Acetazolamide

DB00819

small molecule approved vet_approved

Deskripsi

One of the carbonic anhydrase inhibitors that is sometimes effective against absence seizures. It is sometimes useful also as an adjunct in the treatment of tonic-clonic, myoclonic, and atonic seizures, particularly in women whose seizures occur or are exacerbated at specific times in the menstrual cycle. However, its usefulness is transient often because of rapid development of tolerance. Its antiepileptic effect may be due to its inhibitory effect on brain carbonic anhydrase, which leads to an increased transneuronal chloride gradient, increased chloride current, and increased inhibition. (From Smith and Reynard, Textbook of Pharmacology, 1991, p337)

Struktur Molekul 2D

Berat 222.245
Wujud solid

Peta Jejaring Molekuler
Legenda: ObatTargetGenEnzim(Panah → menunjukkan arah efek / relasi)TransporterCarrier

Profil Farmakokinetik

Waktu Paruh (Half-Life) 3 to 9 hours
Volume Distribusi -
Klirens (Clearance) -

Absorpsi

Data absorpsi tidak tersedia.

Metabolisme

Data metabolisme tidak tersedia.

Rute Eliminasi

Data eliminasi belum tersedia.

Interaksi Makanan

2 Data
  • 1. Drink plenty of fluids.
  • 2. Take with food. Take at least 6 hours before bedtime.

Interaksi Obat

1547 Data
Cyclosporine The serum concentration of Cyclosporine can be increased when it is combined with Acetazolamide.
Buprenorphine Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Buprenorphine.
Doxylamine Doxylamine may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Dronabinol The serum concentration of Dronabinol can be increased when it is combined with Acetazolamide.
Droperidol Droperidol may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Hydrocodone Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Hydrocodone.
Hydroxyzine Hydroxyzine may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Magnesium sulfate The therapeutic efficacy of Acetazolamide can be increased when used in combination with Magnesium sulfate.
Methotrimeprazine Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Methotrimeprazine.
Metyrosine Acetazolamide may increase the sedative activities of Metyrosine.
Minocycline Minocycline may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Mirtazapine Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Mirtazapine.
Nabilone Nabilone may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Orphenadrine Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Orphenadrine.
Paraldehyde Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Paraldehyde.
Perampanel Perampanel may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Pramipexole Acetazolamide may increase the sedative activities of Pramipexole.
Ropinirole Acetazolamide may increase the sedative activities of Ropinirole.
Rotigotine Acetazolamide may increase the sedative activities of Rotigotine.
Rufinamide The risk or severity of adverse effects can be increased when Rufinamide is combined with Acetazolamide.
Sodium oxybate Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Sodium oxybate.
Suvorexant Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Suvorexant.
Tapentadol Tapentadol may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Thalidomide Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Thalidomide.
Zolpidem Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Zolpidem.
Eliglustat The metabolism of Eliglustat can be decreased when combined with Acetazolamide.
Ibrutinib The metabolism of Ibrutinib can be decreased when combined with Acetazolamide.
Nicotine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Nicotine.
Mecamylamine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Mecamylamine.
Pentolinium The risk or severity of adverse effects can be increased when Acetazolamide is combined with Pentolinium.
Trimethaphan The risk or severity of adverse effects can be increased when Acetazolamide is combined with Trimethaphan.
Hexamethonium The risk or severity of adverse effects can be increased when Acetazolamide is combined with Hexamethonium.
Cyclopentamine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Cyclopentamine.
Cilostazol The metabolism of Cilostazol can be decreased when combined with Acetazolamide.
Colchicine The metabolism of Colchicine can be decreased when combined with Acetazolamide.
Fentanyl The risk or severity of CNS depression can be increased when Fentanyl is combined with Acetazolamide.
Iloperidone The metabolism of Iloperidone can be decreased when combined with Acetazolamide.
Retapamulin The metabolism of Retapamulin can be decreased when combined with Acetazolamide.
Tofacitinib The metabolism of Tofacitinib can be decreased when combined with Acetazolamide.
Vardenafil The metabolism of Vardenafil can be decreased when combined with Acetazolamide.
Zopiclone The metabolism of Zopiclone can be decreased when combined with Acetazolamide.
Lovastatin The metabolism of Lovastatin can be decreased when combined with Acetazolamide.
Mefloquine The therapeutic efficacy of Acetazolamide can be decreased when used in combination with Mefloquine.
Mianserin The therapeutic efficacy of Acetazolamide can be decreased when used in combination with Mianserin.
Orlistat Orlistat can cause a decrease in the absorption of Acetazolamide resulting in a reduced serum concentration and potentially a decrease in efficacy.
Topotecan Acetazolamide may increase the excretion rate of Topotecan which could result in a lower serum level and potentially a reduction in efficacy.
Flecainide The excretion of Flecainide can be decreased when combined with Acetazolamide.
Memantine The excretion of Memantine can be decreased when combined with Acetazolamide.
