in combination with Quinidine.
Zopiclone The risk or severity of adverse effects can be increased when Progabide is combined with Zopiclone.
Botulinum toxin type B The risk or severity of CNS depression can be increased when Botulinum toxin type B is combined with Progabide.
Botulinum toxin type A The risk or severity of CNS depression can be increased when Botulinum toxin type A is combined with Progabide.
Baclofen Baclofen may increase the central nervous system depressant (CNS depressant) activities of Progabide.
Ethchlorvynol The risk or severity of CNS depression can be increased when Ethchlorvynol is combined with Progabide.
Succinylcholine The risk or severity of CNS depression can be increased when Succinylcholine is combined with Progabide.
Eletriptan The risk or severity of CNS depression can be increased when Eletriptan is combined with Progabide.
Enflurane The risk or severity of CNS depression can be increased when Enflurane is combined with Progabide.

Target Protein

Gamma-aminobutyric acid type B receptor subunit 2 GABBR2
Gamma-aminobutyric acid receptor subunit alpha-1 GABRA1
Gamma-aminobutyric acid type B receptor subunit 1 GABBR1

Referensi & Sumber

Artikel (PubMed)
  • PMID: 3030072
    Bartholini G, Scatton B, Zivkovic B, Lloyd KG: GABA receptor agonists and extrapyramidal motor function: therapeutic implications for Parkinson's disease. Adv Neurol. 1987;45:79-83.

Contoh Produk & Brand

Produk: 0 • International brands: 2
International Brands
  • Gabren
  • Gabrene — Sanofi S.A.

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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