Methylphenobarbital The serum concentration of Methylphenobarbital can be decreased when it is combined with Acetazolamide.
Phenobarbital The serum concentration of Phenobarbital can be decreased when it is combined with Acetazolamide.
Quinine The excretion of Quinine can be decreased when combined with Acetazolamide.
Methadone The risk or severity of adverse effects can be increased when Methadone is combined with Acetazolamide.
Alfuzosin The metabolism of Alfuzosin can be decreased when combined with Acetazolamide.
Methotrexate The therapeutic efficacy of Methotrexate can be increased when used in combination with Acetazolamide.
Alprazolam The metabolism of Alprazolam can be decreased when combined with Acetazolamide.
Warfarin The serum concentration of Warfarin can be increased when it is combined with Acetazolamide.
Acenocoumarol The serum concentration of Acenocoumarol can be increased when it is combined with Acetazolamide.
(R)-warfarin The serum concentration of (R)-warfarin can be increased when it is combined with Acetazolamide.
R,S-Warfarin alcohol The serum concentration of R,S-Warfarin alcohol can be increased when it is combined with Acetazolamide.
S,R-Warfarin alcohol The serum concentration of S,R-Warfarin alcohol can be increased when it is combined with Acetazolamide.
(S)-Warfarin The serum concentration of (S)-Warfarin can be increased when it is combined with Acetazolamide.
Midazolam The serum concentration of Midazolam can be increased when it is combined with Acetazolamide.
Carbamazepine The serum concentration of Carbamazepine can be increased when it is combined with Acetazolamide.
Metformin The risk or severity of lactic acidosis can be increased when Acetazolamide is combined with Metformin.
Tetracosactide The risk or severity of liver damage can be increased when Tetracosactide is combined with Acetazolamide.
Sodium bicarbonate The risk or severity of adverse effects can be increased when Acetazolamide is combined with Sodium bicarbonate.
Tacrolimus The serum concentration of Tacrolimus can be increased when it is combined with Acetazolamide.
Atorvastatin The metabolism of Atorvastatin can be decreased when combined with Acetazolamide.
Ethanol Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Ethanol.
Azelastine Acetazolamide may increase the central nervous system depressant (CNS depressant) activities of Azelastine.
Brimonidine Brimonidine may increase the central nervous system depressant (CNS depressant) activities of Acetazolamide.
Fluvoxamine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Fluvoxamine.
Citalopram The risk or severity of adverse effects can be increased when Acetazolamide is combined with Citalopram.
Duloxetine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Duloxetine.
Trazodone The risk or severity of adverse effects can be increased when Acetazolamide is combined with Trazodone.
Paroxetine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Paroxetine.
Sertraline The risk or severity of adverse effects can be increased when Acetazolamide is combined with Sertraline.
Sibutramine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Sibutramine.
Nefazodone The risk or severity of adverse effects can be increased when Acetazolamide is combined with Nefazodone.
Escitalopram The risk or severity of adverse effects can be increased when Acetazolamide is combined with Escitalopram.
Zimelidine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Zimelidine.
Dapoxetine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Dapoxetine.
Milnacipran The risk or severity of adverse effects can be increased when Acetazolamide is combined with Milnacipran.
Desvenlafaxine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Desvenlafaxine.
Seproxetine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Seproxetine.
Levomilnacipran Acetazolamide may increase the excretion rate of Levomilnacipran which could result in a lower serum level and potentially a reduction in efficacy.
Indalpine The risk or severity of adverse effects can be increased when Acetazolamide is combined with Indalpine.
Ritanserin The risk or severity of adverse effects can be increased when Acetazolamide is combined with Ritanserin.
Alaproclate The risk or severity of adverse effects can be increased when Acetazolamide is combined with Alaproclate.
Dexketoprofen The risk or severity of adverse effects can be increased when Dexketoprofen is combined with Acetazolamide.
Ketoprofen The risk or severity of adverse effects can be increased when Ketoprofen is combined with Acetazolamide.
Triethylenetetramine The excretion of Triethylenetetramine can be increased when combined with Acetazolamide.
Benzatropine Acetazolamide may increase the excretion rate of Benzatropine which could result in a lower serum level and potentially a reduction in efficacy.
Cyproheptadine The risk or severity of CNS depression can be increased when Cyproheptadine is combined with Acetazolamide.
Amoxapine The risk or severity of CNS depression can be increased when Amoxapine is combined with Acetazolamide.
Propiomazine The risk or severity of CNS depression can be increased when Propiomazine is combined with Acetazolamide.
Propantheline Acetazolamide may increase the excretion rate of Propantheline which could result in a lower serum level and potentially a reduction in efficacy.
Dicyclomine Acetazolamide may increase the excretion rate of Dicyclomine which could result in a lower serum level and potentially a reduction in efficacy.
Maprotiline The risk or severity of CNS depression can be increased when Acetazolamide is combined with Maprotiline.
Flavoxate Acetazolamide may increase the excretion rate of Flavoxate which could result in a lower serum level and potentially a reduction in efficacy.

Target Protein

Carbonic anhydrase 1 CA1
Carbonic anhydrase 2 CA2
Carbonic anhydrase 4 CA4
Carbonic anhydrase 12 CA12
Carbonic anhydrase 14 CA14
Carbonic anhydrase 3 CA3
Carbonic anhydrase 7 CA7
Aquaporin-1 AQP1

Referensi & Sumber

Synthesis reference: Angela C. Potts, Mark Gibson, "Stable ophthalmic preparations containing acetazolamide." U.S. Patent US4888168, issued August, 1981.

Contoh Produk & Brand

Produk: 128 • International brands: 28
Produk
  • Acetazolam
    Tablet • 250 mg • Oral • Canada • Approved
  • AcetaZOLAMIDE
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • AcetaZOLAMIDE
    Tablet • 250 1/1 • Oral • US • Generic • Approved
  • Acetazolamide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Acetazolamide
    Tablet • 125 mg/1 • Oral • US • Generic • Approved
  • Acetazolamide
    Tablet • 125 mg/1 • Oral • US • Generic • Approved
  • Acetazolamide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
  • Acetazolamide
    Tablet • 250 mg/1 • Oral • US • Generic • Approved
Menampilkan 8 dari 128 produk.
International Brands
  • Acemit — Medphano
  • Acemox — Acme
  • Acetak — Akorn
  • Acetamide — Micro Vision
  • Acetazolamax — Pfoshen
  • Azm — Ethical
  • Azol — New Chemical
  • Azomid — Adcock Ingram Pharmaceuticals
  • Carbinib — Edol
  • Défiltran — CSP

Sekuens Gen/Protein (FASTA)

Sekuens dimuat saat dibutuhkan agar halaman tetap ringan.
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